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1
المؤلفون: Stephanie L. Coffing, Victor F. Soliman, Evan Smith, Richard V. Coelho, Jiri Aubrecht, Klaas Schildknegt, Jennifer R. Cheung, Mary E. Lame, Tristan S. Maurer, Phoebe Chiang, Deepak Dalvie, Chandra Vage, Amit S. Kalgutkar, Kim F. McClure
المصدر: Drug Metabolism and Disposition. 35:848-858
مصطلحات موضوعية: Salmonella typhimurium, Pharmacology, Mutagenicity Tests, Stereochemistry, Metabolite, Cyanide, Pharmaceutical Science, Glutathione, medicine.disease_cause, Piperazines, Ames test, Hydroxylation, chemistry.chemical_compound, Piperazine, chemistry, Pyrazines, medicine, Amine gas treating, Obesity, Biotransformation, Serotonin 5-HT2 Receptor Agonists, Genotoxicity
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2
المؤلفون: Swick Andrew Gordon, Judith A. Siuciak, Janice A. Brown, Ravi B. Marala, Terrell A. Patterson, Victor Guanowsky, Phoebe Chiang, Patricia A. Seymour, Sheryl A. McCarthy, Douglas S. Chapin, Philip A. Iredale
المصدر: Neuropharmacology. 52:279-290
مصطلحات موضوعية: Male, Agonist, Dextroamphetamine, medicine.drug_class, medicine.medical_treatment, Hyperkinesis, Motor Activity, Pharmacology, Catalepsy, Piperazines, Mice, Cellular and Molecular Neuroscience, Helplessness, Learned, Extrapyramidal symptoms, Avoidance Learning, Receptor, Serotonin, 5-HT2C, medicine, Animals, Humans, Rats, Wistar, Antipsychotic, Amphetamine, Prepulse inhibition, Behavior, Animal, Dose-Response Relationship, Drug, Amphetamines, medicine.disease, Receptor antagonist, Rats, Serotonin Receptor Agonists, Apomorphine, Disease Models, Animal, Inhibition, Psychological, Psychotic Disorders, Pyrazines, Exploratory Behavior, NIH 3T3 Cells, medicine.symptom, Psychology, Serotonin 5-HT2 Receptor Agonists, Antipsychotic Agents, Protein Binding, medicine.drug
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3
المؤلفون: Paul DaSilva-Jardine, Josephine Spitzer, Michele H. Rosner, Samuel P. Simons, Diane M. Hargrove, Boris A. Chrunyk, Richard F. Hank, Phoebe Chiang, Ernest S. Paight, Swick Andrew Gordon, Robert L. Dow, Peter Cornelius, Gayle K. Schulte, Tate Bonnie Frances, Steven R. Schneider, Terrell A. Patterson, William P. Newsome, Jayvardhan Pandit, Mark Ammirati, Eunsun Lee, Dennis E. Danley, Peter K. LeMotte
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:379-382
مصطلحات موضوعية: Models, Molecular, Thyroid Hormones, Protein Conformation, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Crystallography, X-Ray, Ligands, Biochemistry, Structure-Activity Relationship, Drug Discovery, Humans, Moiety, Uracil, Receptor, Molecular Biology, Receptors, Thyroid Hormone, Thyroid hormone receptor, Chemistry, Molecular Mimicry, Organic Chemistry, Subtype selective, Drug Design, Molecular Medicine, Indicators and Reagents, Protein Binding
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4
المؤلفون: Ravi B. Marala, Stephanie Santucci, Kevin K.-C. Liu, Eunsun Lee, Wendy Werner, Craig Giragossian, Peter Cornelius, Jimmy Kong, Hou Chen, Janice A. Brown, Yuan Zeng, Steven B. Coffey, Phoebe Chiang, Mark A. Dombroski, Terrell A. Patterson, Colleen P. Gibbons, Zane Wenzel, Elizabeth Tomlinson, Bruce Allen Lefker
المصدر: Bioorganicmedicinal chemistry letters. 20(7)
مصطلحات موضوعية: Food intake, Proline, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Pharmacology, Biochemistry, Eating, Structure-Activity Relationship, Dogs, Drug Discovery, Receptor, Serotonin, 5-HT2C, Animals, Humans, Obesity, Receptor, Molecular Biology, Binding selectivity, Chemistry, Organic Chemistry, Brain, Highly selective, Amides, Rats, Orally active, Drug development, Molecular Medicine, Serotonin, Anti-Obesity Agents, Serotonin 5-HT2 Receptor Agonists