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1Academic Journal
المؤلفون: Schimunek J., Seidl P., Elez K., Hempel T., Le T., Noé F., Olsson S., Raich L., Winter R., Gokcan H., Gusev F., Gutkin E. M., Isayev O., Kurnikova M. G., Narangoda C. H., Zubatyuk R., Bosko I. P., Furs K. V., Karpenko A. D., Kornoushenko Y. V., Shuldau M., Yushkevich A., Benabderrahmane M. B., Bousquet-Melou P., Bureau R., Charton B., Cirou B. C., Gil G., Allen W. J., Sirimulla S., Watowich S., Antonopoulos N., Epitropakis N., Krasoulis A., Itsikalis V., Theodorakis S., Kozlovskii I., Maliutin A., Medvedev A., Popov P., Zaretckii M., Eghbal-Zadeh H., Halmich C., Hochreiter S., Mayr A., Ruch P., Widrich M., Berenger F., Kumar A., Yamanishi Y., Zhang K. Y. J., Bengio E., Bengio Y., Jain M. J., Korablyov M., Liu C. H., Marcou G., Glaab E., Barnsley K., Iyengar S. M., Ondrechen M. J., Haupt V. J., Kaiser F., Schroeder M., Pugliese L., Albani S., Athanasiou C., Beccari A., Carloni P., D'Arrigo G., Gianquinto E., Goßen J., Hanke A., Joseph B. P., Kokh D. B., Kovachka S., Manelfi C., Mukherjee G., Muñiz-Chicharro A., Musiani F., Nunes-Alves A., Paiardi G., Rossetti G., Sadiq S. K., Spyrakis F., Talarico C., Tsengenes A., Wade R. C., Copeland C., Gaiser J., Olson D. R., Roy A., Venkatraman V., Wheeler T. J., Arthanari H., Blaschitz K., Cespugli M., Durmaz V., Fackeldey K., Fischer P. D.
المساهمون: Schimunek J., Seidl P., Elez K., Hempel T., Le T., Noé F., Olsson S., Raich L., Winter R., Gokcan H., Gusev F., Gutkin E.M., Isayev O., Kurnikova M.G., Narangoda C.H., Zubatyuk R., Bosko I.P., Furs K.V., Karpenko A.D., Kornoushenko Y.V., Shuldau M., Yushkevich A., Benabderrahmane M.B., Bousquet-Melou P., Bureau R., Charton B., Cirou B.C., Gil G., Allen W.J., Sirimulla S., Watowich S., Antonopoulos N., Epitropakis N., Krasoulis A., Itsikalis V., Theodorakis S., Kozlovskii I., Maliutin A., Medvedev A., Popov P., Zaretckii M., Eghbal-Zadeh H., Halmich C., Hochreiter S., Mayr A., Ruch P., Widrich M., Berenger F., Kumar A., Yamanishi Y., Zhang K.Y.J., Bengio E., Bengio Y., Jain M.J., Korablyov M., Liu C.H., Marcou G., Glaab E., Barnsley K., Iyengar S.M., Ondrechen M.J., Haupt V.J., Kaiser F., Schroeder M., Pugliese L., Albani S., Athanasiou C., Beccari A., Carloni P., D'Arrigo G., Gianquinto E., Goßen J., Hanke A., Joseph B.P., Kokh D.B., Kovachka S., Manelfi C., Mukherjee G., Muñiz-Chicharro A., Musiani F., Nunes-Alves A., Paiardi G., Rossetti G., Sadiq S.K., Spyrakis F., Talarico C., Tsengenes A., Wade R.C., Copeland C., Gaiser J., Olson D.R., Roy A., Venkatraman V., Wheeler T.J., Arthanari H., Blaschitz K., Cespugli M., Durmaz V., Fackeldey K., Fischer P.D.
