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1Academic Journal
المؤلفون: Lake, M Alexandra, Adams, Kristin N, Nie, Feilin, Fowler, Elaine, Verma, Amit K, Dei, Silvia, Teodori, Elisabetta, Sherman, David R, Edelstein, Paul H, Spring, David R, Troll, Mark, Ramakrishnan, Lalita
مصطلحات موضوعية: efflux pump inhibitors, mycobacterial efflux pumps, proton pump inhibitors, tuberculosis rifampicin tolerance, verapamil, Humans, Mycobacterium tuberculosis, Rifampin, Antitubercular Agents, Macrophages, Tuberculosis, Drug Tolerance, Bacterial Proteins, Microbial Sensitivity Tests
وصف الملف: application/pdf
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2Academic Journal
المؤلفون: Braconi, Laura, Dei, Silvia, Contino, Marialessandra, Riganti, Chiara, Bartolucci, Gianluca, Manetti, Dina, Romanelli, Maria Novella, Perrone, Maria Grazia, Colabufo, Nicola Antonio, Guglielmo, Stefano, Teodori, Elisabetta
المساهمون: Università degli Studi di Torino, Università degli Studi di Firenze
المصدر: European Journal of Medicinal Chemistry ; volume 259, page 115716 ; ISSN 0223-5234
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3Academic Journal
المؤلفون: Braconi, Laura, Teodori, Elisabetta, Riganti, Chiara, Coronnello, Marcella, Nocentini, Alessio, Bartolucci, Gianluca, Pallecchi, Marco, Contino, Marialessandra, Manetti, Dina, Romanelli, Maria Novella, Supuran, Claudiu T, Dei, Silvia
المساهمون: Braconi, Laura, Teodori, Elisabetta, Riganti, Chiara, Coronnello, Marcella, Nocentini, Alessio, Bartolucci, Gianluca, Pallecchi, Marco, Contino, Marialessandra, Manetti, Dina, Romanelli, Maria Novella, Supuran, Claudiu T, Dei, Silvia
Relation: info:eu-repo/semantics/altIdentifier/pmid/36269278; info:eu-repo/semantics/altIdentifier/wos/WOS:000877201800001; volume:65; issue:21; firstpage:14655; lastpage:14672; numberofpages:18; journal:JOURNAL OF MEDICINAL CHEMISTRY; https://hdl.handle.net/2318/1885659; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85140853254
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4Academic Journal
المؤلفون: Braconi, Laura, Teodori, Elisabetta, Contino, Marialessandra, Riganti, Chiara, Bartolucci, Gianluca, Manetti, Dina, Romanelli, Maria Novella, Perrone, Maria Grazia, Colabufo, Nicola Antonio, Guglielmo, Stefano, Dei, Silvia
المساهمون: Braconi, Laura, Teodori, Elisabetta, Contino, Marialessandra, Riganti, Chiara, Bartolucci, Gianluca, Manetti, Dina, Romanelli, Maria Novella, Perrone, Maria Grazia, Colabufo, Nicola Antonio, Guglielmo, Stefano, Dei, Silvia
مصطلحات موضوعية: efflux transporters modulator, membrane protein, molecular docking studie, multidrug resistance reverser, structure-activity relationship, ATP Binding Cassette Transporter, Subfamily G, Member 2, ATP-Binding Cassette Transporter, Drug Resistance, Multiple, Neoplasm, Neoplasm Protein, Antineoplastic Agent, Quinazolines
Relation: info:eu-repo/semantics/altIdentifier/pmid/35416421; info:eu-repo/semantics/altIdentifier/wos/WOS:000793926000001; volume:17; issue:12; firstpage:e202200027; lastpage:e202200027; numberofpages:21; journal:CHEMMEDCHEM; https://hdl.handle.net/2318/1881136; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85129869345
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5Academic Journal
المؤلفون: Maach, Soumia, Chiaramonte, Niccolò, Borgonetti, Vittoria, Sarno, Federica, Pierucci, Federica, Dei, Silvia, Teodori, Elisabetta, Altucci, Lucia, Meacci, Elisabetta, Galeotti, Nicoletta, Romanelli, Maria Novella
المساهمون: Associazione Italiana Contro le Leucemie - Linfomi e Mieloma, Fondazione Cassa di Risparmio di Firenze, Regione Campania, Ministero dell’Istruzione, dell’Università e della Ricerca
المصدر: Medicinal Chemistry Research ; volume 31, issue 6, page 960-974 ; ISSN 1054-2523 1554-8120
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6Academic Journal
المؤلفون: Braconi, Laura, Riganti, Chiara, Parenti, Astrid, Cecchi, Marta, Nocentini, Alessio, Bartolucci, Gianluca, Menicatti, Marta, Contino, Marialessandra, Colabufo, Nicola Antonio, Manetti, Dina, Romanelli, Maria Novella, Supuran, Claudiu T., Teodori, Elisabetta
