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1Academic Journal
المؤلفون: Srinivasa P S Rao, Suresh B Lakshminarayana, Jan Jiricek, Marcel Kaiser, Ryan Ritchie, Elmarie Myburgh, Frantisek Supek, Tove Tuntland, Advait Nagle, Valentina Molteni, Pascal Mäser, Jeremy C Mottram, Michael P Barrett, Thierry T Diagana
المصدر: Tropical Medicine and Infectious Disease; Volume 5; Issue 1; Pages: 28
مصطلحات موضوعية: sleeping sickness, drug discovery, Trypanosoma growth inhibitors
وصف الملف: application/pdf
Relation: Neglected and Emerging Tropical Diseases; https://dx.doi.org/10.3390/tropicalmed5010028
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2Supplementary Table 3 from Dual ALK and CDK4/6 Inhibition Demonstrates Synergy against Neuroblastoma
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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3Supplementary Table 1 from Dual ALK and CDK4/6 Inhibition Demonstrates Synergy against Neuroblastoma
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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4
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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5Supplementary Table 4 from Dual ALK and CDK4/6 Inhibition Demonstrates Synergy against Neuroblastoma
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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6
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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7
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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8
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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9
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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10Supplementary Table 2 from Dual ALK and CDK4/6 Inhibition Demonstrates Synergy against Neuroblastoma
المؤلفون: Yaël P. Mossé, Jennifer L. Harris, Nanxin Li, Shiva Krupa, You Qun He, Giordano Caponigro, Sunkyu Kim, Tove Tuntland, Kathryn B. Grandinetti, Edward Ainscow, Timothy R. Smith, Frederick J. King, Lori S. Hart, Theodore D. Hansel, Renata Sano, Nicole R. Infarinato, Hannah T. Ryles, Kateryna Krytska, Andrew C. Wood
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11
المؤلفون: Glen Spraggon, Smith Jeffrey M, Chianelli Donatella, Advait Nagle, Christian Wiesmann, Xiaodong Liu, Yongping Xie, Richard J. Sciotti, Todd Groessl, Kevin Johnson, Xianzhong Liu, Celine Be, Christopher Thompson, Yin H. Lai, Jan Jiricek, Patrick J Rudewicz, Brandon S. Pybus, Casey J. N. Mathison, Valentina Molteni, Honnappa Srinivas, Richard Glynne, Jaime Ballard, Agnes Biggart, Diana Caridha, Andreas Hein, Ashley Mitchell Berman, Mu-Yun Gao, Lauren C. Davis, Michael Shapiro, Michael Gibney, Yen Liang Chen, Vince Yeh, Fabian K. Eggimann, Badry Bursulaya, Mara Kreishman-Deitrick, Lerario Isabelle K, Fang Liang, Shilpi Khare, Wendy Richmond, Srinivasa P. S. Rao, Frantisek Supek, Tove Tuntland, Alexandre Luneau
المصدر: Journal of Medicinal Chemistry
مصطلحات موضوعية: Chagas disease, Antiprotozoal Agents, Drug Annotation, 01 natural sciences, Rats, Sprague-Dawley, Mice, 03 medical and health sciences, Dogs, parasitic diseases, Drug Discovery, medicine, Animals, Humans, African trypanosomiasis, Oxazoles, Leishmania major, 030304 developmental biology, Mice, Inbred BALB C, 0303 health sciences, Chemistry, Leishmania tarentolae, Leishmaniasis, Triazoles, medicine.disease, Virology, Rats, 0104 chemical sciences, 3. Good health, Macaca fascicularis, 010404 medicinal & biomolecular chemistry, Pyrimidines, Visceral leishmaniasis, Liver, Proteasome, Proteasome inhibitor, Leishmaniasis, Visceral, Molecular Medicine, Proteasome Inhibitors, Leishmania donovani, Clearance, medicine.drug
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المؤلفون: W. Perry Gordon, Tove Tuntland, Shelly Meeusen, Leah Clemmer, Sara Da Ros, Laura Bordone, Robert Hill, Thomas Hollenbeck, John W. Fathman, Kenneth Ng, Sheryll Espinola, Xiaohui He, Bo Liu, John Nelson, Maya Iskandar, Xue-Feng Zhu, Vân Nguyen-Tran, Andreas Kreusch, David C.S. Huang, Songchun Jiang, Yong Jia, Badry Bursulaya, Janine E. Baaten, Jian Shi, Mu-Yun Gao, Tao Jiang, Barun Okram, Glen Spraggon, Pierre-Yves Michellys, Hong Liu
