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1Academic Journal
المؤلفون: Frederik F. D. Daeyaert, H. Maarten Vinkers, Marc R. De Jonge, Jan Heeres, M. H. Koymans, Paul J. Lewi, Paul A. J. Janssen
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.84.2580; http://biochempress.com/Files/IECMD_2003/IECMD_2003_037.pdf
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المؤلفون: Muthusamy Venkatraj, Pieter Van der Veken, Jan Heeres, Guy Caljon, Koen Augustyns, Jurgen Joossens, Louis Maes, Paul J. Lewi, Irene G. Salado
المصدر: European journal of medicinal chemistry
مصطلحات موضوعية: 0301 basic medicine, Male, Trypanosoma brucei rhodesiense, Cell Survival, Phenotypic screening, Trypanosoma cruzi, Trypanosoma brucei brucei, Antiprotozoal Agents, Pharmacology, Trypanosoma brucei, 01 natural sciences, 03 medical and health sciences, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Usually fatal, Drug Discovery, medicine, Animals, Humans, African trypanosomiasis, Leishmania infantum, Biology, Triazine, Cell Proliferation, biology, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Triazines, Pharmacology. Therapy, Organic Chemistry, Tsetse fly, General Medicine, Fibroblasts, medicine.disease, biology.organism_classification, Reverse transcriptase, 3. Good health, 0104 chemical sciences, 030104 developmental biology, chemistry, Reverse Transcriptase Inhibitors, Human medicine, Glossina
, Dimerization وصف الملف: pdf
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3
المؤلفون: Pieter Van der Veken, Kevin K. Ariën, Koen Augustyns, Guido Vanham, Paul Cos, Bertrand Dirié, Jan Heeres, Paul J. Lewi, Muthusamy Venkatraj, Johan Michiels, Louis Maes, Jurgen Joossens, Sophie Lyssens
المصدر: Bioorganic and medicinal chemistry
مصطلحات موضوعية: Trypanosoma brucei rhodesiense, Pyrimidine, Anti-HIV Agents, Cell Survival, Trypanosoma brucei brucei, Clinical Biochemistry, Pharmaceutical Science, Microbial Sensitivity Tests, Biochemistry, Cell Line, Nucleoside Reverse Transcriptase Inhibitor, Structure-Activity Relationship, chemistry.chemical_compound, Parasitic Sensitivity Tests, In vivo, Drug Discovery, Humans, Structure–activity relationship, Biology, Molecular Biology, Triazine, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Pharmacology. Therapy, Organic Chemistry, Trypanocidal Agents, HIV Reverse Transcriptase, In vitro, Reverse transcriptase, 3. Good health, HIV-1, Reverse Transcriptase Inhibitors, Molecular Medicine, Nucleoside
وصف الملف: pdf
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المؤلفون: Frans Awouters, Paul J. Lewi
المصدر: Arzneimittelforschung. 57:625-632
مصطلحات موضوعية: medicine.medical_specialty, medicine.drug_class, Atypical antipsychotic, History, 21st Century, Structure-Activity Relationship, Pimozide, Paliperidone Palmitate, Drug Discovery, medicine, Haloperidol, Humans, Paliperidone, Psychiatry, Fluspirilene, Risperidone, business.industry, Isoxazoles, Dopamine receptor binding, History, 20th Century, Pyrimidines, Psychotic Disorders, business, Antipsychotic Agents, medicine.drug
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5
المؤلفون: Kalyan Das, Stephen H. Hughes, Joseph D. Bauman, Eddy Arnold, Aaron J. Shatkin, Arthur D. Clark, Yulia Volovik Frenkel, Paul J. Lewi
المصدر: Proceedings of the National Academy of Sciences. 105:1466-1471
مصطلحات موضوعية: Anti-HIV Agents, Protein Conformation, Stereochemistry, Amino Acid Motifs, Molecular Sequence Data, Mutant, Crystallography, X-Ray, Protein Engineering, chemistry.chemical_compound, Protein structure, Drug Resistance, Viral, Nitriles, Hydrolase, medicine, Humans, Amino Acid Sequence, Enzyme Inhibitors, Polymerase, Diarylpyrimidines, Multidisciplinary, biology, Reverse-transcriptase inhibitor, Rilpivirine, virus diseases, Protein engineering, Biological Sciences, HIV Reverse Transcriptase, Reverse transcriptase, Pyrimidines, chemistry, Drug Design, Mutation, biology.protein, Reverse Transcriptase Inhibitors, medicine.drug
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المؤلفون: Manuel Morrens, Wouter Hulstijn, Paul J. Lewi, Bernard Sabbe
