Academic Journal

Discovery of (2R,4R)‑4-((S)‑2-Amino-3-methylbutanamido)-2-(4-boronobutyl)pyrrolidine-2-carboxylic Acid (AZD0011), an Actively Transported Prodrug of a Potent Arginase Inhibitor to Treat Cancer.

التفاصيل البيبلوغرافية
العنوان: Discovery of (2R,4R)‑4-((S)‑2-Amino-3-methylbutanamido)-2-(4-boronobutyl)pyrrolidine-2-carboxylic Acid (AZD0011), an Actively Transported Prodrug of a Potent Arginase Inhibitor to Treat Cancer.
المؤلفون: Mlynarski, Scott N., Aquila, Brian M., Cantin, Susan, Cook, Steve, Doshi, Aatman, Finlay, M. Raymond V., Gangl, Eric T., Grebe, Tyler, Gu, Chungang, Kawatkar, Sameer P., Petersen, Jens, Pop-Damkov, Petar, Schuller, Alwin G., Shao, Wenlin, Shields, Jason D., Simpson, Iain, Tavakoli, Siavash, Tentarelli, Sharon, Throner, Scott, Wang, Haixia
المصدر: Journal of Medicinal Chemistry; 12/12/2024, Vol. 67 Issue 23, p20827-20841, 15p
قاعدة البيانات: Supplemental Index
الوصف
تدمد:00222623
DOI:10.1021/acs.jmedchem.4c02309