Topical doxycycline monohydrate hydrogel 1% targeting proteases/PAR2 pathway is a novel therapeutic for atopic dermatitis

التفاصيل البيبلوغرافية
العنوان: Topical doxycycline monohydrate hydrogel 1% targeting proteases/PAR2 pathway is a novel therapeutic for atopic dermatitis
المؤلفون: Daniel J. Gibson, Gregory S. Schultz, Anna De Benedetto, Judy Talton, Mingjin Liu, Susmita Datta, James Talton, Mary Bohannon, Peter E. Nadeau
المصدر: Exp Dermatol
سنة النشر: 2020
مصطلحات موضوعية: 0301 basic medicine, Adult, Male, Proteases, Inflammation, Dermatology, Pharmacology, Administration, Cutaneous, Biochemistry, Proof of Concept Study, Severity of Illness Index, Article, Dermatitis, Atopic, 030207 dermatology & venereal diseases, 03 medical and health sciences, Young Adult, 0302 clinical medicine, Immune system, Skin Physiological Phenomena, medicine, Humans, Receptor, PAR-2, Protease Inhibitors, Adverse effect, Molecular Biology, Aged, Doxycycline, business.industry, Pruritus, KLK5, Hydrogels, Atopic dermatitis, Middle Aged, medicine.disease, Clinical trial, 030104 developmental biology, Female, medicine.symptom, business, medicine.drug
الوصف: Atopic Dermatitis (AD) is characterized by skin barrier disruption and an aberrant immune response. Doxycycline are tetracycline antibiotics broadly used systemically to treat inflammatory-dermatologic conditions. Several studies have shown doxycycline have anti-inflammatory and pro-healing properties, mainly by blocking tissue proteolytic activity. It is our hypothesis that daily application of a novel Doxycycline topical formulation in AD subjects will reduce severity of the disease, by blocking cutaneous proteases activity and restoring skin barrier function and inflammation. To test this hypotehsis we performed a proof of concept, open-label clinical study. Subjects enrolled in the study (n=15) applied NanoDOX® Hydrogel 1% daily for four weeks on a chosen eczematous area. Investigational drug was well tolerated, no local or systemic adverse events due to investigational drug were reported. Notably, a significant clinical improvement was observed based on a modified Eczema Area & Severity Index (EASI) score of the treated area from start of treatment to 14 and 28 days post treatment (p
تدمد: 1600-0625
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6395a4472419dc6d6ebf2f5efd495eea
https://pubmed.ncbi.nlm.nih.gov/32997843
Rights: OPEN
رقم الانضمام: edsair.doi.dedup.....6395a4472419dc6d6ebf2f5efd495eea
قاعدة البيانات: OpenAIRE