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1Academic Journal
المصدر: International Journal of Microbiology, Vol 2010 (2010)
مصطلحات موضوعية: Microbiology, QR1-502
وصف الملف: electronic resource
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2Academic Journal
المؤلفون: Vrinda N, Sowmya Bharath, Sheshagiri Gaonkar, B. L. Suresh, B. N. Mahesh, Radha K. Sh, Ramesh Jayaram, Parvinder Kaur, Mycobacteriumciprofloxacin Against
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.623.6980; http://aac.asm.org/content/51/2/576.full.pdf
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3Academic Journal
المؤلفون: Vrinda N, Sowmya Bharath, E. Kantharaj, Parvinder Kaur, B. L. Suresh, B. N. Mahesh, R. Jayashree, Ramesh Jayaram, Radha K. Sh, Sheshagiri Gaonkar
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.514.221; http://aac.asm.org/content/48/8/2951.full.pdf
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4
المؤلفون: V. K. Ramya, Vijender Panduga, Gajanan Shanbhag, Michelle Coulson, Sowmya Bharath, Vaishali Humnabadkar, Prashanti Madhavapeddi, Vasan K. Sambandamurthy, Disha Awasthy, Jim Werngren, Praveena Manjrekar, Chandan Narayan, Vijayashree Achar, Mahesh Kumar Kn, Sunita M. de Sousa, Jitendar Reddy, C. N. Naveen Kumar, Kakoli Mukherjee, Sreenivasaiah Menasinakai, Ugarkar Bheemarao, Samit Ganguly, Umender Sharma, David Waterson, Vikas Patil, Sven Hoffner, Radha Nandishaiah, Sreevalli Sharma, Shahul Hameed P, Uma Arora, Anandkumar Raichurkar, Suresh Solapure, Parvinder Kaur, Jayashree Puttur, Vikas Shinde, Murugan Chinnapattu, Suresh Rudrapatana, Sheshagiri Gaonkar, Anirban Ghosh
المصدر: Journal of Medicinal Chemistry. 57:4889-4905
مصطلحات موضوعية: ERG1 Potassium Channel, hERG, Antitubercular Agents, Administration, Oral, Biological Availability, Microbial Sensitivity Tests, Drug resistance, Pharmacology, DNA gyrase, Microbiology, Mycobacterium tuberculosis, Structure-Activity Relationship, Bacterial Proteins, Piperidines, In vivo, Drug Resistance, Bacterial, Drug Discovery, Animals, Humans, Topoisomerase II Inhibitors, Structure–activity relationship, Tuberculosis, Pulmonary, Mice, Inbred BALB C, biology, Chemistry, Macrophages, Stereoisomerism, biology.organism_classification, Ether-A-Go-Go Potassium Channels, Rats, Molecular Docking Simulation, Protein Subunits, DNA Gyrase, Acute Disease, Chronic Disease, Mutation, biology.protein, Molecular Medicine, Topoisomerase-II Inhibitor, Intracellular, Fluoroquinolones
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5
المؤلفون: P. Ann Boriack-Sjodin, B. K. Kishore Reddy, Ramesh R. Kale, Vijaykamal Ahuja, Sunita M. de Sousa, Krishnan Malolanarasimhan, Sheshagiri Gaonkar, Anandkumar Raichurkar, Sreenivasaiah Menasinakai, Halesha D. Basavarajappa, Prashanti Madhavapeddi, M. R. Manjunatha, Shahul Hameed, David Waterson, Radha Nandishaiah, Vasan K. Sambandamurthy, C. N. Naveen Kumar, Derek Ogg, Vikas Shinde, Vaishali Humnabadkar, Krishna Koushik, Sreevalli Sharma, K. N. Mahesh Kumar, Sandeep R. Ghorpade, Kale Manoj Ganpat, Samit Ganguly, Lalit kumar Jena
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:870-879
مصطلحات موضوعية: Pyridones, Stereochemistry, Clinical Biochemistry, Antitubercular Agents, Administration, Oral, Pharmaceutical Science, Microbial Sensitivity Tests, Biochemistry, DNA gyrase, Hydrophobic effect, Mycobacterium tuberculosis, Inhibitory Concentration 50, Mice, chemistry.chemical_compound, Drug Discovery, Ribose, Animals, Topoisomerase II Inhibitors, Urea, Molecular Biology, IC50, chemistry.chemical_classification, Molecular Structure, biology, Organic Chemistry, Active site, biology.organism_classification, Disease Models, Animal, Thiazoles, Enzyme, chemistry, biology.protein, Molecular Medicine, DNA
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6
