-
1Academic Journal
المؤلفون: Di Maria, Salvatore, Passannanti, Raffaele, Poggialini, Federica, Vagaggini, Chiara, Serafinelli, Alessia, Bianchi, Elena, Governa, Paolo, Botta, Lorenzo, Maga, Giovanni, Crespan, Emmanuele, Manetti, Fabrizio, Dreassi, Elena, Musumeci, Francesca, Carbone, Anna, Schenone, Silvia
المساهمون: Di Maria, Salvatore, Passannanti, Raffaele, Poggialini, Federica, Vagaggini, Chiara, Serafinelli, Alessia, Bianchi, Elena, Governa, Paolo, Botta, Lorenzo, Maga, Giovanni, Crespan, Emmanuele, Manetti, Fabrizio, Dreassi, Elena, Musumeci, Francesca, Carbone, Anna, Schenone, Silvia
مصطلحات موضوعية: Molecular hybridization, Hepatocellular carcinoma, Tyrosine kinases, Src inhibitors, pyrazolo[3,4-d]pyrimidines
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/39406114; info:eu-repo/semantics/altIdentifier/wos/WOS:001336529800001; volume:280; numberofpages:15; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; https://hdl.handle.net/11365/1275614; https://www.sciencedirect.com/science/article/pii/S0223523424008109?via=ihub
-
2Academic Journal
المؤلفون: Cesarini, Silvia, Vicenti, Ilaria, Poggialini, Federica, Filippi, Silvia, Mancin, Eleonora, Fiaschi, Lia, De Marchi, Elisa, Giammarino, Federica, Vagaggini, Chiara, Bizzarri, Bruno Mattia, Saladino, Raffaele, Dreassi, Elena, Zazzi, Maurizio, Botta, Lorenzo
المساهمون: Cesarini, Silvia, Vicenti, Ilaria, Poggialini, Federica, Filippi, Silvia, Mancin, Eleonora, Fiaschi, Lia, De Marchi, Elisa, Giammarino, Federica, Vagaggini, Chiara, Bizzarri, Bruno Mattia, Saladino, Raffaele, Dreassi, Elena, Zazzi, Maurizio, Botta, Lorenzo
مصطلحات موضوعية: anticancer activity, privileged scaffold, pyridine, pyrimidine, scaffold morphing, triazines
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/38611732; info:eu-repo/semantics/altIdentifier/wos/WOS:001201226800001; volume:29; issue:7; numberofpages:20; journal:MOLECULES; https://hdl.handle.net/11365/1262275; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85190364623; https://www.mdpi.com/1420-3049/29/7/1452; https://www.ncbi.nlm.nih.gov/pmc/articles/PMC11013010/
-
3Academic JournalIdentification of Novel Non-Nucleoside Inhibitors of Zika Virus NS5 Protein Targeting MTase Activity
المؤلفون: Fiorucci, Diego, Meaccini, Micaela, Poli, Giulio, Stincarelli, Maria, Alfreda, Vagaggini, Chiara, Giannecchini, Simone, Sutto-Ortiz, Priscila, Canard, Bruno, Decroly, Etienne, Dreassi, Elena, Brai, Annalaura, Botta, Maurizio
المساهمون: Università degli Studi di Siena = University of Siena (UNISI), Università degli Studi di Firenze = University of Florence = Université de Florence (UniFI), Architecture et fonction des macromolécules biologiques (AFMB), Aix Marseille Université (AMU)-Centre National de la Recherche Scientifique (CNRS)-Institut National de Recherche pour l’Agriculture, l’Alimentation et l’Environnement (INRAE)
المصدر: ISSN: 1661-6596.