المصدر: Molecules; Jul2024, Vol. 29 Issue 14, p3290, 32p
مصطلحات موضوعية: CARBONIC anhydrase inhibitors, CARBONIC anhydrase, MULTIDRUG resistance, CYTOTOXINS, CELL lines, PIPERAZINE
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7Academic Journal
المؤلفون: Braconi, Laura, Bartolucci, Gianluca, Contino, Marialessandra, Chiaramonte, Niccolò, Giampietro, Roberta, Manetti, Dina, Perrone, Maria Grazia, Romanelli, Maria Novella, Colabufo, Nicola Antonio, Riganti, Chiara, Dei, Silvia, Teodori, Elisabetta
المساهمون: Braconi, Laura, Bartolucci, Gianluca, Contino, Marialessandra, Chiaramonte, Niccolò, Giampietro, Roberta, Manetti, Dina, Perrone, Maria Grazia, Romanelli, Maria Novella, Colabufo, Nicola Antonio, Riganti, Chiara, Dei, Silvia, Teodori, Elisabetta
مصطلحات موضوعية: MDR reverser, P-gp modulator, Tetrahydroisoquinoline, co-administration assay, cytotoxicity
Relation: info:eu-repo/semantics/altIdentifier/pmid/32253945; info:eu-repo/semantics/altIdentifier/wos/WOS:000526143600001; volume:35; issue:1; firstpage:974; lastpage:992; numberofpages:19; journal:JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY; http://hdl.handle.net/11586/265271; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85083240446
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8Academic Journal
المؤلفون: Casalone, Enrico, Vignolini, Tiziano, Braconi, Laura, Gardini, Lucia, Capitanio, Marco, Pavone, Francesco S., Giovannelli, Lisa, Dei, Silvia, Teodori, Elisabetta
المساهمون: European Union’s Horizon 2020 research and innovation programme, Laserlab-Europe and by EMPIR project MetVBadBugs
المصدر: Journal of Antimicrobial Chemotherapy ; volume 77, issue 2, page 413-424 ; ISSN 0305-7453 1460-2091
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9Academic Journal
المؤلفون: Cantini, Niccolo, Crocetti, Letizia, Guerrini, Gabriella, Vergelli, Claudia, Schepetkin, Igor A., Pallecchi, Marco, Bartolucci, Gianluca, Quinn, Mark T., Teodori, Elisabetta, Giovannoni, Maria Paola
المصدر: Bioorganic & Medicinal Chemistry Letters ; volume 52, page 128380 ; ISSN 0960-894X
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10Academic Journal
المؤلفون: Manetti, Dina, Garifulina, Alexandra, Bartolucci, Gianluca, Bazzicalupi, Carla, Bellucci, Cristina, Chiaramonte, Niccolò, Dei, Silvia, Di Cesare Mannelli, Lorenzo, Ghelardini, Carla, Gratteri, Paola, Spirova, Ekaterina, Shelukhina, Irina, Teodori, Elisabetta, Varani, Katia, Tsetlin, Victor, Romanelli, Maria Novella
المساهمون: Manetti, Dina, Garifulina, Alexandra, Bartolucci, Gianluca, Bazzicalupi, Carla, Bellucci, Cristina, Chiaramonte, Niccolò, Dei, Silvia, Di Cesare Mannelli, Lorenzo, Ghelardini, Carla, Gratteri, Paola, Spirova, Ekaterina, Shelukhina, Irina, Teodori, Elisabetta, Varani, Katia, Tsetlin, Victor, Romanelli, Maria Novella
مصطلحات موضوعية: Acetylcholine receptors, in vitro, quinoline derivates, therapeutic target, ligand efficiency, full agonist, epibatidine
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/30681854; info:eu-repo/semantics/altIdentifier/wos/WOS:000460365600012; volume:62; issue:4; firstpage:1887; lastpage:1901; numberofpages:15; journal:JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/11392/2411948; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85062259340
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11Academic Journal
المؤلفون: Bartolucci, Gianluca, Pallecchi, Marco, Braconi, Laura, Dei, Silvia, Teodori, Elisabetta, Lapolla, Annunziata, Sartore, Giovanni, Traldi, Pietro
المساهمون: Bartolucci, Gianluca, Pallecchi, Marco, Braconi, Laura, Dei, Silvia, Teodori, Elisabetta, Lapolla, Annunziata, Sartore, Giovanni, Traldi, Pietro
مصطلحات موضوعية: mass spectrometry, metformin, reaction of metformin with glucose
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/38203351; volume:25; issue:1; firstpage:1; lastpage:13; numberofpages:13; journal:INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES; https://hdl.handle.net/11577/3503787; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85181900513
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12Academic Journal
