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1Academic Journal
المؤلفون: Bresinsky, Merlin, Strasser, Jessica M., Hubmann, Alexander, Vallaster, Bernadette, McCue, William M., Fuller, Jessica, Singh, Gurpreet, Nelson, Kathryn M., Cuellar, Matthew E., Finzel, Barry C., Ashe, Karen H., Walters, Michael A., Pockes, Steffen
مصطلحات موضوعية: 615 Pharmazie, ddc:615
وصف الملف: application/pdf
Relation: https://epub.uni-regensburg.de/52873/1/Archiv%20der%20Pharmazie%20-%202022%20-%20Bresinsky%20-%20Characterization%20of%20caspase_u20102%20inhibitors%20based%20on%20specific%20sites%20of.pdf; Bresinsky, Merlin, Strasser, Jessica M., Hubmann, Alexander, Vallaster, Bernadette, McCue, William M., Fuller, Jessica, Singh, Gurpreet, Nelson, Kathryn M., Cuellar, Matthew E., Finzel, Barry C., Ashe, Karen H., Walters, Michael A. und Pockes, Steffen (2022) Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis. Archiv der Pharmazie 355 (9), S. 2200095.
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2Academic Journal
المؤلفون: Xue, Lian, Shi, Da-Hua, Harjani, Jitendra R, Huang, Fei, Beveridge, Julia G, Dingjan, Tamir, Ban, Kung, Diab, Sarah, Duffy, Sandra, Lucantoni, Leonardo, Fletcher, Sabine, Chiu, Francis CK, Blundell, Scott, Ellis, Katherine, Ralph, Stuart A, Wirjanata, Grennady, Teguh, Silvia, Noviyanti, Rintis, Chavchich, Marina, Creek, Darren, Price, Ric N, Marfurt, Jutta, Charman, Susan A, Cuellar, Matthew E, Strasser, Jessica M, Dahlin, Jayme L, Walters, Michael A, Edstein, Michael D, Avery, Vicky M, Baell, Jonathan B
مصطلحات موضوعية: Medicinal and biomolecular chemistry, Organic chemistry, Pharmacology and pharmaceutical sciences, Science & Technology, Life Sciences & Biomedicine, Chemistry, Medicinal, Pharmacology & Pharmacy, PLASMODIUM-FALCIPARUM
Relation: Journal of Medicinal Chemistry; Xue, L; Shi, D-H; Harjani, JR; Huang, F; Beveridge, JG; Dingjan, T; Ban, K; Diab, S; Duffy, S; Lucantoni, L; Fletcher, S; Chiu, FCK; Blundell, S; Ellis, K; Ralph, SA; Wirjanata, G; Teguh, S; Noviyanti, R; Chavchich, M; Creek, D; Price, RN; Marfurt, J; Charman, SA; Cuellar, ME; Strasser, JM; Dahlin, JL; Walters, MA; Edstein, MD; Avery, VM; Baell, JB, 3,3 '-Disubstituted 5,5 '-Bi(1,2,4-triazine) Derivatives with Potent in Vitro and in Vivo Antimalarial Activity, Journal of Medicinal Chemistry, 2019, 62 (5), pp. 2485-2498; http://hdl.handle.net/10072/386725
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3Academic Journal
المؤلفون: Dahlin, Jayme L., Nelson, Kathryn M., Strasser, Jessica M., Barsyte-Lovejoy, Dalia, Szewczyk, Magdalena M., Organ, Shawna, Cuellar, Matthew, Singh, Gurpreet, Shrimp, Jonathan H., Nguyen, Nghi, Meier, Jordan L., Arrowsmith, Cheryl H., Brown, Peter J., Baell, Jonathan B., Walters, Michael A.
