المؤلفون: Dominika Pindjakova, Eliska Pilarova, Karel Pauk, Hana Michnova, Jan Hosek, Pratibha Magar, Alois Cizek, Ales Imramovsky, Josef Jampilek

المصدر: International Journal of Molecular Sciences; Volume 23; Issue 19; Pages: 11648

مصطلحات موضوعية: salicylamide, peptidomimetics, antimicrobial activity, cytotoxicity, lipophilicity, structure–activity relationships

جغرافية الموضوع: agris

وصف الملف: application/pdf

Relation: Biochemistry; https://dx.doi.org/10.3390/ijms231911648

الاتاحة: https://doi.org/10.3390/ijms231911648

المؤلفون: Pratibha Magar, Oscar Parravicini, Šárka Štěpánková, Katarina Svrčková, Adriana D. Garro, Izabela Jendrzejewska, Karel Pauk, Jan Hošek, Josef Jampílek, Ricardo D. Enriz, Aleš Imramovský

المصدر: International Journal of Molecular Sciences; Volume 22; Issue 17; Pages: 9447

مصطلحات موضوعية: bioassays, carbamates, cholinesterase inhibitors, molecular modeling, sulfonamides, synthesis

جغرافية الموضوع: agris

وصف الملف: application/pdf

Relation: Molecular Biology; https://dx.doi.org/10.3390/ijms22179447

الاتاحة: https://doi.org/10.3390/ijms22179447

المؤلفون: Šárka Štěpánková, Jan Hošek, Katarína Svrčková, Ricardo D. Enriz, Josef Jampilek, Adriana Garro, Karel Pauk, Izabela Jendrzejewska, Aleš Imramovský, Oscar Parravicini, Pratibha Magar

المصدر: International Journal of Molecular Sciences, Vol 22, Iss 9447, p 9447 (2021)
International Journal of Molecular Sciences
Volume 22
Issue 17

مصطلحات موضوعية: Carbamate, cholinesterase inhibitors, Molecular model, synthesis, Stereochemistry, QH301-705.5, medicine.medical_treatment, sulfoamidy, carbamates, inhibitory cholinesteráz, Molecular Dynamics Simulation, Article, Catalysis, Inorganic Chemistry, Structure-Activity Relationship, chemistry.chemical_compound, Catalytic Domain, sulfonamides, BChE, medicine, Humans, Physical and Theoretical Chemistry, Biology (General), bioassays, Molecular Biology, QD1-999, Spectroscopy, Butyrylcholinesterase, Cholinesterase, chemistry.chemical_classification, Binding Sites, biology, Chemistry, molecular modeling, Organic Chemistry, karbamáty, Active site, General Medicine, Acetylcholinesterase, Computer Science Applications, Sulfonamide, Molecular Docking Simulation, Docking (molecular), biology.protein, AChE

وصف الملف: p. 9447; application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4fe97f9f665fc907bae959315eb34e8e
https://www.mdpi.com/1422-0067/22/17/9447

المؤلفون: Ales Imramovsky, Josef Jampilek, Alois Čížek, Pratibha Magar, Hana Michnová

المصدر: Proceedings of 5th International Electronic Conference on Medicinal Chemistry.

مصطلحات موضوعية: Chemistry, medicine, Salicylamide, Combinatorial chemistry, medicine.drug

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::2241c108d90fbad0c763d2306f903976
https://doi.org/10.3390/ecmc2019-06344

المؤلفون: Aleš Imramovský, Michal Dibus, Radek Jorda, Denisa Hendrychová, Karel Pauk, Eliška Pilařová, Vladimír Kryštof, Pratibha Magar

المصدر: European journal of medicinal chemistry. 188

مصطلحات موضوعية: Cell Survival, Poly ADP ribose polymerase, Phenylalanine, Antineoplastic Agents, Focal adhesion, Structure-Activity Relationship, Leucine, Drug Discovery, Tumor Cells, Cultured, Humans, Cell adhesion, Paxillin, Cell Proliferation, Pharmacology, biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, General Medicine, Dipeptides, HCT116 Cells, Biochemistry, Apoptosis, Cancer cell, biology.protein, Drug Screening Assays, Antitumor

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dbaa1b958f4fd8cfb65ba19c5b2c1934
https://pubmed.ncbi.nlm.nih.gov/31931341

المؤلفون: Eva Řezníčková, Aleš Imramovský, Karel Pauk, Jan Dušek, Radek Jorda, Vladimír Kryštof, Pratibha Magar

المصدر: European journal of medicinal chemistry. 135

مصطلحات موضوعية: 0301 basic medicine, Proteasome Endopeptidase Complex, Phenylalanine, Antineoplastic Agents, Protein degradation, Caspase 7, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Ubiquitin, Leucine, hemic and lymphatic diseases, Cell Line, Tumor, Drug Discovery, Salicylamides, medicine, Humans, Caspase, Cell Proliferation, Pharmacology, biology, Dose-Response Relationship, Drug, Molecular Structure, Bortezomib, Chemistry, Organic Chemistry, General Medicine, Molecular biology, 030104 developmental biology, Biochemistry, Proteasome, Apoptosis, 030220 oncology & carcinogenesis, Cancer cell, biology.protein, Drug Screening Assays, Antitumor, Proteasome Inhibitors, medicine.drug

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cefbfa0864c9e2e65e2a30b14c7872f1
https://pubmed.ncbi.nlm.nih.gov/28441582