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1
المؤلفون: Kirsten Bjergarde, Cécile Delorme, Pierre-Yves Abecassis, Alain Krick, Jean-Paul Nicolas, Gilles Doerflinger, Sébastien Perron, Michel Murer, Houlfa Guizani, Bruno Filoche-Romme, Sylvette Lachaud, Ronan Le Moigne, Céline Prévost, Cécile Combeau, Jacques Mauger, Jean-Christophe Carry, Stéphanie Pouzieux, Laure Delarbre, Laurent Schio, Francois Clerc, Marie-Line Monteiro, Hervé Minoux, Sylvie Monget, Thomas Bertrand, Véronique Crocq-Stuerga, Ma Nina, Francis Gasse, Odile Angouillant-Boniface, Rémi Lebel, Sébastien Maignan, Sylvie Gontier, Anil Nair, Eric Parmantier
المصدر: Journal of medicinal chemistry. 58(1)
مصطلحات موضوعية: Models, Molecular, Aurora inhibitor, Antineoplastic Agents, Mice, SCID, Quinolones, Serine, Small Molecule Libraries, Aurora Kinases, Neoplasms, Drug Discovery, Sf9 Cells, Animals, Aurora Kinase B, Humans, Aurora Kinase C, Mitosis, Protein Kinase Inhibitors, Aurora Kinase A, Molecular Structure, Kinase, Chemistry, HCT116 Cells, Small molecule, Xenograft Model Antitumor Assays, Cell biology, Protein Structure, Tertiary, Models, Chemical, Molecular Medicine, Benzimidazoles, Female, Protein Binding
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2
المؤلفون: Michel Klich, Yannick Benedetti, Periers Anne-Marie, Alain Iltis, Didier Ferroud, Patrick Laurin, Jean-Luc Haesslein, Sylvette Lachaud, Guillaume L’Hermite, Branislav Musicki
المصدر: Tetrahedron Letters. 41:867-871
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Organic Chemistry, Drug Discovery, Grignard reaction, Stereoselectivity, Coumarin, Biochemistry, Combinatorial chemistry, DNA gyrase
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3
المؤلفون: Véronique Loyau, Alain Bonnefoy, Solange Gouin D'ambrieres, A Dussarat, Nicole Tessot, C. Fromentin, Sylvette Lachaud, Patrick Laurin, Jean-Michel Auger, Yannick Benedetti, Francois Bretin, J. F. Chantot, C. Agouridas, A. Denis, Le Martret Odile
المصدر: Journal of Medicinal Chemistry. 41:4080-4100
مصطلحات موضوعية: Male, Models, Molecular, Ketolides, Haemophilus Infections, medicine.drug_class, Staphylococcus, Antibiotics, Colony Count, Microbial, Drug Evaluation, Preclinical, Molecular Conformation, Erythromycin, Crystallography, X-Ray, medicine.disease_cause, Cethromycin, Microbiology, Haemophilus influenzae, Mice, Drug Discovery, medicine, Animals, Respiratory Tract Infections, Ketolide, Antibacterial agent, Chemistry, Streptococcus, Drug Resistance, Microbial, Staphylococcal Infections, Drug Resistance, Multiple, Anti-Bacterial Agents, Penicillin, Streptococcus pneumoniae, Streptococcus pyogenes, Molecular Medicine, Macrolides, Enterococcus, medicine.drug
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4
المؤلفون: Michel Klich, Guillaume L’Hermite, Yannick Benedetti, Periers Anne-Marie, Jean-Luc Haesslein, Sylvette Lachaud, Branislav Musicki, Didier Ferroud, Patrick Laurin, Alain Iltis
المصدر: ChemInform. 31
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Nanotechnology, Stereoselectivity, General Medicine, Coumarin, DNA gyrase, Combinatorial chemistry
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5
المؤلفون: Frank Halley, Céline Amara, Fabienne Châtreau, Gilles Tiraboschi, Pierre-Yves Abecassis, Philippe Bertrand, Sylvette Lachaud, Didier Babin, Gilles Dutruc-Rosset, Alain Chevalier, Alain Krick, Marie-Claude Burgevin, Dominique Lesuisse, Dominique Quarteronet, Thomas Rooney
المصدر: Bioorganicmedicinal chemistry letters. 20(7)
مصطلحات موضوعية: Models, Molecular, Cytochrome P-450 CYP1A2 Inhibitors, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Hydrolysis, Glycogen Synthase Kinase 3, Mice, Pharmacokinetics, In vivo, Cytochrome P-450 CYP1A2, Drug Discovery, Peptide bond, Animals, Humans, Molecular Biology, Protein Kinase Inhibitors, Glycogen Synthase Kinase 3 beta, Kinase, Chemistry, Organic Chemistry, CYP1A2, Metabolic stability, Safety profile, Molecular Medicine
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6
المؤلفون: Nicole Tessot, Jacques Demassey, Periers Anne-Marie, Fabienne Chatreaux, Yannick Benedetti, Jean Khider, Patrick Laurin, Marlene Airault, Michel Klich, Alain Bonnefoy, Pascale Vicat, Branislav Musicki, Didier Ferroud, Patrice Lassaigne, Claudine Dupuis-Hamelin, Jean-Luc Haesslein, Christine Pierre, Alain Iltis, Sylvette Lachaud
المصدر: Bioorganicmedicinal chemistry letters. 10(15)
مصطلحات موضوعية: chemistry.chemical_classification, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biological activity, Microbial Sensitivity Tests, Coumarin, Biochemistry, Chemical synthesis, DNA gyrase, Anti-Bacterial Agents, chemistry.chemical_compound, Anti-Infective Agents, In vivo, Coumarins, Drug Discovery, Molecular Medicine, heterocyclic compounds, Antibacterial activity, Molecular Biology, Lactone, Antibacterial agent, Hexoses