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1Academic Journal
المؤلفون: ANDREW J. POPE, CATHERINE S. V. HOUGE-FRYDRYCH, DAVID J. MCNAIR, JOHN M. BERGE, LUCY MENSAH, NIGEL J. P. BROOM, PETER J. O'HANLON, RICHARD L. JARVEST, STEPHEN RITTENHOUSE
المصدر: The Journal of Antibiotics. 2000, 53(11):1282
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2
المؤلفون: Renae M. Crosby, Xianfeng Li, Yang Liu, Jacob J. Plattner, Joel P. Cooper, Yong-Kang Zhang, Stephen J. Baker, Richard L. Jarvest, Wieslaw M. Kazmierski, Lois L. Wright, Jing-Jing Ji, Suoming Zhang, Wei Bu, Gary K. Smith, Maosheng Duan, Liang Liu, Amy Wang, Charles Z. Ding, Yasheen Zhou, Robert Hamatake, Matthew David Tallant, Katrina L. Creech
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:7351-7356
مصطلحات موضوعية: Carbamate, Serine Proteinase Inhibitors, medicine.medical_treatment, Clinical Biochemistry, Mutant, Pharmaceutical Science, Hepacivirus, Microbial Sensitivity Tests, Viral Nonstructural Proteins, Antiviral Agents, Guanidines, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Amide, Drug Resistance, Viral, Drug Discovery, medicine, Animals, Urea, Structure–activity relationship, Potency, Protease inhibitor (pharmacology), Replicon, Molecular Biology, Oxamic Acid, Dose-Response Relationship, Drug, Molecular Structure, biology, Chemistry, Organic Chemistry, Amides, Enzyme assay, Rats, biology.protein, Molecular Medicine, Carbamates
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3
المؤلفون: Luz H. Carballo, Yasheen Zhou, Máire A. Convery, Julia A. Hubbard, Zhi-Jie Ni, Yang Liu, Richard Martin Grimes, Pamela Nassau, Qun Li, Jon Wright, Dazhong Fan, Lois L. Wright, Wieslaw M. Kazmierski, Pia Thommes, Xuelei Qian, Richard L. Jarvest, Wuxin Zou, Charles Z. Ding, Yong-Kang Zhang, Lewis E. Pennicott, Tadeusz Skarzynski, Katrina L. Creech, Renae M. Crosby, Jacob J. Plattner, Martin John Slater, Xianfeng Li, Gary K. Smith, William McDowell, Suoming Zhang, Stephen J. Baker, Liang Liao
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5695-5700
مصطلحات موضوعية: Boron Compounds, inorganic chemicals, Macrocyclic Compounds, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Hepacivirus, Viral Nonstructural Proteins, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Catalytic Domain, Drug Discovery, medicine, Structure–activity relationship, Protease Inhibitors, Replicon, Molecular Biology, NS3, Binding Sites, Protease, biology, Chemistry, Organic Chemistry, Active site, Boronic Acids, Protease inhibitor (biology), Protein Structure, Tertiary, Enzyme inhibitor, biology.protein, Lactam, Molecular Medicine, medicine.drug
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4
المؤلفون: John Broskey, Sulejman Alihodžić, David J. Holmes, Samra Kapić, Vesna Eraković Haber, Eric Hunt, Roberto Antolović, Hana Čipčić Paljetak, Richard L. Jarvest
المصدر: Bioorganic & Medicinal Chemistry. 18:6569-6577
مصطلحات موضوعية: Stereochemistry, Carboxylic acid, Clinical Biochemistry, Pharmaceutical Science, Ether, Microbial Sensitivity Tests, Azithromycin, Quinolones, tethered macrolides, 6-(x-carboxy)-alkyl-N(1)-ethyl-3- carboxylquinolones, aAntimicrobial activity, structure–activity relationship, Biochemistry, Chemical synthesis, Acylation, Structure-Activity Relationship, chemistry.chemical_compound, Clarithromycin, Drug Discovery, Humans, Molecular Biology, Antibacterial agent, chemistry.chemical_classification, Bicyclic molecule, Organic Chemistry, Antimicrobial, Anti-Bacterial Agents, chemistry, Molecular Medicine, Macrolides, Linker
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5
