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1Academic Journal
المؤلفون: Ying-zi, Xu, Yakushijin, Kenichi, Horne, David A.
المصدر: Tetrahedron Letters ; volume 33, issue 31, page 4385-4388 ; ISSN 0040-4039
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2
المؤلفون: Michael F. Jobling, Donald Rudolph, Karin Regnstrom, Michael P. Bova, Danny Tam, Shendong Yuan, Ying-Zi Xu, David W. G. Wone, Dean R. Artis, Harry Cheung, Hing L. Sham, Zhao Ren, Xiaohua Chen
المصدر: SLAS Discovery. 18:695-704
مصطلحات موضوعية: Streptavidin, High-throughput screening, Hydantoin, Sensitivity and Specificity, Biochemistry, Analytical Chemistry, Small Molecule Libraries, Inhibitory Concentration 50, chemistry.chemical_compound, Biotin, Alzheimer Disease, mental disorders, Amyloid precursor protein, Aspartic Acid Endopeptidases, Humans, Sulfamide, chemistry.chemical_classification, biology, Hydantoins, Ligand binding assay, Combinatorial chemistry, High-Throughput Screening Assays, Enzyme, chemistry, biology.protein, Molecular Medicine, Amyloid Precursor Protein Secretases, Biotechnology
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3
المؤلفون: Anna Liao, Gary Probst, Pamela S. Keim, Kang Hu, Roy K. Hom, David A. Quincy, Michael S. Dappen, Grace T. Kwong, Jenifer Smith, Martin L. Neitzel, Ying-zi Xu, Elizabeth F. Brigham, Kevin P. Quinn, Frédérique Bard, Minghua Sun, Jing Wu, John-Michael Sauer, Dora Kholodenko, Hongbin Zhang, William Wallace, Matthew N. Mattson, Patricia Sacayon, Jacek Jagodzinski, Hing L. Sham, Brian T. Peterson, Simeon Bowers, Jennifer Marugg, Guriqbal S. Basi, Lee H. Latimer, Susanna S. Hemphill, Darren B. Dressen, Karina Wong, Kevin Tanaka, Michael P. Bova, Pamela Santiago, Daniel K. Ness, Anh P. Truong, Wes Zmolek, Lany Ruslim, Christopher Willits, Michael K. Lee, Andrei W. Konradi, Xiaocong M. Ye, Lam Nguyen, Chris M. Semko, Ted A. Yednock, Ruth N. Motter, Albert W. Garofalo, Erich Goldbach, Pearl Tanaka, Danielle L. Aubele
المصدر: Journal of Medicinal Chemistry. 56:5261-5274
مصطلحات موضوعية: Trifluoromethyl, biology, Stereochemistry, Quinoline, In vitro, chemistry.chemical_compound, chemistry, In vivo, Drug Discovery, biology.protein, medicine, Molecular Medicine, Structure–activity relationship, Chirality (chemistry), Amyloid precursor protein secretase, Semagacestat, medicine.drug
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4
المؤلفون: Jennifer S. Smith, Michael A. Pleiss, Caroline Garrido, Ying-Zi Xu, Frank Stappenbeck, Elizabeth Messersmith, Frederique Bard, Bhushan Samant, Linda Mutter, Semko Christopher M, Brent Welch, Brian P. Stupi, Chris Vandervert, Mark Dreyer, Zhenmei Liao, Mike Krimm, Brian Wipke, Ian Gallager, Ted Yednock, Michael S. Dappen, Andrei W. Konradi, Lilibeth Dofiles
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:3070-3074
مصطلحات موضوعية: Models, Molecular, Multiple Sclerosis, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Integrin alpha4beta1, Biochemistry, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, Cell Adhesion, Animals, Humans, Structure–activity relationship, Collagen Type II, Molecular Biology, Sulfonamides, Dose-Response Relationship, Drug, Chemistry, Organic Chemistry, Antagonist, VLA-4, Arthritis, Experimental, Asthma, In vitro, Fibronectins, Rats, Mice, Inbred C57BL, Sprague dawley, Disease Models, Animal, Pyrimidines, Propanoic acid, Rats, Inbred Lew, Antirheumatic Agents, Molecular Medicine, Female, Selectivity
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5
المؤلفون: Gary Probst, Ying-Zi Xu
المصدر: Expert Opinion on Therapeutic Patents. 22:511-540