المصدر: Dahlin , J L , Nelson , K M , Strasser , J M , Barsyte-Lovejoy , D , Szewczyk , M M , Organ , S , Cuellar , M , Singh , G , Shrimp , J H , Nguyen , N , Meier , J L , Arrowsmith , C H , Brown , P J , Baell , J B & Walters , M A 2017 , ' Assay interference and off-target liabilities of reported histone acetyltransferase inhibitors ' , Nature Communications , vol. 8 , no. 1 , 1527 , pp. 1-14 . https://doi.org/10.1038/s41467-017-01657-3
وصف الملف: application/pdf
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4Academic Journal
المؤلفون: Singh, Gurpreet, Liu, Peng, Yao, Katherine R., Strasser, Jessica M., Hlynialuk, Chris, Leinonen-Wright, Kailee, Teravskis, Peter J., Choquette, Jessica M., Ikramuddin, Junaid, Bresinsky, Merlin, Nelson, Kathryn M., Liao, Dezhi, Ashe, Karen H., Walters, Michael A., Pockes, Steffen
مصطلحات موضوعية: 540 Chemie, ddc:540
Relation: Singh, Gurpreet, Liu, Peng, Yao, Katherine R., Strasser, Jessica M., Hlynialuk, Chris, Leinonen-Wright, Kailee, Teravskis, Peter J., Choquette, Jessica M., Ikramuddin, Junaid, Bresinsky, Merlin, Nelson, Kathryn M., Liao, Dezhi, Ashe, Karen H., Walters, Michael A. und Pockes, Steffen (2022) Caspase-2 Inhibitor Blocks Tau Truncation and Restores Excitatory Neurotransmission in Neurons Modeling FTDP-17 Tauopathy. ACS Chemical Neuroscience 13 (10), S. 1549-1557.
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5Academic Journal
المؤلفون: Bresinsky, Merlin, Strasser, Jessica M., Vallaster, Bernadette, Liu, Peng, McCue, William M., Fuller, Jessica, Hubmann, Alexander, Singh, Gurpreet, Nelson, Kathryn M., Cuellar, Matthew E., Wilmot, Carrie M., Finzel, Barry C., Ashe, Karen H., Walters, Michael A., Pockes, Steffen
المساهمون: National Institute on Aging, Lucas Brothers Foundation
المصدر: ACS Pharmacology & Translational Science ; volume 5, issue 1, page 20-40 ; ISSN 2575-9108 2575-9108
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6Academic Journal
المؤلفون: Choi, Si Ho, Bosnakovski, Darko, Strasser, Jessica M., Toso, Erik A., Walters, Michael A., Kyba, Michael
المصدر: SLAS Discovery ; volume 21, issue 7, page 680-688 ; ISSN 2472-5552
الاتاحة: http://dx.doi.org/10.1177/1087057116651868
http://journals.sagepub.com/doi/pdf/10.1177/1087057116651868
http://journals.sagepub.com/doi/full-xml/10.1177/1087057116651868
https://api.elsevier.com/content/article/PII:S2472555222071301?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S2472555222071301?httpAccept=text/plain -
7Academic Journal
المؤلفون: Dahlin, Jayme L., Nissink, J. Willem M., Strasser, Jessica M., Francis, Subhashree, Higgins, LeeAnn, Zhou, Hui, Zhang, Zhiguo, Walters, Michael A.
