Nocarbenzoxazoles A-G, Benzoxazoles Produced by Halophilic Nocardiopsis lucentensis DSM 44048

التفاصيل البيبلوغرافية
العنوان: Nocarbenzoxazoles A-G, Benzoxazoles Produced by Halophilic Nocardiopsis lucentensis DSM 44048
المؤلفون: Huilin Hao, Xiaomei Zhang, Wen-Jun Li, Chunhua Lu, Mingwei Sun
المصدر: Journal of natural products. 78(8)
سنة النشر: 2015
مصطلحات موضوعية: Staphylococcus aureus, Stereochemistry, Nocardiopsis lucentensis, Mycobacterium smegmatis, Pharmaceutical Science, Antineoplastic Agents, Bacillus subtilis, Microbial Sensitivity Tests, Nocardia, Analytical Chemistry, HeLa, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, Candida albicans, Humans, Cytotoxicity, Nuclear Magnetic Resonance, Biomolecular, Pharmacology, Benzoxazoles, Strain (chemistry), biology, Molecular Structure, Organic Chemistry, Hep G2 Cells, Benzoxazole, biology.organism_classification, Halophile, Anti-Bacterial Agents, Complementary and alternative medicine, chemistry, Biochemistry, Pseudomonas aeruginosa, Molecular Medicine, Drug Screening Assays, Antitumor, Two-dimensional nuclear magnetic resonance spectroscopy, Algorithms, HeLa Cells
الوصف: Seven new benzoxazole derivatives, nocarbenzoxazoles A–G (1–7), were isolated from the halophilic strain Nocardiopsis lucentensis DSM 44048. Their structures were elucidated on the basis of 1D and 2D NMR spectroscopic data, HRESIMS, and X-ray single-crystal diffraction. The isolated compounds were assayed for their cytotoxicity against a panel of human tumor cell lines (HepG2, MDA-MB-231, MDA-MB-435, HeLa, and PC3). Compounds 1–6 were found to have modest or no activity. Compound 7 showed selective activity against HepG2 and HeLa with IC50 values of 3 and 1 μM, respectively.
تدمد: 1520-6025
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d561765dcfda7de56af7c43020632af4
https://pubmed.ncbi.nlm.nih.gov/26270803
رقم الانضمام: edsair.doi.dedup.....d561765dcfda7de56af7c43020632af4
قاعدة البيانات: OpenAIRE