مصطلحات موضوعية: Pathology, medicine.medical_specialty, Aspartyl Proteinases, Patent literature, Disease, Bioinformatics, Patents as Topic, Structure-Activity Relationship, Alzheimer Disease, mental disorders, Drug Discovery, Animals, Aspartic Acid Endopeptidases, Humans, Medicine, Protease Inhibitors, Pharmacology, Amyloid beta-Peptides, Molecular Structure, business.industry, Neurodegeneration, Brain, General Medicine, Legislation, Drug, medicine.disease, Small molecule, Biochemistry of Alzheimer's disease, Drug Design, Amyloid Precursor Protein Secretases, business
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6
المؤلفون: Ying Zi Xu, Shan Chai, Li Jun Li, Hong Yan Li, Xian Yue Gang
المصدر: Key Engineering Materials. :692-697
مصطلحات موضوعية: Coupling, Computer science, Mechanical Engineering, Numerical analysis, Mathematical analysis, Mixed finite element method, Boundary knot method, Finite element method, Discrete element method, Computational physics, Mechanics of Materials, General Materials Science, Acoustic radiation, Boundary element method
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7
المؤلفون: Darren B. Dressen, Ying-Zi Xu, Jenifer L. Smith, Xiaocong M. Ye, Elizabeth F. Brigham, Erich Goldbach, Anh P. Truong, Hing L. Sham, Michael P. Bova, Jennifer Marugg, Guriqbal S. Basi, Jacek Jagodzinski, Hongbin Zhang, Michael A. Pleiss, Andrei W. Konradi, Albert W. Garofalo, John-Michael Sauer
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:2195-2199
مصطلحات موضوعية: Models, Molecular, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, Piperidines, Alzheimer Disease, In vivo, Drug Discovery, Pyrazolopyridine, medicine, Amyloid precursor protein, Animals, Humans, Structure–activity relationship, Molecular Biology, chemistry.chemical_classification, Sulfonamides, biology, Organic Chemistry, Sulfonamide (medicine), Biological activity, Enzyme, chemistry, biology.protein, Molecular Medicine, Amyloid Precursor Protein Secretases, Amyloid precursor protein secretase, medicine.drug
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8
المؤلفون: M. Isabel Calaza, and Sean Turner, Ying-zi Xu, Henry Rapoport, Jaesung Choi
المصدر: The Journal of Organic Chemistry. 64:4069-4078
مصطلحات موضوعية: chemistry.chemical_compound, Heptane, chemistry, Bicyclic molecule, Bromide, Intramolecular force, Organic Chemistry, Imine, Regioselectivity, Pyrroline, Medicinal chemistry, Octane
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9
المؤلفون: Robin Barbour, Ying-Zi Xu, Winse Morishige, Gary Probst, Karin Regnstrom, Michael P. Bova, Paul Beroza, Nanhua Yao, Kalyani Mondal, Dean R. Artis
المصدر: Biochemical and biophysical research communications. 441(2)
مصطلحات موضوعية: Aspartic Acid Proteases, Protein Conformation, Enthalpy, Biophysics, Biochemistry, Chemical kinetics, Protein structure, Reaction rate constant, Alzheimer Disease, Amyloid precursor protein, Aspartic Acid Endopeptidases, Humans, Protease Inhibitors, Surface plasmon resonance, Molecular Biology, biology, Chemistry, Cell Biology, Ligand (biochemistry), Enzymes, Immobilized, Crystallography, Kinetics, Ethanolamines, biology.protein, Physical chemistry, Thermodynamics, Amyloid Precursor Protein Secretases, Entropy (order and disorder)
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10
المؤلفون: Gary, Probst, Danielle L, Aubele, Simeon, Bowers, Darren, Dressen, Albert W, Garofalo, Roy K, Hom, Andrei W, Konradi, Jennifer L, Marugg, Matthew N, Mattson, Martin L, Neitzel, Chris M, Semko, Hing L, Sham, Jenifer, Smith, Minghua, Sun, Anh P, Truong, Xiaocong M, Ye, Ying-Zi, Xu, Michael S, Dappen, Jacek J, Jagodzinski, Pamela S, Keim, Brian, Peterson, Lee H, Latimer, David, Quincy, Jing, Wu, Erich, Goldbach, Daniel K, Ness, Kevin P, Quinn, John-Michael, Sauer, Karina, Wong, Hongbin, Zhang, Wes, Zmolek, Elizabeth F, Brigham, Dora, Kholodenko, Kang, Hu, Grace T, Kwong, Michael, Lee, Anna, Liao, Ruth N, Motter, Patricia, Sacayon, Pamela, Santiago, Christopher, Willits, Frédérique, Bard, Michael P, Bova, Susanna S, Hemphill, Lam, Nguyen, Lany, Ruslim, Kevin, Tanaka, Pearl, Tanaka, William, Wallace, Ted A, Yednock, Guriqbal S, Basi
