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1
المؤلفون: Louise Bernier, Gary Chinigo, Chulho Choi, Julien Genovino, Mark W. Bundesmann, Mathieu Frenette, Olugbeminiyi O. Fadeyi, Yohann Gagné, Neal W. Sach, Martins S. Oderinde, Antoine Juneau, Philippe Nuhant, Bhagyashree Khunte, Christophe Allais, Yvette M. Fobian
المصدر: Angewandte Chemie (International ed. in English). 56(48)
مصطلحات موضوعية: chemistry.chemical_classification, Cyclobutanes, Chemistry, 010405 organic chemistry, Iodide, chemistry.chemical_element, General Chemistry, Manganese, General Medicine, Alkylation, Photochemistry, 010402 general chemistry, Redox, Combinatorial chemistry, 01 natural sciences, Catalysis, 0104 chemical sciences, 3. Good health, Alkyl, Minisci reaction
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2
المؤلفون: Anthony Wood, Simon Bailey, David Austen Perry, Heather N. Frost, Yvette M. Fobian, Sylvie K. Sakata, F. Christopher Bi, Xiaolan Ling, Leslie Sloan
المصدر: Drug Discovery Today. 19:289-294
مصطلحات موضوعية: Pharmacology, Underpinning, Drug Industry, Queue management system, Process (engineering), Chemistry, Pharmaceutical, Communication, Research, Contract Services, Work in process, Efficiency, Organizational, Quality Improvement, Workflow, Engineering management, Workflow analysis, Drug Design, Drug Discovery, Humans, Chemistry (relationship), Lean Six Sigma, Productivity
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3eBook
المؤلفون: David C Blakemore, Paul M Doyle, Yvette M Fobian
Resource Type: eBook.
الموضوعات: Drug development
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4eBook
المؤلفون: David C Blakemore, Paul M Doyle, Yvette M Fobian
Resource Type: eBook.
الموضوعات: Drug development
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5
المؤلفون: John Robert Springer, Gina M. Jerome, Hayes Michael J, Michael T. Baratta, Daniel P. Walker, Graciela B. Arhancet, Alexander F. Shaffer, Jaime L. Masferrer, Ben S. Zweifel, Steven E. Heasley, Darin E. Jones, William M. Moore, Jeffrey S. Carter, Yvette M. Fobian, Michael L. Vazquez, Sue Metz
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:1114-1119
مصطلحات موضوعية: Inflammation, Drug discovery, Organic Chemistry, Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Prostaglandin, Benzoxazole, Pharmacology, Biochemistry, In vitro, Bioavailability, Intramolecular Oxidoreductases, Structure-Activity Relationship, chemistry.chemical_compound, chemistry, Pharmacokinetics, In vivo, Drug Discovery, Humans, Molecular Medicine, Structure–activity relationship, Enzyme Inhibitors, Molecular Biology, Prostaglandin-E Synthases
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6
المؤلفون: Daniel P. Walker, Alexander F. Shaffer, William M. Moore, Michael T. Baratta, Sue Metz, Jeffrey A. Scholten, John Robert Springer, Jeffrey S. Carter, Hwang-Fun Lu, Steven E. Heasley, Yvette M. Fobian, Natasha M. Kablaoui, Francisco M. Franco, Li Xing, Shengtian Yang, Hanau Cathleen E, Michael L. Vazquez, Graciela B. Arhancet, Gina M. Jerome
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:1120-1126
مصطلحات موضوعية: Models, Molecular, musculoskeletal diseases, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Acyl glucuronide, Molecular Conformation, Pharmaceutical Science, Biochemistry, Molecular conformation, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Humans, Structure–activity relationship, Enzyme Inhibitors, Molecular Biology, Prostaglandin-E Synthases, Biological evaluation, Benzoxazoles, Organic Chemistry, Benzoxazole, Intramolecular Oxidoreductases, chemistry, Drug Design, Molecular Medicine, lipids (amino acids, peptides, and proteins), Prostaglandin E
