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1Academic Journal
المؤلفون: Vásquez, Ivana Raquel, Riafrecha, Leonardo Ezequiel, Martínez Heredia, Leandro, Echeverría, Gustavo Alberto, Piro, Oscar Enrique, Lavecchia, Martín José, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: Química, Imines, Cancer, Enzyme inhibitor
وصف الملف: application/pdf
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2Academic Journal
المؤلفون: Riafrecha, Leonardo Ezequiel, Le Pors, Macarena, Lavecchia, Martín José, Bua, Silvia, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: Química, Vanillin, Carbonic anhydrase, Enzyme inhibitors, Molecular docking, Enones
وصف الملف: application/pdf; 2118-2127
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3Dissertation/ Thesis
المؤلفون: Riafrecha, Leonardo Ezequiel
المساهمون: Colinas, Pedro Alfonso, Arenas, Yésica Soledad
مصطلحات موضوعية: Química, Educación, Taller de escritura, Trabajo final, Química orgánica
وصف الملف: application/pdf
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4Academic Journal
مصطلحات موضوعية: Bioquímica, C-cinamoilglicosidos, Anhidrasa carbónica, DFT
وصف الملف: application/pdf
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5Academic Journal
المؤلفون: Zaro, María José, Bortolotti, Ana, Riafrecha, Leonardo Ezequiel, Concellón, Analía, Morbidoni, Héctor R., Colinas, Pedro Alfonso
مصطلحات موضوعية: Química, Dual mechanism, Glycomimetic, Tuberculosis
وصف الملف: application/pdf; 1726-1730
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6Academic Journal
المؤلفون: Riafrecha, Leonardo Ezequiel, Vullo, Daniela, Ouahrani-Bettache, Safia, Köhler, Stephan, Dumy, Pascal, Winum, Jean-Yves, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: Química, Antibacterial, Carbohydrate, Carbonic anhydrase
وصف الملف: application/pdf; 1017-1020
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7Academic Journal
مصطلحات موضوعية: Ciencias Exactas, Carbohydrate, carbonic anhydrase, pathogen
وصف الملف: application/pdf; 857-861
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8Dissertation/ Thesis
المؤلفون: Riafrecha, Leonardo Ezequiel
المساهمون: Colinas, Pedro Alfonso
مصطلحات موضوعية: Ciencias Exactas, Química, Glicósidos, Anhidrasas Carbónicas, Compuestos Químicos
وصف الملف: application/pdf
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9Academic Journal
المؤلفون: Riafrecha, Leonardo Ezequiel, Vullo, Daniela, Ouahrani Bettache, Safia, Köhler, Stephan, Dumy, Pascal, Winum, Jean Yves, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: ANTIBACTERIAL, CARBOHYDRATE, CARBONIC ANHYDRASE, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: http://hdl.handle.net/11336/39664; Riafrecha, Leonardo Ezequiel; Vullo, Daniela; Ouahrani Bettache, Safia; Köhler, Stephan; Dumy, Pascal; et al.; Inhibition of β-carbonic anhydrases from Brucella suis with C-cinnamoyl glycosides incorporating the phenol moiety; Taylor & Francis Ltd; Journal of Enzyme Inhibition and Medicinal Chemistry; 30; 6; 11-2015; 1017-1020; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/39664
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10Academic Journal
مصطلحات موضوعية: CARBONIC aNHYDRASES, C-GLYCOSYL SULFAMATES, CARBOHYDRATE, PHARMACOPHORE, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: info:eu-repo/semantics/altIdentifier/url/https://www.sciencedirect.com/science/article/pii/S0045206817306387; http://hdl.handle.net/11336/99690; Riafrecha, Leonardo Ezequiel; Bua, Silvia; Supuran, Claudiu T.; Colinas, Pedro Alfonso; Improving the carbonic anhydrase inhibition profile of the sulfamoylphenyl pharmacophore by attachment of carbohydrate moieties; Academic Press Inc Elsevier Science; Bioorganic Chemistry; 76; 2-2018; 61-66; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/99690
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11Academic Journal
مصطلحات موضوعية: Carbohydrate, Carbonic Anhydrase, Pathogen, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: http://hdl.handle.net/11336/53460; Riafrecha, Leonardo Ezequiel; Vullo, Daniela; Supuran, Claudiu T.; Colinas, Pedro Alfonso; C-glycosides incorporating the 6-methoxy-2-naphthyl moiety are selective inhibitors of fungal and bacterial carbonic anhydrases; Taylor & Francis; Journal of Enzyme Inhibition and Medicinal Chemistry; 30; 5; 9-2015; 857-861; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/53460
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12Academic Journal
المؤلفون: Riafrecha, Leonardo Ezequiel, Le Pors, Macarena Soledad, Lavecchia, Martín José, Bua, Silvia, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: VANILLIN, CARBONIC ANHYDRASE, MOLECULAR DOCKING, ENONES, ENZYME INHIBITORS, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: http://hdl.handle.net/11336/155128; Riafrecha, Leonardo Ezequiel; Le Pors, Macarena Soledad; Lavecchia, Martín José; Bua, Silvia; Supuran, Claudiu T.; et al.; Vanillin enones as selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII: The out of the active site pocket for the design of selective inhibitors?; Taylor & Francis Ltd; Journal of Enzyme Inhibition and Medicinal Chemistry; 36; 1; 4-10-2021; 2118-2127; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/155128
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13Academic Journal