مصطلحات موضوعية: COVID-19, SARS-CoV-2, drug discovery, machine learning
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/37833243; volume:43; issue:1; firstpage:1; lastpage:19; numberofpages:19; journal:MOLECULAR INFORMATICS; https://hdl.handle.net/11585/955638; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85176949170
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2Academic Journal
المؤلفون: Bersani M., Failla M., Vascon F., Gianquinto E., Bertarini L., Baroni M., Cruciani G., Verdirosa F., Sannio F., Docquier J. D., Cendron L., Spyrakis F., Lazzarato L., Tondi D.
المساهمون: Bersani, M., Failla, M., Vascon, F., Gianquinto, E., Bertarini, L., Baroni, M., Cruciani, G., Verdirosa, F., Sannio, F., Docquier, J. D., Cendron, L., Spyrakis, F., Lazzarato, L., Tondi, D.
مصطلحات موضوعية: 1,2,4-triazole-3-thione, NDM-1, competitive inhibitor, resistance, structure-based drug design
Relation: info:eu-repo/semantics/altIdentifier/pmid/38139809; info:eu-repo/semantics/altIdentifier/wos/WOS:001130773700001; volume:16; issue:12; firstpage:2; lastpage:22; journal:PHARMACEUTICALS; https://hdl.handle.net/11380/1330267; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85180662931
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3Academic Journal
المؤلفون: Guardigni M., Pruccoli L., Santini A., Simone A. D., Bersani M., Spyrakis F., Frabetti F., Uliassi E., Andrisano V., Pagliarani B., Fernández-Gómez P., Palomo V., Bolognesi M. L., Tarozzi A., Milelli A.
المساهمون: Guardigni M., Pruccoli L., Santini A., Simone A.D., Bersani M., Spyrakis F., Frabetti F., Uliassi E., Andrisano V., Pagliarani B., Fernández-Gómez P., Palomo V., Bolognesi M.L., Tarozzi A., Milelli A.
مصطلحات موضوعية: Alzheimer’s disease, chemical knockdown, glycogen synthase kinase 3β, protein degradation, proteolysis targeting chimeras
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/37218653; info:eu-repo/semantics/altIdentifier/wos/WOS:001016482200001; volume:14; issue:11; firstpage:1963; lastpage:1970; numberofpages:8; journal:ACS CHEMICAL NEUROSCIENCE; https://hdl.handle.net/11585/934799; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85162827353
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4Conference
المؤلفون: Lazzarato, L., Failla, M., Gianquinto, E., Bersani, M., Bertarini, L., Verri, A., Vascon, F., Sannio, F., Verdirosa, F., Beatrice, N., De Luca, F., Costi, M. P., Cruciani, G., Docquier, J. D., Cendron, L., Spyrakis, F., Tondi, D.
المساهمون: Lazzarato, L., Failla, M., Gianquinto, E., Bersani, M., Bertarini, L., Verri, A., Vascon, F., Sannio, F., Verdirosa, F., Beatrice, N., De Luca, F., Costi, M.P., Cruciani, G., Docquier, J.D., Cendron, L., Spyrakis, F., Tondi, D.
Relation: ispartofbook:Book of abstracts of XXVII National Meeting on Medicinal Chemistry; XXVII National Meeting on Medicinal Chemistry; firstpage:42; lastpage:42; numberofpages:1; http://hdl.handle.net/2318/1874226
الاتاحة: http://hdl.handle.net/2318/1874226
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5Academic Journal
المؤلفون: Pippione, A.C., Kilic-Kurt, Z., Kovachka, S., Sainas, S., Rolando, B., Denasio, E., Pors, Klaus, Adinolfi, S., Zonari, D., Bagnati, R., Lolli, M.L., Spyrakis, F., Oliaro-Bosso, S., Boschi, D.
