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1
المؤلفون: Nicholas A. Meanwell, Ravi Kumar Trivedi, Tatyana Zvyaga, Richard Rampulla, Sarkunam Kandhasamy, Debarati Mazumder Tagore, Sureshbabu Vishwakrishnan, Arvind Mathur, Sunitha Puttaswamy, Abhijith Rao, Hua Fang, Sankar Sivaprasad, Susan Jenkins, Eric Mull, Kathy Mosure, Kaushik Ghosh, Barbara Zheng, Subba Reddy, Fiona McPhee, Chaoqun Chen, Bowsher Michael S, James Loy, Ying-Kai Wang, Amit Kumar, Ramkumar Rajamani, Kishore Rendunchintala, Paul Michael Scola, Gillis Eric P, Salil D. Desai, Li-Qiang Sun, Rushith Kumar Anumula, Nagalakshmi Pulicharla, Sheldon Hiebert, Venkata Rao Baratam, Paul Falk, Sarmistha Sinha, Stanley D'andrea
المصدر: Journal of Medicinal Chemistry. 63:14740-14760
مصطلحات موضوعية: Serine Proteinase Inhibitors, viruses, Hepatitis C virus, CHO Cells, Hepacivirus, Microbial Sensitivity Tests, Tripeptide, Viral Nonstructural Proteins, medicine.disease_cause, Antiviral Agents, Peptides, Cyclic, 01 natural sciences, Structure-Activity Relationship, 03 medical and health sciences, Cricetulus, Drug Stability, Drug Discovery, Genotype, medicine, Animals, 030304 developmental biology, 0303 health sciences, NS3, Molecular Structure, Chemistry, virus diseases, Virology, digestive system diseases, Third generation, Rats, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Microsomes, Liver, Molecular Medicine, Ns3 4a protease
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2
المؤلفون: Priyadeep Bhutani, John F. Kadow, Rambabu Arla, Sarmistha Sinha, Murugaiah A. M. Subbaiah, Susan Jenkins, Murali Subramanian, Salil D. Desai, Shweta Padmanabhan, Sandhya Mandlekar, Nicholas A. Meanwell, Lakshumanan Subramani, Srikanth Sridhar, Mark Krystal, Thangeswaran Ramar
المصدر: European Journal of Medicinal Chemistry. 207:112749
مصطلحات موضوعية: Alkylation, Tertiary amine, Atazanavir Sulfate, Biological Availability, 01 natural sciences, 03 medical and health sciences, Drug Stability, HIV Protease, HIV-1 protease, Drug Discovery, medicine, Humans, Prodrugs, Amines, Amino Acids, 030304 developmental biology, Pharmacology, chemistry.chemical_classification, 0303 health sciences, biology, 010405 organic chemistry, Chemistry, Organic Chemistry, HIV Protease Inhibitors, General Medicine, Prodrug, Combinatorial chemistry, 0104 chemical sciences, Bioavailability, Atazanavir, Amino acid, biology.protein, Amine gas treating, Linker, medicine.drug
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3
المؤلفون: George Crull, Ipsit Kundu, Balvinder S. Vig, Varia Sailesh Amilal, Salil D. Desai, Hemant Bhutani, Narayana P. Swamy, Ravi P. Shah, Chiranjeevi Venkatesh, Sridhar Desikan, Sherif Badawy, Duohai Pan, Junshu Zhao
المصدر: European Journal of Pharmaceutical Sciences. 152:105429
مصطلحات موضوعية: Vinyl alcohol, Materials science, Polymers, Pharmaceutical Science, Ether, Hydrochloric acid, 02 engineering and technology, engineering.material, 030226 pharmacology & pharmacy, Excipients, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Coating, Dissolution, chemistry.chemical_classification, Aqueous solution, Polymer, 021001 nanoscience & nanotechnology, Acid strength, chemistry, Chemical engineering, Polyvinyl Alcohol, engineering, 0210 nano-technology, Tablets
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4
المؤلفون: Mathiazhagan Annadurai, Ramakanth Sarabu, Salil D. Desai, John F. Kadow, Nicholas A. Meanwell, Sarmistha Sinha, Susan Jenkins, Murali Subramanian, Rambabu Arla, Murugaiah A. M. Subbaiah, Thangeswaran Ramar, Shweta Padmanabhan, Priyadeep Bhutani, Mark Krystal, Chunfu Wang, Sandhya Mandlekar, Lakshumanan Subramani, Srikanth Sridhar
المصدر: Journal of medicinal chemistry. 61(9)
