المؤلفون: Marchetti*, Kathryn A, Merrill, Nathan, Vandecan, Nathalie, Bao, Liwei, Cheng, Xu, Udager, Aaron, Herrel, Lindsey A, Montgomery, Jeffery, Hafez, Khaled, Morgan, Todd, Weizer, Alon, Alva, Ajjai, Soellner, Matthew, Merajver, Sofia, Kaffenberger, Samuel

المصدر: Journal of Urology ; volume 203, issue Supplement 4 ; ISSN 0022-5347 1527-3792

الاتاحة: http://dx.doi.org/10.1097/ju.0000000000000934.011
http://journals.lww.com/10.1097/JU.0000000000000934.011

المؤلفون: Mao, Wuxiang, Vandecan, Nathalie M., Bingham, Christopher R., Tsang, Pui Ki, Ulintz, Peter, Sexton, Rachel, Bochar, Daniel A., Merajver, Sofia D., Soellner, Matthew B.

المصدر: ACS Chemical Biology; 1/19/2024, Vol. 19 Issue 1, p110-116, 7p

المؤلفون: Mao, Wuxiang, Vandecan, Nathalie M., Bingham, Christopher R., Tsang, Pui Ki, Ulintz, Peter, Sexton, Rachel, Bochar, Daniel A., Merajver, Sofia D., Soellner, Matthew B.

المساهمون: National Institute of General Medical Sciences

المصدر: ACS Chemical Biology ; volume 19, issue 1, page 110-116 ; ISSN 1554-8929 1554-8937

الاتاحة: http://dx.doi.org/10.1021/acschembio.3c00548
https://pubs.acs.org/doi/pdf/10.1021/acschembio.3c00548

المؤلفون: Johnson, Taylor K., Bochar, Daniel A., Vandecan, Nathalie M., Furtado, Jessica, Agius, Michael P., Phadke, Sameer, Soellner, Matthew B.

مصطلحات موضوعية: Antagonism, Asciminib, Kinase, Chemical Engineering, Chemistry, Materials Science and Engineering, Engineering, Science

وصف الملف: application/pdf

Relation: Johnson, Taylor K.; Bochar, Daniel A.; Vandecan, Nathalie M.; Furtado, Jessica; Agius, Michael P.; Phadke, Sameer; Soellner, Matthew B. (2022). "Reply to Correspondence on “Synergy and Antagonism between Allosteric and Active-Site Inhibitors of Abl Tyrosine Kinase”." Angewandte Chemie 134(46): n/a-n/a.; https://hdl.handle.net/2027.42/175174; Angewandte Chemie; H. Huang, R. Zhao, B. M. Dickson, R. D. Skeel, C. B. Post, J. Phys. Chem. B 2012, 116, 4465 – 4475.; X. Wang, A. Roy, A. Hochhaus, H. M. Kantarjian, T.-T. Chen, N. P. Shah, Clin. Pharmacol. 2013, 5, 85 – 97.; A. Brown, Int. J. Mol. Sci. 2009, 10, 3457 – 3477.; D. Li, L. Chen, R. Wang, R. Liu, G. Ge, Anal. Chem. 2017, 89, 7130 – 7138.; T. P. Hughes, M. J. Maure, J. E. Cortes, et al., N. Engl. J. Med. 2019, 381, 2315 – 2326.; F. J. Adrián, Q. Ding, T. Sim, et al., Nat. Chem. Biol. 2006, 2, 95 – 102.; T.-C. Chou, Pharmacol. Rev. 2006, 58, 621 – 681.; T. K. Johnson, D. A. Bochar, N. M. Vandecan, J. Furtado, M. P. Agius, S. Phadke, M. B. Soellner, Angew. Chem. Int. Ed. 2021, 60, 20196 – 20199; Angew. Chem. 2021, 133, 20358 – 20361.; F. E. Kwarcinski, K. R. Brandvold, S. Phadke, O. M. Beleh, T. K. Johnson, J. L. Meagher, M. A. Seeliger, J. A. Stuckey, M. B. Soellner, ACS Chem. Biol. 2016, 11, 1296 – 1304.; M. P. Agius, K. S. Ko, T. K. Johnson, F. E. Kwarcinski, S. Phadke, E. J. Lachacz, M. B. Soellner, ACS Chem. Biol. 2019, 14, 1556 – 1563.; M. A. Seeliger, B. Nagar, F. Frank, X. Cao, M. N. Henderson, J. Kuriyan, Structure 2007, 15, 299 – 311.; B. J. Druker, M. Talpaz, D. J. Resta, et al., N. Engl. J. Med. 2001, 344, 1031 – 1037.; L. Skora, J. Mestan, D. Fabbro, W. Jahnke, S. Grzsiek, Proc. Natl. Acad. Sci. USA 2013, 110, E4437 – E4445.; Asciminib (SCEMBLIX®) prescribing information, Reference ID: 4880647, https://www.accessdata.fda.gov/drugsatfda_docs/label/2021/215358s000Orig1lbl.pdf (accessed June 29, 2022).; A. B. Patel, T. O’Hare, M. W. Deininger, Hematol. Oncol. Clin. North Am. 2017, 31, 589 – 612.; C. A. Eide, M. S. Zabriskie, S. L. S. Stevens, et al., Cancer Cell 2019, 36, 431 – 443.; H. J. G. Lindstrom, R. Friedman, BMC Cancer 2020, 20, 397.; J. D. Vasta, C. R. Corona, J. Wilkinson, et al., Cell Chem. Biol. 2018, 25, 206 – 214.; Cancer Dependency Map, https://depmap.org/portal/cell line/ACH-000983?tab=mutation (accessed June 29, 2022).

