Strategic Application and Transformation of ortho-Disubstituted Phenyl and Cyclopropyl Ketones To Expand the Scope of Hydrogen Borrowing Catalysis

التفاصيل البيبلوغرافية
العنوان: Strategic Application and Transformation of ortho-Disubstituted Phenyl and Cyclopropyl Ketones To Expand the Scope of Hydrogen Borrowing Catalysis
المؤلفون: James R, Frost, Choon Boon, Cheong, Wasim M, Akhtar, Dimitri F J, Caputo, Neil G, Stevenson, Timothy J, Donohoe
المصدر: Journal of the American Chemical Society. 137(50)
سنة النشر: 2015
الوصف: The application of an iridium-catalyzed hydrogen borrowing process to enable the formation of α-branched ketones with higher alcohols is described. In order to facilitate this reaction, ortho-disubstituted phenyl and cyclopropyl ketones were recognized as crucial structural motifs for C-C bond formation. Having optimized the key catalysis step, the ortho-disubstituted phenyl products could be further manipulated by a retro-Friedel-Crafts acylation reaction to produce synthetically useful carboxylic acid derivatives. In contrast, the cyclopropyl ketones underwent homoconjugate addition with several nucleophiles to provide further functionalized branched ketone products.
تدمد: 1520-5126
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::7ab89d93b59f0ede63110edb53120dd8
https://pubmed.ncbi.nlm.nih.gov/26654947
رقم الانضمام: edsair.pmid..........7ab89d93b59f0ede63110edb53120dd8
قاعدة البيانات: OpenAIRE