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7
المؤلفون: David C. Blakemore, Alexandria P. Taylor, Ralph P. Robinson, Yvette M. Fobian, Lyn H. Jones, Olugbeminiyi O. Fadeyi
المصدر: ChemInform. 47
مصطلحات موضوعية: Drug development, Drug discovery, business.industry, Chemistry, Rapid access, General Medicine, Biochemical engineering, business, Chemical space, Pharmaceutical industry
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8
المؤلفون: Lyn H. Jones, Yvette M. Fobian, Alexandria P. Taylor, David C. Blakemore, Olugbeminiyi O. Fadeyi, Ralph P. Robinson
المصدر: Organicbiomolecular chemistry. 14(28)
مصطلحات موضوعية: 010405 organic chemistry, Drug discovery, business.industry, Chemistry, Organic Chemistry, Nanotechnology, Oxidation reduction, Stereoisomerism, Chemistry Techniques, Synthetic, 010402 general chemistry, Photochemical Processes, 01 natural sciences, Biochemistry, Chemical space, 0104 chemical sciences, Drug development, Heterocyclic Compounds, Drug Discovery, Rapid access, Humans, Physical and Theoretical Chemistry, business, Oxidation-Reduction, Pharmaceutical industry
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9
المؤلفون: Joe T. Collins, Steven E. Heasley, Hwang-Fun Lu, Yvette M. Fobian, Allison MacInnes, Michael K. Mao, Tizah Evelyn Anjeh, Michael L. Vazquez, Daniel P. Walker
المصدر: Synlett. 2011:2959-2962
مصطلحات موضوعية: Chemistry, Organic Chemistry, Organic chemistry, Chiral resolution
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10
المؤلفون: Michael A. Tones, Paul A. Bradley, Graham L. Smith, Lee R. Roberts, Geoff E. Gymer, Katherine S. England, Fox David Nathan Abraham, Steven E. Heasley, Michelle Schmidt, Mark E. Bunnage, Yvette M. Fobian, Jerome Molette, David Fairman, Dack Kevin Neil
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:6515-6518
مصطلحات موضوعية: chemistry.chemical_classification, GUCY1B3, Organic Chemistry, Clinical Biochemistry, GUCY1A3, Triazole, Guanylate Cyclase Stimulators, Enzyme Activators, Receptors, Cytoplasmic and Nuclear, Pharmaceutical Science, Triazoles, Biochemistry, chemistry.chemical_compound, Soluble Guanylyl Cyclase, Enzyme, chemistry, Guanylate Cyclase, Drug Discovery, Molecular Medicine, Organic chemistry, Molecule, Acids, Molecular Biology
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11
المؤلفون: Sandra W. Curtiss, D. Joseph Rogier, Alan MacInnes, Brown David L, Mike B. Tollefson, Brian R. Bond, Yvette M. Fobian, Maddux Todd Michael, Dafydd R. Owen, Jeanne M. Rumsey, Brent V. Mischke, Jerry W. Cubbage, Alan G. Benson, Robert Hughes, Lena L Zhang, E. Jon Jacobsen, Steven E. Heasley, Joseph B. Moon, Ying Yu, John M. Molyneaux, Yi Zheng, Brad A. Acker, Blevis-Bal Radhika M, John N. Freskos, John K. Walker, Jennie L. Walgren
المصدر: Journal of Medicinal Chemistry. 53:2656-2660
مصطلحات موضوعية: Stereochemistry, Chemistry, Pharmacology, chemistry.chemical_compound, Spontaneously hypertensive rat, Orally active, Design synthesis, In vivo, cGMP-specific phosphodiesterase type 5, Drug Discovery, Molecular Medicine, Potency, Penetrant (biochemical), Biological evaluation
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12