الاتاحة: https://hdl.handle.net/2027.42/175174
https://doi.org/10.1002/ange.202209518

المؤلفون: Phadke, Sameer, Lopez-Barcons, Lluis, Vandecan, Nathalie, Wu, Zhifen, Johnson, Taylor K., Lachacz, Eric J., Merajver, Sofia D., Soellner, Matthew B.

المساهمون: Breast Cancer Research Foundation, National Institutes of Health

المصدر: RSC Medicinal Chemistry ; volume 13, issue 1, page 64-71 ; ISSN 2632-8682

الاتاحة: http://dx.doi.org/10.1039/d1md00296a
http://pubs.rsc.org/en/content/articlepdf/2022/MD/D1MD00296A

المؤلفون: Johnson, Taylor K., Bochar, Daniel A., Vandecan, Nathalie M., Furtado, Jessica, Agius, Michael P., Phadke, Sameer, Soellner, Matthew B.

مصطلحات موضوعية: Abl, allostery, inhibitors, kinase, synergy, Materials Science and Engineering, Chemistry, Chemical Engineering, Engineering, Science

وصف الملف: application/pdf

Relation: Johnson, Taylor K.; Bochar, Daniel A.; Vandecan, Nathalie M.; Furtado, Jessica; Agius, Michael P.; Phadke, Sameer; Soellner, Matthew B. (2021). "Synergy and Antagonism between Allosteric and Active‐Site Inhibitors of Abl Tyrosine Kinase." Angewandte Chemie 133(37): 20358-20361.; https://hdl.handle.net/2027.42/169317; Angewandte Chemie; T. O’Hare, C. A. Eide, M. W. Deininger, Clin. Lymphoma Myeloma Leuk. 2017, 7, S120 – S130.; J. E. Cortes, D. W. Kim, J. Pinilla-Ibarz, P. le Coutre, R. Paquette, C. Chuah, F. E. Nicolini, J. F. Apperley, H. J. Khoury, M. Talpaz, J. DiPersio, J. D. DeAngelo, E. Abruzzese, D. Rea, M. Baccarani, M. C. Müller, C. Gambacorti-Passerini, S. Wong, S. Lustgarten, V. M. Rivera, T. Clackson, C. D. Turner, F. G. Haluska, F. Guilhot, M. W. Deininger, A. Hochhaus, T. Hughes, J. M. Goldman, N. P. Shah, H. Kantarjian, N. Engl. J. Med. 2013, 369, 1783 – 1796.; F. J. Adrián, Q. Ding, T. Sim, A. Velentza, C. Sloan, Y. Liu, G. Zhang, W. Hur, S. Ding, P. Manley, J. Mestan, D. Fabbro, N. S. Gray, Nat. Chem. Biol. 2006, 2, 95 – 102.; R. E. Iacob, J. Zhang, N. S. Gray, J. R. Engen, PLoS One 2011, 6, e15929.; J. Zhang, F. J. Adrián, W. Jahnke, S. W. Cowan-Jacob, A. G. Li, R. E. Iacob, T. Sim, J. Powers, C. Dierks, F. Sun, G. R. Guo, Q. Ding, B. Okram, Y. Choi, A. Wojciechowski, X. Deng, G. Liu, G. Fendrich, A. Strauss, N. Vajpai, S. Grzesiek, T. Tuntland, Y. Liu, B. Bursulaya, M. Azam, P. W. Manley, J. R. Engen, G. Q. Daley, M. Warmuth, N. S. Gray, Nature 2010, 463, 501 – 506.; B. Nagar, O. Hantschel, M. A. Young, K. Scheffzek, D. Veach, W. Bornmann, B. Clarkson, G. Superti-Furga, J. Kuriyan, Cell 2003, 112, 859 – 871.; T.