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1Academic JournalAugmented Antitumor Activity for Novel Dual PI3K/BDR4 Inhibitors, SF2523 and SF1126 in Ewing Sarcoma
المصدر: Journal of Pediatric Hematology/Oncology. 43(3)
مصطلحات موضوعية: Biomedical and Clinical Sciences, Oncology and Carcinogenesis, Pediatric Research Initiative, Pediatric, Pediatric Cancer, Stem Cell Research, Rare Diseases, Cancer, 5.1 Pharmaceuticals, Development of treatments and therapeutic interventions, Animals, Antineoplastic Agents, Cell Cycle Proteins, Cell Line, Tumor, Cell Survival, Chromones, Humans, Mice, Morpholines, Oligopeptides, Phosphoinositide-3 Kinase Inhibitors, Phosphorylation, Pyrans, Sarcoma, Ewing, Transcription Factors, Ewing sarcoma, dual inhibition, phosphoinositide-3 kinase (PI3K) pathway, bromodomain and extraterminal domain (BET) proteins, SF1126, SF2523, Cardiorespiratory Medicine and Haematology, Oncology & Carcinogenesis, Cardiovascular medicine and haematology
وصف الملف: application/pdf
URL الوصول: https://escholarship.org/uc/item/5vm2r5rx
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2Augmented Antitumor Activity for Novel Dual PI3K/BDR4 Inhibitors, SF2523 and SF1126 in Ewing Sarcoma
المصدر: Journal of pediatric hematology/oncology, vol 43, iss 3
مصطلحات موضوعية: Cell Cycle Proteins, Cardiorespiratory Medicine and Haematology, Mice, 0302 clinical medicine, Phosphorylation, Phosphoinositide-3 Kinase Inhibitors, Cancer, Pediatric, Tumor, Kinase, Bone cancer, Sarcoma, Hematology, phosphoinositide-3 kinase (PI3K) pathway, Oncology, 5.1 Pharmaceuticals, 030220 oncology & carcinogenesis, Oligopeptides, Pediatric Research Initiative, Cell Survival, Pediatric Cancer, Morpholines, bromodomain and extraterminal domain (BET) proteins, Antineoplastic Agents, Sarcoma, Ewing, SF2523, Cell Line, 03 medical and health sciences, Rare Diseases, Cell Line, Tumor, Ewing, medicine, Animals, Humans, Viability assay, Oncology & Carcinogenesis, Protein kinase B, PI3K/AKT/mTOR pathway, Pyrans, business.industry, dual inhibition, SF1126, medicine.disease, Stem Cell Research, Bromodomain, Chromones, Pediatrics, Perinatology and Child Health, Cancer research, business, Ewing sarcoma, 030215 immunology, Transcription Factors
وصف الملف: application/pdf
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المؤلفون: Ryota Takahashi, Keisuke Tateishi, Yasuo Tanaka, Yousuke Nakai, Kiyoshi Hasegawa, Yoshihiro Sakamoto, Yotaro Kudo, Mariko Tanaka, Takuma Nakatsuka, Hideaki Ijichi, Hiroaki Fujiwara, Hiroyuki Isayama, Koji Miyabayashi, Taku Aoki, Kazuhiko Koike, Keisuke Yamamoto, Yasuyuki Morishita, Norihiro Kokudo, Masashi Fukayama, Mayumi Hoshikawa
المصدر: Oncotarget
مصطلحات موضوعية: 0301 basic medicine, Male, Pathology, endocrine system diseases, Transcription, Genetic, Mice, SCID, pancreatic ductal adenocarcinoma (PDAC), Epigenesis, Genetic, cancer-associated fibroblast (CAF), Mice, Cancer-Associated Fibroblasts, Mice, Inbred NOD, Transforming Growth Factor beta, Medicine, STAT3, biology, Molecular pathology, Azepines, Immunohistochemistry, Oncology, Disease Progression, Cytokines, Research Paper, Carcinoma, Pancreatic Ductal, Signal Transduction, STAT3 Transcription Factor, medicine.medical_specialty, Chromatin Immunoprecipitation, Stromal cell, bromodomain and extraterminal domain (BET) proteins, JQ1, Primary Cell Culture, BET inhibitor, 03 medical and health sciences, Pancreatic cancer, Cell Line, Tumor, Animals, Humans, Hedgehog Proteins, Protein kinase B, Pancreas, Cell Proliferation, epigenetics, business.industry, Proteins, Triazoles, medicine.disease, Xenograft Model Antitumor Assays, Actins, Bromodomain, Pancreatic Neoplasms, 030104 developmental biology, Cancer research, biology.protein, business, Chromatin immunoprecipitation
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المؤلفون: Bikash R. Pattnaik, Pawan K Shahi, Jun Li, Mengxue Zhang, Jonathan N. Ouellette, Jyoti J. Watters, Yingmei Fu, Lei Zhao, Wai T. Wong, Lian-Wang Guo, Bowen Wang
المصدر: Journal of Neuroinflammation
مصطلحات موضوعية: 0301 basic medicine, Retinal degeneration, Bromodomain and extraterminal domain (BET) proteins, JQ1, Immunology, Mice, Transgenic, Nerve Tissue Proteins, Receptors, Cell Surface, Biology, Epigenetic readers, Proinflammatory cytokine, Epigenesis, Genetic, 03 medical and health sciences, chemistry.chemical_compound, Mice, Cellular and Molecular Neuroscience, PDE6B, Retinitis pigmentosa, rd10 mice, medicine, Animals, Microglial activation, Photoreceptor Cells, Retina, General Neuroscience, Research, Neurodegeneration, Retinal Degeneration, Retinal, medicine.disease, Bromodomain, Cell biology, Mice, Inbred C57BL, Disease Models, Animal, 030104 developmental biology, medicine.anatomical_structure, chemistry, Neurology, Retinitis Pigmentosa