Effect of Drug Loading and Process Temperature on Physicochemical Properties of Manidipine Hydrochloride Solid Dispersion

التفاصيل البيبلوغرافية
العنوان: Effect of Drug Loading and Process Temperature on Physicochemical Properties of Manidipine Hydrochloride Solid Dispersion
المؤلفون: Benchawan Chamsai, Pornsak Sriamornsak
المصدر: Advanced Materials Research. 1060:176-179
بيانات النشر: Trans Tech Publications, Ltd., 2014.
سنة النشر: 2014
مصطلحات موضوعية: Chromatography, Materials science, Organic solvent, General Engineering, Polyethylene glycol, Amorphous solid, chemistry.chemical_compound, Chemical engineering, chemistry, Scientific method, PEG ratio, Manidipine hydrochloride, Dispersion (chemistry), Solid solution
الوصف: Binary solid dispersions of manidipine hydrochloride (MDP) and polyethylene glycol (PEG) 4000 are prepared by melting method. Drug loading and process temperature are varied in the range of 5-30% and 150-210°C, respectively. After melting, only the formulation using 5% MDP and process temperature of 210°C showed yellow clear solution and halo pattern of powder X-ray diffractograms with the absence of peaks. These results indicated that the higher process temperature (210°C) can melt all MDP powders and provide the amorphous product. Moreover, only the higher carrier content can change the crystalline form of MDP to the amorphous form. A clear, solid solution could not be prepared when the drug loading was higher than 5%. In this study, the melting technique avoiding the use of organic solvent was successfully applied to prepared binary solid dispersion.
تدمد: 1662-8985
DOI: 10.4028/www.scientific.net/amr.1060.176
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::c35579c5b29b72fd58f8ab349a311ee6
https://doi.org/10.4028/www.scientific.net/amr.1060.176
Rights: CLOSED
رقم الانضمام: edsair.doi...........c35579c5b29b72fd58f8ab349a311ee6
قاعدة البيانات: OpenAIRE
الوصف
تدمد:16628985
DOI:10.4028/www.scientific.net/amr.1060.176