المساهمون: National Institute of Diabetes and Digestive and Kidney Diseases, Pharmaceutical Research and Manufacturers of America Foundation, National Institute of General Medical Sciences, Mayo Foundation for Medical Education and Research, Minnesota Partnership for Biotechnology and Medical Genomics
المصدر: Journal of Medicinal Chemistry ; volume 58, issue 5, page 2091-2113 ; ISSN 0022-2623 1520-4804
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8Academic Journal
المؤلفون: Bosnakovski, Darko, Choi, Si Ho, Strasser, Jessica M, Toso, Erik A, Walters, Michael A, Kyba, Michael
المصدر: Skeletal Muscle ; volume 4, issue 1 ; ISSN 2044-5040
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9Academic Journal
المؤلفون: Dahlin, Jayme L., Sinville, Rondedrick, Solberg, Jonathan, Zhou, Hui, Han, Junhong, Francis, Subhashree, Strasser, Jessica M., John, Kristen, Hook, Derek J., Walters, Michael A., Zhang, Zhiguo
المساهمون: Thomas, Tim
المصدر: PLoS ONE ; volume 8, issue 11, page e78877 ; ISSN 1932-6203
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10Academic Journal
المؤلفون: Priebbenow, Daniel L., Leaver, David J., Nguyen, Nghi, Cleary, Benjamin, Lagiakos, H. Rachel, Sanchez, Julie, Xue, Lian, Huang, Fei, Sun, Yuxin, Mujumdar, Prashant, Mudududdla, Ramesh, Varghese, Swapna, Teguh, Silvia, Charman, Susan A., White, Karen L., Shackleford, David M., Katneni, Kasiram, Cuellar, Matthew, Strasser, Jessica M., Dahlin, Jayme L., Walters, Michael A., Street, Ian P., Monahan, Brendon J., Jarman, Kate E., Jousset Sabroux, Helene, Falk, Hendrik, Chung, Matthew C., Hermans, Stefan J., Downer, Natalie L., Parker, Michael W., Voss, Anne K., Thomas, Tim, Baell, Jonathan B.
المساهمون: Department of Education, Employment and Workplace Relations, Australian Government, National Health and Medical Research Council, State Government of Victoria
المصدر: Journal of Medicinal Chemistry ; volume 63, issue 9, page 4655-4684 ; ISSN 0022-2623 1520-4804
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11Academic Journal
المؤلفون: Xie, Yiyue, Tummala, Padmaja, Oakley, Aaron J., Deora, Girdhar Singh, Nakano, Yuji, Rooke, Melissa, Cuellar, Matthew E., Strasser, Jessica M., Dahlin, Jayme L., Walters, Michael A., Casarotto, Marco G., Board, Philip G., Baell, Jonathan B.
المساهمون: National Health and Medical Research Council
المصدر: Journal of Medicinal Chemistry ; volume 63, issue 6, page 2894-2914 ; ISSN 0022-2623 1520-4804
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12Academic Journal
المؤلفون: Leaver, David J., Cleary, Benjamin, Nguyen, Nghi, Priebbenow, Daniel L., Lagiakos, H. Rachel, Sanchez, Julie, Xue, Lian, Huang, Fei, Sun, Yuxin, Mujumdar, Prashant, Mudududdla, Ramesh, Varghese, Swapna, Teguh, Silvia, Charman, Susan A., White, Karen L., Katneni, Kasiram, Cuellar, Matthew, Strasser, Jessica M., Dahlin, Jayme L., Walters, Michael A., Street, Ian P., Monahan, Brendon J., Jarman, Kate E., Sabroux, Helene Jousset, Falk, Hendrik, Chung, Matthew C., Hermans, Stefan J., Parker, Michael W., Thomas, Tim, Baell, Jonathan B.
المساهمون: National Health and Medical Research Council
المصدر: Journal of Medicinal Chemistry ; volume 62, issue 15, page 7146-7159 ; ISSN 0022-2623 1520-4804
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13Academic Journal
المؤلفون: Dahlin, Jayme L., Cuellar, Matthew, Singh, Gurpreet, Nelson, Kathryn M., Strasser, Jessica M., Rappe, Todd, Xia, Youlin, Veglia, Gianluigi, Walters, Michael A.
المصدر: Current Protocols in Chemical Biology ; volume 10, issue 1, page 91-117 ; ISSN 2160-4762 2160-4762
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14Academic Journal
المؤلفون: Dahlin, Jayme L.1,2, Nissink, J. Willem M.3, Francis, Subhashree4, Strasser, Jessica M.4, John, Kristen4, Zhang, Zhiguo5, Walters, Michael A.4 mwalters@umn.edu
المصدر: Bioorganic & Medicinal Chemistry Letters. Nov2015, Vol. 25 Issue 21, p4740-4752. 13p.
مصطلحات موضوعية: *NUCLEAR magnetic resonance, *DRUG development, *ETHYLENEDIAMINETETRAACETIC acid, *SERUM albumin, *IN vitro studies