المصدر: ACS Medicinal Chemistry Letters. 8:1048-1053
مصطلحات موضوعية: 0301 basic medicine, Kinase, Organic Chemistry, Pattern recognition receptor, Biology, Biochemistry, digestive system diseases, RIPK2, Serine, 03 medical and health sciences, 030104 developmental biology, In vivo, NOD2, Drug Discovery, Tyrosine kinase, Ex vivo
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المؤلفون: Yael P. Mosse, You Qun He, Hannah T. Ryles, Renata Sano, Lori S. Hart, Nicole R. Infarinato, Theodore D. Hansel, Kateryna Krytska, Giordano Caponigro, Timothy R. Smith, Kathryn B. Grandinetti, Frederick J. King, Edward K. Ainscow, Sunkyu Kim, Shiva Krupa, Tove Tuntland, Andrew C. Wood, Jennifer L. Harris, Nanxin Li
المصدر: Clinical Cancer Research. 23:2856-2868
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, biology, Ceritinib, Cyclin-dependent kinase 4, medicine.drug_class, Pharmacology, medicine.disease, Pediatric cancer, ALK inhibitor, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Oncology, hemic and lymphatic diseases, 030220 oncology & carcinogenesis, Neuroblastoma, biology.protein, medicine, Anaplastic lymphoma kinase, Cyclin-dependent kinase 6, Combination drug, medicine.drug
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المؤلفون: Thierry T. Diagana, Valentina Molteni, Advait Nagle, Jeremy C. Mottram, Pascal Mäser, Jan Jiricek, Ryan Ritchie, Srinivasa P. S. Rao, Frantisek Supek, Elmarie Myburgh, Marcel Kaiser, Suresh B. Lakshminarayana, Michael P. Barrett, Tove Tuntland
المصدر: Tropical Medicine and Infectious Disease; Volume 5; Issue 1; Pages: 28
Tropical Medicine and Infectious Disease, Vol 5, Iss 1, p 28 (2020)
Tropical Medicine and Infectious Diseaseمصطلحات موضوعية: 0301 basic medicine, Chagas disease, sleeping sickness, 030231 tropical medicine, lcsh:Medicine, drug discovery, Trypanosoma growth inhibitors, Pharmacology, Article, 03 medical and health sciences, 0302 clinical medicine, In vivo, parasitic diseases, Medicine, Potency, African trypanosomiasis, trypanosoma growth inhibitors, Mode of action, General Immunology and Microbiology, business.industry, lcsh:R, Public Health, Environmental and Occupational Health, Trypanosoma brucei rhodesiense, medicine.disease, In vitro, 3. Good health, 030104 developmental biology, Infectious Diseases, Proteasome, business
وصف الملف: application/pdf
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المؤلفون: Advait Nagle, Ben G. Wen, Srinivasa P. S. Rao, Monique Stinson, Glenn C. Federe, Richard Glynne, Yin H. Lai, Ianne C. Rivera, Ansgar Brock, Michael Shapiro, Hazel X. Y. Koh, John D. Venable, Jaime Ballard, J. Robert Gillespie, Badry Bursulaya, Glen Spraggon, Xianzhong Liu, Mu-Yun Gao, Vince Yeh, Tove Tuntland, Fang Liang, S. Whitney Barnes, Todd Groessl, Shilpi Khare, Elmarie Myburgh, Agnes Biggart, Lauren C. Davis, Jocelyn Tan, Pranab Mishra, Frantisek Supek, Casey J. N. Mathison, Valentina Molteni, Jeremy C. Mottram, Frederick S. Buckner, John R. Walker
المصدر: Nature
مصطلحات موضوعية: 0301 basic medicine, Chagas disease, Proteasome Endopeptidase Complex, 030106 microbiology, Trypanosoma brucei, Article, 03 medical and health sciences, Inhibitory Concentration 50, Mice, Species Specificity, parasitic diseases, medicine, Animals, Chymotrypsin, Humans, Chagas Disease, Molecular Targeted Therapy, Kinetoplastida, Trypanosoma cruzi, Leishmaniasis, Multidisciplinary, biology, Molecular Structure, Triazoles, Leishmania, biology.organism_classification, medicine.disease, Virology, 3. Good health, Disease Models, Animal, 030104 developmental biology, Pyrimidines, Trypanosomiasis, African, Proteasome, Parasitology, Female, Trypanosomiasis, Proteasome Inhibitors
وصف الملف: application/pdf
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المؤلفون: Nanxin Li, Loren Jon, Fangxian Sun, Van Phung, AnneMarie Culazzo, Bin Hu, Jennifer L. Harris, Allen G. Li, Min Lu, Bo Liu, Zhicheng Wang, Yi Fan, Francisco Adrian, Susan McCormack, Ha-Soon Choi, Francois Gessier, Pamela A. Albaugh, Mahavir Prashad, Celine Tompkins, Andreas Kreusch, Chopiuk Greg, Valentina Molteni, Yong Jia, Tami Hood, Guoxun Liu, Apurva Chaudhary, Auzon Steffy, Tove Tuntland, H. Martin Seidel, Paul Vincent Rucker, Jianwei Che, Jie Li
المصدر: ACS Medicinal Chemistry Letters. 6:562-567