مصطلحات موضوعية: Aldo-keto reductase 1C3 (AKR1C3), Castration Resistant Prostate Cancer (CRPC), Bioisosteric modulation, Hydroxytriazole scaffold
الاتاحة: http://hdl.handle.net/10454/19070
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6Academic Journal
المؤلفون: Pippione A. C., Kilic-Kurt Z., Kovachka S., Sainas S., Rolando B., Denasio E., Pors K., Adinolfi S., Zonari D., Bagnati R., Lolli M. L., Spyrakis F., Oliaro-Bosso S., Boschi D.
المساهمون: Pippione A.C., Kilic-Kurt Z., Kovachka S., Sainas S., Rolando B., Denasio E., Pors K., Adinolfi S., Zonari D., Bagnati R., Lolli M.L., Spyrakis F., Oliaro-Bosso S., Boschi D.
مصطلحات موضوعية: AKR1C3 inhibitors, prostate cancer, triazoles, aldo-keto reductase
Relation: info:eu-repo/semantics/altIdentifier/pmid/35447434; info:eu-repo/semantics/altIdentifier/wos/WOS:000793638500009; volume:237; firstpage:114366; lastpage:114384; numberofpages:19; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/2318/1859921; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85128267024; https://www-scopus-com.bibliopass.unito.it/record/display.uri?eid=2-s2.0-85128267024&origin=resultslist&sort=plf-f&src=s&st1=10.1016/j.ejmech.2022.114366&sid=07f6cd37fbeafef783a3f166320d8feb&sot=b&sdt=b&sl=33&s=DOI(10.1016/j.ejmech.2022.114366)&relpos=0&citeCnt=0&searchTerm=&featureToggles=FEATURE_NEW_DOC_DETAILS_EXPORT:1
الاتاحة: http://hdl.handle.net/2318/1859921
https://doi.org/10.1016/j.ejmech.2022.114366
https://www-scopus-com.bibliopass.unito.it/record/display.uri?eid=2-s2.0-85128267024&origin=resultslist&sort=plf-f&src=s&st1=10.1016/j.ejmech.2022.114366&sid=07f6cd37fbeafef783a3f166320d8feb&sot=b&sdt=b&sl=33&s=DOI(10.1016/j.ejmech.2022.114366)&relpos=0&citeCnt=0&searchTerm=&featureToggles=FEATURE_NEW_DOC_DETAILS_EXPORT:1 -
7Academic Journal
المؤلفون: Dahdouh, E, Allander, L, Falgenhauer, L, Iorga, BI, Lorenzetti, S, Marcos-Alcalde, I, Martin, NI, Martinez-Martinez, L, Mingorance, J, Naas, T, Rubin, JE, Spyrakis, F, Tangden, T, Gomez-Puertas, P
المساهمون: Dahdouh, E, Allander, L, Falgenhauer, L, Iorga, BI, Lorenzetti, S, Marcos-Alcalde, I, Martin, NI, Martinez-Martinez, L, Mingorance, J, Naas, T, Rubin, JE, Spyrakis, F, Tangden, T, Gomez-Puertas, P
مصطلحات موضوعية: inhibitors of carbapenemase, virtual screening, approach rationalization
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:000852846600001; volume:23; issue:17; firstpage:9746; lastpage:9751; numberofpages:6; journal:INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES; https://hdl.handle.net/2318/1880320; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85137593402
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8Academic Journal
المؤلفون: Gianquinto E., Sodano F., Rolando B., Kostrzewa M., Allara M., Mahmoud A. M., Kumar P., Spyrakis F., Ligresti A., Chegaev K.
المساهمون: Gianquinto, E., Sodano, F., Rolando, B., Kostrzewa, M., Allara, M., Mahmoud, A. M., Kumar, P., Spyrakis, F., Ligresti, A., Chegaev, K.
مصطلحات موضوعية: cannabinoid receptor, drug design, hCB2R selective ligand, in silico simulation, mechanism of receptor activation
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:000897397600001; volume:27; issue:23; firstpage:8152; journal:MOLECULES; https://hdl.handle.net/11588/950134; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85143614156
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9Academic Journal
المؤلفون: Tiburtini, G. A., Bertarini, L., Bersani, M., Dragani, T. A., Rolando, B., Binello, A., Barge, A., Spyrakis, F.
