The c-Cbl Ubiquitin Ligase Regulates Nuclear β-Catenin and Angiogenesis by Its Tyrosine Phosphorylation Mediated through the Wnt Signaling Pathway*

التفاصيل البيبلوغرافية
العنوان: The c-Cbl Ubiquitin Ligase Regulates Nuclear β-Catenin and Angiogenesis by Its Tyrosine Phosphorylation Mediated through the Wnt Signaling Pathway*
المؤلفون: Jean M. Francis, Rosana D. Meyer, Vipul C. Chitalia, Moshe Shashar, Nader Rahimi, Chrystelle Kiang, Itrat Harrold, Elazer R. Edelman, Hui Feng, Qing Zhao, Sowmya Shivanna
بيانات النشر: American Society for Biochemistry and Molecular Biology, 2015.
سنة النشر: 2015
مصطلحات موضوعية: Angiogenesis, Mutation, Missense, Neovascularization, Physiologic, macromolecular substances, environment and public health, Biochemistry, chemistry.chemical_compound, Ubiquitin, hemic and lymphatic diseases, Human Umbilical Vein Endothelial Cells, Animals, Humans, Proto-Oncogene Proteins c-cbl, Tyrosine, Phosphorylation, Molecular Biology, Wnt Signaling Pathway, Zebrafish, beta Catenin, Cell Nucleus, biology, Chemistry, fungi, Wnt signaling pathway, Tyrosine phosphorylation, Cell Biology, Zebrafish Proteins, Ubiquitin ligase, Cell biology, enzymes and coenzymes (carbohydrates), Amino Acid Substitution, Catenin, Proteolysis, biology.protein, Cancer research, Protein Multimerization
الوصف: Wnt signaling plays important roles in both the tumor-induced angiogenesis and tumorigenesis through the transcriptionally active nuclear β-catenin. Recently, c-Cbl was identified as a unique E3 ubiquitin ligase targeting the active nuclear β-catenin. However, little is known about the molecular mechanisms by which c-Cbl regulates ubiquitination and degradation of active β-catenin. Here, we demonstrate that Wnt activation promotes the phosphorylation of c-Cbl at tyrosine 731(Tyr-731), which increases c-Cbl dimerization and binding to β-catenin. Tyr-731 phosphorylation and dimerization mediate c-Cbl nuclear translocation and lead to the degradation of nuclearly active β-catenin in the Wnt-on phase. c-Cbl activation also inhibits expression of the pro-angiogenic Wnt targets, IL-8 and VEGF. Phospho-Tyr-731-inactive mutant c-Cbl (Y731F) enhances and phosphomimetic mutant c-Cbl (Y731E) suppresses angiogenesis in zebrafish. Taken together, we have identified a novel mechanism for the regulation of active nuclear β-catenin by c-Cbl and its critical role in angiogenesis. This mechanism can be further explored to modulate both the pathological angiogenesis and the tumorigenesis.
اللغة: English
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2ee3f06504627e9e19686f493a68a6a3
https://europepmc.org/articles/PMC4432275/
Rights: OPEN
رقم الانضمام: edsair.doi.dedup.....2ee3f06504627e9e19686f493a68a6a3
قاعدة البيانات: OpenAIRE