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1Academic Journal
المؤلفون: Nina Kerres, Steffen Steurer, Stefanie Schlager, Gerd Bader, Helmut Berger, Maureen Caligiuri, Christian Dank, John R. Engen, Peter Ettmayer, Bernhard Fischerauer, Gerlinde Flotzinger, Daniel Gerlach, Thomas Gerstberger, Teresa Gmaschitz, Peter Greb, Bingsong Han, Elizabeth Heyes, Roxana E. Iacob, Dirk Kessler, Heike Kölle, Lyne Lamarre, David R. Lancia, Simon Lucas, Moriz Mayer, Katharina Mayr, Nikolai Mischerikow, Katja Mück, Christoph Peinsipp, Oliver Petermann, Ulrich Reiser, Dorothea Rudolph, Klaus Rumpel, Carina Salomon, Dirk Scharn, Renate Schnitzer, Andreas Schrenk, Norbert Schweifer, Diane Thompson, Elisabeth Traxler, Roland Varecka, Tilman Voss, Alexander Weiss-Puxbaum, Sandra Winkler, Xiaozhang Zheng, Andreas Zoephel, Norbert Kraut, Darryl McConnell, Mark Pearson, Manfred Koegl
المصدر: Cell Reports, Vol 20, Iss 12, Pp 2860-2875 (2017)
مصطلحات موضوعية: oncogene, transcription factor, drug target, drug discovery, cancer, lymphoma, BTB domain, ubiquitin, Biology (General), QH301-705.5
وصف الملف: electronic resource
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2Academic Journal
المؤلفون: Juergen Ramharter (2163022), Dirk Kessler (2556022), Peter Ettmayer (3013665), Marco H. Hofmann (10304398), Thomas Gerstberger (2556016), Michael Gmachl (10304401), Tobias Wunberg (3346658), Christiane Kofink (2739130), Michael Sanderson (3241353), Heribert Arnhof (1947235), Gerd Bader (2556040), Klaus Rumpel (2436175), Andreas Zöphel (10304404), Renate Schnitzer (3346640), Jark Böttcher (10304407), Jonathan C. O’Connell (8508444), Rachel L. Mendes (4257835), David Richard (10304410), Nikolai Pototschnig (10304413), Irene Weiner (10304416), Wolfgang Hela (10304419), Katja Hauer (10304422), Daniela Haering (7245806), Lyne Lamarre (7861718), Bernhard Wolkerstorfer (4481332), Christian Salamon (10304425), Patrick Werni (10304428), Silvia Munico-Martinez (10304431), Reiner Meyer (10304434), Matthew D. Kennedy (10304437), Norbert Kraut (10304440), Darryl B. McConnell (2685361)
مصطلحات موضوعية: Biophysics, Biochemistry, Molecular Biology, Pharmacology, Cancer, Hematology, Chemical Sciences not elsewhere classified, BI -3406, colorectal tumor cells, KRAS G 13D, PPI, contact surface area, 1-KRAS, probe SOS 1 biology, EGFR inhibitor afatinib, interaction, SOS 1 inhibitors, SOS 1 activators, Y 884 SOS 1
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3
المؤلفون: Jürgen Moll, Natarajan Muthusamy, Norbert Kraut, Darryl B. McConnell, Mark Pearson, Segundo Gonzalez, Peter Ettmayer, Sumithira Vasu, Swagata Goswami, Girish Rajgolikar, Michael P. Sanderson, Thomas Gerstberger, Renate Schnitzer, Andreas Zoephel, Heribert Arnhof, Dirk Scharn, Jark Böttcher, Seila Lorenzo-Herrero, Marc Kerenyi, Sebastian Carotta, Maria A. Impagnatiello, Harald Engelhardt, Rajeswaran Mani, Marco H. Hofmann
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4
المؤلفون: Jürgen Moll, Natarajan Muthusamy, Norbert Kraut, Darryl B. McConnell, Mark Pearson, Segundo Gonzalez, Peter Ettmayer, Sumithira Vasu, Swagata Goswami, Girish Rajgolikar, Michael P. Sanderson, Thomas Gerstberger, Renate Schnitzer, Andreas Zoephel, Heribert Arnhof, Dirk Scharn, Jark Böttcher, Seila Lorenzo-Herrero, Marc Kerenyi, Sebastian Carotta, Maria A. Impagnatiello, Harald Engelhardt, Rajeswaran Mani, Marco H. Hofmann
