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المصدر: The Medicinal Chemist's Guide to Solving ADMET Challenges ISBN: 9781788012270
مصطلحات موضوعية: Drug, Cytochrome, biology, Chemistry, media_common.quotation_subject, Endogeny, SUPERFAMILY, Metabolism, Pharmacology, Inhibitory postsynaptic potential, digestive system, biology.protein, Drug metabolism, media_common
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المؤلفون: Peter J. Bungay, Martin Corless, Sarah Elizabeth Skerratt, Joseph S. Warmus, Sharan K. Bagal, C. Elizabeth Payne, Miller Duncan Charles, Kemp Mark Ian, David R. Fenwick, Paul Blackwell, Yoshihisa Murata, Bruce Brown, Laia Malet Sanz, David Fengas, James Michael Crawforth, Victoria Gray, Wolfgang Klute, Alan Daniel Brown, David C. Blakemore, Edward B. Stevens
المصدر: Bioorganic & Medicinal Chemistry. 27:230-239
مصطلحات موضوعية: Benzimidazole, 010405 organic chemistry, Sodium channel, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Inflammatory pain, Highly selective, 01 natural sciences, Biochemistry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, Safety profile, chemistry, Drug Discovery, NAV1, Molecular Medicine, Molecular Biology, ADME
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المصدر: ACS Symposium Series ISBN: 9780841234321
ACS Symposium Seriesمصطلحات موضوعية: business.industry, Trk receptor, Medicine, Pharmacology, business
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المؤلفون: Michelle Tran-Dubé, Bruce M. Bechle, Michelle Kraus, Ciarán N. Cronin, Kim James, Joseph S. Warmus, Fen Wang, Jianmin Sun, Indrawan James Mcalpine, Sacha Ninkovic, Jianwei Bian, Samantha Elizabeth Greasley, Neil J. Flanagan, Matthew Corbett, Rebecca Dias, Andrews Mark David, Asako Nagata, John F. Braganza, Linda Kitching, David C. Blakemore, Eric Johnson, Sarah Elizabeth Skerratt, Kiyoyuki Omoto, Sharan K. Bagal, Jingrong Jean Cui, James Bilsland, Peter J. Bungay, Rachel L. Grimley, Stephanie Scales, Gareth Waldron
المصدر: Journal of medicinal chemistry. 61(15)
مصطلحات موضوعية: 0301 basic medicine, animal structures, Protein Conformation, Pyridines, Pain, Tropomyosin receptor kinase B, Neurotrophin-3, Pharmacology, Tropomyosin receptor kinase A, Ligands, 030226 pharmacology & pharmacy, Tropomyosin receptor kinase C, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Drug Discovery, Animals, Humans, Tissue Distribution, Protein Kinase Inhibitors, Brain-derived neurotrophic factor, biology, Chemistry, Receptor Protein-Tyrosine Kinases, Rats, Molecular Docking Simulation, 030104 developmental biology, Nerve growth factor, nervous system, Solubility, Trk receptor, biology.protein, Molecular Medicine, Neurotrophin
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المؤلفون: Sarah Elizabeth Skerratt, Xiaohe Tong, Lei Zhao, Rita Ferreira, Joe Warmus, Sarah A. Nickolls, Sian Humphreys, Csilla C. Jorgensen
المصدر: MedChemComm. 7:1564-1571
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, biology, High-throughput screening, Organic Chemistry, Ferroportin, Pharmaceutical Science, medicine.disease, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Iron homeostasis, chemistry, High-content screening, Drug Discovery, medicine, biology.protein, Molecular Medicine, BODIPY, Hemochromatosis
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المصدر: MedChemComm. 7:813-819
مصطلحات موضوعية: 0301 basic medicine, Stereochemistry, Binding pocket, Pharmaceutical Science, urologic and male genital diseases, Biochemistry, Homology (biology), 03 medical and health sciences, Oxidoreductase, Drug Discovery, Progesterone receptor, heterocyclic compounds, Pharmacology, chemistry.chemical_classification, biology, Chemistry, organic chemicals, Organic Chemistry, Antagonist, Active site, respiratory system, Sulfonamide, enzymes and coenzymes (carbohydrates), 030104 developmental biology, biology.protein, Molecular Medicine, Pharmacophore
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المؤلفون: Joseph S. Warmus, Sarah Elizabeth Skerratt, Steven M Reister, David C. Pryde, Thomas Ryckmans, J. Turner, Karen M. Padilla, Katrina E. Yoger, A. C. Gerlach, Nigel Alan Swain, G. Amato, Peter J. Cox, C. G. West, Brian E. Marron, David C. Blakemore
المصدر: MedChemComm. 7:2145-2158
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, medicine.drug_class, Chemistry, Organic Chemistry, Pharmaceutical Science, Carboxamide, Atopic dermatitis, medicine.disease, Biochemistry, Combinatorial chemistry, 03 medical and health sciences, 030104 developmental biology, Pharmacokinetics, Drug Discovery, medicine, Molecular Medicine
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المؤلفون: Christopher William West, Sarah Elizabeth Skerratt
المصدر: Channels. 9:344-351