المصدر: Psychiatry research
Psychiatry Research, 161, 1, pp. 121-125
Psychiatry Research, 161, 121-125مصطلحات موضوعية: Adult, Male, Nosology, medicine.medical_specialty, Psychosis, Catatonia, Neuropsychological Tests, behavioral disciplines and activities, Diagnosis, Differential, Discrimination Learning, Reaction Time, medicine, Humans, Psychiatry, Biological Psychiatry, Psychomotor learning, Schizophrenia, Catatonic, Action, intention, and motor control, Perception, Action and Control [DI-BCB_DCC_Theme 2], Cognition, medicine.disease, Psychiatry and Mental health, Stereotypy (non-human), Pattern Recognition, Visual, Schizophrenia, Female, Human medicine, Psychomotor Disorders, Stereotyped Behavior, Cognition Disorders, Psychomotor disorder, Psychology, Psychomotor Performance, psychological phenomena and processes, Antipsychotic Agents, Clinical psychology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9ae79b68d43f695ec6b2b9f215deb5a8
https://doi.org/10.1016/j .psychres.2008.01.017 -
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المؤلفون: Johan Michiels, Sergey Sergeyev, Paul J. Lewi, Philippe Franck, Guido Vanham, Jan Heeres, Kevin K. Ariën, Christophe M. L. Vande Velde, Ashok K. Yadav, Bert U. W. Maes, Hans De Winter
المصدر: Journal of medicinal chemistry
مصطلحات موضوعية: 0301 basic medicine, Pyrimidine, Anti-HIV Agents, Pyridines, Stereochemistry, Mutant, Human immunodeficiency virus (HIV), Nanotechnology, Microbial Sensitivity Tests, medicine.disease_cause, 01 natural sciences, Cell Line, Nucleoside Reverse Transcriptase Inhibitor, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Moiety, Structure–activity relationship, Aniline Compounds, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Chemistry, Pharmacology. Therapy, HIV Reverse Transcriptase, Reverse transcriptase, In vitro, 0104 chemical sciences, Fluorobenzenes, 030104 developmental biology, HIV-1, Reverse Transcriptase Inhibitors, Molecular Medicine
وصف الملف: pdf
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المؤلفون: Paul J. Lewi, Johanna Smeyers-Verbeke
المساهمون: Analytical Chemistry and Pharmaceutical Technology
المصدر: Journal of Chemometrics. 21:252-256
مصطلحات موضوعية: Work (electrical), Operations research, Computer science, Applied Mathematics, Perspective (graphical), Engineering ethics, Prof. D.L.Massart, Analytical Chemistry
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المؤلفون: Manuel Morrens, Wouter Hulstijn, Paul J. Lewi, Marc De Hert, Bernard Sabbe
المصدر: Schizophrenia Research, 84, 2/3, pp. 397-404
Schizophrenia research
Schizophrenia Research, 84, 397-404مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, Perseveration, Stereotypic Movement Disorder, Neuropsychological Tests, Audiology, Severity of Illness Index, Developmental psychology, Wisconsin Card Sorting Test, medicine, Humans, Biological Psychiatry, California Verbal Learning Test, Action, intention, and motor control, Neuropsychology, Cognition, medicine.disease, Diagnostic and Statistical Manual of Mental Disorders, Stereotypic movement disorder, Psychiatry and Mental health, Stereotypy (non-human), Cognitive inhibition, Schizophrenia, Female, medicine.symptom, Cognition Disorders, Psychology
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::61981e3b1c5879b838d4f53ffcf551e8
https://doi.org/10.1016/j .schres.2006.01.024 -
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المؤلفون: Paul J. Lewi, Eddy Arnold, Stephen H. Hughes, Kalyan Das
المصدر: Progress in Biophysics and Molecular Biology. 88:209-231
مصطلحات موضوعية: Gene Expression Regulation, Viral, Drug, Molecular model, Anti-HIV Agents, Protein Conformation, Stereochemistry, media_common.quotation_subject, Dapivirine, Biophysics, Etravirine, Biology, Structure-Activity Relationship, chemistry.chemical_compound, Drug Delivery Systems, Drug Resistance, Multiple, Viral, medicine, Animals, Humans, Molecular Biology, media_common, Diarylpyrimidines, Flexibility (engineering), Acquired Immunodeficiency Syndrome, Crystallography, Genetic Variation, virus diseases, Adaptation, Physiological, HIV Reverse Transcriptase, Reverse transcriptase, chemistry, Drug Design, HIV-1, Reverse Transcriptase Inhibitors, Nucleoside, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6cc84498852bfc0bc6296de615be12bd
