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المؤلفون: Whitney Kilu, Dieter Steinhilber, Daniel Merk, Jan Heering, Ewgenij Proschak
المصدر: The Journal of Biological Chemistry
مصطلحات موضوعية: 0301 basic medicine, PPARγ, Peroxisome proliferator-activated receptor, PPAR, peroxisome proliferator-activated receptor, Ligands, Biochemistry, Benzoates, drug target, Nuclear Receptor Coactivator 1, LBD, ligand-binding domain, heterodimer, TETRAC, non-classical thyroid hormone 3,3',5,5'-tetraiodothyroacetic acid, homogeneous time-resolved FRET (HTRF), Tb-SA, terbium cryptate conjugated to streptavidin, chemistry.chemical_classification, allostery, Protein Stability, cofactor recruitment, NR, nuclear receptor, Ligand (biochemistry), CREB-Binding Protein, Cell biology, Research Article, Transcriptional Activation, homodimer, RXR, retinoid X receptor, Allosteric regulation, Retinoid X receptor, Rosiglitazone, 03 medical and health sciences, Retinoids, CBP-1, CREB-binding protein coactivator motif 1, FXR, farnesoid X receptor, Protein Domains, Coactivator, RXRα, Humans, HTRF, homogeneous time-resolved FRET, Molecular Biology, Retinoid X Receptor alpha, 030102 biochemistry & molecular biology, SRC1-2, steroid receptor coactivator 1 motif 2, Reproducibility of Results, sGFP, super folder green fluorescent protein, Cell Biology, PPAR gamma, Retinoic acid receptor, 030104 developmental biology, HEK293 Cells, chemistry, Nuclear receptor, DBD, DNA-binding domain, Mutation, Farnesoid X receptor, Protein Multimerization, AF-2, activation function 2