مصطلحات موضوعية: NS5, non-nucleoside inhibitors, ZIKV, DENV, antiviral agents, LD50, [CHIM.THER]Chemical Sciences/Medicinal Chemistry, [SDV.MHEP.ME]Life Sciences [q-bio]/Human health and pathology/Emerging diseases, [SDV.MHEP.MI]Life Sciences [q-bio]/Human health and pathology/Infectious diseases, [SDV.MP.VIR]Life Sciences [q-bio]/Microbiology and Parasitology/Virology
-
4Academic Journal
المؤلفون: Di Stefano, Miriana, Masoni, Samuele, Bononi, Giulia, Poli, Giulio, Galati, Salvatore, Gado, Francesca, Manzi, Simone, Vagaggini, Chiara, Brai, Annalaura, Caligiuri, Isabella, Asif, Kanwal, Rizzolio, Flavio, Macchia, Marco, Chicca, Andrea, Sodi, Andrea, Di Bussolo, Valeria, Minutolo, Filippo, Meier, Philip, Gertsch, Jürg, Granchi, Carlotta, Dreassi, Elena, Tuccinardi, Tiziano
المصدر: Di Stefano, Miriana; Masoni, Samuele; Bononi, Giulia; Poli, Giulio; Galati, Salvatore; Gado, Francesca; Manzi, Simone; Vagaggini, Chiara; Brai, Annalaura; Caligiuri, Isabella; Asif, Kanwal; Rizzolio, Flavio; Macchia, Marco; Chicca, Andrea; Sodi, Andrea; Di Bussolo, Valeria; Minutolo, Filippo; Meier, Philip; Gertsch, Jürg; Granchi, Carlotta; . (2024). Design, synthesis, ADME and biological evaluation of benzylpiperidine and benzylpiperazine derivatives as novel reversible monoacylglycerol lipase (MAGL) inhibitors. European journal of medicinal chemistry, 263(115916), p. 115916. Elsevier 10.1016/j.ejmech.2023.115916
مصطلحات موضوعية: 570 Life sciences, biology, 610 Medicine & health
وصف الملف: application/pdf
Relation: https://boris.unibe.ch/189143/
-
5Academic Journal
المؤلفون: Saletti, Mario, Paolino, Marco, Venditti, Jacopo, Bonechi, Claudia, Giuliani, Germano, Lamponi, Stefania, Tassone, Giusy, Boccia, Antonella, Botta, Chiara, Blancafort, Lluís, Poggialini, Federica, Vagaggini, Chiara, Cappelli, Andrea
المساهمون: Ministero dell'Università e della Ricerca, Università degli Studi di Siena
المصدر: ChemBioChem ; volume 25, issue 8 ; ISSN 1439-4227 1439-7633
-
6Academic Journal
المؤلفون: Vagaggini, Chiara, Petroni, Debora, D'Agostino, Ilaria, Poggialini, Federica, Cavallini, Chiara, Cianciusi, Annarita, Salis, Annalisa, D'Antona, Lucia, Francesconi, Valeria, Manetti, Fabrizio, Damonte, Gianluca, Musumeci, Francesca, Menichetti, Luca, Dreassi, Elena, Carbone, Anna, Schenone, Silvia
المصدر: Drug Development Research ; volume 85, issue 1 ; ISSN 0272-4391 1098-2299
-
7Academic Journal
المؤلفون: Maresca, Luisa, Crivaro, Enrica, Migliorini, Francesca, Anichini, Giulia, Giammona, Alessandro, Pepe, Sara, Poggialini, Federica, Vagaggini, Chiara, Giannini, Giuseppe, Sestini, Serena, Borgognoni, Lorenzo, Lapucci, Andrea, Dreassi, Elena, Taddei, Maurizio, Manetti, Fabrizio, Petricci, Elena, Stecca, Barbara
المساهمون: Maresca, Luisa, Crivaro, Enrica, Migliorini, Francesca, Anichini, Giulia, Giammona, Alessandro, Pepe, Sara, Poggialini, Federica, Vagaggini, Chiara, Giannini, Giuseppe, Sestini, Serena, Borgognoni, Lorenzo, Lapucci, Andrea, Dreassi, Elena, Taddei, Maurizio, Manetti, Fabrizio, Petricci, Elena, Stecca, Barbara
مصطلحات موضوعية: GLI transcription factor, cancer, melanoma, small molecule inhibitors