المؤلفون: R. Jayashree, Sowmya Bharath, Ramesh Jayaram, Parvinder Kaur, B. L. Suresh, Radha Shandil, Sheshagiri Gaonkar, V. Balasubramanian, Vrinda Nandi, B. N. Mahesh
المصدر: Antimicrobial Agents and Chemotherapy. 51:576-582
مصطلحات موضوعية: Ofloxacin, Time Factors, Moxifloxacin, Antitubercular Agents, Drug Evaluation, Preclinical, Microbial Sensitivity Tests, Pharmacology, Biology, Microbiology, Mycobacterium tuberculosis, Mice, Ciprofloxacin, Predictive Value of Tests, In vivo, medicine, Animals, Tuberculosis, Experimental Therapeutics, Pharmacology (medical), Antibacterial agent, Aza Compounds, Mice, Inbred BALB C, Dose-Response Relationship, Drug, biology.organism_classification, Anti-Bacterial Agents, Infectious Diseases, Sparfloxacin, Pharmacodynamics, Quinolines, Fluoroquinolones, medicine.drug
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7
المؤلفون: E. Kantharaj, Ramesh Jayaram, B. L. Suresh, V. Balasubramanian, Radha Shandil, Vrinda Nandi, B. N. Mahesh, R. Jayashree, Sheshagiri Gaonkar, Parvinder Kaur, Sowmya Bharath
المصدر: Antimicrobial Agents and Chemotherapy. 48:2951-2957
مصطلحات موضوعية: Male, Tuberculosis, medicine.drug_class, Antitubercular Agents, Microbial Sensitivity Tests, In Vitro Techniques, Pharmacology, Antimycobacterial, Cell Line, Mice, Pharmacokinetics, Isoniazid, Animals, Humans, Medicine, Experimental Therapeutics, Pharmacology (medical), Chromatography, High Pressure Liquid, Antibacterial agent, Aerosols, Mice, Inbred BALB C, Dose-Response Relationship, Drug, business.industry, Macrophages, Dose fractionation, Blood Proteins, Mycobacterium tuberculosis, medicine.disease, Dose–response relationship, Infectious Diseases, Area Under Curve, Pharmacodynamics, Immunology, Female, business, Protein Binding, medicine.drug
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8
المؤلفون: E. Kantharaj, Parvinder Kaur, R. Jayashree, Ramesh Jayaram, B. L. Suresh, Radha Shandil, Sheshagiri Gaonkar, V. Balasubramanian, B. N. Mahesh, Sowmya Bharat, Vrinda Nandi
المصدر: Antimicrobial Agents and Chemotherapy. 47:2118-2124
مصطلحات موضوعية: Male, medicine.drug_class, Antibiotics, Microbial Sensitivity Tests, In Vitro Techniques, Biology, Cell Line, Microbiology, Mycobacterium tuberculosis, Mice, Pharmacokinetics, In vivo, medicine, Animals, Potency, Experimental Therapeutics, Pharmacology (medical), Antibiotics, Antitubercular, Tuberculosis, Pulmonary, Aerosols, Pharmacology, Mice, Inbred BALB C, Dose-Response Relationship, Drug, Macrophages, biology.organism_classification, Disease Models, Animal, Dose–response relationship, Infectious Diseases, Pharmacodynamics, Female, Rifampin, Rifampicin, medicine.drug
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9
المؤلفون: Sheshagiri Gaonkar, Naveen Kumar, David Melnick, Scott Butler, V. Balasubramanian, Sowmya Bharath, K. N. Mahesh, Jitender Reddy, Radha Shandil, Abhijeet Deshpande, Lindsay Wright, Suresh Solapure
مصطلحات موضوعية: Drug, Tuberculosis, media_common.quotation_subject, Microbial Sensitivity Tests, Pharmacology, Mycobacterium tuberculosis, Mice, Pharmacokinetics, Oral administration, Drug Resistance, Multiple, Bacterial, medicine, Extracellular, Animals, Pharmacology (medical), Experimental Therapeutics, Drug Dosage Calculations, Tuberculosis, Pulmonary, Oxazolidinones, media_common, Mice, Inbred BALB C, Lung, biology, Dose-Response Relationship, Drug, business.industry, medicine.disease, biology.organism_classification, Disease Models, Animal, Infectious Diseases, medicine.anatomical_structure, Pharmacodynamics, Area Under Curve, Immunology, business
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10
