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1Academic Journal
المؤلفون: Jia, Ruifang, Zhang, Jiwei, Zhang, Jian, Bertagnin, Chiara, Bonomini, Anna, Guizzo, Laura, Gao, Zhen, Ji, Xiangkai, Li, Zhuo, Liu, Chuanfeng, Ju, Han, Ma, Xiuli, Loregian, Arianna, Huang, Bing, Zhan, Peng, Liu, Xinyong
المساهمون: Jia, Ruifang, Zhang, Jiwei, Zhang, Jian, Bertagnin, Chiara, Bonomini, Anna, Guizzo, Laura, Gao, Zhen, Ji, Xiangkai, Li, Zhuo, Liu, Chuanfeng, Ju, Han, Ma, Xiuli, Loregian, Arianna, Huang, Bing, Zhan, Peng, Liu, Xinyong
مصطلحات موضوعية: 150-cavity, boronic acid, influenza, neuraminidase inhibitor, oseltamivir derivative, Amino Acid, Animal, Antiviral Agent, Boron, Drug Resistance, Viral, Enzyme Inhibitor, Mice, Molecular Docking Simulation, Neuraminidase, Oseltamivir, Influenza A Virus, H1N1 Subtype, H5N1 Subtype
Relation: info:eu-repo/semantics/altIdentifier/pmid/36234966; info:eu-repo/semantics/altIdentifier/wos/WOS:000867983100001; volume:27; issue:19; firstpage:6426; journal:MOLECULES; http://hdl.handle.net/11577/3459859; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85139811458
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المؤلفون: Zhang, J., Natarajan Arul, Murugan, Tian, Y., Bertagnin, C., Fang, Z., Kang, D., Kong, X., Jia, H., Sun, Z., Jia, R., Gao, P., Poongavanam, V., Loregian, A., Xu, W., Ma, X., Ding, X., Huang, B., Zhan, P., Liu, X.
المصدر: Journal of Medicinal Chemistry. 61(22):9976-9999
مصطلحات موضوعية: 4 acetamido 3 (pentan 3 yloxy) 5 [(4 phenoxybenzyl)amino]cyclohex 1 ene 1 carboxylic acid, 4 acetamido 3 (pentan 3 yloxy) 5 [[4 (pentan 3 yloxy)benzyl]amino]cyclohex 1 ene 1 carboxylic acid, 4 acetamido 3 (pentan 3 yloxy) 5 [[4 (phenylsulfonyl)benzyl]amino]cyclohex 1 ene 1 carboxylic acid, 4 acetamido 3 (pentan 3 yloxy) 5 [[4 (phenylthio)benzyl]amino]cyclohex 1 ene 1 carboxylic acid, 4 acetamido 3 (pentan 3 yloxy) 5 [[4 (thiophen 2 yl thio)benzyl]amino]cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 amino 3 (1 ethylpropoxy) 1 cyclohexene 1 carboxylic acid, 4 acetamido 5 [(4 benzoylbenzyl)amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [(4 benzylbenzyl)amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [(4 ethylbenzyl)amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [(4 isopropylbenzyl)amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [(4 methoxybenzyl)amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [[3 (cyclopentyl)benzyl]amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [[3 (sec butylthio)benzyl]amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [[4 (benzo[b]thiophen 2 yl)benzyl)amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [[4 (cyclohexylthio)benzyl]amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [[4 (cyclopentyl)benzyl]amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [[4 (isobutylthio)benzyl]amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, 4 acetamido 5 [[4 (sec butylthio)benzyl]amino] 3 (pentan 3 yloxy)cyclohex 1 ene 1 carboxylic acid, antivirus agent, diclofenac, ethyl 4 acetamido 3 (pentan 3 yloxy) 5 [[4 (phenylthio)benzyl]amino]cyclohex 1 ene 1 carboxylate, ethyl 4 acetamido 5 [[4 (benzo[b]thiophen 5 yl)benzyl]amino] 3 (pentan 3 yloxy) cyclohex 1 ene 1 carboxylate, oseltamivir, oseltamivir derivative, propafenone, ribavirin, testosterone, unclassified drug, unindexed drug, virus sialidase, zanamivir, animal experiment, animal model, antiviral activity, area under the curve, Article, bioassay, controlled study, drug clearance, drug half life, drug potency, drug stability, drug structure, drug synthesis, human, human cell, Influenza A virus, Influenza A virus (H3N2), Influenza A virus (H5N1), Influenza A virus (H5N2), Influenza A virus (H5N6), Influenza A virus (H5N8), maximum concentration, MDCK cell line, metabolic stability, molecular model, nonhuman, pharmacokinetic parameters, plasma concentration-time curve, rat, time to maximum plasma concentration
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