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/37473878; info:eu-repo/semantics/altIdentifier/wos/WOS:001055429300001; volume:195; numberofpages:15; journal:PHARMACOLOGICAL RESEARCH; https://hdl.handle.net/11365/1239754; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85165911129; https://www.sciencedirect.com/science/article/pii/S1043661823002141
-
8Academic Journal
المؤلفون: Poggialini, Federica, Vagaggini, Chiara, Brai, Annalaura, Pasqualini, Claudia, Crespan, Emmanuele, Maga, Giovanni, Perini, Cecilia, Cabella, Noemi, Botta, Lorenzo, Musumeci, Francesca, Frosini, Maria, Schenone, Silvia, Dreassi, Elena
المساهمون: Poggialini, Federica, Vagaggini, Chiara, Brai, Annalaura, Pasqualini, Claudia, Crespan, Emmanuele, Maga, Giovanni, Perini, Cecilia, Cabella, Noemi, Botta, Lorenzo, Musumeci, Francesca, Frosini, Maria, Schenone, Silvia, Dreassi, Elena
مصطلحات موضوعية: ADME, antiproliferative activity, c-Src/Abl dual inhibitor, glioblastoma, pyrazolo[3,4-d]pyrimidine, tyrosine kinase
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/36839775; info:eu-repo/semantics/altIdentifier/wos/WOS:000939969900001; volume:15; issue:2; journal:PHARMACEUTICS; https://hdl.handle.net/11365/1259735; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85149125372; https://www.mdpi.com/1999-4923/15/2/453
-
9Academic Journal
المؤلفون: Brai, Annalaura, Poggialini, Federica, Vagaggini, Chiara, Pasqualini, Claudia, Simoni, Sauro, Francardi, Valeria, Dreassi, Elena
المساهمون: Brai, Annalaura, Poggialini, Federica, Vagaggini, Chiara, Pasqualini, Claudia, Simoni, Sauro, Francardi, Valeria, Dreassi, Elena
مصطلحات موضوعية: 3R principle, LD50, Tenebrio molitor, animal model, antiviral, metabolism, toxicity assessment
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/36768618; info:eu-repo/semantics/altIdentifier/wos/WOS:000929606300001; volume:24; issue:3; firstpage:1; lastpage:11; numberofpages:11; journal:INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES; https://hdl.handle.net/11365/1236077; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85147901944; https://www.mdpi.com/1422-0067/24/3/2296; https://www.ncbi.nlm.nih.gov/pmc/articles/PMC9917132/
-
10Academic Journal
المؤلفون: Brai, Annalaura, Brogi, Edoardo, Tarchi, Franca, Poggialini, Federica, Vagaggini, Chiara, Simoni, Sauro, Francardi, Valeria, Dreassi, Elena
المصدر: Foods; Jan2025, Vol. 14 Issue 2, p325, 14p
-
11Academic Journal
المؤلفون: Murthy, Sudarshan, Nizi, Maria Giulia, Venkannagari, Harikanth, Prunskaite-Hyyryläinen, Renata, Dreassi, Elena, Lüscher, Bernhard, Korn, Patricia, Tabarrini, Oriana, Lehtiö, Lari, Maksimainen, Mirko M., Massari, Serena, Alaviuhkola, Juho, Lippok, Barbara E., Vagaggini, Chiara, Sowa, Sven T., Galera-Prat, Albert, Ashok, Yashwanth
المصدر: Journal of medicinal chemistry 66(2), 1301-1320 (2023). doi:10.1021/acs.jmedchem.2c01460
مصطلحات موضوعية: info:eu-repo/classification/ddc/610
جغرافية الموضوع: DE