مصطلحات موضوعية: Drug, medicine.medical_treatment, media_common.quotation_subject, Atazanavir Sulfate, Administration, Oral, Biological Availability, Pharmacology, 030226 pharmacology & pharmacy, Rats, Sprague-Dawley, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, HIV-1 protease, In vivo, Drug Discovery, medicine, Animals, Prodrugs, Tissue Distribution, media_common, Protease, biology, Symporters, Chemistry, HIV Protease Inhibitors, Prodrug, Fatty Acid Transport Proteins, Atazanavir, Bioavailability, Rats, 030220 oncology & carcinogenesis, biology.protein, Molecular Medicine, medicine.drug
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5
المؤلفون: Salil D. Desai, Lee E. Kirsch
المصدر: International Journal of Chemical Kinetics. 47:471-488
مصطلحات موضوعية: Steric effects, chemistry.chemical_classification, Base (chemistry), Organic Chemistry, Inorganic chemistry, Substituent, Biochemistry, Inorganic Chemistry, chemistry.chemical_compound, Acid catalysis, Hydrolysis, chemistry, Sodium hydroxide, Hydroxide, Physical and Theoretical Chemistry, Alkaline hydrolysis
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6
المؤلفون: Zhixin Zong, Lee E. Kirsch, Salil D. Desai, Aditya Mohan Kaushal, Eric J. Munson, Raj Suryanarayanan, Dewey H. Barich, Kassibla Elodie Dempah
المصدر: AAPS PharmSciTech. 14:19-28
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Cyclohexanecarboxylic Acids, Analytical chemistry, Pharmaceutical Science, Aquatic Science, Spectrophotometry, Drug Discovery, medicine, Dehydration, Amines, Cellulose, Chromatography, High Pressure Liquid, gamma-Aminobutyric Acid, Ecology, Evolution, Behavior and Systematics, Polymorphism, Genetic, Ecology, medicine.diagnostic_test, Chemistry, Recrystallization (metallurgy), General Medicine, Nuclear magnetic resonance spectroscopy, medicine.disease, Polymorphism (materials science), Solid-state nuclear magnetic resonance, Spray drying, Spectrophotometry, Ultraviolet, Gabapentin, Agronomy and Crop Science, Powder Diffraction, Powder diffraction, Research Article
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7
المؤلفون: Lee E. Kirsch, Hong Shian Huang, Raj Suryanarayanan, Eric J. Munson, Salil D. Desai, Dewey H. Barich, Zhixin Zong, Aditya Mohan Kaushal
المصدر: AAPS PharmSciTech. 12
مصطلحات موضوعية: Cyclohexanecarboxylic Acids, Surface Properties, Analytical chemistry, Pharmaceutical Science, Aquatic Science, complex mixtures, Annealing (glass), Hydrolysis, chemistry.chemical_compound, Drug Stability, X-Ray Diffraction, Spectroscopy, Fourier Transform Infrared, Drug Discovery, Technology, Pharmaceutical, Spiro Compounds, Relative humidity, Amines, Particle Size, gamma-Aminobutyric Acid, Ecology, Evolution, Behavior and Systematics, Aza Compounds, Chromatography, Reverse-Phase, Ecology, Moisture, Chemistry, digestive, oral, and skin physiology, technology, industry, and agriculture, Water, food and beverages, Humidity, General Medicine, respiratory tract diseases, Lactam, Degradation (geology), Anticonvulsants, Particle size, Gabapentin, Powders, Agronomy and Crop Science, Research Article, Nuclear chemistry
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8
المؤلفون: Hong Shian Huang, Eric J. Munson, Lee E. Kirsch, Aditya Mohan Kaushal, Zhixin Zong, Salil D. Desai, Raj Suryanarayanan, Dewey H. Barich
المصدر: AAPS PharmSciTech. 12:1465-1465
مصطلحات موضوعية: Ecology, Pharmacology toxicology, Solid-state, Pharmaceutical Science, General Medicine, Aquatic Science, Quality by Design, Food and drug administration, Engineering management, Pharmaceutical technology, Drug Discovery, Business, Erratum, Agronomy and Crop Science, Ecology, Evolution, Behavior and Systematics