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1Academic Journal
المساهمون: Berry, Edward
المصدر: Journal of Biological Chemistry; 281; 9; Other Information: Journal Publication Date: 03/03/2006
وصف الملف: Medium: ED
URL الوصول: http://www.osti.gov/scitech/servlets/purl/891223
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2Academic Journal
المؤلفون: Huang, Li-shar, Sun, Gang, Cobessi, David, Wang, Andy C., Shen, John T., Tung, Eric Y., Anderson, Vernon E., Berry, Edward A.
مصطلحات موضوعية: Basic biological sciences, Complex II succinate dehydrogenase respiratory chain binding site suicide inhibitor 3-nitropropionic acid nitroalkene
وصف الملف: application/pdf
URL الوصول: https://escholarship.org/uc/item/49p301zw
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3Academic Journal
المؤلفون: Reihill M., Guazzelli L., Remaut H., Oscarson S.
المساهمون: Reihill, M., Guazzelli, L., Remaut, H., Oscarson, S.
Relation: info:eu-repo/semantics/altIdentifier/pmid/32961972; info:eu-repo/semantics/altIdentifier/wos/WOS:000580032100001; volume:25; issue:18; numberofpages:18; journal:MOLECULES; http://hdl.handle.net/11568/1064868; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85091602219; https://www.mdpi.com/1420-3049/25/18/4281
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4Academic Journal
المؤلفون: Caccia Sonia, Ricagno Stefano, Bolognesi Martino
المصدر: Biomolecular Concepts, Vol 1, Iss 2, Pp 117-130 (2010)
مصطلحات موضوعية: α1-antitrypsin, crystal structure, dementia, familial encephalopathy with ns inclusion bodies (fenib), neuroserpin (ns), polymer, protease inhibitor, serine protease, serpinopathies, suicide inhibitor, Biology (General), QH301-705.5
وصف الملف: electronic resource
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5Academic Journal
المصدر: Proceedings of the National Academy of Sciences of the United States of America, 1990 Oct 01. 87(20), 7930-7934.
URL الوصول: https://www.jstor.org/stable/2355448
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6Academic Journal
المؤلفون: S. Caccia, S. Ricagno, M. Bolognesi
المساهمون: S. Caccia, S. Ricagno, M. Bolognesi
مصطلحات موضوعية: a1-antitrypsin, crystal structure, dementia, familial encephalopathy with NS inclusion bodies (FENIB), neuroserpin (NS), polymer, protease inhibitor, serine protease, serpinopathie, suicide inhibitor, Settore BIO/11 - Biologia Molecolare, Settore BIO/10 - Biochimica
Relation: info:eu-repo/semantics/altIdentifier/pmid/25961991; volume:1; issue:2; firstpage:117; lastpage:130; numberofpages:14; journal:BIOMOLECULAR CONCEPTS; http://hdl.handle.net/2434/147279; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-83555179759
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7Academic Journal
المؤلفون: Alahuhta, Markus, Salin, Mikko, Casteleijn, Marco G., Kemmer, Christian, El-Sayed, Ibrahim, Augustyns, Koen, Neubauer, Peter, Wierenga, Rik K.
المصدر: Alahuhta , M , Salin , M , Casteleijn , M G , Kemmer , C , El-Sayed , I , Augustyns , K , Neubauer , P & Wierenga , R K 2008 , ' Structure-based protein engineering efforts with a monomeric TIM variant : The importance of a single point mutation for generating an active site with suitable binding properties ' , Protein Engineering, Design and Selection , vol. 21 , no. 4 , pp. 257-266 . https://doi.org/10.1093/protein/gzn002
مصطلحات موضوعية: Citrate, Monomeric TIM, Protein design, Suicide inhibitor, Transition state analog, /dk/atira/pure/sustainabledevelopmentgoals/good_health_and_well_being, name=SDG 3 - Good Health and Well-being
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8Academic Journal
المؤلفون: Silvestri I., Lyu H., Fata F., Banta P. R., Mattei B., Ippoliti R., Bellelli A., Pitari G., Ardini M., Petukhova V., Thatcher G. R. J., Petukhov P. A., Williams D. L., Angelucci F.
المساهمون: Silvestri I, Lyu H, Fata F, Banta PR, Mattei B, Ippoliti R, Bellelli A, Pitari G, Ardini M, Petukhova V, Thatcher GRJ, Silvestri, I., Lyu, H., Fata, F., Banta, P. R., Mattei, B., Ippoliti, R., Bellelli, A., Pitari, G., Ardini, M., Petukhova, V., Thatcher, G. R. J., Petukhov, P. A., Williams, D. L., Angelucci, F.