-C. Chou, Cancer Res. 2010, 70, 440 – 446.; M. P. Agius, K. S. Ko, T. K. Johnson, F. E. Kwarcinski, S. Phadke, E. J. Lachacz, M. B. Soellner, ACS Chem. Biol. 2019, 14, 1556 – 1563.; T.-C. Chou, Pharmacol. Rev. 2007, 58, 621 – 681.; L. Skora, J. Mestan, D. Fabbro, W. Jahnke, S. Grzesiek, Proc. Natl. Acad. Sci. USA 2013, 110, E4437 - E4445.; D. Fabbro, P. W. Manley, W. Jahnke, J. Liebetanz, A. Szyttenholm, G. Fendrich, A. Strauss, J. Zhang, N. S. Gray, F. Adrian, M. Warmuth, X. Pelle, R. Grotzfeld, F. Berst, A. Marzinzik, S. W. Cowan-Jacob, P. Furet, J. Mestan, Biochim. Biophys. Acta Proteins Proteomics 2010, 1804, 454 – 462.; M. Khateb, N. Ruimi, H. Khamisie, Y. Najajreh, A. Mian, A. Metodieva, M. Ruthardt, J. Mahajna, BMC Cancer 2012, 12, 563 – 572.; R. Kurzrock, J. U. Gutterman, M. Talpaz, N. Engl. J. Med. 1988, 319, 990 – 998.; B. J. Druker, F. Guilhot, S. G. O’Brien, I. Gathmann, H. Kantarjian, N. Gattermann, M. W. N. Deininger, R. T. Silver, J. M. Goldman, R. M. Stone, F. Cervantes, A. Hochhaus, B. L. Powell, J. L. Gabrilove, P. Rousselot, J. Reiffers, J. J. Cornelissen, T. Hughes, H. Agis, T. Fischer, G. Verhoef, J. Shepherd, G. Saglio, A. Gratwohl, J. L. Nielsen, J. P. Radich, B. Simonsson, K. Taylor, M. Baccarani, L. Letvak, R. A. Larson, N. Engl. J. Med. 2006, 355, 2408 – 2417.; V. Prasad, S. Mailankody, JAMA J. Am. Med. Assoc. 2014, 311, 353 – 354.; F. E. Kwarcinski, K. R. Brandvold, S. Phadke, O. M. Beleh, T. K. Johnson, J. L. Meagher, M. A. Seeliger, J. A. Stuckey, M. B. Soellner, ACS Chem. Biol. 2016, 11, 1296 – 1304.; O. Hantschel, B. Nagar, S. Guettler, J. Kretzschmar, K. Dorey, J. Kuriyan, G. Superti-Furga, Cell 2003, 112, 845 – 857.; S. Panjarianm, R. E. Iacob, S. Chen, T. E. Wales, J. R. Engen, T. E. Smithgall, J. Biol. Chem. 2013, 288, 6116 – 6129.; F. Grebien, O. Hantschel, J. Wojcik, I. Kaupe, B. Kovacic, A. M. Wyrzucki, G. D. Gish, S. Cerny-Reiterer, A. Koide, H. Beug, T. Pawson, P. Valent, S. Koide, G. Superti-Furga, Cell 2011, 147, 306 – 319.; P. Filippakopoulos, M. Kofler, O. Hantschel, G. D. Gish, F. Grebien, E. Salah, P. Neudecker, L. E. Kay, B. E. Turk, G. Superti-Furga, T. Pawson, S. Knapp, Cell 2016, 134, 793 – 803.; T.-C. Chou, P. Talalay, Adv. Enzyme Regul. 1984, 22, 27 – 55.

