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1Academic Journal
المؤلفون: Morteza Abdoli, Alessandro Bonardi, Paola Gratteri, Claudiu T. Supuran, Raivis Žalubovskis
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 39, Iss 1 (2024)
مصطلحات موضوعية: Carbonic anhydrase, inhibitors, hydantoins, phthalimides, docking studies, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2Academic Journal
المؤلفون: Alessio Nocentini, Anna Di Porzio, Alessandro Bonardi, Carla Bazzicalupi, Andrea Petreni, Tarita Biver, Silvia Bua, Simona Marzano, Jussara Amato, Bruno Pagano, Nunzia Iaccarino, Stefano De Tito, Stefano Amente, Claudiu T. Supuran, Antonio Randazzo, Paola Gratteri
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 39, Iss 1 (2024)
مصطلحات موضوعية: G-Quadruplex, carbonic anhydrase, multitarget-directed ligands, tumours, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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3Academic JournalDiscovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors
المؤلفون: Simone Giovannuzzi, Alessandro Bonardi, Paola Gratteri, Alessio Nocentini, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)
مصطلحات موضوعية: Drug design, metalloenzyme, inhibition, click chemistry, hCA III, molecular dynamics, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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4Academic Journal
المؤلفون: Nora Astrain-Redin, Niccolò Paoletti, Daniel Plano, Alessandro Bonardi, Paola Gratteri, Andrea Angeli, Carmen Sanmartin, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)
مصطلحات موضوعية: Selenium, carbonic anhydrase, inhibitors, NSAIDs, tumours, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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5Academic Journal
المؤلفون: Waleed A. Badawi, Mahmoud Rashed, Alessio Nocentini, Alessandro Bonardi, Mohammad M. Abd-Alhaseeb, Sara T. Al-Rashood, Giri Babu Veerakanellore, Taghreed A. Majrashi, Eslam B. Elkaeed, Bahaa Elgendy, Paola Gratteri, Claudiu T. Supuran, Wagdy M. Eldehna, Mohamed Elagawany
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)
مصطلحات موضوعية: Analgesic, Synthesis, Pyridazinone, Sulphonates, Molecular modelling, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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6Academic Journal
المؤلفون: Alessandro Bonardi, Silvia Bua, Jacob Combs, Carrie Lomelino, Jacob Andring, Sameh Mohamed Osman, Alessandra Toti, Lorenzo Di Cesare Mannelli, Paola Gratteri, Carla Ghelardini, Robert McKenna, Alessio Nocentini, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 930-939 (2022)
مصطلحات موضوعية: Tail approach, carbonic anhydrase, inhibitor, X-ray crystallography, hypoxic tumour, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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7Academic Journal
المؤلفون: Alessio Nocentini, Alessandro Bonardi, Simone Pratesi, Paola Gratteri, Carlo Dani, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 37, Iss 1, Pp 487-501 (2022)
مصطلحات موضوعية: bilirubin, hyperbilirubinaemia, jaundice, antioxidant, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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8Academic Journal
المؤلفون: Alessandro Bonardi, Alessio Nocentini, Sameh Mohamed Osman, Fatmah Ali Alasmary, Tahani Mazyad Almutairi, Dalal Saied Abdullah, Paola Gratteri, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 36, Iss 1, Pp 469-479 (2021)
مصطلحات موضوعية: resistance, virulence, metalloenzyme, inhibition, md, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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9Academic Journal
المؤلفون: Morteza Abdoli, Alessandro Bonardi, Niccolò Paoletti, Ashok Aspatwar, Seppo Parkkila, Paola Gratteri, Claudiu T. Supuran, Raivis Žalubovskis
المصدر: Molecules, Vol 28, Iss 10, p 4020 (2023)
مصطلحات موضوعية: carbonic anhydrase, inhibitors, sulfonamides, bacterial enzymes, Mycobacterium tuberculosis, in silico studies, Organic chemistry, QD241-441
وصف الملف: electronic resource
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10Academic Journal
المؤلفون: Davide Ialongo, Antonella Messore, Valentina Noemi Madia, Valeria Tudino, Alessio Nocentini, Paola Gratteri, Simone Giovannuzzi, Claudiu T. Supuran, Alice Nicolai, Susanna Scarpa, Samanta Taurone, Michele Camarda, Marco Artico, Veronica Papa, Francesco Saccoliti, Luigi Scipione, Roberto Di Santo, Roberta Costi
المصدر: Pharmaceuticals, Vol 16, Iss 2, p 188 (2023)
مصطلحات موضوعية: metalloenzyme, carbonic anhydrase, diketo acids, carbonic anhydrase inhibitors, breast cancer, tongue squamous cell carcinoma, Medicine, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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11Academic Journal
