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1Academic Journal
المؤلفون: Albertini, C, Salerno, A, Atzenti, S, Uliassi, E, Massenzio, F, Maruca, A, Rocca, R, Mecava, M, Silva, FSG, Mena, D, Valente, P, Duarte, AI, Chavarria, D, Bissaro, M, Moro, S, Federico, S, Spalluto, G, Soukup, O, Borges, F, Alcaro, S, Monti, B, Oliveira, PJ, Menendez, JC, Bolognesi, ML
المساهمون: Albertini, C, Salerno, A, Atzenti, S, Uliassi, E, Massenzio, F, Maruca, A, Rocca, R, Mecava, M, Silva, FSG, Mena, D, Valente, P, Duarte, AI, Chavarria, D, Bissaro, M, Moro, S, Federico, S, Spalluto, G, Soukup, O, Borges, F, Alcaro, S, Monti, B, Oliveira, PJ, Menendez, JC, Bolognesi, ML
مصطلحات موضوعية: Polypharmacology, MTDL, ALS, benzothiazole, MAO, riluzole, rasagiline
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/35868251; info:eu-repo/semantics/altIdentifier/wos/WOS:000838605400001; volume:13; issue:15; firstpage:2252; lastpage:2260; numberofpages:9; journal:ACS CHEMICAL NEUROSCIENCE; https://hdl.handle.net/11585/894854; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85135596285
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2Academic Journal
المؤلفون: Spinaci A., Lambertucci C., Cui C., Buccioni M., Marucci G., Cescon E., Federico S., Spalluto G., Dal Ben D., Volpini R.
المساهمون: Spinaci, A., Lambertucci, C., Cui, C., Buccioni, M., Marucci, G., Cescon, E., Federico, S., Spalluto, G., Dal Ben, D., Volpini, R.
مصطلحات موضوعية: CK1 delta inhibitors, Adenine derivatives, Casein kinase 1 delta, Synthesis of purine derivatives, Molecular modeling, Medicinal chemistry
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:001175151400001; volume:33; issue:4; firstpage:611; lastpage:619; numberofpages:9; journal:MEDICINAL CHEMISTRY RESEARCH; https://hdl.handle.net/11581/487511
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3Academic Journal
المؤلفون: Calenda S., Catarzi D., Varano F., Vigiani E., Volpini R., Lambertucci C., Spinaci A., Trevisan L., Grieco I., Federico S., Spalluto G., Novello G., Salmaso V., Moro S., Colotta V.
المساهمون: Calenda, S., Catarzi, D., Varano, F., Vigiani, E., Volpini, R., Lambertucci, C., Spinaci, A., Trevisan, L., Grieco, I., Federico, S., Spalluto, G., Novello, G., Salmaso, V., Moro, S., Colotta, V.
مصطلحات موضوعية: benzimidazole derivatives, CK1δ inhibitors, molecular modeling
Relation: info:eu-repo/semantics/altIdentifier/pmid/38675428; info:eu-repo/semantics/altIdentifier/wos/WOS:001210237700001; volume:17; issue:4; journal:PHARMACEUTICALS; https://hdl.handle.net/11581/487512
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4Academic Journal
المؤلفون: Grieco I., Bissaro M., Tiz D. B., Perez D. I., Perez C., Martinez A., Redenti S., Mariotto E., Bortolozzi R., Viola G., Cozza G., Spalluto G., Moro S., Federico S.
المساهمون: Grieco, I., Bissaro, M., Tiz, D. B., Perez, D. I., Perez, C., Martinez, A., Redenti, S., Mariotto, E., Bortolozzi, R., Viola, G., Cozza, G., Spalluto, G., Moro, S., Federico, S.
مصطلحات موضوعية: BBB-PAMPA assay, Kinase molecular modeling, Neurodegenerative disease, Protein kinase CK1 delta, [1,2,4]triazolo[1,5-a][1,3,5]triazine, [1,2,4]triazolo[1,5-c]pyrimidine, Binding Site, Blood-Brain Barrier, Casein Kinase Idelta, Cell Line, Cell Survival, Drug Design, Human, Kinetic, Molecular Docking Simulation, Protein Kinase Inhibitor, Pyrimidine, Static Electricity, Structure-Activity Relationship, Thermodynamic, Triazine, Triazoles
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/33721670; info:eu-repo/semantics/altIdentifier/wos/WOS:000637742700030; volume:216; firstpage:-; lastpage:-; numberofpages:27; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/11368/2991414; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85102293647; https://www.sciencedirect.com/science/article/pii/S022352342100180X?via=ihub
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5Book
المؤلفون: Prencipe F., Da Ros T., Cescon E., Grieco I., Persico M., Spalluto G., Federico S.