المصدر: Archives of Toxicology; Sep2024, Vol. 98 Issue 9, p3035-3047, 13p
مصطلحات موضوعية: CHEMICAL transportation, ORGANIC anion transporters, BIOMOLECULES, CARRIER proteins, FLUOROALKYL compounds, FLUOROCARBONS
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10Academic Journal
المؤلفون: Failla M., Molaro M. C., Schiano M. E., Serafini M., Tiburtini G. A., Gianquinto E., Scoccia R., Battisegola C., Rimoli M. G., Chegaev K., Ercolano G., Lazzarato L., Spyrakis F., Sodano F.
المساهمون: Failla, M., Molaro, M. C., Schiano, M. E., Serafini, M., Tiburtini, G. A., Gianquinto, E., Scoccia, R., Battisegola, C., Rimoli, M. G., Chegaev, K., Ercolano, G., Lazzarato, L., Spyrakis, F., Sodano, F.
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:001359019600001; volume:67; issue:22; firstpage:19988; lastpage:20021; numberofpages:34; journal:JOURNAL OF MEDICINAL CHEMISTRY; https://hdl.handle.net/11588/989088
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11Academic Journal
المؤلفون: Cozzi M., Failla M., Gianquinto E., Kovachka S., Buoli Comani V., Compari C., De Bei O., Giaccari R., Marchesani F., Marchetti M., Ronda L., Rolando B., Baroni M., Cruciani G., Campanini B., Bettati S., Faggiano S., Lazzarato L., Spyrakis F.
المساهمون: Cozzi, M., Failla, M., Gianquinto, E., Kovachka, S., Buoli Comani, V., Compari, C., De Bei, O., Giaccari, R., Marchesani, F., Marchetti, M., Ronda, L., Rolando, B., Baroni, M., Cruciani, G., Campanini, B., Bettati, S., Faggiano, S., Lazzarato, L., Spyrakis, F.
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:001199822700079; volume:14; issue:1; journal:SCIENTIFIC REPORTS; https://hdl.handle.net/11381/2977973; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85189896105
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12Academic Journal
المؤلفون: Santini A., Tassinari E., Poeta E., Loi M., Ciani E., Trazzi S., Piccarducci R., Daniele S., Martini C., Pagliarani B., Tarozzi A., Bersani M., Spyrakis F., Danková D., Olsen C. A., Soldati R., Tumiatti V., Montanari S., De Simone A., Milelli A.
المساهمون: Santini A., Tassinari E., Poeta E., Loi M., Ciani E., Trazzi S., Piccarducci R., Daniele S., Martini C., Pagliarani B., Tarozzi A., Bersani M., Spyrakis F., Danková D., Olsen C.A., Soldati R., Tumiatti V., Montanari S., De Simone A., Milelli A.
مصطلحات موضوعية: Alzheimer’s disease, Glycogen Synthase Kinase 3β, Histone Deacetylase, Multitarget Drug, Neuroprotection
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/38747979; info:eu-repo/semantics/altIdentifier/wos/WOS:001226132400001; volume:15; issue:11; firstpage:2099; lastpage:2111; numberofpages:13; journal:ACS CHEMICAL NEUROSCIENCE; https://hdl.handle.net/11585/973360; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85193466667
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13Academic Journal
المؤلفون: D'arrigo G., Gianquinto E., Rossetti G., Cruciani G., Lorenzetti S., Spyrakis F.
المساهمون: D'arrigo G., Gianquinto E., Rossetti G., Cruciani G., Lorenzetti S., Spyrakis F.