Relation: info:eu-repo/semantics/altIdentifier/issn/0022-2623; info:eu-repo/semantics/altIdentifier/issn/0095-9065; info:eu-repo/semantics/altIdentifier/issn/1943-2992; info:eu-repo/semantics/altIdentifier/wos/WOS:000910959600001; info:eu-repo/semantics/altIdentifier/issn/1520-4804; info:eu-repo/semantics/altIdentifier/pmid/pmid:36598465; https://publications.rwth-aachen.de/record/949222; https://publications.rwth-aachen.de/search?p=id:%22RWTH-2023-01636%22
-
12Academic Journal
المؤلفون: Murthy, Sudarshan, Nizi, Maria Giulia, Maksimainen, Mirko M., Massari, Serena, Alaviuhkola, Juho, Lippok, Barbara E., Vagaggini, Chiara, Sowa, Sven T., Galera-Prat, Albert, Ashok, Yashwanth, Venkannagari, Harikanth, Prunskaite-Hyyryläinen, Renata, Dreassi, Elena, Lüscher, Bernhard, Korn, Patricia, Tabarrini, Oriana, Lehtiö, Lari
المساهمون: Sigrid Jus?liuksen S??ti, Deutsche Forschungsgemeinschaft, Jane ja Aatos Erkon S??ti, Magnus Ehrnroothin S??ti
المصدر: Journal of Medicinal Chemistry ; volume 66, issue 2, page 1301-1320 ; ISSN 0022-2623 1520-4804
-
13Conference
المؤلفون: Vezzoli Miriana, Orro Alessandro, Trombetti Gabriele, Poggialini Francesca, Vagaggini Chiara, Dreassi Elena, Schenone Silvia, Fossa Paola, Carbone Anna, D’Ursi Pasqualina
المساهمون: Vezzoli, Miriana, Orro, Alessandro, Trombetti, Gabriele, Poggialini, Francesca, Vagaggini, Chiara, Dreassi, Elena, Schenone, Silvia, Fossa, Paola, Carbone, Anna, D’Ursi, Pasqualina
مصطلحات موضوعية: Rational design, AI assisted drug design
وصف الملف: ELETTRONICO
Relation: ispartofbook:Abstract Book 20th Annual Meeting of the Bioinformatics Italian Society; 20th Annual Meeting of the Bioinformatics Italian Society; firstpage:1; lastpage:1; numberofpages:1; https://hdl.handle.net/11567/1174676
الاتاحة: https://hdl.handle.net/11567/1174676
-
14Academic Journal
المؤلفون: Bononi, Giulia, Di Stefano, Miriana, Poli, Giulio, Ortore, Gabriella, Meier, Philip, Masetto, Francesca, Caligiuri, Isabella, Rizzolio, Flavio, Macchia, Marco, Chicca, Andrea, Avan, Amir, Giovannetti, Elisa, Vagaggini, Chiara, Brai, Annalaura, Dreassi, Elena, Valoti, Massimo, Minutolo, Filippo, Granchi, Carlotta, Gertsch, Jürg, Tuccinardi, Tiziano
المساهمون: Bononi, Giulia, Di Stefano, Miriana, Poli, Giulio, Ortore, Gabriella, Meier, Philip, Masetto, Francesca, Caligiuri, Isabella, Rizzolio, Flavio, Macchia, Marco, Chicca, Andrea, Avan, Amir, Giovannetti, Elisa, Vagaggini, Chiara, Brai, Annalaura, Dreassi, Elena, Valoti, Massimo, Minutolo, Filippo, Granchi, Carlotta, Gertsch, Jürg, Tuccinardi, Tiziano
Relation: info:eu-repo/semantics/altIdentifier/pmid/35522977; info:eu-repo/semantics/altIdentifier/wos/WOS:000808007900009; volume:65; issue:10; firstpage:7118; lastpage:7140; numberofpages:23; journal:JOURNAL OF MEDICINAL CHEMISTRY; https://hdl.handle.net/11568/1162652; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85131106451
-
15Academic Journal
المؤلفون: Marinacci, Beatrice, D'Agostino, Ilaria, Angeli, Andrea, Carradori, Simone, Melfi, Francesco, Grande, Rossella, Corsiani, Micol, Ferraroni, Marta, Agamennone, Mariangela, Tondo, Anna Rita, Zara, Susi, Puca, Valentina, Pellegrini, Benedetta, Vagaggini, Chiara, Dreassi, Elena, Patrauchan, Marianna A., Capasso, Clemente, Nicolotti, Orazio, Carta, Fabrizio, Supuran, Claudiu T.