المؤلفون: Zhi-Jie Ni, Qun Li, Martin John Slater, Wuxin Zou, Linos Lazarides, Yang Liu, Lois L. Wright, Paul Rowland, Liang Liao, Charles Z. Ding, Tadeusz Skarzynski, Jacob J. Plattner, Jackie E. Mordaunt, Don O. Somers, Xianfeng Li, Colin M. Edge, Yong-Kang Zhang, Gemma Victoria White, Malcolm Ellis, Jon Wright, Stephen J. Baker, Dazhong Fan, Wieslaw M. Kazmierski, Gary K. Smith, Pia Thommes, Lewis E. Pennicott, Julia A. Hubbard, Richard L. Jarvest, Bill McDowell, Yasheen Zhou, Xuelei Qian, Pamela Nassau, Richard Martin Grimes
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:3550-3556
مصطلحات موضوعية: Stereochemistry, viruses, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Peptide, Hepacivirus, Viral Nonstructural Proteins, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Catalytic Domain, Drug Discovery, Serine, medicine, Molecular Biology, chemistry.chemical_classification, Serine protease, NS3, Protease, Molecular Structure, biology, Organic Chemistry, virus diseases, Active site, Boronic Acids, digestive system diseases, Protease inhibitor (biology), chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, medicine.drug
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6
المؤلفون: Sula Anne Armstrong, Pamela Brown, Darren Jason Mitchell, Stephen Rittenhouse, Dieter Hamprecht, Andrew Keith Forrest, Royston C. B. Copley, Peter J. O'Hanlon, John S. Elder, Richard L. Jarvest, Murray J. B. Brown, John M. Berge, David R. Witty
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:3937-3941
مصطلحات موضوعية: Models, Molecular, Methionine—tRNA ligase, medicine.drug_class, Stereochemistry, Staphylococcus, Clinical Biochemistry, Pharmaceutical Science, Context (language use), Methionine-tRNA Ligase, Microbial Sensitivity Tests, Quinolones, Biochemistry, Structure-Activity Relationship, Drug Discovery, Enterococcus faecalis, medicine, Enzyme Inhibitors, Molecular Biology, Antibacterial agent, Molecular Structure, Bicyclic molecule, Chemistry, Organic Chemistry, Biological activity, Quinolone, Anti-Bacterial Agents, Kinetics, Molecular Medicine, Pharmacophore, Antibacterial activity
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7
المؤلفون: David Leese, Alan C. Spivey, Fujiang Zhu, Stephen Davey, Richard L. Jarvest
المصدر: Tetrahedron. 60:4513-4525
مصطلحات موضوعية: Atropisomer, Organic Chemistry, Absolute configuration, Enantioselective synthesis, Substituent, General Medicine, Combinatorial chemistry, Biochemistry, Catalysis, Kinetic resolution, Acylation, chemistry.chemical_compound, Nucleophile, chemistry, Drug Discovery, Organic chemistry, Selectivity, Chirality (chemistry)
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8
المؤلفون: Michael J. Stanhope, Karen A. Ingraham, James R. Brown, David J. Holmes, Richard L. Jarvest, Peter J. O'Hanlon, Stephen Rittenhouse, Daniel R. Gentry
المصدر: Antimicrobial Agents and Chemotherapy. 47:1784-1789
مصطلحات موضوعية: DNA, Bacterial, Molecular Sequence Data, Methionine-tRNA Ligase, Microbial Sensitivity Tests, medicine.disease_cause, Polymerase Chain Reaction, Isozyme, Microbiology, Mechanisms of Resistance, Drug Resistance, Bacterial, Streptococcus pneumoniae, medicine, Pharmacology (medical), Amino Acid Sequence, Enzyme Inhibitors, Gene, Antibacterial agent, Pharmacology, Genetics, chemistry.chemical_classification, Base Sequence, biology, biology.organism_classification, Isoenzymes, Infectious Diseases, Enzyme, chemistry, Mutagenesis, Staphylococcus aureus, Horizontal gene transfer, Sequence Alignment, Bacteria
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9
المؤلفون: David R. Witty, Dieter Hamprecht, Ashley E. Fenwick, Paul S. Carter, Richard L. Jarvest, Murray J. B. Brown, Peter J. O'Hanlon, Martin Hibbs, Andrew J. Pope, Lucy Mensah, Christine M. Richardson, Peter Henry Milner, Andrew West, Andrew P. Fosberry
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:3171-3174