المساهمون: Vittoria Colotta, Claudiu T. Supuran, Prencipe, F., Da Ros, T., Cescon, E., Grieco, I., Persico, M., Spalluto, G., Federico, S.
مصطلحات موضوعية: Adenosine receptor, Binding, Carbon nanotube, Dendrimer, Fluorescent ligand, GPCR, Preladenant, Probe, Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine, Radioligand, Radiotracer, SCH442416, SCH58261
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/isbn/978-3-031-39724-0; info:eu-repo/semantics/altIdentifier/isbn/978-3-031-39725-7; ispartofbook:Purinergic Receptors and their Modulators; volume:41; firstpage:47; lastpage:87; numberofpages:41; serie:TOPICS IN MEDICINAL CHEMISTRY; alleditors:Vittoria Colotta, Claudiu T. Supuran; https://hdl.handle.net/11368/3067479; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85175088933
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6Academic Journal
المؤلفون: Cescon E., Bolcato G., Federico Stephanie, Bissaro M., Valentini A., Ferlin M. G., Spalluto G., Sturlese M., Moro S.
المساهمون: Cescon, E., Bolcato, G., Federico, Stephanie, Bissaro, M., Valentini, A., Ferlin, M. G., Spalluto, G., Sturlese, M., Moro, S.
مصطلحات موضوعية: Casein kinase 1 δ, consensus docking, scaffold repurposing, virtual screening
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/32550997; info:eu-repo/semantics/altIdentifier/wos/WOS:000541747800018; volume:11; issue:6; firstpage:1168; lastpage:1174; numberofpages:7; journal:ACS MEDICINAL CHEMISTRY LETTERS; http://hdl.handle.net/11577/3349043; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85087087230
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7Academic Journal
المؤلفون: Federico S., Lassiani L., Spalluto G.
المساهمون: Federico, S., Lassiani, L., Spalluto, G.
مصطلحات موضوعية: Adenosine receptor, Covalent ligand, Fluorescent ligand, GPCR probe, Radioligand, Radiotracers
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/31726680; info:eu-repo/semantics/altIdentifier/wos/WOS:000505739800024; volume:12; issue:4; firstpage:168; lastpage:168; numberofpages:1; journal:PHARMACEUTICALS; http://hdl.handle.net/11368/2955003; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85075088071; https://www.mdpi.com/1424-8247/12/4/168
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8Academic Journal
المؤلفون: Tan A., Babak M. V., Venkatesan G., Lim C., Klotz K. -N., Herr D. R., Cheong S. L., Federico S., Spalluto G., Ong W. -Y., Chen Y. Z., Loo J. S. E., Pastori G.
المساهمون: Tan, A., Babak, M. V., Venkatesan, G., Lim, C., Klotz, K. -N., Herr, D. R., Cheong, S. L., Federico, S., Spalluto, G., Ong, W. -Y., Chen, Y. Z., Loo, J. S. E., Pastori, G.
مصطلحات موضوعية: Gastrointestinal cancer, HA, AR, Indolylpyrimidylpiperazine, Partial agonists
Time: 3
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/31614517; info:eu-repo/semantics/altIdentifier/wos/WOS:000496249500030; volume:24; issue:20; firstpage:1; lastpage:16; numberofpages:16; journal:MOLECULES; http://hdl.handle.net/11368/2954606; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85073481666; https://www.mdpi.com/1420-3049/24/20/3661
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9Academic Journal
المؤلفون: Federico S., Persico M., Trevisan L., Biasinutto C., Bolcato G., Salmaso V., Da Ros T., Gianferrara T., Prencipe F., Kachler S., Klotz K. -N., Pacor S., Moro S., Spalluto G.
المساهمون: Federico, S., Persico, M., Trevisan, L., Biasinutto, C., Bolcato, G., Salmaso, V., Da Ros, T., Gianferrara, T., Prencipe, F., Kachler, S., Klotz, K. -N., Pacor, S., Moro, S., Spalluto, G.
مصطلحات موضوعية: A3, adenosine receptor, antagonist, cancer, GPCR, [1,2,4]triazolo[1,5-c]pyrimidine
وصف الملف: ELETTRONICO
Relation: info:eu-repo/semantics/altIdentifier/pmid/37675643; info:eu-repo/semantics/altIdentifier/wos/WOS:001071135000001; volume:18/2023; issue:21; firstpage:"-"; lastpage:"-"; numberofpages:15; journal:CHEMMEDCHEM; https://hdl.handle.net/11368/3067475; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85171738153
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10Academic Journal
المؤلفون: Tan, A., Babak, M.V., Venkatesan, G., Lim, C., Klotz, K.-N., Herr, D.R., Cheong, S.L., Federico, S., Spalluto, G., Ong, W.-Y., Chen, Y.Z., Loo, J.S.E., Pastori, G.
