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1
المؤلفون: Cheryl L. Walker, Richard C. Winneker, Magid Abou-Gharbia, Jerauld S. Skotnicki, Wenling Kao, Eugene L. Brown, Russell R. Broaddus, Bhuvanesh Dave, Adrienne S. McCampbell, Wei Liu, Kathryn A. Saraf, Ewa Wilson, Michelle L. Kimberland, Monette M. Cotreau, Sung E. Choe, Heather A. Harris, Scott A. Jelinsky, Judy S. Crabtree
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2
المؤلفون: Cheryl L. Walker, Richard C. Winneker, Magid Abou-Gharbia, Jerauld S. Skotnicki, Wenling Kao, Eugene L. Brown, Russell R. Broaddus, Bhuvanesh Dave, Adrienne S. McCampbell, Wei Liu, Kathryn A. Saraf, Ewa Wilson, Michelle L. Kimberland, Monette M. Cotreau, Sung E. Choe, Heather A. Harris, Scott A. Jelinsky, Judy S. Crabtree
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3
المؤلفون: Cheryl L. Walker, Richard C. Winneker, Magid Abou-Gharbia, Jerauld S. Skotnicki, Wenling Kao, Eugene L. Brown, Russell R. Broaddus, Bhuvanesh Dave, Adrienne S. McCampbell, Wei Liu, Kathryn A. Saraf, Ewa Wilson, Michelle L. Kimberland, Monette M. Cotreau, Sung E. Choe, Heather A. Harris, Scott A. Jelinsky, Judy S. Crabtree
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4
المؤلفون: Cheryl L. Walker, Richard C. Winneker, Magid Abou-Gharbia, Jerauld S. Skotnicki, Wenling Kao, Eugene L. Brown, Russell R. Broaddus, Bhuvanesh Dave, Adrienne S. McCampbell, Wei Liu, Kathryn A. Saraf, Ewa Wilson, Michelle L. Kimberland, Monette M. Cotreau, Sung E. Choe, Heather A. Harris, Scott A. Jelinsky, Judy S. Crabtree
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5
المؤلفون: Cheryl L. Walker, Richard C. Winneker, Magid Abou-Gharbia, Jerauld S. Skotnicki, Wenling Kao, Eugene L. Brown, Russell R. Broaddus, Bhuvanesh Dave, Adrienne S. McCampbell, Wei Liu, Kathryn A. Saraf, Ewa Wilson, Michelle L. Kimberland, Monette M. Cotreau, Sung E. Choe, Heather A. Harris, Scott A. Jelinsky, Judy S. Crabtree
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6
المؤلفون: Lloyd M. Garrick, John F. Mehlmann, Diane B. Hauze, Joshua E. Cottom, Daniel M. Green, Jeffrey C. Pelletier, Murty Chengalvala, Irene Feingold, Joseph T. Lundquist, John F. Rogers, Charles William Mann, Linda Shanno, Jay E. Wrobel, Christine Huselton, Wenling Kao, Kees Kenneth L
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:1986-1990
مصطلحات موضوعية: medicine.medical_specialty, Benzimidazole, Time Factors, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Gonadotropin-releasing hormone, Peptide hormone, Biochemistry, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, Heterocyclic Compounds, Oral administration, Internal medicine, Drug Discovery, medicine, Animals, Receptor, Molecular Biology, Volume of distribution, Chemistry, Organic Chemistry, Antagonist, Luteinizing Hormone, Rats, Bioavailability, Endocrinology, Models, Animal, Molecular Medicine, Benzimidazoles, Receptors, LHRH
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7
المؤلفون: Murty V. Chengalvala, Linda Shanno, Charles William Mann, Josh Cottom, Diane B. Hauze, Jay E. Wrobel, Irene Feingold, Jeffrey C. Pelletier, Gregory S. Kopf, Daniel M. Green, John A. Rogers, Wenling Kao, Christine Huselton, John F. Mehlmann, Joseph T. Lundquist, Lloyd M. Garrick, James W. Jetter
المصدر: Bioorganic & Medicinal Chemistry. 16:6617-6640
مصطلحات موضوعية: Male, endocrine system, medicine.medical_specialty, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Gonadotropin-releasing hormone, Methylation, Biochemistry, Piperazines, Gonadotropin-releasing hormone antagonist, Rats, Sprague-Dawley, Structure-Activity Relationship, Prostate cancer, In vivo, Internal medicine, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Receptor, Piperazine, Molecular Biology, Leuteinizing hormone, Molecular Structure, Chemistry, Organic Chemistry, Antagonist, Luteinizing Hormone, medicine.disease, Glycolates, Rats, Cross-Linking Reagents, Endocrinology, Molecular Medicine, Benzimidazoles, Receptors, LHRH, hormones, hormone substitutes, and hormone antagonists
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8
المؤلفون: Jill L. Hardenburg, John Rogers, Darlene C. Deecher, Francisco J. López, Emily S. Shen, Brian J. Arey, Jay Wrobel, James W Jetter, M. Claudia Perez, Daniel M. Green, Wenling Kao
المصدر: Bioorganic & Medicinal Chemistry. 10:639-656
مصطلحات موضوعية: Male, endocrine system, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Nitro compound, Pharmaceutical Science, Carboxamide, Sulfonic acid, Transfection, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, Inhibitory Concentration 50, Mice, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Thyroid-stimulating hormone, Testis, Drug Discovery, Cyclic AMP, Tumor Cells, Cultured, medicine, Animals, Humans, Receptor, Molecular Biology, Progesterone, Benzoic acid, chemistry.chemical_classification, Granulosa Cells, Chemistry, Organic Chemistry, Estrogen Antagonists, Receptors, Thyrotropin, Progesterone secretion, Rats, Benzamides, Receptors, FSH, Molecular Medicine, Female, Follicle Stimulating Hormone, Sulfonic Acids, Dimerization
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9
المؤلفون: Daniel M. Green, Wenling Kao, Jay E. Wrobel, John Rogers
المصدر: Synthetic Communications. 32:2695-2704
مصطلحات موضوعية: chemistry.chemical_classification, Follicle-stimulating hormone, Chemistry, Organic Chemistry, Antagonist, Organic chemistry, Moiety, Sulfonic acid, Protecting group, Isopropyl
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10
المؤلفون: John A. Rogers, Jamin Chi, Gi-Chung Chen, Li Di, James W. Jetter, M. Claudia Perez, Emily S. Shen, Wenling Kao, Jay E. Wrobel
المصدر: Bioorganicmedicinal chemistry. 14(16)
مصطلحات موضوعية: Agonist, endocrine system, Alkylation, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Substituent, Pharmaceutical Science, Hamster, CHO Cells, Biochemistry, Chemical synthesis, Cell Line, chemistry.chemical_compound, Follicle-stimulating hormone, Structure-Activity Relationship, Cricetinae, Drug Discovery, medicine, Cyclic AMP, Animals, Humans, Luciferases, Molecular Biology, Chinese hamster ovary cell, Organic Chemistry, Ovary, Biological activity, Recombinant Proteins, chemistry, Molecular Medicine, Receptors, FSH, Female, Thiazolidinediones, Follicle Stimulating Hormone, Follicle-stimulating hormone receptor
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11
المؤلفون: Richard W. Rees, Wenling Kao
المصدر: Prostaglandins. 16(3)
مصطلحات موضوعية: Thioketal, Prostaglandins E, Synthetic, chemistry.chemical_compound, Chemistry, Endocrinology, chemistry, Chemical Phenomena, Stereochemistry, Guinea Pigs, Animals, lipids (amino acids, peptides, and proteins), Biological Assay, Biochemistry