المؤلفون: Paolo Guglielmi, Giulia Rotondi, Daniela Secci, Andrea Angeli, Paola Chimenti, Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Simone Carradori, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 1891-1905 (2020)
مصطلحات موضوعية: saccharin, acesulfame, triazole, docking, carbonic anhydrase inhibitors, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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12Academic JournalThe antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors
المؤلفون: Aleksandrs Pustenko, Alessio Nocentini, Paola Gratteri, Alessandro Bonardi, Igor Vozny, Raivis Žalubovskis, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 1011-1020 (2020)
مصطلحات موضوعية: carbonic anhydrase inhibitors, molecular dynamics, furagin, hydantoin, synthesis, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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13Academic Journal
المؤلفون: Alessio Nocentini, Sameh M. Osman, Igor A. Rodrigues, Veronica S. Cardoso, Fatmah Ali S. Alasmary, Zeid AlOthman, Alane B. Vermelho, Paola Gratteri, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 34, Iss 1, Pp 1164-1171 (2019)
مصطلحات موضوعية: carbonic anhydrase, chagas disease, leishmania, trypanosoma, nitroaromatics, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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14Academic Journal
المؤلفون: Alessio Nocentini, Alessandro Bonardi, Paola Gratteri, Bruno Cerra, Antimo Gioiello, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 33, Iss 1, Pp 1453-1459 (2018)
مصطلحات موضوعية: Carbonic anhydrase, inhibitor, steroids, phenol, bile acid, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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15Academic Journal
المؤلفون: Alessio Nocentini, Daniela Vullo, Sonia Del Prete, Sameh M. Osman, Fatmah A.S. Alasmary, Zeid AlOthman, Clemente Capasso, Fabrizio Carta, Paola Gratteri, Claudiu T. Supuran
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 32, Iss 1, Pp 1064-1070 (2017)
مصطلحات موضوعية: Carbonic anhydrase, β-CA-class enzyme, monothiocarbamate, inhibitor, Malassezia globosa, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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16Academic Journal
المؤلفون: Matteo Savastano, Matteo Fiaschi, Giovanni Ferraro, Paola Gratteri, Palma Mariani, Antonio Bianchi, Carla Bazzicalupi
المصدر: Molecules, Vol 25, Iss 6, p 1355 (2020)
مصطلحات موضوعية: chemosensor, zinc, fluorescence, scorpiand, azamacrocycles, anion binding, supramolecular interactions, Organic chemistry, QD241-441
وصف الملف: electronic resource
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17Academic Journal
المؤلفون: Matteo Savastano, Celeste García-Gallarín, Claudia Giorgi, Paola Gratteri, Maria Dolores López de la Torre, Carla Bazzicalupi, Antonio Bianchi, Manuel Melguizo
المصدر: Molecules, Vol 24, Iss 12, p 2247 (2019)
مصطلحات موضوعية: s-tetrazines, anion complexes, anion–π interactions, lone pair–π interactions, H bonding, supramolecular forces, crystal structures, stability constants, complexation enthalpy, Organic chemistry, QD241-441
وصف الملف: electronic resource
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18Academic Journal
المؤلفون: Matteo Savastano, Carla Bazzicalupi, Giovanni Ferraro, Emiliano Fratini, Paola Gratteri, Antonio Bianchi
المصدر: Molecules, Vol 24, Iss 11, p 2098 (2019)
مصطلحات موضوعية: desferrioxamine, zirconium, chelates, molecular modelling, stability constants, Organic chemistry, QD241-441
وصف الملف: electronic resource
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19Academic Journal
المؤلفون: Luca Guandalini, Elisabetta Martini, Paola Gratteri, Carla Ghelardini, Katia Varani, Maria Novella Romanelli
المصدر: ARKIVOC, Vol 2006, Iss 8, Pp 50-65 (2006)
مصطلحات موضوعية: Organic chemistry, QD241-441
وصف الملف: electronic resource
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20Academic Journal
المؤلفون: Simone Giovannuzzi, Daniel Chavarria, Gustavo Provensi, Manuela Leri, Monica Bucciantini, Simone Carradori, Alessandro Bonardi, Paola Gratteri, Fernanda Borges, Alessio Nocentini, Claudiu T. Supuran
مصطلحات موضوعية: Biochemistry, Medicine, Cell Biology, Neuroscience, Pharmacology, Biological Sciences not elsewhere classified, Chemical Sciences not elsewhere classified, reactive oxygen species, predict admet properties, lead optimization led, cholinergic system disruption, brain carbonic anhydrases, 7 – 32, 1 – 90, classical ca inhibitors, induced neuronal toxicity, methazolamide prevent amyloid, amyloid plaque formation, first dual inhibitors, reverted ros formation, highly effective cais, 6 nm ), 50 sub, dual inhibitors, related toxicity, k <, sub, target drugs, significant set, ros production