المؤلفون: Maddux Todd Michael, Yvette M. Fobian, Alan G. Benson, Dafydd R. Owen, Brian R. Bond, Christopher Phillips, Brad A. Acker, E. Jon Jacobsen, Michael John Palmer, D. Joseph Rogier, John M. Molyneaux, Brent V. Mischke, John N. Freskos, Tracy J. Ringer, Andrew Simon Bell, Blevis-Bal Radhika M, Robert Hughes, David G. Brown, Steve E. Heasley, Joseph B. Moon, John K. Walker, Brown David L, William C. Stallings, Michael B. Tollefson, Alan MacInnes, Jerry W. Cubbage, Yung Yu, Margarita Rodriquez-Lens, Fox David Nathan Abraham
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:4088-4091
مصطلحات موضوعية: medicine.drug_mechanism_of_action, Phosphodiesterase Inhibitors, Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Pharmaceutical Science, Crystallographic data, Crystallography, X-Ray, Biochemistry, Chemical synthesis, QH301, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, 3',5'-Cyclic-GMP Phosphodiesterases, Catalytic Domain, Drug Discovery, Hydrolase, medicine, Animals, Humans, QD, Molecular Biology, Cyclic Nucleotide Phosphodiesterases, Type 5, chemistry.chemical_classification, Cyclic Nucleotide Phosphodiesterases, Type 6, biology, Bicyclic molecule, Phosphoric Diester Hydrolases, Chemistry, Organic Chemistry, Hydrogen-Ion Concentration, Phosphodiesterase 5 Inhibitors, Protein Structure, Tertiary, Rats, Enzyme, Enzyme inhibitor, Drug Design, Pyrazines, biology.protein, Lactam, Molecular Medicine, Phosphodiesterase 5 inhibitor
وصف الملف: application/pdf
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13
المؤلفون: David Price, Enoch S. Huang, Yao Zhang, Larry Whiteley, Yvette M. Fobian, Julian Blagg, Jens Loesel, Michael E. Gibbs, Teresa Krieger-Burke, Travis T. Wager, Nigel Greene, Rajesh V. Devraj, Richard W. Gilles, Simon Bailey, Decrescenzo Gary A, Jason D. Hughes, Edmund L. Ellsworth
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:4872-4875
مصطلحات موضوعية: Male, Drug, Drug-Related Side Effects and Adverse Reactions, media_common.quotation_subject, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Pharmacology, Biochemistry, Polar surface area, Structure-Activity Relationship, Dogs, In vivo, Drug Discovery, Animals, Humans, Molecular Biology, Drug toxicity, media_common, Chemistry, Organic Chemistry, Chemical space, Rats, Pharmaceutical Preparations, Lipophilic efficiency, Toxicity, Lipophilicity, Molecular Medicine, Female
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14
المؤلفون: John N. Freskos, Yvette M. Fobian, Timothy E. Benson, Michael J. Bienkowski, David L. Brown, Thomas L. Emmons, Robert Heintz, Alice Laborde, Joseph J. McDonald, Brent V. Mischke, John M. Molyneaux, Joseph B. Moon, Patrick B. Mullins, D. Bryan Prince, Donna J. Paddock, Alfredo G. Tomasselli, Gregory Winterrowd
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:73-77
مصطلحات موضوعية: Sulfonamides, Molecular Structure, Protein Conformation, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Structure-Activity Relationship, Alzheimer Disease, Drug Design, Drug Discovery, Humans, Molecular Medicine, Protease Inhibitors, Sulfones, Amyloid Precursor Protein Secretases, Molecular Biology
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15
المؤلفون: Jane L. Wang, Michael B. Tollefson, Margaret L. Grapperhaus, James A. Sikorski, Richard C. Durley, Monica B. Norton, Michele A. Promo, Michele A. Melton, Mark A. Massa, Emily J. Reinhard, Brian S. Hickory, William F. Vernier, Mark E. Smith, Yvette M. Fobian, Karen Regina, Bryan J. Witherbee, Daniel T. Connolly
المصدر: Journal of Medicinal Chemistry. 46:2152-2168
مصطلحات موضوعية: biology, Stereochemistry, Chemistry, Stereoisomerism, Chemical synthesis, Drug Discovery, Cholesterylester transfer protein, biology.protein, Molecular Medicine, Structure–activity relationship, Potency, lipids (amino acids, peptides, and proteins), Enantiomer, IC50, CETP inhibitor