المساهمون: PHARMACY, PHARMACOLOGY, ANATOMY
المصدر: Scopus OA2019
مصطلحات موضوعية: Gastrointestinal cancer, HA3AR, Indolylpyrimidylpiperazines, Partial agonists
Relation: Tan, A., Babak, M.V., Venkatesan, G., Lim, C., Klotz, K.-N., Herr, D.R., Cheong, S.L., Federico, S., Spalluto, G., Ong, W.-Y., Chen, Y.Z., Loo, J.S.E., Pastori, G. (2019). Design, synthesis and evaluation of new indolylpyrimidylpiperazines for gastrointestinal cancer therapy. Molecules 24 (20) : 3661. ScholarBank@NUS Repository. https://doi.org/10.3390/molecules24203661; https://scholarbank.nus.edu.sg/handle/10635/211662
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11Academic Journal
المؤلفون: Shao, Y.M., Ma, X., Paira, P., Tan, A., Herr, D.R., Lim, K.L., Ng, C.H., Venkatesan, G., Klotz, K.N., Federico, S., Spalluto, G., Cheong, S.L., Chen, Y.Z., Pastorin, G.
المساهمون: Blum, D.
مصطلحات موضوعية: CHO Cells, Animals, Genetically Modified, Humans, Cricetulus, Drosophila, Parkinsonian Disorders, Parkinson Disease, Piperazines, Pyrimidines, Receptors, Dopamine D2, Receptor, Adenosine A2A, Dopamine Agonists, Antiparkinson Agents, Radioligand Assay, Drug Evaluation, Preclinical, Drug Discovery, Adenosine A2 Receptor Antagonists, Support Vector Machine, Adenylyl Cyclase Inhibitors
Relation: PLoS One, 2018; 13(1):e0188212-e0188212; http://hdl.handle.net/2440/124495; Tan, A. [0000-0002-8935-0773]
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12Academic Journal
المؤلفون: Vimercati L., Cavone D., Delfino M. C., De Maria L., Caputi A., Sponselli S., Corrado V., Bruno V., Spalluto G., Eranio G., Ferri G. M.
المساهمون: Vimercati, L., Cavone, D., Delfino, M. C., De Maria, L., Caputi, A., Sponselli, S., Corrado, V., Bruno, V., Spalluto, G., Eranio, G., Ferri, G. M.
مصطلحات موضوعية: Earthquake, Exposure detector, Lung cancer estimation software, Radon, Residential building
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:000715407200001; volume:12; issue:10; firstpage:1342; journal:ATMOSPHERE; http://hdl.handle.net/11586/379763; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85117614869
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13Academic Journal
المؤلفون: Federico S., Margiotta E., Moro S., Kachler S., Klotz K. -N., Spalluto G.
المساهمون: Federico, S., Margiotta, E., Moro, S., Kachler, S., Klotz, K. -N., Spalluto, G.
مصطلحات موضوعية: pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine, adenosine receptor, adenosine receptor antagonist, A3AR, GPCR probe
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/34046614; info:eu-repo/semantics/altIdentifier/wos/WOS:000625239200009; volume:12; issue:2; firstpage:254; lastpage:262; numberofpages:9; journal:RSC MEDICINAL CHEMISTRY; http://hdl.handle.net/11368/2991410; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85102069105; https://pubs.rsc.org/en/content/articlelanding/2021/md/d0md00380h#!divAbstract
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14Academic Journal
المؤلفون: Pineux F., Federico S., Klotz K. -N., Kachler S., Michiels C., Sturlese M., Prato M., Spalluto G., Moro S., Bonifazi D.
المساهمون: Pineux, F., Federico, S., Klotz, K. -N., Kachler, S., Michiels, C., Sturlese, M., Prato, M., Spalluto, G., Moro, S., Bonifazi, D.
مصطلحات موضوعية: A3, adenosine receptor, carbon nanotube, docking, G protein-coupled receptor, magnetic cell sorting, theranostics
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/32706529; info:eu-repo/semantics/altIdentifier/wos/WOS:000566814900001; volume:15; issue:20; firstpage:1909; lastpage:1920; numberofpages:12; journal:CHEMMEDCHEM; http://hdl.handle.net/11368/2991406; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85090443351
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15Academic Journal
المؤلفون: Federico S., Margiotta E., Moro S., Kozma E., Gao Z. -G., Jacobson K. A., Spalluto G.
المساهمون: Federico, S., Margiotta, E., Moro, S., Kozma, E., Gao, Z. -G., Jacobson, K. A., Spalluto, G.