المصدر: Journal of Medicinal Chemistry; 11/14/2024, Vol. 67 Issue 21, p19077-19102, 26p
-
16Academic Journal
المؤلفون: Brai, Annalaura, Neri, Cassia, Tarchi, Franca, Poggialini, Federica, Vagaggini, Chiara, Frosinini, Riccardo, Simoni, Sauro, Francardi, Valeria, Dreassi, Elena
المصدر: Foods; Nov2024, Vol. 13 Issue 21, p3450, 16p
مصطلحات موضوعية: EDIBLE insects, METABOLITES, FOOD industry, TENEBRIO molitor, MONOUNSATURATED fatty acids, TREHALOSE
-
17Academic Journal
المؤلفون: Maramai, Samuele, Saletti, Mario, Paolino, Marco, Giuliani, Germano, Cazzola, Jessica, Spaiardi, Paolo, Talpo, Francesca, Frosini, Maria, Pifferi, Alice, Ballarotto, Marco, Carotti, Andrea, Poggialini, Federica, Vagaggini, Chiara, Dreassi, Elena, Giorgi, Gianluca, Dondio, Giulio, Cappelli, Andrea, Rosario Biella, Gerardo, Anzini, Maurizio
المساهمون: Maramai, Samuele, Saletti, Mario, Paolino, Marco, Giuliani, Germano, Cazzola, Jessica, Spaiardi, Paolo, Talpo, Francesca, Frosini, Maria, Pifferi, Alice, Ballarotto, Marco, Carotti, Andrea, Poggialini, Federica, Vagaggini, Chiara, Dreassi, Elena, Giorgi, Gianluca, Dondio, Giulio, Cappelli, Andrea, Rosario Biella, Gerardo, Anzini, Maurizio
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:001298108400001; volume:112; journal:BIOORGANIC & MEDICINAL CHEMISTRY; https://hdl.handle.net/11391/1579815; https://www.sciencedirect.com/science/article/pii/S0968089624002864?via=ihub
-
18Academic Journal
المؤلفون: Balestri, Lorenzo J. I., D’Agostino, Ilaria, Rango, Enrico, Vagaggini, Chiara, Marchitiello, Rosalba, Mariotti, Melinda, Casian, Alexandru, Deodato, Davide, Truglio, Giuseppina I., Orofino, Francesco, Sanguinetti, Maurizio, Bugli, Francesca, Botta, Lorenzo, Dreassi, Elena
المصدر: Molecular Diversity ; volume 26, issue 6, page 3399-3409 ; ISSN 1381-1991 1573-501X
-
19Periodical
المؤلفون: Marinacci, Beatrice, D’Agostino, Ilaria, Angeli, Andrea, Carradori, Simone, Melfi, Francesco, Grande, Rossella, Corsiani, Micol, Ferraroni, Marta, Agamennone, Mariangela, Tondo, Anna Rita, Zara, Susi, Puca, Valentina, Pellegrini, Benedetta, Vagaggini, Chiara, Dreassi, Elena, Patrauchan, Marianna A., Capasso, Clemente, Nicolotti, Orazio, Carta, Fabrizio, Supuran, Claudiu T.
المصدر: Journal of Medicinal Chemistry; November 2024, Vol. 67 Issue: 21 p19077-19102, 26p
-
20Academic Journal
المصدر: International Journal of Molecular Sciences; Jul2024, Vol. 25 Issue 14, p7588, 17p
مصطلحات موضوعية: FOOD chemistry, ESSENTIAL amino acids, FUNCTIONAL analysis, UNSATURATED fatty acids, METABOLITES, MARINE algae, FLAXSEED
مصطلحات جغرافية: ASIA