مصطلحات موضوعية: Nociception, Chemistry, Drug discovery, Sodium channel, Biophysics, Complex disease, Pain, Voltage-Gated Sodium Channels, Review, Pharmacology, Biochemistry, Tolerability, Ion channel modulation, Animals, Humans, Effective treatment, Neuroscience, Ion channel, Anesthetics, Sodium Channel Blockers
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المؤلفون: Sarah Elizabeth Skerratt, R. Ian Storer
مصطلحات موضوعية: business.industry, In vivo, Kinase, Medicine, Penetration (firestop), business, Neuroscience, Design space
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المؤلفون: Yuya Maruyama, Sarah E. Johnston, Emma Armstrong, Csilla C. Jorgensen, Rubben Torella, Parul Choudhary, Caroline L. Benn, R. Ian Storer, Maria Barthmes, John S. Janiszewski, Sarah Elizabeth Skerratt, Mary Piotrowski
المصدر: Frontiers in Molecular Neuroscience
مصطلحات موضوعية: 0301 basic medicine, Phenotypic screening, solute carrier, Allosteric regulation, Biology, SLC5A7, 03 medical and health sciences, Cellular and Molecular Neuroscience, 0302 clinical medicine, medicine, Molecular Biology, Original Research, mass spectrometry, Virtual screening, SSM electrophysiology, phenotypic screening, Transporter, acetylcholine, small molecule screening, Solute carrier family, Choline transporter, 030104 developmental biology, Biochemistry, HACU (high affinity choline uptake), Cholinergic, Neuroscience, 030217 neurology & neurosurgery, Acetylcholine, medicine.drug
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المصدر: MedChemComm. 4:244-251
مصطلحات موضوعية: Pharmacology, Series (mathematics), business.industry, Computer science, Organic Chemistry, Bayesian probability, Pharmaceutical Science, Machine learning, computer.software_genre, Biochemistry, Triage, Rapid identification, Identification (information), Drug Discovery, False positive paradox, Molecular Medicine, Artificial intelligence, business, computer
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المؤلفون: Russell Jones, Inaki Morao, Colin Robinson, Stupple Paul Anthony, Susan Cole, David G. Brown, Karl Richard Gibson, Angus N. R. Nedderman, Gareth Waldron, Sarah Elizabeth Skerratt, James Bilsland, Andrews Mark David, Kiyoyuki Omoto, Peter J. Bungay, Kimberly Skinner, Sharan K. Bagal, Thomas Ryckmans
المصدر: Journal of medicinal chemistry. 59(22)
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Druggability, Pain, Quantitative Structure-Activity Relationship, Neurotrophin-3, Pharmacology, 01 natural sciences, Receptor tyrosine kinase, 03 medical and health sciences, Drug Discovery, medicine, Humans, Pyrroles, Protein Kinase Inhibitors, Brain-derived neurotrophic factor, biology, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Chronic pain, medicine.disease, 0104 chemical sciences, 030104 developmental biology, Nerve growth factor, Pyrimidines, nervous system, Trk receptor, QD431, biology.protein, Molecular Medicine, Protein Kinases, Neurotrophin
وصف الملف: application/pdf
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مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Dihydropyran, Organic Chemistry, Drug Discovery, Organic chemistry, Biochemistry
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المؤلفون: Thomas Ryckmans, James Edward John Mills, Mark E. Bunnage, Miller Duncan Charles, Alan Daniel Brown, C M Barker, Sarah Elizabeth Skerratt
المصدر: Med. Chem. Commun.. 3:174-178
مصطلحات موضوعية: Pharmacology, Series (mathematics), Computer science, Organic Chemistry, Pharmaceutical Science, Context (language use), computer.software_genre, Biochemistry, Empirical research, Drug Discovery, Molecular Medicine, Pairwise comparison, Data mining, computer
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المصدر: Tetrahedron Letters. 50:7141-7143
مصطلحات موضوعية: chemistry.chemical_compound, Formal synthesis, chemistry, Dihydropyran, Stereochemistry, Organic Chemistry, Drug Discovery, Organic chemistry, Indolizidine, Biochemistry, Quinolizidines
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المؤلفون: Robert M. Owen, Sharan K. Bagal, David C. Pryde, Edward B. Stevens, Peter J. Cox, Kiyoyuki Omoto, R. Ian Storer, Sarah Elizabeth Skerratt, Alan Daniel Brown, Benjamin Sidders, Nigel Alan Swain
المصدر: Journal of medicinal chemistry. 56(3)
مصطلحات موضوعية: Models, Molecular, Drug discovery, Functional features, Computational biology, Biology, Pharmacology, Ion Channels, Membrane protein, Drug Discovery, Molecular Medicine, Humans, Tissue distribution, Ion channel, High potential, Phylogeny
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المصدر: Organic letters. 13(22)
مصطلحات موضوعية: Models, Molecular, Vinyl Compounds, Bicyclic molecule, Molecular Structure, Stereochemistry, Chemistry, Organic Chemistry, Biochemistry, Combinatorial chemistry, Cyclization, Core (graph theory), Urea, Physical and Theoretical Chemistry, Curtius rearrangement, Pyrrolizidine Alkaloids