مصطلحات موضوعية: Staphylococcus aureus, Indoles, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Tryptophan-tRNA Ligase, Microbial Sensitivity Tests, Tryptophan—tRNA ligase, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Structure–activity relationship, Enzyme Inhibitors, Molecular Biology, Antibacterial agent, chemistry.chemical_classification, Natural product, Bacteria, Hydrolysis, Organic Chemistry, Stereoisomerism, Biological activity, Antimicrobial, Anti-Bacterial Agents, Enzyme, chemistry, Molecular Medicine, Indicators and Reagents, Antibacterial activity
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10
المؤلفون: Andrew Keith Forrest, Murray J. B. Brown, Martin Hibbs, Valerie Berry, Robert J. Sheppard, Deborah Dee Jaworski, John S. Elder, Courtney Slater-Radosti, Peter J. O'Hanlon, Helen F. Boyd, John M. Berge, Richard L. Jarvest, Andrew J. Pope, Angela Worby, Andrew P. Fosberry, Daniel R. Gentry, Stephen Rittenhouse
المصدر: Journal of Medicinal Chemistry. 45:1959-1962
مصطلحات موضوعية: Staphylococcus aureus, Micrococcaceae, medicine.drug_class, Staphylococcus, Antibiotics, Methionine-tRNA Ligase, Quinolones, medicine.disease_cause, Microbiology, Rats, Sprague-Dawley, Structure-Activity Relationship, Staphylococcus epidermidis, Drug Resistance, Bacterial, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Antibacterial agent, biology, Chemistry, Biological activity, biology.organism_classification, Abscess, Anti-Bacterial Agents, Rats, Biochemistry, Molecular Medicine, Antibacterial activity, Enterococcus, Bacteria
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11
المصدر: Macrocycles in Drug Discovery ISBN: 9781849737012
مصطلحات موضوعية: Simeprevir, chemistry.chemical_classification, Protease, medicine.medical_treatment, Hepatitis C virus, virus diseases, Biology, medicine.disease_cause, Telaprevir, chemistry.chemical_compound, Enzyme, Biochemistry, chemistry, RNA polymerase, Boceprevir, medicine, NS5B, medicine.drug
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12Synthetic analogues of SB-219383. Novel C-glycosyl peptides as inhibitors of tyrosyl tRNA synthetase
المؤلفون: Pamela Brown, Peter J. O'Hanlon, Richard L. Jarvest, Lucy Mensah, Andrew J. Pope, Drake S. Eggleston, R. Curtis Haltiwanger
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:711-714
مصطلحات موضوعية: Models, Molecular, Staphylococcus aureus, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Peptide, environment and public health, Biochemistry, chemistry.chemical_compound, Hydroxylamine, Bacterial Proteins, Tyrosine-tRNA Ligase, parasitic diseases, Drug Discovery, Moiety, Glycosyl, Enzyme Inhibitors, Furans, Molecular Biology, Pyrans, Antibacterial agent, chemistry.chemical_classification, Dipeptide, Molecular Structure, Organic Chemistry, Bridged Bicyclo Compounds, Heterocyclic, enzymes and coenzymes (carbohydrates), Enzyme, Tyrosine—tRNA ligase, chemistry, Molecular Medicine, hormones, hormone substitutes, and hormone antagonists
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13
المؤلفون: Ivan Leo Pinto, Richard L. Jarvest, Halina T. Serafinowska
المصدر: Tetrahedron Letters. 41:1597-1600
مصطلحات موضوعية: chemistry.chemical_compound, Four component, Chemistry, Organic Chemistry, Drug Discovery, Polymer chemistry, Alkoxy group, Thiophene, Condensation reaction, Biochemistry
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14
المؤلفون: Christine E. Dabrowski, Richard L. Jarvest, A V Fernandez, Patrick Lavery, Ivan Leo Pinto, L J Jennings, David G. Tew, S M Ashman
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:443-448
مصطلحات موضوعية: Proteases, medicine.drug_class, viruses, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Oxazines, medicine.disease_cause, Antiviral Agents, Biochemistry, Chemical synthesis, Virus, Cell Line, Drug Discovery, medicine, Protease Inhibitors, Molecular Biology, Herpesviridae, chemistry.chemical_classification, Protease, Chemistry, Organic Chemistry, Varicella zoster virus, In vitro, Molecular Medicine
