المؤلفون: Dittrich, Birger, Connor, Lauren, Fabbiani, Francesca, Piechon, Philippe

Relation: Dittrich, Birger, Connor, Lauren, Fabbiani, Francesca and Piechon, Philippe (2024) Linking solid-state phenomena via energy differences in `archetype crystal structures'. IUCrJ. ISSN 2052-2525

الاتاحة: https://oak.novartis.com/52212/
https://doi.org/10.1107/S2052252524002641

المؤلفون: Sager, Emine, Tzvetkova, Pavleta, Gossert, Alvar D., Piechon, Philippe, Luy, Burkhard

المصدر: Chemistry - a European journal, 26 (63), 14435–14444 ; ISSN: 0947-6539, 1521-3765

مصطلحات موضوعية: ddc:540, Chemistry & allied sciences, info:eu-repo/classification/ddc/540

وصف الملف: application/pdf

Relation: info:eu-repo/semantics/altIdentifier/wos/000573975600001; info:eu-repo/semantics/altIdentifier/issn/0947-6539; info:eu-repo/semantics/altIdentifier/issn/1521-3765; https://publikationen.bibliothek.kit.edu/1000128315; https://publikationen.bibliothek.kit.edu/1000128315/124505480; https://doi.org/10.5445/IR/1000128315

الاتاحة: https://publikationen.bibliothek.kit.edu/1000128315
https://publikationen.bibliothek.kit.edu/1000128315/124505480
https://doi.org/10.5445/IR/1000128315

المؤلفون: Lapointe, Guillaume, Skepper, Colin K, Holder, Lauren M, Armstrong, Duncan, Bellamacina, Cornelia, Blais, Johanne, Bussiere, Dirksen, Bian, Jianwei, Cepura, Cody, Chan, Helen, Dean, Charles R, De Pascale, Gianfranco, Dhumale, Bhavesh, Fisher, L Mark, Fulsunder, Mangesh, Kantariya, Bhavin, Kim, Julie, King, Sean, Kossy, Lauren, Kulkarni, Upendra, Lakshman, Jay, Leeds, Jennifer A, Ling, Xiaolan, Lvov, Anatoli, Ma, Sylvia, Malekar, Swapnil, McKenney, David, Mergo, Wosenu, Metzger, Louis, Mhaske, Keshav, Moser, Heinz E, Mostafavi, Mina, Namballa, Sunil, Noeske, Jonas, Osborne, Colin, Patel, Ashish, Patel, Darshit, Patel, Tushar, Piechon, Philippe, Polyakov, Valery, Prajapati, Krunal, Prosen, Katherine R, Reck, Folkert, Richie, Daryl L, Sanderson, Mark R, Satasia, Shailesh, Savani, Bhautik, Selvarajah, Jogitha, Sethuraman, Vijay, Shu, Wei, Tashiro, Kyuto, Thompson, Katherine V, Vaarla, Krishniah, Vala, Lakhan, Veselkov, Dennis A, Vo, Jason, Vora, Bhavesh, Wagner, Trixie, Wedel, Laura, Williams, Sarah L, Yendluri, Satya, Yue, Qin, Yifru, Aregahegn, Zhang, Yong, Rivkin, Alexey

المصدر: Lapointe , G , Skepper , C K , Holder , L M , Armstrong , D , Bellamacina , C , Blais , J , Bussiere , D , Bian , J , Cepura , C , Chan , H , Dean , C R , De Pascale , G , Dhumale , B , Fisher , L M , Fulsunder , M , Kantariya , B , Kim , J , King , S , Kossy , L , Kulkarni , U , Lakshman , J , Leeds , J A , Ling , X , Lvov ....