مصطلحات موضوعية: Kinase, Melanoma, Organic Chemistry, Biology, Tropomyosin receptor kinase A, medicine.disease, medicine.disease_cause, Biochemistry, Tropomyosin, Molecular biology, nervous system, Trk receptor, Drug Discovery, medicine, Cancer research, biology.protein, Receptor, Carcinogenesis, Neurotrophin
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المؤلفون: Loren Jon, Valentina Molteni, Nanxin Li, W. Perry Gordon, Garrett M. Brodeur, Tove Tuntland, Jamie L. Croucher, Radhika Iyer, Bo Liu
المصدر: Cancer Chemotherapy and Pharmacology. 75:131-141
مصطلحات موضوعية: Cancer Research, Cell Survival, Mice, Nude, Antineoplastic Agents, Pharmacology, Biology, Irinotecan, Toxicology, Article, Neuroblastoma, chemistry.chemical_compound, In vivo, Cell Line, Tumor, Antineoplastic Combined Chemotherapy Protocols, Temozolomide, medicine, Animals, Humans, Receptor, trkB, Pharmacology (medical), Phosphorylation, Protein Kinase Inhibitors, Membrane Glycoproteins, Dose-Response Relationship, Drug, Drugs, Investigational, Protein-Tyrosine Kinases, medicine.disease, Survival Analysis, Xenograft Model Antitumor Assays, Neoplasm Proteins, Tumor Burden, Dacarbazine, Oncology, chemistry, Trk receptor, Toxicity, Camptothecin, Growth inhibition, Protein Processing, Post-Translational, Half-Life, medicine.drug
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المؤلفون: Chek Shik Lim, Advait Nagle, Chun Li, Clemens H. M. Kocken, Pranab Mishra, Tove Tuntland, Wei Lin Sandra Sim, Rachel Borboa, Case W. McNamara, Seh Yong Leong, Nobutaka Kato, Christophe Bodenreider, Anne-Marie Zeeman, Prasuna Guntapalli, Kelli Kuhen, Thomas Hollenbeck, Thierry T. Diagana, Arnab K. Chatterjee, Elizabeth A. Winzeler, Liying Jocelyn Tan, Jonathan Chang, Siti Nurdiana Abas, Paul W. Smith, Bryan K. S. Yeung, Yong Cheng Tan, David C. Tully, Jason Roland, Suresh B. Lakshminarayana, Bin Zou, Kerstin Gagaring
المصدر: ACS Medicinal Chemistry Letters. 5:947-950
مصطلحات موضوعية: 0303 health sciences, Imidazopyridine, 030306 microbiology, Phenotypic screening, Organic Chemistry, Cell, Biology, Simian, Bioinformatics, biology.organism_classification, Biochemistry, Virology, Plasmodium, 3. Good health, 03 medical and health sciences, medicine.anatomical_structure, In vivo, parasitic diseases, Drug Discovery, medicine, Structure–activity relationship, Parasite hosting, 030304 developmental biology
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19
المؤلفون: Young Kim, Tove Tuntland, H. Martin Seidel, Thomas H. Marsilje, Nanxin Li, Wei Pei, You-Qun He, Xiaoming Cui, Wendy Richmond, Markus Warmuth, Auzon Steffy, Alex Aycinena, Sungjoon Kim, W. Perry Gordon, Donald S. Karanewsky, AnneMarie Culazzo Pferdekamper, Jin Yunho, Jonathan Chang, Ruo Steensma, Jennifer L. Harris, Bo Liu, Sean B. Joseph, Yelena Sarkisova, Christian C. Lee, Todd Groessl, Bei Chen, Wenshuo Lu, Chopiuk Greg, Tao Jiang, Kevin Johnson, Tetsuo Uno, Pierre-Yves Michellys, Jiqing Jiang, Andrew Phimister, Allen G. Li, Nathanael S. Gray, Badry Bursulaya, Frank Sun, Yongqin Wan, Jie Li
المصدر: Journal of Medicinal Chemistry. 56:5675-5690
مصطلحات موضوعية: Pyrimidine, Brigatinib, Ceritinib, Chemistry, medicine.drug_class, Rational design, Pharmacology, ALK inhibitor, chemistry.chemical_compound, In vivo, hemic and lymphatic diseases, Drug Discovery, medicine, Molecular Medicine, Anaplastic lymphoma kinase, Structure–activity relationship, medicine.drug
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20
المؤلفون: Weijia Ou, Hugo D. Urbina, Reynand Pacoma, Jennifer L. Harris, Alana Althage, Daniel E. Mason, Andrew M. Schumacher, Juliano Alves, Gus Welzel, Tove Tuntland, Eric C. Peters, James Watson, Laura H. Jacobson, Bo Liu, John R. Walker
المصدر: The Journal of Neuroscience. 33:2457-2464
مصطلحات موضوعية: Male, Genetically modified mouse, medicine.medical_specialty, Proteases, medicine.medical_treatment, Molecular Sequence Data, Mice, Transgenic, Amyloid beta-Protein Precursor, Mice, Route of administration, Downregulation and upregulation, Internal medicine, Amyloid precursor protein, Animals, Humans, Medicine, Amino Acid Sequence, Neprilysin, Metalloproteinase, Amyloid beta-Peptides, Protease, Dose-Response Relationship, Drug, biology, business.industry, General Neuroscience, fungi, Brain, Articles, Mice, Inbred C57BL, Endocrinology, Proteolysis, biology.protein, Female, business