المصدر: Journal of medicinal chemistry. 56(13)
مصطلحات موضوعية: Male, Time Factors, Gene Expression, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, Dogs, Drug Stability, Basic Helix-Loop-Helix Transcription Factors, Animals, Humans, RNA, Messenger, Enzyme Inhibitors, Homeodomain Proteins, Sulfonamides, Amyloid beta-Peptides, Dose-Response Relationship, Drug, Molecular Structure, Receptors, Notch, Rats, Models, Chemical, Area Under Curve, Drug Design, Microsomes, Liver, Quinolines, Pyrazoles, Transcription Factor HES-1, Amyloid Precursor Protein Secretases, Heterocyclic Compounds, 3-Ring
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11
المؤلفون: Angie Wadsworth, Wenxian Mao, Stellanie Simmonds, Eric Peterson, Christopher Vandevert, F. Bong San Pablo, Ted Yednock, Ying-Zi Xu, David A. Quincy, Carlos Lorenzana, Andrei W. Konradi, Kassandra Inez Rossiter, Michael S. Dappen, Michael A. Pleiss, Frederique Bard, Elizabeth Messersmith, Brian Wipke, Caroline Garrido, Jenifer L. Smith, Christopher M. Semko, Jacek Jagodzinski, Lilibeth Dofiles
المصدر: Bioorganicmedicinal chemistry letters. 23(14)
مصطلحات موضوعية: Injections, Subcutaneous, Integrin alpha4, Clinical Biochemistry, Pharmaceutical Science, Cleavage (embryo), Biochemistry, α4β7 integrin, Polyethylene Glycols, Jurkat Cells, In vivo, Drug Discovery, PEG ratio, Animals, Humans, α4 integrin, α4β1 integrin, Molecular Biology, Chemistry, Organic Chemistry, Antibodies, Monoclonal, Esters, Rats, Molecular Medicine, Conjugate, Half-Life
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12
المؤلفون: Bhushan Samant, Mark Shoemaker, Michael Krimm, Elizabeth Messersmith, Brent Welch, John-Michael Sauer, Linda Chen, Michael S. Dappen, Wenxian Mao, Zhenmei Liao, Ted Yednock, Jenifer L. Smith, Carrol Henschel, Nancy G. Wehner, Lilibeth Dofiles, Ian Gallager, Linda Mutter, Michael A. Pleiss, Mark Dreyer, David A. Quincy, Andrei W. Konradi, Hongbin Zhang, Christopher M. Semko, Kassandra Inez Rossiter, Eric Petersen, George Shopp, Juri Y Fukuda, Brian Wipke, Christopher Vandevert, Frederique Bard, Judevin Lugar, Ying-Zi Xu
المصدر: Bioorganicmedicinal chemistry letters. 23(15)
مصطلحات موضوعية: Integrins, Clinical Biochemistry, Rat model, Pharmaceutical Science, Arthritis, Administration, Oral, Pharmacology, Integrin alpha4beta1, Biochemistry, Jurkat cells, α4β7 integrin, Arthritis, Rheumatoid, Jurkat Cells, Crohn Disease, Drug Discovery, Area under curve, medicine, Animals, Humans, Molecular Biology, Chemistry, Organic Chemistry, medicine.disease, Rats, Disease Models, Animal, Liver metabolism, Rheumatoid arthritis, Area Under Curve, Microsomes, Liver, Molecular Medicine, Half-Life
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13
المؤلفون: K. Yakushijin, David A. Horne, Ying-zi Xu
المصدر: Tetrahedron Letters. 37:8121-8124
مصطلحات موضوعية: chemistry.chemical_compound, Olefin fiber, Chemistry, Alkaloid, Organic Chemistry, Drug Discovery, Regioselectivity, Imidazole, Organic chemistry, Biochemistry, Stevensine, Pyrrole
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14
المؤلفون: Hing L. Sham, Ying-Zi Xu, Zhao Ren, Shendong Yuan, Julie Lougheed, Eric Brecht, Wayman Chan, Roy K. Hom, Lany Ruslim, Paul Beroza, Michael P. Bova, Dean R. Artis, Yong L. Zhu, Jiangli Yan, Simeon Bowers, Danny Tam, Hu Pan, Nanhua Yao
المصدر: Bioorganicmedicinal chemistry letters. 23(10)
