Synthesis and Antidepressant activity of pyrazoline based MAO-inhibitors

التفاصيل البيبلوغرافية
العنوان: Synthesis and Antidepressant activity of pyrazoline based MAO-inhibitors
المؤلفون: Alok Kumar, Ashok Kumar Pattnaik, Vishnu Nayak Badavath, Venkatesan Jayaprakash, Surender Singh Jadav, Barij Nayan Sinha
المصدر: Journal of Pharmaceutical Chemistry. 3:1-3
بيانات النشر: Vensel Publications, 2016.
سنة النشر: 2016
مصطلحات موضوعية: Elevated plus maze, medicine.drug_class, Chemistry, MAO inhibitors, Pyrazoline, Pharmacology, 01 natural sciences, Anxiolytic, Tail suspension test, 030227 psychiatry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, medicine, Antidepressant, Behavioural despair test
الوصف: A series of nine 3-(2-hydroxyphenyl)-5-aryl-N-phenyl-4,5-dihydropyrazole-1-carbothioamide derivative s (3a-3i) that were earlier reported as potent rMAO-A inhibitors were evaluated for their antidepressant activity in Porsolt's behavioral despair test (forced swim test) and Tail Suspension test activity, among them, compounds (3e and 3h) were found to have potent antidepressant activity. Reduction in duration of immobility was significant for all the compounds in Porsolts swim test compared with tail suspension test. 3h was further evaluated for anxiolytic activity in Elevated plus maze and was found to be devoid of it.
تدمد: 2349-5731
DOI: 10.14805/jphchem.2016.art45
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::33f1664a18c0e05254ed69fd305cc451
https://doi.org/10.14805/jphchem.2016.art45
رقم الانضمام: edsair.doi...........33f1664a18c0e05254ed69fd305cc451
قاعدة البيانات: OpenAIRE
الوصف
تدمد:23495731
DOI:10.14805/jphchem.2016.art45