وصف الملف: application/pdf

الاتاحة: https://kclpure.kcl.ac.uk/portal/en/publications/675d57ab-71d9-4244-886c-019cc57306cd
https://doi.org/10.1021/acs.jmedchem.1c00375
https://kclpure.kcl.ac.uk/ws/files/152730155/Discovery_and_Optimization_of_LAPOINTE_Epub30Apr2021_GREEN_VoR.pdf
http://www.scopus.com/inward/record.url?scp=85106542493&partnerID=8YFLogxK

المؤلفون: Cho, Hyelim, Shen, Qiong, Zhang, Lydia H., Okumura, Mikiko, Kawakami, Akinori, Ambrose, Jessi, Sigoillot, Frederic, Miller, Howard R., Gleim, Scott, Cobos-Correa, Amanda, Wang, Ying, Piechon, Philippe, Roma, Guglielmo, Eggimann, Fabian, Moore, Charles, Aspesi, Peter, Mapa, Felipa A., Burks, Heather, Ross, Nathan T., Krastel, Philipp, Hild, Marc, Maimone, Thomas J., Fisher, David E., Nomura, Daniel K., Tallarico, John A., Canham, Stephen M., Jenkins, Jeremy L., Forrester, William C.

المساهمون: National Institutes of Health

المصدر: Cell Chemical Biology ; volume 28, issue 10, page 1407-1419.e6 ; ISSN 2451-9456

الاتاحة: http://dx.doi.org/10.1016/j.chembiol.2021.03.004
https://api.elsevier.com/content/article/PII:S2451945621001434?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S2451945621001434?httpAccept=text/plain

المؤلفون: Sager, Emine, Tzvetkova, Pavleta, Gossert, Alvar D., Piechon, Philippe, Luy, Burkhard

المصدر: Chemistry - A European Journal, 26 (63)

مصطلحات موضوعية: molecular dynamics, natural products, quinolizidine, reserpine, residual dipolar couplings, structure elucidation

وصف الملف: application/application/pdf

Relation: info:eu-repo/semantics/altIdentifier/wos/000573975600001; http://hdl.handle.net/20.500.11850/445836

الاتاحة: https://hdl.handle.net/20.500.11850/445836
https://doi.org/10.3929/ethz-b-000445836

المؤلفون: Thoma, Gebhard, Vangrevelinghe, Eric, Luneau, Alexandre, Piechon, Philippe, Beerli, Christian, Zerwes, Hans Guenter

Relation: Thoma, Gebhard, Vangrevelinghe, Eric, Luneau, Alexandre, Piechon, Philippe, Beerli, Christian and Zerwes, Hans Guenter (2023) Novel Concept for Super-Soft Topical Drugs: Deactivation by an Enzyme-Induced Switch into an Inactive Conformation. ACS medicinal chemistry letters, 14. ISSN 1948-5875; https://doi.org/10.1021/acsmedchemlett.3c00169

الاتاحة: https://oak.novartis.com/50267/
https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.3c00169
https://doi.org/10.1021/acsmedchemlett.3c00169

المؤلفون: Fouché, Marianne, Schäfer, Michael, Berghausen, Jörg, Desrayaud, Sandrine, Blatter, Markus, Piéchon, Philippe, Dix, Ina, Martin Garcia, Aimar, Roth, Hans‐Jörg

المصدر: ChemMedChem ; volume 11, issue 10, page 1108-1108 ; ISSN 1860-7179 1860-7187

الاتاحة: http://dx.doi.org/10.1002/cmdc.201600230
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fcmdc.201600230
https://onlinelibrary.wiley.com/doi/full/10.1002/cmdc.201600230

المؤلفون: Bill, Anke, Hall, Michelle Lynn, Borawski, Jason, Hodgson, Catherine, Jenkins, Jeremy, Piechon, Philippe, Popa, Oana, Rothwell, Christopher, Tranter, Pamela, Tria, Scott, Wagner, Trixie, Whitehead, Lewis, Gaither, L.Alex

المصدر: Journal of Biological Chemistry ; volume 289, issue 16, page 11029-11041 ; ISSN 0021-9258

الاتاحة: http://dx.doi.org/10.1074/jbc.m114.549188
https://api.elsevier.com/content/article/PII:S0021925820483231?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0021925820483231?httpAccept=text/plain
https://syndication.highwire.org/content/doi/10.1074/jbc.M114.549188

المؤلفون: Velcicky, Juraj, Wilcken, Rainer, Cotesta, Simona, Janser, Philipp, Schlapbach, Achim, Piechon, Philippe, Villard, Frederic, Bouhelal, Rochdi, Piller, Fabian, Harlfinger, Stephanie, Stringer, Rowan, Fehlmann, Dominique, Kaupmann, Klemens, Littlewood-Evans, Amanda, Haffke, Matthias, Gommermann, Nina

