6-Sulfooxymethylbenzo[a]pyrene Is an Ultimate Electrophilic and Carcinogenic Form of the Intermediary Metabolite 6-Hydroxymethylbenzo[a]pyrene

التفاصيل البيبلوغرافية
العنوان: 6-Sulfooxymethylbenzo[a]pyrene Is an Ultimate Electrophilic and Carcinogenic Form of the Intermediary Metabolite 6-Hydroxymethylbenzo[a]pyrene
المؤلفون: James W. Flesher, Jamie Horn, Andreas F. Lehner
المصدر: Biochemical and Biophysical Research Communications. 234:554-558
بيانات النشر: Elsevier BV, 1997.
سنة النشر: 1997
مصطلحات موضوعية: Stereochemistry, Metabolite, Biophysics, Mutagen, medicine.disease_cause, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, Mice, chemistry.chemical_compound, 6-sulfooxymethylbenzo(a)pyrene, medicine, Animals, Benzopyrenes, Molecular Biology, Carcinogen, Cell Biology, Rats, Intermediary metabolite, Liver, chemistry, Electrophile, Carcinogens, Pyrene, Female, Sarcoma, Experimental
الوصف: Previous experiments have demonstrated that the intermediary metabolite 6-hydroxymethylbenzo[a] pyrene (HMBP) can be activated to the electrophilic mutagen, 6-sulfooxymethylbenzo[a]pyrene (SMBP), by rat and mouse liver PAPS-dependent sulfotransferase activity or by chemical synthesis. This aralkylating metabolite and 6-hydroxymethylbenzo[a]pyrene were individually administered to groups of 12 female Sprague-Dawley rats, at a 0.2 μmol dose three times weekly for 20 doses. SMBP induced sarcomas at the site of injection in 12 of 12 rats by 33 weeks, whereas HMBP induced sarcomas at the site of injection in 12 of 12 rats by 31 weeks. These results, taken together with the results of previous studies, strongly support the hypothesis that the electrophilic mutagen SMBP accounts for most, if not all, of the complete carcinogenicity of the intermediary metabolite HMBP and probably at least some of the complete carcinogenicity of 6-methylbenzo[a]pyrene (MBP), 6-formylbenzo[a]pyrene (formylBP), and even benzo[a]pyrene (BP), all of which are metabolized to HMBP.
تدمد: 0006-291X
DOI: 10.1006/bbrc.1997.6679
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2fb84309afe89261d2c60d8bb3ebfd0b
https://doi.org/10.1006/bbrc.1997.6679
Rights: CLOSED
رقم الانضمام: edsair.doi.dedup.....2fb84309afe89261d2c60d8bb3ebfd0b
قاعدة البيانات: OpenAIRE
الوصف
تدمد:0006291X
DOI:10.1006/bbrc.1997.6679