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5
المؤلفون: Segundo Gonzalez, Dirk Scharn, Mark Pearson, Sebastian Carotta, Swagata Goswami, Natarajan Muthusamy, Heribert Arnhof, Sumithira Vasu, Norbert Kraut, Seila Lorenzo-Herrero, Harald Engelhardt, Michael P. Sanderson, Marc Kerenyi, Maria Antonietta Impagnatiello, Rajeswaran Mani, Renate Schnitzer, Jark Böttcher, Peter Ettmayer, Girish Rajgolikar, Marco H. Hofmann, Jürgen Moll, Andreas Zoephel, Darryl B. McConnell, Thomas Gerstberger
المصدر: Mol Cancer Ther
مصطلحات موضوعية: Cytotoxicity, Immunologic, 0301 basic medicine, Cancer Research, Melanoma, Experimental, Apoptosis, Breast Neoplasms, Mice, SCID, Article, GZMB, Mice, 03 medical and health sciences, 0302 clinical medicine, Mice, Inbred NOD, Tumor Cells, Cultured, medicine, Animals, Humans, Phosphorylation, Protein Kinase Inhibitors, Cell Proliferation, biology, Chemistry, Degranulation, Cancer, Cyclin-Dependent Kinase 8, Acquired immune system, medicine.disease, Xenograft Model Antitumor Assays, Cyclin-Dependent Kinases, Killer Cells, Natural, Mice, Inbred C57BL, Granzyme B, Leukemia, Myeloid, Acute, STAT1 Transcription Factor, 030104 developmental biology, Oncology, Perforin, 030220 oncology & carcinogenesis, Cancer cell, Cancer research, biology.protein, Female, Antibody
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6
المؤلفون: Zhulin Tan, Nitinchandra D. Patel, Harald Engelhardt, Mark Petronczki, Georg Egger, Elisabeth Grondal, Lyne Lamarre, Joyce C. Leung, Bernadette Sharps, Nizar Haddad, Anke Baum, Andreas Bergner, Andreas Schrenk, Renate Schnitzer, Eugene Chong, Tobias Wunberg, Moriz Mayer, Thomas Gerstberger, Dietrich Böse, Andreas Zoephel, Darryl B. McConnell, Christian Engelhardt, Monika Kriz, Nina C. Gonnella, Mariusz Krawiec, Heinz Stadtmüller, Peter Ettmayer, Jonathan T. Reeves, Julian E. Fuchs, Barbara Hopfgartner, Dirk Scharn, Andreas Grimm, Biljana Peric Simov, Flavio Solca, Gerd Bader, Sandra Döbel, Roland Kousek
المصدر: Journal of Medicinal Chemistry. 62:10272-10293
مصطلحات موضوعية: Lung Neoplasms, Protein Conformation, Entropy, Transgene, Antineoplastic Agents, Mice, Transgenic, Crystallography, X-Ray, medicine.disease_cause, 01 natural sciences, Mice, Structure-Activity Relationship, 03 medical and health sciences, T790M, Carcinoma, Non-Small-Cell Lung, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Epidermal growth factor receptor, Protein Kinase Inhibitors, 030304 developmental biology, 0303 health sciences, Mutation, biology, Chemistry, Xenograft Model Antitumor Assays, respiratory tract diseases, 0104 chemical sciences, ErbB Receptors, 010404 medicinal & biomolecular chemistry, Protein kinase domain, Cyclization, Cell culture, Hepatocytes, Cancer research, biology.protein, Molecular Medicine, Benzimidazoles, Female, Tyrosine kinase
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7