الاتاحة: https://hdl.handle.net/2027.42/169317
https://doi.org/10.1002/ange.202105351

المؤلفون: Merrill, Nathan M., Lachacz, Eric J., Vandecan, Nathalie M., Ulintz, Peter J., Bao, Liwei, Lloyd, John P., Yates, Joel A., Morikawa, Aki, Merajver, Sofia D., Soellner, Matthew B.

المساهمون: Breast Cancer Relief Foundation, National Cancer Institute

المصدر: Breast Cancer Research and Treatment ; volume 179, issue 2, page 337-347 ; ISSN 0167-6806 1573-7217

الاتاحة: http://dx.doi.org/10.1007/s10549-019-05473-9
http://link.springer.com/content/pdf/10.1007/s10549-019-05473-9.pdf
http://link.springer.com/article/10.1007/s10549-019-05473-9/fulltext.html

المؤلفون: Phadke, Sameer, Lopez-Barcons, Lluis, Vandecan, Nathalie, Wu, Zhifen, Johnson, Taylor K., Lachacz, Eric J., Merajver, Sofia D., Soellner, Matthew B.

المصدر: MedChemComm; 2022, Vol. 13 Issue: 1 p64-71, 8p

المؤلفون: Merrill, Nathan M., Lachacz, Eric J., Vandecan, Nathalie M., Ulintz, Peter J., Bao, Liwei, Lloyd, John P., Yates, Joel A., Morikawa, Aki, Merajver, Sofia D., Soellner, Matthew B.

المصدر: Breast Cancer Research & Treatment; Jan2020, Vol. 179 Issue 2, p337-347, 11p

المؤلفون: Merrill, Nathan M.^1,2 (AUTHOR), Kaffenberger, Samuel D.¹ (AUTHOR), Bao, Liwei² (AUTHOR), Vandecan, Nathalie³ (AUTHOR), Goo, Laura^1,2 (AUTHOR), Apfel, Athena² (AUTHOR), Cheng, Xu² (AUTHOR), Qin, Zhaoping² (AUTHOR), Liu, Chia-Jen² (AUTHOR), Bankhead, Armand^4,5 (AUTHOR), Wang, Yin² (AUTHOR), Kathawate, Varun² (AUTHOR), Tudrick, Lila² (AUTHOR), Serhan, Habib A.² (AUTHOR), Farah, Zackariah² (AUTHOR), Ellimoottil, Chad⁶ (AUTHOR), Hafez, Khaled S.⁶ (AUTHOR), Herrel, Lindsey A.^1,6 (AUTHOR), Montgomery, Jeffrey S.^1,6 (AUTHOR), Morgan, Todd M.^1,6 (AUTHOR)

المصدر: European Urology. Nov2024, Vol. 86 Issue 5, p434-444. 11p.

مصطلحات موضوعية: *PEARSON correlation (Statistics), *CANCER invasiveness, *DRUG use testing, *INVESTIGATIONAL therapies, *MEDICAL screening, *BLADDER cancer