Crystallinity, hygroscopicity and dissolution of moricizine hydrochloride hemihydrate

التفاصيل البيبلوغرافية
العنوان: Crystallinity, hygroscopicity and dissolution of moricizine hydrochloride hemihydrate
المؤلفون: Lei-Shu Wu, Christopher A. Koval, Christine Gerard, Munir A. Hussain, Susan M. Rowe
المصدر: Journal of pharmaceutical and biomedical analysis. 12(8)
سنة النشر: 1994
مصطلحات موضوعية: Thermogravimetric analysis, Calorimetry, Differential Scanning, Chemistry, Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Pharmaceutical Science, Humidity, Moricizine, Analytical Chemistry, Granulation, Crystallinity, Moricizine Hydrochloride, Polymorphism (materials science), Solubility, X-Ray Diffraction, Drug Discovery, Thermogravimetry, Anhydrous, Water of crystallization, Crystallization, Dissolution, Spectroscopy, Nuclear chemistry
الوصف: A typical anhydrous moricizine hydrochloride, an antiarrhythmic agent, is a non-hygroscopic crystalline material. Three lots of moricizine hydrochloride were found to deliquesce within a day at 85% relative humidity, exhibit different X-ray powder diffraction (XRPD) patterns and have more rapid dissolution rate than that of typical anhydrous material. No change in XRPD pattern was observed when the solvent (ethanol) was removed from these lots by heating to 80 degrees C. A two-step water release was observed by thermogravimetric analysis (TGA): a surface water release and a water of hydration release, for these heated samples. The stoichiometry of the water of hydration suggests that it is a hemihydrate. The dissolution rate of the hemihydrate was faster than that of typical anhydrous material. This hemihydrate could be converted to a typical anhydrous material by heating to 90 degrees C. The granules obtained by a simulated wet granulation process on typical lots and typical lots containing up to 20% of hemihydrate exhibited similar physical behaviour to that of typical anhydrous material.
تدمد: 0731-7085
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::58b54a4fb72a10e127a291b9ca8653e9
https://pubmed.ncbi.nlm.nih.gov/7819378
Rights: CLOSED
رقم الانضمام: edsair.doi.dedup.....58b54a4fb72a10e127a291b9ca8653e9
قاعدة البيانات: OpenAIRE