المؤلفون: Yvonne Scherbantin, Gerd Bader, thomas Fett, Harald Weinstabl, Sophie Mitzner, Tuncay Ciftci, Bernhard Wolkerstorfer, Jens Bruchhaus, Xiaobing Lv, Dongyang Li, Bernadette Sharps, Daniela Haering, Heribert Arnhof, Nikolai Mischerikow, Geraldine Garavel, Andreas Schrenk, Joerg Rinnenthal, Roland Kousek, Thomas Gerstberger, Guido Scholz, Stephan Karl Zahn, Paola Martinelli, Jens Quant, Renate Schnitzer, Andreas Zoephel, Darryl B. McConnell, Moriz Mayer, Dirk Kessler, Xuechun Zhang, Michelle Burkard, Mark Pearson, Karin S. Hofbauer, Alicia Du, Matthias Treu, Christoph Harrer, Yali Li, Fabio Savarese, Klaus Rumpel, Biljana Peric-Simov, Georg Dahmann, Wolfgang Sommergruber, Peter Ettmayer
المصدر: Journal of Medicinal Chemistry. 62:7976-7997
مصطلحات موضوعية: chemistry.chemical_classification, 0303 health sciences, biology, Dehydrogenase, Prodrug, Nicotinamide adenine dinucleotide, 01 natural sciences, Cofactor, 0104 chemical sciences, Serine, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, chemistry, Biochemistry, Oxidoreductase, Drug Discovery, biology.protein, Molecular Medicine, NAD+ kinase, Phosphoglycerate dehydrogenase, 030304 developmental biology
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8
المؤلفون: Birgit Wilding, Dirk Scharn, Dietrich Böse, Anke Baum, Valeria Santoro, Paolo Chetta, Renate Schnitzer, Dana A. Botesteanu, Christoph Reiser, Stefan Kornigg, Petr Knesl, Alexandra Hörmann, Anna Köferle, Maja Corcokovic, Simone Lieb, Guido Scholz, Jens Bruchhaus, Markus Spina, Josef Balla, Biljana Peric-Simov, Jasmin Zimmer, Sophie Mitzner, Thomas N. Fett, Alexandra Beran, Lyne Lamarre, Thomas Gerstberger, Daniel Gerlach, Markus Bauer, Andreas Bergner, Andreas Schlattl, Gerd Bader, Matthias Treu, Harald Engelhardt, Stephan Zahn, Julian E. Fuchs, Johannes Zuber, Peter Ettmayer, Mark Pearson, Mark Petronczki, Norbert Kraut, Darryl B. McConnell, Flavio Solca, Ralph A. Neumüller
المصدر: Nature cancer. 3(7)
مصطلحات موضوعية: ErbB Receptors, Cancer Research, Lung Neoplasms, Oncology, Receptor, ErbB-2, Carcinoma, Non-Small-Cell Lung, Humans, Exons, Genes, erbB-2, Protein Kinase Inhibitors
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9
المؤلفون: Reiner Meyer, Heribert Arnhof, Daniela Haering, Rachel L Mendes, David J. Richard, Irene Weiner, Norbert Kraut, Wolfgang Hela, Christian Salamon, Klaus Rumpel, Gerd Bader, Michael Gmachl, Andreas Dr. Zöphel, Renate Schnitzer, Peter Ettmayer, Jark Böttcher, Matthew D Kennedy, Juergen Ramharter, Michael P. Sanderson, Darryl B. McConnell, Nikolai Pototschnig, Dirk Kessler, Silvia Munico-Martinez, Tobias Wunberg, Marco H. Hofmann, Katja Hauer, Thomas Gerstberger, Lyne Lamarre, Patrick Werni, Christiane Kofink, Jonathan O’Connell, Bernhard Wolkerstorfer
المصدر: Journal of medicinal chemistry. 64(10)
مصطلحات موضوعية: Afatinib, Mutagenesis (molecular biology technique), Molecular Dynamics Simulation, medicine.disease_cause, 01 natural sciences, Proto-Oncogene Proteins p21(ras), 03 medical and health sciences, Allosteric Regulation, Catalytic Domain, Drug Discovery, medicine, Humans, Protein Interaction Maps, Colorectal tumor, 030304 developmental biology, EGFR inhibitors, 0303 health sciences, Binding Sites, Chemistry, 0104 chemical sciences, ErbB Receptors, 010404 medicinal & biomolecular chemistry, Cancer research, SOS1, Mutagenesis, Site-Directed, Quinazolines, Molecular Medicine, KRAS, Colorectal Neoplasms, SOS1 Protein, medicine.drug, Foot-in-the-door technique
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10