Relation: Velcicky, Juraj, Wilcken, Rainer, Cotesta, Simona, Janser, Philipp, Schlapbach, Achim, Piechon, Philippe, Villard, Frederic, Bouhelal, Rochdi, Piller, Fabian, Harlfinger, Stephanie, Stringer, Rowan, Fehlmann, Dominique, Kaupmann, Klemens, Littlewood-Evans, Amanda, Haffke, Matthias and Gommermann, Nina (2020) Discovery And Optimization of Novel SUCNR1 Inhibitors: Design of Zwitterionic Derivatives with Salt-Bridge for Improvement of Oral Exposure. Journal of Medicinal Chemistry, 63 (17). pp. 9856-9875. ISSN 0022-26231520-4804

الاتاحة: https://oak.novartis.com/42931/
https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c01020
https://doi.org/10.1021/acs.jmedchem.0c01020

المؤلفون: Gu, Wayne, Zhao, Jibin, Li, Yunzhong, Yu, Bo, Tian, Xiangguang, Min, Jacob, Xu, Su, Gu, Huijuan, Sun, Junjie, Wang, Xufan, Ye, Shengqing, Yang, Hongwei, Tian, Yingtao, Gao, Feng, Gai, Yu, Wang, Yan, Zhang, Xuesong, Luo, Xi, Schenkel, Berthold, Venturoni, Francesco, Filipponi, Paolo, Guelat, Bertrand, Allmendinger, Thomas, Hoehn, Pascale, Kovacic, Nikola, Hermann, Luca, Schlama, Thierry, Ruch, Thomas, Derrien, Nadine, Piechon, Philippe, Kleinbeck-Riniker, Florian, Chen, Like, Wang, Huaimin, Wietfeld, Bernhard, Zhao, Stephen, Chang, Tommy, Lu, Xiaoquan, Zhang, Jianghua, Wu, Jingjing, Jia, Guanghua, Liu, Weichun, Gu, Xin, Hai, Dong

Relation: Gu, Wayne, Zhao, Jibin, Li, Yunzhong, Yu, Bo, Tian, Xiangguang, Min, Jacob, Xu, Su, Gu, Huijuan, Sun, Junjie, Wang, Xufan, Ye, Shengqing, Yang, Hongwei, Tian, Yingtao, Gao, Feng, Gai, Yu, Wang, Yan, Zhang, Xuesong, Luo, Xi, Schenkel, Berthold, Venturoni, Francesco, Filipponi, Paolo, Guelat, Bertrand, Allmendinger, Thomas, Hoehn, Pascale, Kovacic, Nikola, Hermann, Luca, Schlama, Thierry, Ruch, Thomas, Derrien, Nadine, Piechon, Philippe, Kleinbeck-Riniker, Florian, Chen, Like, Wang, Huaimin, Wietfeld, Bernhard, Zhao, Stephen, Chang, Tommy, Lu, Xiaoquan, Zhang, Jianghua, Wu, Jingjing, Jia, Guanghua, Liu, Weichun, Gu, Xin and Hai, Dong (2020) Application of Transition-Metal Catalysis, Biocatalysis and Flow Chemistry as State-of-the-Art Technologies in the Synthesis of LCZ696. The Journal of Organic Chemistry. ISSN 0022-32631520-6904

الاتاحة: https://oak.novartis.com/40789/
https://doi.org/10.1021/acs.joc.0c00473

المؤلفون: Sager, Emine, Tzvetkova, Pavleta, Gossert, Alvar D., Piechon, Philippe, Luy, Burkhard

المصدر: Chemistry-a European journal, 26 (63), 14435–14444
Chemistry-A European Journal, 26 (63)

مصطلحات موضوعية: reserpine, natural products, quinolizidine, Chemistry & allied sciences, structure elucidation, ddc:540, molecular dynamics, residual dipolar couplings

وصف الملف: application/pdf; application/application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::568f27825cff6db8efbce7e726e02c4d

المؤلفون: Reggane, Maude, Wiest, Johannes, Saedtler, Marco, Harlacher, Cornelius, Gutmann, Marcus, Zottnick, Sven, Piechon, Philippe, Dix, Ina, Müller-Buschbaum, Klaus, Holzgrabe, Ulrike, Meinel, Lorenz, Galli, Bruno