المؤلفون: Buchieri, María Virginia, Riafrecha, Leonardo Ezequiel, Rodríguez, Oscar Mariano, Vullo, Daniela, Morbidoni, Héctor Ricardo, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: C-Glycosides, Mycobacterium Tuberculosis, Carbonic Anhydrase, Anti-Tubercular Activity, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: info:eu-repo/semantics/altIdentifier/url/http://www.sciencedirect.com/science/article/pii/S0960894X12015375; http://hdl.handle.net/11336/24754; Buchieri, María Virginia; Riafrecha, Leonardo Ezequiel; Rodríguez, Oscar Mariano; Vullo, Daniela; Morbidoni, Héctor Ricardo; et al.; Inhibition of the β-carbonic anhydrases from Mycobacterium tuberculosis with C-cinnamoyl glycosides: Identification of the first inhibitor with anti-mycobacterial activity; Pergamon-Elsevier Science Ltd.; Bioorganic & Medicinal Chemistry Letters; 23; 3; 1-2013; 740-743; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/24754
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14Academic Journal
المؤلفون: Riafrecha, Leonardo Ezequiel, Rodríguez, Oscar Mariano, Vullo, Daniela, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: Glycomimetics, Enzyme Inhibitors, Cancer, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: info:eu-repo/semantics/altIdentifier/url/http://www.sciencedirect.com/science/article/pii/S0968089614005768; http://hdl.handle.net/11336/32829; Rodríguez, Oscar Mariano; Colinas, Pedro Alfonso; Supuran, Claudiu T.; Vullo, Daniela; Riafrecha, Leonardo Ezequiel; Attachment of carbohydrates to methoxyaryl moieties leads to highly selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII; Pergamon-Elsevier Science Ltd.; Bioorganic & Medicinal Chemistry; 22; 19; 8-2014; 5308-5314; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/32829
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15Academic Journal
المؤلفون: Riafrecha, Leonardo Ezequiel, Rodríguez, Oscar Mariano, Vullo, Daniela, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: C-Glycosides, Carbonic Anhydrase, Phenol, Enzyme Inhibition, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: info:eu-repo/semantics/altIdentifier/url/http://www.sciencedirect.com/science/article/pii/S0968089612006992; http://hdl.handle.net/11336/22550; Riafrecha, Leonardo Ezequiel; Rodríguez, Oscar Mariano; Vullo, Daniela; Supuran, Claudiu T.; Colinas, Pedro Alfonso; Synthesis of C-cinnamoyl glycosides and their inhibitory activity against mammalian carbonic anhydrases; Elsevier; Bioorganic & Medicinal Chemistry; 21; 6; 9-2012; 1489-1494; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/22550
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16Academic Journal
المؤلفون: Zaro, Maria Jose, Bortolotti, Ana, Riafrecha, Leonardo Ezequiel, Concellón, Analía, Morbidoni, Héctor Ricardo, Colinas, Pedro Alfonso
مصطلحات موضوعية: ABTS, DPPH, MYCOBACTERIUM TUBERCULOSIS, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: http://hdl.handle.net/11336/112280; Zaro, Maria Jose; Bortolotti, Ana; Riafrecha, Leonardo Ezequiel; Concellón, Analía; Morbidoni, Héctor Ricardo; et al.; Anti-tubercular and antioxidant activities of C-glycosyl carbonic anhydrase inhibitors: towards the development of novel chemotherapeutic agents against Mycobacterium tuberculosis; Taylor & Francis Ltd; Journal of Enzyme Inhibition and Medicinal Chemistry; 31; 5-2016; 1726-1730; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/112280
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17Academic Journal
المؤلفون: Vasquez, Ivana Raquel, Riafrecha, Leonardo Ezequiel, Martinez Heredia, Leandro, Echeverría, Gustavo Alberto, Piro, Oscar Enrique, Lavecchia, Martín José, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: glucoimines, enzyme inhibitor, docking, X-ray, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: info:eu-repo/semantics/altIdentifier/url/https://linkinghub.elsevier.com/retrieve/pii/S0022286024022877; http://hdl.handle.net/11336/243946; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/243946
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18Academic Journal
المؤلفون: Barri, Ivan Alejandro, Riafrecha, Leonardo Ezequiel, Echeverría, Gustavo Alberto, Piro, Oscar Enrique, Colinas, Pedro Alfonso
مصطلحات موضوعية: Carbohydrates, Cycloaddition, Diastereomer, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: info:eu-repo/semantics/altIdentifier/url/https://linkinghub.elsevier.com/retrieve/pii/S0022286024007725; http://hdl.handle.net/11336/234867; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/234867
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19Academic Journal
المؤلفون: Le Pors, Macarena Soledad, Santa Maria de la Parra, Lucía, Riafrecha, Leonardo Ezequiel, Vullo, Daniela, Leon, Ignacio Esteban, Supuran, Claudiu T., Colinas, Pedro Alfonso
مصطلحات موضوعية: CANCER, ENZYME INHIBITORS, ISOXAZOLES, O-GLYCOSIDES, TARGETED THERAPY, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: http://hdl.handle.net/11336/223156; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/223156
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20Academic Journal
المؤلفون: Le Pors, Macarena Soledad, Barri, Ivan Alejandro, Riafrecha, Leonardo Ezequiel, Echeverría, Gustavo Alberto, Piro, Oscar Enrique, Colinas, Pedro Alfonso
مصطلحات موضوعية: Click-chemistry, Cycloaddition, O-Glycosides, https://purl.org/becyt/ford/1.4, https://purl.org/becyt/ford/1
وصف الملف: application/pdf
Relation: http://hdl.handle.net/11336/215161; CONICET Digital; CONICET
الاتاحة: http://hdl.handle.net/11336/215161