المؤلفون: Andreas Schrenk, Daniela Häring, Silke Fischer, Stefan Kornigg, Alex G. Waterson, Andreas Mantoulidis, Manfred Koegl, Markus Zeeb, Thomas Gerstberger, Mark Pearson, Wolfgang Hela, Andreas Zoephel, Darryl B. McConnell, Michael Gmachl, Bernadette Sharps, Jale Karolyi-Oezguer, Johann Hoffmann, Franziska Moser, Jason Phan, Teresa Gmaschitz, David Covini, Bernhard Wolkerstorfer, Qi Sun, Lyne Lamarre, Gabriella Siszler, Renate Schnitzer, Moriz Mayer, Dirk Kessler, Katharina Schipany, Petr Knesl, Christian Salamon, Peter Greb, Stephen W. Fesik, Andreas Gollner, Yvonne Scherbantin, Silvia Munico-Martinez, Craig M. Goodwin, Roland Kousek, Jörg Rinnenthal, Jiqing Sai, Christoph Peinsipp, Laetitia J. Martin
المصدر: Proceedings of the National Academy of Sciences of the United States of America
مصطلحات موضوعية: Neuroblastoma RAS viral oncogene homolog, Models, Molecular, Druggability, GTPase, medicine.disease_cause, Proto-Oncogene Proteins p21(ras), 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, KRAS, medicine, Humans, HRAS, Letters, neoplasms, 030304 developmental biology, 0303 health sciences, Multidisciplinary, Oncogene, Chemistry, Drug discovery, Effector, Cell Biology, Biological Sciences, fragment-based drug design, NMR, digestive system diseases, 3. Good health, PNAS Plus, Pharmaceutical Preparations, 030220 oncology & carcinogenesis, oncology, Physical Sciences, Cancer research, structure-based drug design, Nanoparticles, Guanosine Triphosphate
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11
المؤلفون: Simon Wöhrle, Tom Owen-Hughes, Jale Karolyi-Oezguer, Teresa Gmaschitz, Steffen Steurer, Bernadette Sharps, Heribert Arnhof, Gerd Bader, Joerg Rinnenthal, Thomas Gerstberger, Peter Greb, Manfred Koegl, Johannes Wachter, Michael Galant, Klaus Rumpel, Carina Riedmueller, William Farnaby, David Zollman, Peter Ettmayer, Meng-Ying Wu, Michael J. Roy, Emelyne Diers, Andreas Zoephel, Nicole Trainor, Darryl B. McConnell, Nicola Wiechens, Mark Pearson, Guido Boehmelt, Oliver Petermann, Alessio Ciulli, Renate Schnitzer, Harald Weinstabl, Christian Dank, Katharina Ehrenhöfer-Wölfer, Alexander Weiss-Puxbaum, Claire Whitworth, Elisabeth Traxler
المصدر: Nature chemical biology
مصطلحات موضوعية: Chromatin remodeling, Article, 03 medical and health sciences, 0302 clinical medicine, Humans, Molecular Biology, Ternary complex, Cells, Cultured, 030304 developmental biology, Cell Proliferation, 0303 health sciences, biology, Molecular Structure, Chemistry, Cell growth, Proteolysis targeting chimera, Myeloid leukemia, Nuclear Proteins, Cell Biology, Chromatin Assembly and Disassembly, 3. Good health, Cell biology, Bromodomain, Ubiquitin ligase, DNA-Binding Proteins, Leukemia, Myeloid, Acute, 030220 oncology & carcinogenesis, Cancer cell, biology.protein
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12
المؤلفون: David R. Lancia, John R. Engen, Elizabeth Heyes, Katharina Mayr, Lyne Lamarre, Mark Pearson, Carina Salomon, Simon Lucas, Steffen Steurer, Alexander Weiss-Puxbaum, Klaus Rumpel, Gerlinde Flotzinger, Norbert Kraut, Xiaozhang Zheng, Daniel Gerlach, Katja Mück, Sandra Winkler, Heike Kölle, Peter Ettmayer, Nikolai Mischerikow, Christian Dank, Ulrich Reiser, Dirk Scharn, Bingsong Han, Teresa Gmaschitz, Andreas Schrenk, Nina Kerres, Norbert Schweifer, Dirk Kessler, Tilman Voss, Renate Schnitzer, Manfred Koegl, Roland Varecka, Moriz Mayer, Dorothea Rudolph, Oliver Petermann, Diane Thompson, Thomas Gerstberger, Christoph Peinsipp, Roxana E. Iacob, Stefanie Schlager, Gerd Bader, Helmut Berger, Peter Greb, Maureen Caligiuri, Elisabeth Traxler, Bernhard Fischerauer, Andreas Zoephel, Darryl B. McConnell