المؤلفون: David Waterson, Vijender Panduga, Gajanan Shanbhag, Jim Werngren, Sheshagiri Gaonkar, Manjunatha R, Gulebahar Sheikh, Prashanti Madhavapeddi, Reetobrata Basu, Kakoli Mukherjee, Radha Shandil, Jitendar Reddy, Vrinda Nandi, Mahesh Kumar, Suresh Solapure, Venkita Subbulakshmi, Anirban Ghosh, Disha Awasthy, Praveena Manjrekar, Jon Read, Meenakshi Balganesh, Abhijeet Deshpande, Vaishali Humnabadkar, Anand Kumar V. Raichurkar, Sven Hoffner, Helen H.J. McMiken, Shahul Hameed P, Vasan K. Sambandamurthy, Sreevalli Sharma, Jayashree Puttur, Murugan Chinnapattu
المصدر: Antimicrobial agents and chemotherapy. 58(1)
مصطلحات موضوعية: Antitubercular Agents, DNA gyrase, Microbiology, Cell Line, Mycobacterium tuberculosis, Mice, Structure-Activity Relationship, Structure–activity relationship, Animals, Humans, Tuberculosis, Pharmacology (medical), Experimental Therapeutics, Mode of action, chemistry.chemical_classification, Pharmacology, biology, Errata, Mycobacterium smegmatis, Point mutation, biochemical phenomena, metabolism, and nutrition, biology.organism_classification, bacterial infections and mycoses, Enzyme, Infectious Diseases, chemistry, Biochemistry, DNA supercoil, bacteria
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11
المؤلفون: Sunita M. de Sousa, C. N. Naveen Kumar, Anandkumar Raichurkar, Kale Manoj Ganpat, Krishna Koushik, M. R. Manjunatha, David Waterson, Vasan K. Sambandamurthy, Vikas Shinde, K. N. Mahesh Kumar, Jitendar Reddy, Julie A. Tucker, Prashanti Madhavapeddi, Derek Ogg, Sandeep R. Ghorpade, Shubhada Barde, Halesha D. Basavarajappa, Shahul Hameed P, Samit Ganguly, V. K. Ramya, Lalit kumar Jena, Vijender Panduga, Vijaykamal Ahuja, Prakash Vachaspati, David C. McKinney, Jayashree Giridhar, Anirban Ghosh, Sheshagiri Gaonkar, Supreeth Guptha, P. Ann Boriack-Sjodin, Suresh Rudrapatna, Sreevalli Sharma, Usha Kranthi, Vaishali Humnabadkar
المصدر: Journal of medicinal chemistry. 56(21)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Pyridines, Antitubercular Agents, DNA gyrase, Mycobacterium tuberculosis, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Drug Discovery, Ribose, Structure–activity relationship, Animals, Topoisomerase II Inhibitors, Tuberculosis, Urea, Homology modeling, IC50, Mice, Inbred BALB C, biology, Dose-Response Relationship, Drug, Molecular Structure, biochemical phenomena, metabolism, and nutrition, biology.organism_classification, In vitro, Disease Models, Animal, chemistry, Biochemistry, DNA Gyrase, Molecular Medicine, Pharmacophore
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12
المؤلفون: Suresh Solapure, Samit Ganguly, Vijender Panduga, Naveen Kumar, George L. Drusano, K. G. Vishwas, Radha Shandil, V. Balasubramanian, Sheshagiri Gaonkar, K. N. Mahesh Kumar, Jitendar Reddy, Abhijeet Deshpande, Arnold Louie
مصطلحات موضوعية: Tuberculosis, Moxifloxacin, Antitubercular Agents, Pharmacology, Mycobacterium tuberculosis, Mice, Oral administration, In vivo, medicine, Animals, Pharmacology (medical), Experimental Therapeutics, Tuberculosis, Pulmonary, Aza Compounds, Mice, Inbred BALB C, Lung, biology, business.industry, biochemical phenomena, metabolism, and nutrition, medicine.disease, biology.organism_classification, Infectious Diseases, medicine.anatomical_structure, Pharmacodynamics, Immunology, Quinolines, Rifampin, Antagonism, business, medicine.drug, Fluoroquinolones
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13Academic Journal
المؤلفون: Vadim Makarov, Giulia Manina, Katarina Mikusova, Ute Möllmann, Olga Ryabova, Brigitte Saint-Joanis, Neeraj Dhar, Maria Rosalia Pasca, Silvia Buroni, Anna Paola Lucarelli, Anna Milano, Edda De Rossi, Martina Belanova, Adela Bobovska, Petronela Dianiskova, Jana Kordulakova, Claudia Sala, Elizabeth Fullam, Patricia Schneider, John D McKinney, Priscille Brodin, Thierry Christophe, Simon Waddell, Philip Butcher, Jakob Albrethsen, Ida Rosenkrands, Roland Brosch, Vrinda Nandi, Sowmya Bharath, Sheshagiri Gaonkar, Radha K Shandil, Venkataraman Balasubramanian, Tanjore Balganesh, Sandeep Tyagi, Jacques Grosset, Giovanna Riccardi, Stewart T Cole