مصطلحات موضوعية: Androgen, Estrogen, Flavonoid, G protein-coupled receptor, Genomic action, Molecular docking, Non-genomic action, Nuclear receptor, Cell Nucleu, Estradiol, Estrogen Receptor alpha, Estrogen Receptor beta, Human, Molecular Docking Simulation, Protein Binding, Receptors, Cell Surface, Testosterone
Relation: info:eu-repo/semantics/altIdentifier/pmid/33799482; info:eu-repo/semantics/altIdentifier/wos/WOS:000645400400001; volume:26; issue:1613; firstpage:1; lastpage:24; numberofpages:24; journal:MOLECULES; http://hdl.handle.net/2318/1806800; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85103863063
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14Academic Journal
المؤلفون: Parisi C., Failla M., Fraix A., Menilli L., Moret F., Reddi E., Rolando B., Spyrakis F., Lazzarato L., Fruttero R., Gasco A., Sortino S.
المساهمون: Parisi C., Failla M., Fraix A., Menilli L., Moret F., Reddi E., Rolando B., Spyrakis F., Lazzarato L., Fruttero R., Gasco A., Sortino S.
Relation: info:eu-repo/semantics/altIdentifier/pmid/34163730; info:eu-repo/semantics/altIdentifier/wos/WOS:000637925000007; volume:12; issue:13; firstpage:4740; lastpage:4746; numberofpages:7; journal:CHEMICAL SCIENCE; http://hdl.handle.net/2318/1794858; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85103917275
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15Academic Journal
المؤلفون: Marverti G., Marraccini C., Martello A., D'Arca D., Pacifico S., Guerrini R., Spyrakis F., Gozzi G., Lauriola A., Santucci M., Cannazza G., Tagliazucchi L., Cazzato A. S., Losi L., Ferrari S., Ponterini G., Costi M. P.
المساهمون: Marverti G., Marraccini C., Martello A., D'Arca D., Pacifico S., Guerrini R., Spyrakis F., Gozzi G., Lauriola A., Santucci M., Cannazza G., Tagliazucchi L., Cazzato A.S., Losi L., Ferrari S., Ponterini G., Costi M.P.
مصطلحات موضوعية: Antineoplastic Agent, Catalytic Domain, Cell Line, Tumor, Cell Proliferation, Drug Delivery System, Enzyme Inhibitor, Female, Folate Receptor 1, Folic Acid, Human, Models, Molecular, Ovarian Neoplasm, Peptide, Thymidylate Synthase
Relation: info:eu-repo/semantics/altIdentifier/pmid/33710891; info:eu-repo/semantics/altIdentifier/wos/WOS:000635440600024; volume:64; issue:6; firstpage:3204; lastpage:3221; numberofpages:18; journal:JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/2318/1806796; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85103469735
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16Academic Journal
المؤلفون: Gastaldi S., Boscaro V., Gianquinto E., Sandall C. F., Giorgis M., Marini E., Blua F., Gallicchio M., Spyrakis F., Macdonald J. A., Bertinaria M.
المساهمون: Gastaldi S., Boscaro V., Gianquinto E., Sandall C.F., Giorgis M., Marini E., Blua F., Gallicchio M., Spyrakis F., Macdonald J.A., Bertinaria M.
مصطلحات موضوعية: ATP hydrolysi, Interleukin-1β, MD simulation, NLRP3 inhibitor, Pyroptosi, Human, Inflammasome, Interleukin-1beta, Macrophage, NLR Family, Pyrin Domain-Containing 3 Protein, THP-1 Cell, Imidazoles
Relation: info:eu-repo/semantics/altIdentifier/pmid/34209843; info:eu-repo/semantics/altIdentifier/wos/WOS:000671249300001; volume:26; issue:13; firstpage:1; lastpage:35; numberofpages:35; journal:MOLECULES; http://hdl.handle.net/2318/1798199; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85109365476; https://www.mdpi.com/1420-3049/26/13/3975
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17Academic Journal
المؤلفون: Santucci M., Luciani R., Gianquinto E., Pozzi C., Di Pisa F., Dello Iacono L., Landi G., Tagliazucchi L., Mangani S., Spyrakis F., Costi M. P.