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15
المؤلفون: Michele M Gorczyca, David G. Tew, Andrew West, Patrick Lavery, Christine E. Dabrowski, Edmund J. Sternberg, Richard L. Jarvest, Ivan Leo Pinto, L.John Jennings, Ashley E. Fenwick, B. Clarke
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:449-452
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, Alkylation, Cell Survival, Stereochemistry, Acylation, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Spectrometry, Mass, Fast Atom Bombardment, Biochemistry, Oxazines, Drug Discovery, medicine, Moiety, Molecular Biology, Protease, biology, Chemistry, Serine Endopeptidases, Organic Chemistry, Enzyme inhibitor, Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization, Michael reaction, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins), Cysteine
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16
المؤلفون: J.N. Champness, Richard L. Jarvest, William C. Summers, Piet Herdewijn, Erik De Clercq, Mark R. Sanderson, Rob Visse, Matthew S. Bennett, Frank Wien, Tomasz Ostrowski
المصدر: Proteins: Structure, Function, and Genetics. 32:350-361
مصطلحات موضوعية: biology, Nucleoside analogue, Kinase, Active site, Biochemistry, Enzyme structure, chemistry.chemical_compound, chemistry, Structural Biology, Thymidine kinase, Penciclovir, biology.protein, medicine, Binding site, Thymidine, Molecular Biology, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3fc7c796f5cdf6613a7ec3e51a0a0d6c
https://doi.org/10.1002/(sici)1097-0134(19980815)32:3<350::aid-prot10>3.0.co;2-8 -
17
المؤلفون: Richard L. Jarvest, L.John Jennings, Susan C. Connor, Halina T. Serafinowska, Joselina G. Gorniak, Andrew West
المصدر: Bioorganic & Medicinal Chemistry Letters. 7:1733-1738
مصطلحات موضوعية: chemistry.chemical_classification, Proteases, Protease, biology, Chemistry, medicine.medical_treatment, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, biology.organism_classification, Biochemistry, In vitro, Virus, Enzyme, Betaherpesvirinae, Enzyme inhibitor, Drug Discovery, medicine, biology.protein, Molecular Medicine, Protease inhibitor (pharmacology), Molecular Biology
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18
المؤلفون: Anthony G. DiLella, Richard L. Jarvest, Daniel J. O'Shannessy, Andrew West, Christine Debouck, Arunbai Patel, Ivan Leo Pinto, Kevin O'Donnell, Joselina G. Gorniak
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:2467-2472
مصطلحات موضوعية: Proteases, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Mechanism based, Biochemistry, Combinatorial chemistry, Serine, Covalent bond, Drug Discovery, Molecular Medicine, Molecular Biology
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19
المؤلفون: Joselina G. Gorniak, Martin J. Parratt, Richard L. Jarvest, James E. Strickler, Christine Debouck, Halina T. Serafinowska, L.John Jennings
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:2463-2466
مصطلحات موضوعية: Protease, Stereochemistry, Benzoxazinones, Chemistry, medicine.medical_treatment, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Mechanism based, HSL and HSV, Mass spectrometry, Biochemistry, Drug Discovery, medicine, Molecular Medicine, Molecular Biology
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20Academic Journal
المؤلفون: Xianfeng Li, Yong-Kang Zhang, Yang Liu, Charles Z Ding, Yasheen Zhou, Qun Li, Jacob J Plattner, Stephen J Baker, Suoming Zhang, Wieslaw M Kazmierski, Lois L Wright, Gary K Smith, Richard M Grimes, Renae M Crosby, Katrina L Creech, Luz H Carballo, Martin J Slater, Richard L Jarvest, Pia Thommes, Julia A Hubbard, Maire A Convery, Pamela M Nassau, William McDowell, Tadeusz J Skarzynski, Xuelei Qian, Dazhong Fan, Liang Liao, Zhi-Jie Ni, Lewis E Pennicott, Wuxin Zou, Jon Wright
مصطلحات موضوعية: Uncategorised value