Academic Journal
Bioisosteric Discovery of NPA101.3, a Second-Generation RET/VEGFR2 Inhibitor Optimized for Single-Agent Polypharmacology
العنوان: | Bioisosteric Discovery of NPA101.3, a Second-Generation RET/VEGFR2 Inhibitor Optimized for Single-Agent Polypharmacology |
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المؤلفون: | Moccia, Marialuisa, Frett, Brendan, Zhang, Lingtian, Lakkaniga, Naga Rajiv, Briggs, David C., Chauhan, Rakhee, Brescia, Annalisa, Federico, Giorgia, Yan, Wei, Santoro, Massimo, McDonald, Neil Q., Li, Hong-yu, Carlomagno, Francesca |
المساهمون: | National Cancer Institute, European Commission, Ministero dell?Istruzione, dell?Universit? e della Ricerca, Associazione Italiana per la Ricerca sul Cancro, University of Arkansas for Medical Sciences, Wellcome Trust, American Thyroid Association, National Institute of General Medical Sciences, Regione Campania, Cancer Research UK, Association for Multiple Endocrine Neoplasia Disorders |
المصدر: | Journal of Medicinal Chemistry ; volume 63, issue 9, page 4506-4516 ; ISSN 0022-2623 1520-4804 |
بيانات النشر: | American Chemical Society (ACS) |
سنة النشر: | 2020 |
نوع الوثيقة: | article in journal/newspaper |
اللغة: | English |
DOI: | 10.1021/acs.jmedchem.9b01336 |
الاتاحة: | http://dx.doi.org/10.1021/acs.jmedchem.9b01336 http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b01336 https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b01336 |
Rights: | https://creativecommons.org/licenses/by/4.0/ |
رقم الانضمام: | edsbas.D648ADC2 |
قاعدة البيانات: | BASE |
DOI: | 10.1021/acs.jmedchem.9b01336 |
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