المصدر: Cell Reports, Vol 20, Iss 12, Pp 2860-2875 (2017)
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Proteasome Endopeptidase Complex, Protein family, Druggability, Repressor, lymphoma, Biology, medicine.disease_cause, General Biochemistry, Genetics and Molecular Biology, drug target, drug discovery, 03 medical and health sciences, Inhibitory Concentration 50, Structure-Activity Relationship, 0302 clinical medicine, Protein Domains, Transcription (biology), immune system diseases, oncogene, hemic and lymphatic diseases, Cell Line, Tumor, ubiquitin, medicine, cancer, Humans, BTB domain, Transcription factor, lcsh:QH301-705.5, transcription factor, Cell Proliferation, Drug discovery, Ubiquitination, DNA, BCL6, Gene Expression Regulation, Neoplastic, Kinetics, 030104 developmental biology, HEK293 Cells, Pyrimidines, lcsh:Biology (General), 030220 oncology & carcinogenesis, Proteolysis, Cancer research, Proto-Oncogene Proteins c-bcl-6, Carcinogenesis, Protein Binding
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13
المؤلفون: Michael Gmachl, Thomas Gerstberger, Heinz Stadtmueller, Heribert Arnhof, Christiane Kofink, Marco H. Hofmann, Juergen Moll, David Richard, Adrian Saldanha, Rachel L Mendes, Mark Pearson, Peter Ettmayer, Darryl B. McConnell, Norbert Kraut, Michael P. Sanderson, Fabio Savarese, Dana-Adriana Botesteanu, Tobias Wunberg, Daniel Gerlach, Francesca Trapani, Renate Schnitzer, Dirk Kessler, Jonathan O’Connell, Jürgen Ramharter
المصدر: Molecular Cancer Therapeutics. 18:C133-C133
مصطلحات موضوعية: MAPK/ERK pathway, Cancer Research, Oncogene, business.industry, MEK inhibitor, Cancer, Context (language use), medicine.disease_cause, medicine.disease, Oncology, medicine, Cancer research, SOS1, Guanine nucleotide exchange factor, KRAS, business
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14
المؤلفون: Jale Karolyi-Oezguer, Renate Schnitzer, Heribert Arnhof, Emelyne Diers, Andreas Zoephel, Harald Weinstabl, Bernadette Sharps, Darryl B. McConnell, Katharina Ehrenhöfer-Wölfer, Peter Ettmayer, David Zollman, Joerg Rinnenthal, Guido Boehmelt, Michael J. Roy, Meng-Ying Wu, Alessio Ciulli, Thomas Gerstberger, Klaus Rumpel, William Farnaby, Carina Riedmueller, Alexander Weiss-Puxbaum, Nicole Trainor, Peter Greb, Mark Pearson, Johannes Wachter, Michael Galant, Steffen Steurer, Tom Owen-Hughes, Oliver Petermann, Simon Wöhrle, Manfred Koegl, Nicola Wiechens, Elisabeth Traxler, Gerd Bader, Teresa Gmaschitz, Christian Dank, Claire Whitworth
المصدر: Nature Chemical Biology. 15:846-846
مصطلحات موضوعية: 0303 health sciences, Chemistry, DNA repair, 030302 biochemistry & molecular biology, Cell Biology, Chromatin remodeling, Cell biology, Bromodomain, Chromatin, 03 medical and health sciences, chemistry.chemical_compound, Transcription (biology), SMARCA4, Nucleosome, Molecular Biology, DNA, 030304 developmental biology
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15
