ChemInform Abstract: Preparation of Phosphoglycerides by Phosphoramidite Chemistry

التفاصيل البيبلوغرافية
العنوان: ChemInform Abstract: Preparation of Phosphoglycerides by Phosphoramidite Chemistry
المؤلفون: Christopher McGuigan, Bernadette Swords, Michael S. Anson
المصدر: ChemInform. 23
بيانات النشر: Wiley, 2010.
سنة النشر: 2010
مصطلحات موضوعية: Hydrolysis, Phosphoramidite, Chemistry, Yield (chemistry), Organic chemistry, Phosphoramidate, General Medicine, Spectral data, Cleavage (embryo)
الوصف: Phosphoglycerides have been prepared in high yield by a three-step procedure utilising phosphoramidite intermediates. 2-Chloro-3-methyl-1,3,2-oxazaphosphospholidine 5 reacts with diacylglycerols to give cyclic phosphoramidites in near-quantitative yield. These are oxidised to the corresponding phosphates in very high yield with N2O4. The phosphates hydrolyse in water at ambient temperature, via exclusive P–N cleavage, to yield the target phospholipids. Similarly prepared from 2-chloro-1,3-dimethyl-1,3,2-diazaphospholidine 1 were the phosphoramidate lipid analogues. Spectral data on the intermediates and products are included and discussed.
تدمد: 0931-7597
DOI: 10.1002/chin.199247259
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::66e5ca6c8cb686811bc69098763a2a94
https://doi.org/10.1002/chin.199247259
Rights: CLOSED
رقم الانضمام: edsair.doi...........66e5ca6c8cb686811bc69098763a2a94
قاعدة البيانات: OpenAIRE
الوصف
تدمد:09317597
DOI:10.1002/chin.199247259