https://doi.org/10.1016/j .pbiomolbio.2004.07.001 -
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المؤلفون: Paul J. Lewi
المصدر: Journal of Chemometrics. 19:282-287
مصطلحات موضوعية: Scientific enterprise, Engineering, business.industry, Applied Mathematics, media_common.quotation_subject, Perspective (graphical), Foundation (evidence), Case description, Genius, Analytical Chemistry, Statistics, Charisma, business, media_common
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المؤلفون: Paul J. Lewi
المصدر: Chemometrics and Intelligent Laboratory Systems. 77:215-223
مصطلحات موضوعية: Multivariate analysis, Biplot, Process Chemistry and Technology, Bivariate analysis, computer.software_genre, Column (database), Computer Science Applications, Analytical Chemistry, Weighting, Factorization, Statistics, Leverage (statistics), Data mining, Raw data, computer, Spectroscopy, Software, Mathematics
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4d4ca388e384edc8a4580f8080709bcd
https://doi.org/10.1016/j .chemolab.2004.07.010 -
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المؤلفون: Eddy Arnold, Kalyan Das, Yulia Volovik Frenkel, Paul A. J. Janssen,⊥,† and, Arthur D. Clark, Paul J. Lewi, Yuh-Hwa Wang
المصدر: Journal of Medicinal Chemistry. 48:1974-1983
مصطلحات موضوعية: Absorption (pharmacology), Chemical Phenomena, Light, Administration, Oral, Biological Availability, Concentration effect, Models, Biological, Absorption, Microscopy, Electron, Transmission, Dynamic light scattering, Drug Discovery, Animals, Humans, Scattering, Radiation, Molecule, Organic chemistry, Aqueous solution, Chemistry, Physical, Triazines, Chemistry, Hydrogen-Ion Concentration, Rats, Bioavailability, Gastrointestinal Tract, Solutions, Pyrimidines, Lipophilicity, Biophysics, Reverse Transcriptase Inhibitors, Molecular Medicine, Particle size, Hydrophobic and Hydrophilic Interactions, Half-Life
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المؤلفون: Harr F Njai, Paul J Lewi, Cornelus GM Janssen, Sergio Garcia, Katrien Fransen, Luc Kestens, Guido Vanham, Paul AJ Janssen
المصدر: Antiviral Therapy. 10:255-262
مصطلحات موضوعية: Pharmacology, Infectious Diseases, virus diseases, Pharmacology (medical)
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المؤلفون: Lucien Maria Henricus Koymans, Frits Daeyaert, Paul Adriaan Jan Janssen, Vinkers Hm, de Jonge Mr, Paul J. Lewi, Jan Heeres
المصدر: Journal of Medicinal Chemistry. 48:2176-2183
مصطلحات موضوعية: Models, Molecular, Molecular model, Anti-HIV Agents, Molecular Conformation, Human immunodeficiency virus (HIV), Quantitative Structure-Activity Relationship, Computational biology, medicine.disease_cause, Approximation error, Drug Discovery, medicine, Databases, Protein, chemistry.chemical_classification, Binding Sites, Molecular Structure, biology, Reverse-transcriptase inhibitor, Interaction energy, HIV Reverse Transcriptase, Reverse transcriptase, Enzyme, chemistry, Biochemistry, Enzyme inhibitor, biology.protein, Reverse Transcriptase Inhibitors, Molecular Medicine, medicine.drug
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المؤلفون: Paul L. Boyer, H. Maarten Vinkers, Robert W. Kavash, Marie Pierre de Béthune, Eddy Arnold, Patrick K. Clark, Jan Heeres, Donald William Ludovici, Paul A. J. Janssen, Lucien Maria Henricus Koymans, Michael J. Kukla, Koen Andries, Mark A. Lichtenstein, Rudi Pauwels, Paul J. Lewi, Bart De Corte, Chih Y. Ho, Hong Ye, Marc René De Jonge, Kalyan Das, Arthur D. Clark, Frederik Frans Desire Daeyaert, Stephen H. Hughes
المصدر: Journal of medicinal chemistry