مصطلحات موضوعية: Models, Molecular, Clinical Biochemistry, Pharmaceutical Science, Thiophenes, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, mental disorders, Drug Discovery, Thiophene, Structure–activity relationship, Organic chemistry, Aspartic Acid Endopeptidases, Humans, Protease Inhibitors, Molecular Biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Highly selective, Isoquinolines, Combinatorial chemistry, Drug Design, Molecular Medicine, Structure based, Amyloid Precursor Protein Secretases
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15
المؤلفون: Gary Probst, Nanhua Yao, Danny Tam, Julie Lougheed, Zhao Ren, Hu Pan, Ying-Zi Xu, Wayman Chan, Dean R. Artis, Lany Ruslim, Shendong Yuan, Roy K. Hom, Yong L. Zhu, Paul Beroza, Andrei W. Konradi, Eric Brecht, Michael P. Bova, Hing L. Sham, Simeon Bowers
المصدر: Bioorganicmedicinal chemistry letters. 23(7)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Catalysis, Structure-Activity Relationship, Drug Discovery, Aspartic Acid Endopeptidases, Humans, Protease Inhibitors, Molecular Biology, chemistry.chemical_classification, Aspartic Acid, Dose-Response Relationship, Drug, Molecular Structure, Hydrogen bond, Chemistry, Organic Chemistry, Isoquinolines, Drug Design, Molecular Medicine, Structure based, Efflux, Amyloid Precursor Protein Secretases
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16
المؤلفون: Ying-zi Xu, Kenichi Yakushijin, David A. Horne, Giao Phan
المصدر: Tetrahedron Letters. 35:351-354
مصطلحات موضوعية: Coupling (electronics), chemistry.chemical_compound, Chemical coupling, Bicyclic molecule, Computational chemistry, Stereochemistry, Chemistry, Organic Chemistry, Drug Discovery, Lactam, Biochemistry
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17
المؤلفون: Ying-Zi Xu, Eric Sandberg, Frederique Bard, Lan K. Nguyen, Caroline Garrido, Kelly Cockcroft, William A Wallace, Michael P. Bova, Chris M. Semko
المصدر: Journal of biomolecular screening. 16(5)
مصطلحات موضوعية: Integrins, Integrin, Immunoglobulins, Biochemistry, Jurkat cells, Analytical Chemistry, Cell Line, Small Molecule Libraries, Jurkat Cells, Mucoproteins, Addressin, Cell Adhesion, Humans, Cell adhesion, Receptor, biology, Dose-Response Relationship, Drug, Chemistry, Cell adhesion molecule, Adhesion, Ligand (biochemistry), Cell biology, High-Throughput Screening Assays, Kinetics, HEK293 Cells, Metals, biology.protein, Molecular Medicine, Cell Adhesion Molecules, Biotechnology
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18
المؤلفون: Ying-zi Xu, David A. Horne, K. Yakushijin
المصدر: Tetrahedron Letters. 34:6981-6984
مصطلحات موضوعية: chemistry.chemical_compound, Schiff base, chemistry, Organic Chemistry, Drug Discovery, Intermolecular force, Organic chemistry, Biochemistry, Cycloaddition
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19
المؤلفون: Judevin Lugar, Kevin P. Quinn, Anna Liao, Darren B. Dressen, Linda Chen, Thomas N. Thompson, Elizabeth J. Holsztynska, Francine S. Farouz, Whitney Dunn, Christopher Vandevert, Ying-Zi Xu, Michael Jefferies, Thorsett Eugene D, Mark Dreyer, Michael A. Pleiss, Ted Yednock, Andrei W. Konradi, Stephen B. Freedman, Linda Mutter, Semko Christopher M
المصدر: Bioorganicmedicinal chemistry letters. 21(6)
مصطلحات موضوعية: Pyrimidine, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Biological Availability, Pharmacology, Integrin alpha4beta1, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Pharmacokinetics, immune system diseases, Oral administration, Drug Discovery, Animals, Molecular Biology, Sheep, Drug discovery, Organic Chemistry, Antagonist, Biological activity, Asthma, Bioavailability, Disease Models, Animal, Pyrimidines, chemistry, Molecular Medicine
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20
المؤلفون: K. Yakushijin, David A. Horne, Ying-zi Xu
المصدر: ChemInform. 23
مصطلحات موضوعية: Chemistry, Organic chemistry, General Medicine, Link (knot theory)