مصطلحات موضوعية: Quinone methide, Redox metabolism, Schistosomiasi, Secondary site, Suicide inhibitor
Relation: info:eu-repo/semantics/altIdentifier/pmid/31870799; info:eu-repo/semantics/altIdentifier/wos/WOS:000506882400019; volume:147; firstpage:200; lastpage:211; numberofpages:12; journal:FREE RADICAL BIOLOGY & MEDICINE; http://hdl.handle.net/11575/107098; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85076825399; www.elsevier.com/locate/freeradbiomed
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9Academic Journal
المؤلفون: Khosrow Aghaiypour, Er Wlodawer, Jacek Lubkowski
المساهمون: The Pennsylvania State University CiteSeerX Archives
مصطلحات موضوعية: Bacterial L-asparaginase, Enzymatic mechanism, X-ray crystallography, Suicide inhibitor
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.374.9612; http://mcl1.ncifcrf.gov/wlo_pubs/200.pdf
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10Academic Journal
المؤلفون: Atsushi Tabata, Hiroyasu Kinemuchi, Kensuke Kisara, Lars Oreland, Masato Jinbo, Takeshi Tadano, Yoshie Toyoshima, Yuichiro Arai
المصدر: The Japanese Journal of Pharmacology. 2000, 83(2):164
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11
المؤلفون: Paumann-Page, Martina, Furtmüller, Paul G., Hofbauer, Stefan, Paton, Louise N., Obinger, Christian, Kettle, Anthony J.
المصدر: Archives of Biochemistry and Biophysics
مصطلحات موضوعية: Mechanism-based inhibition, Myeloperoxidase, Oxidative modification, Neutrophils, Temperature, Biophysics, Heme, Hydrogen Peroxide, Biochemistry, Article, Protein Structure, Secondary, Protein Structure, Tertiary, Enzyme Activation, Kinetics, Protein Subunits, Oxidative stress, Suicide inhibitor, Enzyme Stability, Humans, Molecular Biology, ComputingMethodologies_COMPUTERGRAPHICS, Peroxidase, Protein Unfolding
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12
المؤلفون: Sonia Caccia, Martino Bolognesi, Stefano Ricagno
المصدر: Biomolecular Concepts, Vol 1, Iss 2, Pp 117-130 (2010)
مصطلحات موضوعية: crystal structure, QH301-705.5, medicine.medical_treatment, polymer, serine protease, Synaptogenesis, Serpin, neuroserpin (ns), serpinopathies, General Biochemistry, Genetics and Molecular Biology, familial encephalopathy with ns inclusion bodies (fenib), protease inhibitor, Cellular and Molecular Neuroscience, Neuroserpin, medicine, Biology (General), Reactive center, Serine protease, chemistry.chemical_classification, Protease, biology, Chemistry, General Medicine, Protein superfamily, Cell biology, Amino acid, biology.protein, suicide inhibitor, α1-antitrypsin, dementia
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13
المؤلفون: Francesca De Maria, Anna Maria Caccuri, Angela Bullo, Paola Turella, Giuseppe Filomeni, Giorgio Federici, Giovanni Antonini, Lorenzo Stella, Giorgio Ricci
المساهمون: Giorgio, Ricci, FRANCESCA DE, Maria, Antonini, Giovanni, Paola, Turella, Angela, Bullo, Lorenzo, Stella, Giuseppe, Filomeni, Giorgio, Federici, ANNA MARIA, Caccuri
المصدر: Journal of Biological Chemistry. 280:26397-26405
مصطلحات موضوعية: non-GSH peptidomimetic compound, biology, Chemistry, Peptidomimetic, Stereochemistry, Active site, Enzyme inhibitor, Cell Biology, Plasma protein binding, Glutathione, Biochemistry, chemistry.chemical_compound, Mechanism of action, Docking (molecular), enzyme kinetics, biology.protein, medicine, suicide inhibitor, Enzyme kinetics, medicine.symptom, Binding site, Molecular Biology, Glutathione S-Transferase
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14Academic Journal
المؤلفون: ROTILI, Dante, De Luca A, Tarantino D, Pezzola S, FORGIONE, MARIANTONIETTA, Morozzo Della Rocca B, Falconi M, MAI, Antonello, Caccuri A.M.
المساهمون: Rotili, Dante, De Luca, A, Tarantino, D, Pezzola, S, Forgione, Mariantonietta, Morozzo Della Rocca, B, Falconi, M, Mai, Antonello, Caccuri, A. M.
