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المؤلفون: Roberto Dal Zuffo, Manuela Villa, Biagina Marrocco, Sergio Valente, Paolo Trifiro, Giuseppe Meroni, Mario Varasi, Oronza A. Botrugno, Anna Cappa, Paola Dessanti, Andrea Mattevi, Ciro Mercurio, Giulia Stazi, Saverio Minucci, Paola Vianello, Florian Thaler, Antonello Mai
المصدر: Journal of Medicinal Chemistry. 59:1501-1517
مصطلحات موضوعية: LSD1 epigenetics, monoamine-oxidase-b, breast-cancer, cyclopropylamine derivatives, modifying enzymes, LSD1 inhibition, methylation, cells, proteins, complex, targets, 0301 basic medicine, Acute promyelocytic leukemia, Administration, Oral, Antineoplastic Agents, Pharmacology, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Leukemia, Promyelocytic, Acute, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Humans, Structure–activity relationship, Enzyme Inhibitors, Clonogenic assay, Histone Demethylases, Acute leukemia, Chemistry, KDM1A, Biological activity, medicine.disease, Leukemia, 030104 developmental biology, 030220 oncology & carcinogenesis, Molecular Medicine, Tranylcypromine