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المؤلفون: Stephen Joseph Johnson, Shelly A. Glase, Suzanne R. Kesten, Peter J. Manley, Lawrence D. Wise, Jon Wright, Thomas G. Heffner, Thomas A. Pugsley, Robert G. MacKenzie, Hyacinth C. Akunne
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:1361-1366
مصطلحات موضوعية: Chemistry, Aryl, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Stimulation, Pharmacology, Biochemistry, Partial agonist, chemistry.chemical_compound, Dopamine receptor D1, Dopamine receptor D3, Dopamine, Dopamine receptor D2, Drug Discovery, medicine, Molecular Medicine, Receptor, Molecular Biology, medicine.drug
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2
المؤلفون: Walter H. Moos, Stephen Joseph Johnson, Sharie L. Myers, Michael R. Pavia, Suzanne R. Kesten, Roy D. Schwarz, Robert E. Davis, Sheila H. Hobbs, Linda L. Coughenour, David T. Dudley
المصدر: ChemInform. 22
مصطلحات موضوعية: Biochemistry, Pilocarpine, Chemistry, medicine, Cholinergic, General Medicine, Pharmacology, Muscarinic agonist, medicine.drug, Acetylcholine receptor
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3
المؤلفون: Michael R. Pavia, Roy D. Schwarz, Robert E. Davis, Linda L. Coughenour, Stephen Joseph Johnson, Sharie L. Myers, David T. Dudley, Walter H. Moss, Sheila H. Hobbs, Suzanne R. Kesten
المصدر: Bioorganic & Medicinal Chemistry Letters. 1:147-150
مصطلحات موضوعية: Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Alpha (ethology), Pharmacology, Biochemistry, Muscarinic agonist, In vitro, Pilocarpine, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Molecular Medicine, Cholinergic, Molecular Biology, medicine.drug, Acetylcholine receptor
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4
المؤلفون: Jon L. Wright, Tracy F. Gregory, Suzanne R. Kesten, Peter A. Boxer, Kevin A. Serpa, Leonard T. Meltzer, Lawrence D. Wise, Stephen A. Espitia, Christopher S. Konkoy, Edward R. Whittemore, Richard M. Woodward
المصدر: Journal of medicinal chemistry. 43(18)
مصطلحات موضوعية: Cerebral Cortex, Male, Patch-Clamp Techniques, Receptors, Dopamine D2, Administration, Oral, In Vitro Techniques, Transfection, Receptors, N-Methyl-D-Aspartate, Corpus Striatum, Rats, Antiparkinson Agents, Rats, Sprague-Dawley, Radioligand Assay, Xenopus laevis, Piperidines, Receptors, Adrenergic, alpha-1, Drug Discovery, Oocytes, Molecular Medicine, Animals, Benzimidazoles, Excitatory Amino Acid Antagonists
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5
المؤلفون: Sui Xiong Cai, Christina T. Shipp, Zhang-Lin Zhou, Jon L. Wright, John F. W. Keana, Manuel Acosta-Burruel, Suzanne R. Kesten, Minhtam Tran, Edward R. Whittemore, Jon E. Hawkinson, Amir P. Tamiz, Anthony P. Guzikowski, Richard M. Woodward, Soo Hong-Bae
المصدر: Journal of medicinal chemistry. 43(5)
مصطلحات موضوعية: Male, Pyrrolidines, Stereochemistry, Substituent, In Vitro Techniques, Chemical synthesis, Receptors, N-Methyl-D-Aspartate, Pyrrolidine, Receptors, Dopamine, Rats, Sprague-Dawley, chemistry.chemical_compound, Mice, Radioligand Assay, Xenopus laevis, Piperidines, Seizures, Receptors, Adrenergic, alpha-1, Drug Discovery, Ifenprodil, Phenyl group, Animals, Receptor, Cerebral Cortex, Electroshock, Corpus Striatum, Rats, chemistry, Oocytes, Molecular Medicine, NMDA receptor, Anticonvulsants, Piperidine, Excitatory Amino Acid Antagonists
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المؤلفون: Suzanne R. Kesten, Jonathan Wright, Lawrence D. Wise, Thomas G. Heffner, Thomas A. Pugsley, Stephen Joseph Johnson
المصدر: Journal of medicinal chemistry. 42(18)
مصطلحات موضوعية: Reflex, Startle, Dopamine, CHO Cells, Pharmacology, Motor Activity, Chemical synthesis, Piperazines, chemistry.chemical_compound, Mice, Structure-Activity Relationship, In vivo, Cricetinae, Drug Discovery, medicine, Structure–activity relationship, Animals, Humans, Benzopyrans, Receptor, Chemistry, Chinese hamster ovary cell, Receptors, Dopamine D4, Antagonist, Rats, Dopamine D2 Receptor Antagonists, Drug Design, Schizophrenia, Molecular Medicine, Dopamine Antagonists, Thymidine, medicine.drug, Antipsychotic Agents, Protein Binding
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المؤلفون: J. R. Rubin, Lawrence D. Wise, A E Corbin, David Juergen Wustrow, Thomas G. Heffner, Kim T. Zoski, Steven Z. Whetzel, Suzanne R. Kesten, Thomas A. Pugsley, Wouter A. Brink, Thomas R. Belliotti
المصدر: Bioorganicmedicinal chemistry letters. 8(12)
مصطلحات موضوعية: Indoles, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Stereoisomerism, Motor Activity, Biochemistry, Chemical synthesis, Structure-Activity Relationship, X-Ray Diffraction, Dopamine, Drug Discovery, medicine, Moiety, Structure–activity relationship, Animals, Receptor, Molecular Biology, Chemistry, Receptors, Dopamine D2, Organic Chemistry, Receptors, Dopamine D4, Ligand (biochemistry), Rats, Receptors, Serotonin, Molecular Medicine, Enantiomer, medicine.drug