Plasmin Overcomes Resistance to Prostaglandin E2 in Fibrotic Lung Fibroblasts by Reorganizing Protein Kinase A Signaling

التفاصيل البيبلوغرافية
العنوان: Plasmin Overcomes Resistance to Prostaglandin E2 in Fibrotic Lung Fibroblasts by Reorganizing Protein Kinase A Signaling
المؤلفون: Katsuhide Okunishi, Marc Peters-Golden, Thomas H. Sisson, Steven K. Huang, Cory M. Hogaboam, Richard Simon
المصدر: Journal of Biological Chemistry. 286:32231-32243
بيانات النشر: Elsevier BV, 2011.
سنة النشر: 2011
مصطلحات موضوعية: Pulmonary Fibrosis, Drug Resistance, A Kinase Anchor Proteins, Biology, Biochemistry, Dinoprostone, Bleomycin, Mice, Fibrosis, Oxytocics, Cyclic AMP, medicine, Animals, Humans, Fibrinolysin, Protein Phosphatase 2, Protein kinase A signaling, Protein kinase A, Fibroblast, Lung, Molecular Biology, Cell Nucleus, Mice, Knockout, Antibiotics, Antineoplastic, Cell Biology, Lipid signaling, Protein phosphatase 2, Fibroblasts, medicine.disease, Cyclic AMP-Dependent Protein Kinases, Cell biology, Cytoskeletal Proteins, medicine.anatomical_structure, Signal transduction, Microtubule-Associated Proteins, Signal Transduction
الوصف: Collagen deposition by fibroblasts contributes to scarring in fibrotic diseases. Activation of protein kinase A (PKA) by cAMP represents a pivotal brake on fibroblast activation, and the lipid mediator prostaglandin E(2) (PGE(2)) exerts its well known anti-fibrotic actions through cAMP signaling. However, fibrotic fibroblasts from the lungs of patients with idiopathic pulmonary fibrosis, or of mice with bleomycin-induced fibrosis, are resistant to the normal collagen-inhibiting action of PGE(2). In this study, we demonstrate that plasminogen activation to plasmin restores PGE(2) sensitivity in fibrotic lung fibroblasts from human and mouse. This involves amplified PKA signaling resulting from the promotion of new interactions between AKAP9 and PKA regulatory subunit II in the perinuclear region as well as from the inhibition of protein phosphatase 2A. This is the first report to show that an extracellular mediator can dramatically reorganize and amplify the intracellular PKA-A-kinase anchoring protein signaling network and suggests a new strategy to control collagen deposition by fibrotic fibroblasts.
تدمد: 0021-9258
DOI: 10.1074/jbc.m111.235606
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1f9327537fb27d1e2f1939bff0e8a165
https://doi.org/10.1074/jbc.m111.235606
Rights: OPEN
رقم الانضمام: edsair.doi.dedup.....1f9327537fb27d1e2f1939bff0e8a165
قاعدة البيانات: OpenAIRE
الوصف
تدمد:00219258
DOI:10.1074/jbc.m111.235606