Relation: Reggane, Maude, Wiest, Johannes, Saedtler, Marco, Harlacher, Cornelius, Gutmann, Marcus, Zottnick, Sven, Piechon, Philippe, Dix, Ina, Müller-Buschbaum, Klaus, Holzgrabe, Ulrike, Meinel, Lorenz and Galli, Bruno (2018) Bioinspired co-crystals of Imatinib providing enhanced kinetic solubility. European Journal of Pharmaceutics and Biopharmaceutics, 128. pp. 290-299. ISSN 18733441

الاتاحة: https://oak.novartis.com/35107/
https://doi.org/10.1016/j.ejpb.2018.05.012

المؤلفون: Velcicky, Juraj, Wilcken, Rainer, Cotesta, Simona, Janser, Philipp, Schlapbach, Achim, Wagner, Trixie, Piechon, Philippe, Villard, Frederic, Bouhelal, Rochdi, Piller, Fabian, Harlfinger, Stephanie, Stringer, Rowan, Fehlmann, Dominique, Kaupmann, Klemens, Littlewood-Evans, Amanda, Haffke, Matthias, Gommermann, Nina

المصدر: Journal of Medicinal Chemistry; 9/10/2020, Vol. 63 Issue 17, p9856-9875, 20p

المؤلفون: Pillong, Max, Marx, Corinne, Piechon, Philippe, Wicker, Jerome GP, Cooper, Richard I, Wagner, Beatrix

Relation: Pillong, Max, Marx, Corinne, Piechon, Philippe, Wicker, Jerome GP, Cooper, Richard I and Wagner, Beatrix (2017) A publicly available crystallisation data set and its application in machine learning. CrystEngComm, 19 (27). pp. 3737-3745.

الاتاحة: https://oak.novartis.com/32776/
http://pubs.rsc.org/en/content/articlelanding/2017/ce/c7ce00738h#!divAbstract
https://doi.org/10.1039/c7ce00738h

المؤلفون: Fouche, Marianne, Roth, Hans-Joerg, Schaefer, Michael, Berghausen, Joerg, Desrayaud, Sandrine, Blatter, Markus, Piechon, Philippe, Dix, Ina, Martin Garcia, Aimar

Relation: Fouche, Marianne, Roth, Hans-Joerg, Schaefer, Michael, Berghausen, Joerg, Desrayaud, Sandrine, Blatter, Markus, Piechon, Philippe, Dix, Ina and Martin Garcia, Aimar (2016) Design and Development of a Cyclic Decapeptide Scaffold with Suitable Properties for Bioavailability and Oral Exposure. ChemMedChem.

الاتاحة: https://oak.novartis.com/28435/

المؤلفون: Gu, Xingxian, Zhao, Jibin, Chen, Like, Li, Yunzhong, Yu, Bo, Tian, Xiangguang, Min, Zhongcheng, Xu, Su, Gu, Huijuan, Sun, Junjie, Lu, Xiaoquan, Chang, Meng, Wang, Xufan, Zhao, Liqun, Ye, Shengqing, Yang, Hongwei, Tian, Yingtao, Gao, Feng, Gai, Yu, Jia, Guanghua, Wu, Jingjing, Wang, Yan, Zhang, Jianghua, Zhang, Xuesong, Liu, Weichun, Gu, Xin, Luo, Xi, Dong, Hai, Wang, Huaimin, Schenkel, Berthold, Venturoni, Francesco, Filipponi, Paolo, Guelat, Bertrand, Allmendinger, Thomas, Wietfeld, Bernhard, Hoehn, Pascale, Kovacic, Nikola, Hermann, Luca, Schlama, Thierry, Ruch, Thomas, Derrien, Nadine, Piechon, Philippe, Kleinbeck, Florian

المصدر: The Journal of Organic Chemistry; June 2020, Vol. 85 Issue: 11 p6844-6853, 10p

المؤلفون: Kayser, Hartmut, Eilinger, Philipp, Piechon, Philippe, Wagner, Trixie

المصدر: Archives of Biochemistry and Biophysics ; volume 513, issue 1, page 27-35 ; ISSN 0003-9861

الاتاحة: http://dx.doi.org/10.1016/j.abb.2011.06.011
https://api.elsevier.com/content/article/PII:S0003986111002463?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0003986111002463?httpAccept=text/plain