مصطلحات موضوعية: Mycobacterium, Tuberculosis, Drug discovery, Transcriptional profiling, Infection
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14
المؤلفون: Sowmya Bharath, Disha Awasthy, Umender Sharma, Venkita Subbulakshmi, Sheshagiri Gaonkar, Nimi Marcel, Radha Shandil, Reena Yadav
المصدر: Microbiology (Reading, England). 155(Pt 9)
مصطلحات موضوعية: Auxotrophy, Branched-chain amino acid, Cell Culture Techniques, Vaccines, Attenuated, Microbiology, chemistry.chemical_compound, Mice, Valine, Animals, Tuberculosis Vaccines, Tuberculosis, Pulmonary, Amino acid synthesis, chemistry.chemical_classification, Acetolactate synthase, Mice, Inbred BALB C, biology, Virulence, Macrophages, Mycobacterium tuberculosis, Amino acid, Acetolactate Synthase, chemistry, Biochemistry, Genes, Bacterial, biology.protein, Leucine, Isoleucine, Amino Acids, Branched-Chain, Gene Deletion
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15
المؤلفون: V. Balasubramanian, Radha Shandil, Vadim Makarov, Patricia Schneider, Martina Belanova, Anna Milano, Priscille Brodin, Tanjore S. Balganesh, Claudia Sala, Sandeep Tyagi, Katarína Mikušová, Thierry Christophe, Adela Bobovská, Edda De Rossi, Anna Paola Lucarelli, Ute Möllmann, Giulia Manina, Petronela Dianišková, Elizabeth Fullam, Roland Brosch, O. B. Ryabova, Simon J. Waddell, Maria Rosalia Pasca, Ida Rosenkrands, Brigitte Saint-Joanis, Jana Korduláková, Sheshagiri Gaonkar, Silvia Buroni, Jacques H. Grosset, Jakob Albrethsen, Philip D. Butcher, Stewart T. Cole, John D. McKinney, Sowmya Bharath, Neeraj Dhar, Vrinda Nandi, Giovanna Riccardi
مصطلحات موضوعية: Identification, Tuberculosis, Molecular Sequence Data, Antitubercular Agents, Racemases and Epimerases, Thiazines, SQ109, Microbial Sensitivity Tests, Article, Mycobacterium, Microbiology, Mycobacterium tuberculosis, Mice, chemistry.chemical_compound, Cell Wall, Polysaccharides, Drug Resistance, Bacterial, medicine, Animals, Spiro Compounds, Amino Acid Sequence, Enzyme Inhibitors, Ethambutol, chemistry.chemical_classification, Mice, Inbred BALB C, QR0075, Multidisciplinary, Molecular Structure, biology, Gene Expression Regulation, Bacterial, biology.organism_classification, medicine.disease, Arabinose, R1, Cell-Wall, In vitro, Enzyme, chemistry, Genes, Bacterial, Ex vivo, medicine.drug
وصف الملف: application/pdf
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16Academic Journal
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.1041.1140; http://downloads.hindawi.com/journals/ijmicro/2010/426035.pdf
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17Academic Journal
المؤلفون: Sowmya Bharat, R. K. Sh, E. Kantharaj, L. Suresh, B. N. Mahesh, R. Jayashree, Vrinda N, Ramesh Jayaram, Sheshagiri Gaonkar, Parvinder Kaur
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.527.2164; http://aac.asm.org/content/47/7/2118.full.pdf
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18Academic Journal
المساهمون: The Pennsylvania State University CiteSeerX Archives
المصدر: ftp://ftp.ncbi.nlm.nih.gov/pub/pmc/df/ee/Int_J_Microbiol_2010_Mar_18_2010_426035.tar.gz
وصف الملف: application/zip
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19Academic Journal
المؤلفون: Awasthy, Disha1, Sheshagiri Gaonkar1, Shandil, R. K.1, Yadav, Reena1, Bharath, Sowmya1, Marcel, Nimi1, Subbulakshmi, Venkita1, Sharma, Umender1 umender.sharma@astrazeneca.com
المصدر: Microbiology (13500872). Sep2009, Vol. 155 Issue 9, p2978-2987. 10p.
مصطلحات موضوعية: *PHYSIOLOGICAL effects of enzymes, *BRANCHED chain amino acids, *MYCOBACTERIUM tuberculosis, *LABORATORY mice, *MICROBIAL virulence