مصطلحات موضوعية: Adenosine receptor, Fluorescent ligand, G protein-coupled receptor, Molecular modeling, Molecular probes
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/31787357; info:eu-repo/semantics/altIdentifier/wos/WOS:000509616800031; volume:186; firstpage:1; lastpage:16; numberofpages:16; journal:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY; http://hdl.handle.net/11368/2955016; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85075902118; https://www.sciencedirect.com/science/article/pii/S0223523419310384?via=ihub
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16Academic Journal
المؤلفون: Cacciari B., Crepaldi P., Cheng C. Y., Bossi E., Spalluto G., Federico S., Jacobson K. A., Cattaneo M.
المساهمون: Cacciari, B., Crepaldi, P., Cheng, C. Y., Bossi, E., Spalluto, G., Federico, S., Jacobson, K. A., Cattaneo, M.
مصطلحات موضوعية: 4-amino-2-thiopyrimidine-5-carboxylic acid, 6-amino-2-thio-3H-pyrimin-4-one, clopidogrel, platelet aggregation inhibition, Substituted 4-amino-2-thiopyrimidine, synthesis, Platelet Aggregation, Platelet Aggregation Inhibitor, Pyrimidine, Structure-Activity Relationship
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/30734681; info:eu-repo/semantics/altIdentifier/wos/WOS:000497706100004; volume:15; issue:8; firstpage:863; lastpage:872; numberofpages:10; journal:MEDICINAL CHEMISTRY; http://hdl.handle.net/11368/2955011; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85063860151; http://www.eurekaselect.com/169801/article
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17Academic Journal
المؤلفون: Federico S., Spalluto G.
المساهمون: Federico, S., Spalluto, G.
مصطلحات موضوعية: adenosine receptor, dendrimer, fluorescent ligand, functionalized ligand, GPCR, irreversible ligand, multitarget ligand, multivalent ligand, nanoparticle, theranostic
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/pmid/31317789; info:eu-repo/semantics/altIdentifier/wos/WOS:000492205700002; volume:11; issue:14; firstpage:1673; lastpage:1677; numberofpages:5; journal:FUTURE MEDICINAL CHEMISTRY; http://hdl.handle.net/11368/2955005; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85071995351
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18Academic Journal
المؤلفون: FEDERICO, SALVATORE, Margiotta E., Paoletta S., Kachler S., Klotz K. -N., Jacobson K. A., Pastorin G., Moro S., Spalluto G.
المساهمون: Federico, Salvatore, Margiotta, E., Paoletta, S., Kachler, S., Klotz, K. -N., Jacobson, K. A., Pastorin, G., Moro, S., Spalluto, G.
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:000475806000020; volume:10; issue:7; firstpage:1094; lastpage:1108; numberofpages:15; journal:MEDCHEMCOMM; http://hdl.handle.net/11577/3308009; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85069459931; http://pubs.rsc.org/en/journals/journal/md
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19Academic Journal
المؤلفون: Redenti S., Marcovich I., DE VITA, TIZIANA, Perez C., De Zorzi R., Demitri N., Perez D. I., BOTTEGONI, GIOVANNI, Bisignano P., Bissaro M., Moro S., Martinez A., Storici P., Spalluto G., CAVALLI, ALESSANDRO, Federico S.
المساهمون: Redenti, S., Marcovich, I., DE VITA, Tiziana, Perez, C., De Zorzi, R., Demitri, N., Perez, D. I., Bottegoni, Giovanni, Bisignano, P., Bissaro, M., Moro, S., Martinez, A., Storici, P., Spalluto, G., Cavalli, Alessandro, Federico, S.
مصطلحات موضوعية: casein kinase 1δ, glycogen synthase kinase 3β, neuroinflammation, Parkinson's disease, thia-Michael reaction
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/wos/WOS:000458432600003; volume:14; issue:3; firstpage:310; lastpage:314; numberofpages:5; journal:CHEMMEDCHEM; http://hdl.handle.net/11577/3308003; info:eu-repo/semantics/altIdentifier/scopus/2-s2.0-85060180817; http://onlinelibrary.wiley.com/journal/10.1002/(ISSN)1860-7187
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20Book
المؤلفون: Dell’Osso G. R., Pierucci A., Spalluto G.
المساهمون: Giuseppe Alaimo, Angelo Ciribini, Bruno Daniotti, Guido Dell’Osso, Maria Antonietta Esposito, Dell’Osso, G. R., Pierucci, A., Spalluto, G.
وصف الملف: STAMPA
Relation: info:eu-repo/semantics/altIdentifier/isbn/978-88-387-6164-5; ispartofbook:The missing brick: towards a 21st Century built environment industry = Il mattone mancante: verso l'industria dell'ambiente costruito del 21mo secolo; firstpage:332; lastpage:351; numberofpages:20; serie:POLITECNICA; alleditors:Giuseppe Alaimo, Angelo Ciribini, Bruno Daniotti, Guido Dell’Osso, Maria Antonietta Esposito; http://hdl.handle.net/11589/122772
الاتاحة: http://hdl.handle.net/11589/122772