المؤلفون: Matucci, Rosanna, Bellucci, Cristina, Martino, Maria Vittoria, Nesi, Marta, Manetti, Dina, Welzel, Jessica, Bartz, Ulrike, Holze, Janine, Tränkle, Christian, Mohr, Klaus, Mazzolari, Angelica, Vistoli, Giulio, Dei, Silvia, Teodori, Elisabetta, Romanelli, Maria Novella
المساهمون: R. Matucci, C. Bellucci, M.V. Martino, M. Nesi, D. Manetti, J. Welzel, U. Bartz, J. Holze, C. Tränkle, K. Mohr, A. Mazzolari, G. Vistoli, S. Dei, E. Teodori, M.N. Romanelli
مصطلحات موضوعية: Acethylcholine chloride, Allosteric modulation, Atropine sulphate, Carbachol chloride, Carbachol dimer, Gallamine triethiodide, Hexamethonium chloride, McN-A-343 chloride, Muscarinic acetylcholine receptor (mAChR), PubChem CID: 5831, PubChem CID: 5926, PubChem CID: 6060, PubChem CID: 6172, PubChem CID: 64663, PubChem CID: 93550, Settore CHIM/08 - Chimica Farmaceutica
Relation: info:eu-repo/semantics/altIdentifier/pmid/32534072; info:eu-repo/semantics/altIdentifier/wos/WOS:000569368800003; volume:883; firstpage:1; lastpage:9; numberofpages:9; journal:EUROPEAN JOURNAL OF PHARMACOLOGY; http://hdl.handle.net/2434/740370; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85088794475
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13Academic Journal
المؤلفون: Chiaramonte, Niccolò, Maach, Soumia, Biliotti, Caterina, Angeli, Andrea, Bartolucci, Gianluca, Braconi, Laura, Dei, Silvia, Teodori, Elisabetta, Supuran, Claudiu T., Romanelli, Maria Novella
المساهمون: University of Florence
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry ; volume 35, issue 1, page 1003-1010 ; ISSN 1475-6366 1475-6374
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14Academic Journal
المؤلفون: Romanelli, Maria Novella, Braconi, Laura, Gabellini, Alessio, Manetti, Dina, Marotta, Giambattista, Teodori, Elisabetta
المصدر: Molecules; Jan2024, Vol. 29 Issue 1, p68, 49p
مصطلحات موضوعية: DRUG approval, MOIETIES (Chemistry), PIPERAZINE, KINASE inhibitors, MOLECULES
الشركة/الكيان: UNITED States. Food & Drug Administration
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15Academic Journal
المؤلفون: Bartolucci, Gianluca, Pallecchi, Marco, Braconi, Laura, Dei, Silvia, Teodori, Elisabetta, Lapolla, Annunziata, Sartore, Giovanni, Traldi, Pietro
المصدر: International Journal of Molecular Sciences; Jan2024, Vol. 25 Issue 1, p180, 13p
مصطلحات موضوعية: METFORMIN, LIQUID chromatography-mass spectrometry, MASS spectrometry, TANDEM mass spectrometry, GLUCOSE, DRUG target
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16Academic Journal
المصدر: Cancer Drug Resistance
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17Academic Journal
المؤلفون: Crocetti, Letizia, Giovannoni, Maria Paola, Schepetkin, Igor A., Quinn, Mark T., Khlebnikov, Andrei I., Cantini, Niccolò, Guerrini, Gabriella, Iacovone, Antonella, Teodori, Elisabetta, Vergelli, Claudia
المساهمون: Montana Agricultural Experiment Station, Tomsk Polytechnic University, National Institutes of Health, Ministry of Education and Science of the Russian Federation, National Institute of Food and Agriculture
المصدر: Bioorganic & Medicinal Chemistry ; volume 26, issue 21, page 5583-5595 ; ISSN 0968-0896
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18Academic Journal
المؤلفون: Pallecchi, Marco, Lucio, Luigi, Braconi, Laura, Menicatti, Marta, Dei, Silvia, Teodori, Elisabetta, Bartolucci, Gianluca
المصدر: International Journal of Molecular Sciences; Jul2023, Vol. 24 Issue 13, p11155, 18p
مصطلحات موضوعية: ION traps, ISOMERS, TANDEM mass spectrometry, MASS spectrometry, ALGORITHMS
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19Academic Journal
المؤلفون: Teodori, Elisabetta, Dei, Silvia, Bartolucci, Gianluca, Perrone, Maria Grazia, Manetti, Dina, Romanelli, Maria Novella, Contino, Marialessandra, Colabufo, Nicola Antonio
المصدر: ChemMedChem ; volume 12, issue 16, page 1369-1379 ; ISSN 1860-7179 1860-7187
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20Academic Journal
المؤلفون: Romanelli, Maria Novella, Manetti, Dina, Braconi, Laura, Dei, Silvia, Gabellini, Alessio, Teodori, Elisabetta
المصدر: Expert Opinion on Drug Discovery ; volume 17, issue 9, page 969-984 ; ISSN 1746-0441 1746-045X