مصطلحات موضوعية: Models, Molecular, Anti-HIV Agents, Protein Conformation, Stereochemistry, Etravirine, Crystallography, X-Ray, Nucleoside Reverse Transcriptase Inhibitor, chemistry.chemical_compound, Protein structure, Drug Resistance, Viral, Nitriles, Drug Discovery, medicine, Diarylpyrimidines, Reverse-transcriptase inhibitor, biology, Chemistry, Wild type, HIV Reverse Transcriptase, Pyridazines, Discovery and development of non-nucleoside reverse-transcriptase inhibitors, Pyrimidines, Enzyme inhibitor, Mutation, biology.protein, Reverse Transcriptase Inhibitors, Molecular Medicine, medicine.drug
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المؤلفون: Marc René De Jonge, Paul J. Lewi, Yulia Volovik, Luc Koymans, Marie Pierre de Béthune, Walter Van den Broeck, Frits Daeyaert, Frédéric Vanhoutte, Jan Heeres, Paul A. J. Janssen, Maarten Vinkers, Jef Peeters, Herman Borghys, Kaylan Das, Hilde Bohets, Edward Arnold, Koen Andries, Jos Leempoels, Arthur D. Clark, Gerben Albert Eleutherius Van 'T Klooster, Philip Timmerman
المساهمون: Analytical Chemistry and Pharmaceutical Technology
المصدر: Drugs in R & D. 5:245-257
مصطلحات موضوعية: Models, Molecular, Anti-HIV Agents, Anti-HIV Agents/chemistry, Biological Availability, Pharmacology, Polar surface area, Nucleoside Reverse Transcriptase Inhibitor, Structure-Activity Relationship, Dogs, Pharmacokinetics, In vivo, Sasa, Animals, Humans, biology, Triazines, Chemistry, biology.organism_classification, Rats, Bioavailability, Pyrimidines, HIV-1/drug effects, Intestinal Absorption, Area Under Curve, Anti-HIV Agents/pharmacokinetics, Lipophilicity, HIV-1, Reverse Transcriptase Inhibitors, Lymph, Caco-2 Cells, Drug metabolism
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المؤلفون: Jan Heeres, Marc René De Jonge, Frits Daeyaert, Maarten Vinkers, Luc Koymans, Paul Adriaan Jan Janssen, Paul J. Lewi
المصدر: Proteins: Structure, Function, and Bioinformatics. 54:526-533
مصطلحات موضوعية: Lead Finder, Chemistry, Biochemistry, Combinatorial chemistry, Protein structure, Protein–ligand docking, Structural Biology, Docking (molecular), Searching the conformational space for docking, Target protein, Binding site, Pharmacophore, Molecular Biology, Algorithm
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المؤلفون: Marc René De Jonge, Henk Timmerman, Lucien Maria Henricus Koymans, Frederik Frans Desire Daeyaert, Koen Jeanne Alfons Van Aken, Paul J. Lewi, Joop H. van Lenthe, Jan Heeres, Paul A. J. Janssen, H. Maarten Vinkers
المصدر: Journal of Medicinal Chemistry. 46:2765-2773
مصطلحات موضوعية: Quantitative structure–activity relationship, Fitness function, Databases, Factual, Molecular Structure, Molecular model, Combinatorial Chemistry Techniques, Anti-HIV Agents, Stereochemistry, Quantitative Structure-Activity Relationship, Moment (mathematics), chemistry.chemical_compound, Electric dipole moment, Dipole, Pharmaceutical Preparations, chemistry, Drug Design, Drug Discovery, Reverse Transcriptase Inhibitors, Molecular Medicine, Organic synthesis, Biological system, Software
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المؤلفون: Bart De Corte, Hong Ye, Chih Y. Ho, Donald William Ludovici, Marc René De Jonge, Hilde Azijn, Paul J. Lewi, Michael J. Kukla, Paul Adriaan Jan Janssen, Mark A. Lichtenstein, Lucien Maria Henricus Koymans, Koen Jeanne Alfons Van Aken, Edward Arnold, Rudi Pauwels, Marie Pierre de Béthune, Frederik Frans Desire Daeyaert, Robert W. Kavash, Koen Andries, Jan Heeres, Kalyan Das
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:2235-2239
مصطلحات موضوعية: Anti-HIV Agents, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Human immunodeficiency virus (HIV), Pharmaceutical Science, medicine.disease_cause, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Nitriles, Drug Discovery, medicine, Anti-hiv drugs, Inhibitory concentration 50, Structure–activity relationship, Molecular Biology, Diarylpyrimidines, biology, Chemistry, Organic Chemistry, virus diseases, biology.organism_classification, Virology, HIV Reverse Transcriptase, Reverse transcriptase, Pyrimidines, Mutation, Lentivirus, HIV-1, Reverse Transcriptase Inhibitors, Molecular Medicine