Co-relationship of physical stability of amorphous dispersions with enthalpy relaxation

التفاصيل البيبلوغرافية
العنوان: Co-relationship of physical stability of amorphous dispersions with enthalpy relaxation
المؤلفون: S S, Bansal, A M, Kaushal, A K, Bansal
المصدر: Die Pharmazie. 63(11)
سنة النشر: 2008
مصطلحات موضوعية: Sulfonamides, Calorimetry, Differential Scanning, Cyclooxygenase 2 Inhibitors, Drug Stability, Drug Storage, Pharmaceutic Aids, Temperature, Povidone, Thermodynamics, Isoxazoles, Crystallization, Algorithms
الوصف: Physical stability studies of valdecoxib (VLB) and its solid dispersions with PVP (1, 2, 5, 10, 15 and 20% w/w) were carried out by Differential Scanning Calorimetry (DSC). Change in specific heat with time was measured to determine the degree of crystallinity of amorphous drug and its binary dispersions after storage at 40 degrees C and 75% RH. The rate of crystallization was found to decrease with increasing PVP concentration and time for 10% crystallization (t90%) was found to increase significantly for the amorphous drug when formulated as PVP dispersions. Enthalpy relaxation was found to be inversely correlated with t90% (min) values and was found to be a good predictor of devitrification tendency and hence stability of amorphous VLB.
تدمد: 0031-7144
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::422017dafe8a9d993a50ba48ad252cc2
https://pubmed.ncbi.nlm.nih.gov/19069241
رقم الانضمام: edsair.pmid..........422017dafe8a9d993a50ba48ad252cc2
قاعدة البيانات: OpenAIRE