مصطلحات موضوعية: glutathione-S-transferase, nitrobenzoxadiazole, sigma-complex, suicide inhibitor, water solubility
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:000348003500017; volume:89; firstpage:156; lastpage:171; numberofpages:16; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; https://hdl.handle.net/11590/493071
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15
المصدر: Journal of Biotechnology. 101(1):19-28
مصطلحات موضوعية: EXPRESSION, HYDROLASE, Bacillus subtilis lipase, phosphonate suicide inhibitor, BETA-LACTAMASE MUTANTS, DIRECTED MOLECULAR EVOLUTION, GENE, IN-VITRO SELECTION, MICROBIAL LIPASES, CATALYTIC ACTIVITY, phage display, PSEUDOMONAS LIPASES, 2-O-isopropylidene-sn-glycerol, LIPOLYTIC ENZYMES
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16
المؤلفون: Anna Maria Caccuri, Antonello Mai, Silvia Pezzola, Domenico Tarantino, Blasco Morozzo della Rocca, Mattia Falconi, Dante Rotili, Mariantonietta Forgione, Anastasia De Luca
مصطلحات موضوعية: Models, Molecular, Glutathione-S-transferase, Stereochemistry, Thio, Antineoplastic Agents, Naphthalenes, chemistry.chemical_compound, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, Structure–activity relationship, Humans, Enzyme Inhibitors, Settore BIO/10, Cytotoxicity, Alkyl, Cell Proliferation, nitrobenzoxadiazole, sigma-complex, suicide inhibitor, water solubility, Pharmacology, chemistry.chemical_classification, biology, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Imidazoles, General Medicine, Glutathione, Bioavailability, Glutathione S-transferase, chemistry, Glutathione S-Transferase pi, biology.protein, Selectivity
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17Academic Journal
المؤلفون: Huang, Li-shar, Sun, Gang, Cobessi, David, Wang, Andy C., Shen,John T., Tung, Eric Y., Anderson, Vernon E., Berry, Edward A.
المساهمون: USDOE Director, Office of Science. Office of Basic EnergySciences, National Institutes of Health
المصدر: Journal Name: Journal of Biological Chemistry; Journal Volume: 281; Journal Issue: 9; Related Information: Journal Publication Date: 03/03/2006
مصطلحات موضوعية: Oxidation, Arginine, Residues, Adducts, Fragmentation, Respiration, Protons, Toxins, Enzymes, Ubiquinone Complex Ii Succinate Dehydrogenase Respiratory Chain Bindingsite Suicide Inhibitor 3-Nitropropionic Acid Nitroalkene, Cleavage, Resolution, Trypsin, Decarboxylation, Modifications, 59 Basic Biological Sciences, Dehydrogenation, Complex Ii Succinate Dehydrogenase Respiratory Chain Bindingsite Suicide Inhibitor 3-Nitropropionic Acid Nitroalkene, Catalysts, 72 Physics Of Elementary Particles And Fields, Catalysis, Substrates
وصف الملف: Text
Relation: rep-no: LBNL--59358; grantno: DE-AC02-05CH11231; grantno: NIHR01GM62563; osti: 891223; https://digital.library.unt.edu/ark:/67531/metadc876632/; ark: ark:/67531/metadc876632
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18Academic Journal
المؤلفون: Alonso, Hernan, Kleifeld, Oded, Yeheskel, Adva, Ong, Poh C., Liu, Yu C., Stok, Jeanette E., De Voss, James J., Roujeinikova, Anna
مصطلحات موضوعية: Alkane hydroxylase (AlkB), Alkyne, Enzyme inactivation, Mono-oxygenase, Pseudomonas putida, Suicide inhibitor, 1303 Biochemistry, 1307 Cell Biology, 1312 Molecular Biology
Relation: orcid:0000-0002-8759-3931; orcid:0000-0002-2659-5140; BF040030; DP130101930
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19
المؤلفون: Axel T. Brunger, Betty W Shen, Sapan A Shah
المصدر: Structure. 5:1067-1075
مصطلحات موضوعية: Models, Molecular, Cyclohexanecarboxylic Acids, Stereochemistry, Ornithine aminotransferase, Molecular Sequence Data, Arginine, Crystallography, X-Ray, 010402 general chemistry, 01 natural sciences, Cofactor, 03 medical and health sciences, chemistry.chemical_compound, Gabaculine, Structural Biology, Gyrate Atrophy, Humans, Transferase, Enzyme Inhibitors, Molecular Biology, Transaminases, 030304 developmental biology, chemistry.chemical_classification, 0303 health sciences, Binding Sites, Ornithine-Oxo-Acid Transaminase, biology, ornithine aminotransferase, substrate recognition, Aminobutyrates, Active site, Glutamic acid, Ornithine, 0104 chemical sciences, Enzyme, chemistry, Biochemistry, Pyridoxal Phosphate, pyridoxal -5′-phosphate, biology.protein, Tyrosine, suicide inhibitor, X-ray structure
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20
المؤلفون: Henning D. Mootz, Uwe Linne, Nadine D. Weikart, Stefanie Sommer
المصدر: Bioorganicmedicinal chemistry. 21(9)
مصطلحات موضوعية: Proteases, SENP1, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, SUMO enzymes, Cysteine Proteinase Inhibitors, Biochemistry, Deubiquitinating enzyme, Cysteine peptidase, Mice, Structure-Activity Relationship, Suicide inhibitor, Drug Discovery, Catalytic triad, Endopeptidases, medicine, Tumor Cells, Cultured, Animals, Sulfhydryl Compounds, Molecular Biology, Medicine(all), Protease, biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Cysteine Endopeptidases, Electrophile, Alkynes, biology.protein, Molecular Medicine, Posttranslational modification, Oxyanion hole