المؤلفون: Jark Boettcher, Mark Pearson, Segundo Gonzalez, Rajeswaran Mani, Maria Antonietta Impagnatiello, Marco H. Hofmann, Heribert Arnhof, Girish Rajgolikar, Andreas Zoephel, Darryl B. McConnell, Juergen Moll, Sumithira Vasu, Sebastian Carotta, Marc Kerenyi, Harald Engelhardt, Seila Lorenzo-Herrero, Natarajan Muthusamy, Norbert Kraut, Peter Ettmayer, Renate Schnitzer, Thomas Gerstberger, Dirk Scharn, Swagata Goswami
المصدر: Cancer Research. 79:510-510
مصطلحات موضوعية: Cancer Research, biology, Chemistry, Melanoma, Cancer, medicine.disease, Acquired immune system, Granzyme B, Cytolysis, Oncology, Perforin, medicine, biology.protein, Cancer research, Cytotoxic T cell, Receptor
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16
المؤلفون: Peter Ettmayer, Herbert Nar, Andreas Bergner, Renate Schnitzer
مصطلحات موضوعية: 0301 basic medicine, Virtual screening, Engineering, Drug discovery, business.industry, Nanotechnology, Entry point, Hit to lead, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Lead (geology), Risk analysis (engineering), 030220 oncology & carcinogenesis, business
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17
المؤلفون: Mark Pearson, David R. Lancia, Daniel Gerlach, John R. Engen, Andreas Zoephel, Darryl B. McConnell, Nina Kerres, Christian Dank, Xiaozhang Zheng, Stefanie Schlager, Gerd Bader, Tilman Voss, Nikolai Mischerikow, Renate Schnitzer, Norbert Kraut, Mayer Moriz, Thomas Gerstberger, Maureen Caligiuri, Manfred Koegl, Bingsong Han, Peter Ettmayer, Klaus Rumpel, Roxana E. Iacob, Dirk Kessler, Steffen Steurer
المصدر: Cancer Research. 78:3354-3354
مصطلحات موضوعية: Cancer Research, Oncology, immune system diseases, hemic and lymphatic diseases, Research community, Philosophy, medicine, Cancer research, Repressor, Carcinogenesis, medicine.disease_cause, BCL6, Transcription factor
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18
المؤلفون: William Farnaby, Alessio Ciulli, Peter Ettmayer, Manfred Koegl, Renate Schnitzer, Claire Whitworth, Steffen Steurer
المصدر: ESMO Open. 3:A198
مصطلحات موضوعية: Streptavidin, Cancer Research, Lysis, biology, Chemistry, Context (language use), law.invention, Ubiquitin ligase, chemistry.chemical_compound, Oncology, law, Biotinylation, Recombinant DNA, biology.protein, Biophysics, Ternary operation, Ternary complex
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19
المؤلفون: Moritz Mayer, Darryl B. McConnell, Gerhard Gmaschitz, Sebastian Carotta, Heribert Arnhof, Marc Kerenyi, Mark Pearson, Jürgen Moll, Christian Engelhardt, Michael P. Sanderson, Dirk Scharn, Georg Egger, Harald Engelhardt, Marco H. Hofmann, Renate Schnitzer, Norbert Kraut, Maria Antonietta Impagnatiello
المصدر: Cancer Research. 77:4630-4630
مصطلحات موضوعية: Cancer Research, biology, Kinase, Chemistry, Granzyme B, Oncology, Perforin, Cell culture, Cancer cell, biology.protein, STAT protein, Cancer research, Cytotoxic T cell, STAT1
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20
المؤلفون: Renate Schnitzer, Gerhard Loeber
المصدر: Genetic Engineering ISBN: 9781489917416
مصطلحات موضوعية: Drug, Reporter gene, Structural biology, Drug discovery, Computer science, Cellular Assay, media_common.quotation_subject, Laboratory automation, Drug design, Identification (biology), Computational biology, media_common