المساهمون: Santucci M., Luciani R., Gianquinto E., Pozzi C., Di Pisa F., Dello Iacono L., Landi G., Tagliazucchi L., Mangani S., Spyrakis F., Costi M.P.
مصطلحات موضوعية: DHFR-TS, Drug discovery, GSK Kinetobox, Leishmaniasi, Medium throughput screening, Molecular modelling, PTR1, Trypanosomiasis
Relation: info:eu-repo/semantics/altIdentifier/pmid/34959646; volume:14; issue:12; firstpage:1246; lastpage:1246; numberofpages:1; journal:PHARMACEUTICALS; info:eu-repo/grantAgreement/EC/FP7/603240; http://hdl.handle.net/2318/1829160; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85120403715
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18Academic Journal
المؤلفون: Gossen J., Albani S., Hanke A., Joseph B. P., Bergh C., Kuzikov M., Costanzi E., Manelfi C., Storici P., Gribbon P., Beccari A. R., Talarico C., Spyrakis F., Lindahl E., Zaliani A., Carloni P., Wade R. C., Musiani F., Kokh D. B., Rossetti G.
المساهمون: Gossen J., Albani S., Hanke A., Joseph B.P., Bergh C., Kuzikov M., Costanzi E., Manelfi C., Storici P., Gribbon P., Beccari A.R., Talarico C., Spyrakis F., Lindahl E., Zaliani A., Carloni P., Wade R.C., Musiani F., Kokh D.B., Rossetti G.
مصطلحات موضوعية: conformational space, druggability, molecular dynamics simulation, Mpro, protein binding site flexibility, SARS-CoV-2, virtual screening
Relation: info:eu-repo/semantics/altIdentifier/pmid/34136757; info:eu-repo/semantics/altIdentifier/wos/WOS:000662229400006; volume:4; issue:3; firstpage:1079; lastpage:1095; numberofpages:17; journal:ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE; http://hdl.handle.net/2318/1806794; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85103514869
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19Academic Journal
المؤلفون: Ronda L., Tonelli A., Sogne E., Autiero I., Spyrakis F., Pellegrino S., Abbiati G., Maffioli E., Schulte C., Piano R., Cozzini P., Mozzarelli A., Bettati S., Clerici F., Milani P., Lenardi C., Tedeschi G., Gelmi M. L.
المساهمون: Ronda L., Tonelli A., Sogne E., Autiero I., Spyrakis F., Pellegrino S., Abbiati G., Maffioli E., Schulte C., Piano R., Cozzini P., Mozzarelli A., Bettati S., Clerici F., Milani P., Lenardi C., Tedeschi G., Gelmi M.L.
مصطلحات موضوعية: Biosensor, Circular dichroism, Fluorescence, Molecular dynamic, Nanostructured surface, Point-of-care detection, Staphylococcus aureus
Relation: info:eu-repo/semantics/altIdentifier/pmid/32887407; info:eu-repo/semantics/altIdentifier/wos/WOS:000569787700001; volume:20; issue:17; firstpage:1; lastpage:22; numberofpages:22; journal:SENSORS; http://hdl.handle.net/2318/1765347; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85090099945
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20Academic Journal
المؤلفون: Spyrakis F., Santucci M., Maso L., Cross S., Gianquinto E., Sannio F., Verdirosa F., De Luca F., Docquier J. -D., Cendron L., Tondi D., Venturelli A., Cruciani G., Costi M. P.
المساهمون: Spyrakis F., Santucci M., Maso L., Cross S., Gianquinto E., Sannio F., Verdirosa F., De Luca F., Docquier J.-D., Cendron L., Tondi D., Venturelli A., Cruciani G., Costi M.P.
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:000556388300017; volume:10; issue:12763; firstpage:1; lastpage:15; numberofpages:15; journal:SCIENTIFIC REPORTS; http://hdl.handle.net/2318/1765330; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85088710021