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16
المؤلفون: Michele A Melton, Nigam P. Rath, Ming Zeng, Margaret L. Grapperhaus, Brian S Hickory, Jane L Wang, Elaine S. Krul, Deborah M. Heuvelman, Mark E. Smith, Kevin C. Glenn, Richard C Durley, Deborah A. Mischke, Bryan J. Witherbee, Daniel T. Connolly, Dale P Spangler, Dorothy D. Honda, Yvette M. Fobian, James A. Sikorski, Mark A. Massa, Barry L. Parnas
المصدر: Journal of Medicinal Chemistry. 45:3891-3904
مصطلحات موضوعية: Male, Models, Molecular, Stereochemistry, Substituent, Stereoisomerism, Lipoproteins, VLDL, Alkylation, Crystallography, X-Ray, Chemical synthesis, Propanolamines, Acylation, Propanol, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Cricetinae, Drug Discovery, Animals, Combinatorial Chemistry Techniques, Humans, Structure–activity relationship, Serum Albumin, Glycoproteins, Aniline Compounds, Mesocricetus, Molecular Structure, Phenyl Ethers, Cholesterol Ester Transfer Proteins, Lipoproteins, LDL, Mice, Inbred C57BL, chemistry, Molecular Medicine, Enantiomer, Carrier Proteins, Lipoproteins, HDL, Protein Binding
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17
المؤلفون: James R. Kiefer, Barta Thomas E, Heintz Robert M, Yvette M. Fobian, Daniel P. Becker, Grace E. Munie, Patrick B. Mullins, John M. Molyneaux, Brent V. Mischke, Darren J. Kassab, Louis J. Bedell, John N. Freskos
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2823-2825
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Ether, Carboxamide, Matrix Metalloproteinase Inhibitors, Hydroxamic Acids, Biochemistry, Chemical synthesis, Substrate Specificity, Sulfone, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Amide, Drug Discovery, medicine, Humans, Structure–activity relationship, Protease Inhibitors, Molecular Biology, Hydroxamic acid, Molecular Structure, Organic Chemistry, Amides, chemistry, Molecular Medicine, Selectivity
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18
المؤلفون: D. André d’Avignon, Yvette M. Fobian, Kevin D. Moeller
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:315-318
مصطلحات موضوعية: chemistry.chemical_classification, Bicyclic molecule, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Substrate (chemistry), Peptide, Ring (chemistry), Biochemistry, Combinatorial chemistry, chemistry.chemical_compound, Peptide backbone, chemistry, Derivative (finance), Amide, Drug Discovery, Molecular Medicine, Nonane, Molecular Biology
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19
المؤلفون: Yvette M. Fobian, Fabrice Cornille, Kevin D. Moeller, Denise D. Beusen, Garland R. Marshall, Urszula Slomczynska
المصدر: Tetrahedron Letters. 35:6989-6992
مصطلحات موضوعية: chemistry.chemical_classification, Dipeptide, Bicyclic molecule, Organic Chemistry, Peptide, Electrochemistry, Biochemistry, Combinatorial chemistry, Amino acid, chemistry.chemical_compound, chemistry, Amide, Drug Discovery, Lactam, Selectivity
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20APPLICATION OF HMBC AND HMQC-TOCSY NMR METHODS TO ASSIGN THE STRUCTURES OF BICYCLIC-PEPTIDE MIMETICS
المصدر: Journal of Coordination Chemistry. 32:135-144
مصطلحات موضوعية: chemistry.chemical_classification, Proton, Bicyclic molecule, Chemistry, Carbon-13 NMR satellite, Stereochemistry, Nuclear Theory, Heteroatom, Peptide, Protonation, Proton spin crisis, Materials Chemistry, Physics::Accelerator Physics, Organic chemistry, Molecule, Physical and Theoretical Chemistry, Nuclear Experiment