نتائج البحث - "Nimje, Roshan Y."

1

Academic Journal

Mass spectrometric‐based investigation of differentially protected azatryptophan derivatives using Orbitrap mass spectrometry: Differentiation of positional isomers under protonation and alkali‐cationization conditions

المؤلفون: Gajjela, Raju, Kandula, Ravikanth Reddy, Kuppusamy, Prakasam, Nimje, Roshan Y., Gupta, Anuradha, Bagadi, Muralidhararao, Mathur, Arvind

المساهمون: Bristol-Myers Squibb Canada

المصدر: Rapid Communications in Mass Spectrometry ; volume 36, issue 5 ; ISSN 0951-4198 1097-0231

الاتاحة: http://dx.doi.org/10.1002/rcm.9239
https://onlinelibrary.wiley.com/doi/pdf/10.1002/rcm.9239
https://onlinelibrary.wiley.com/doi/full-xml/10.1002/rcm.9239

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2

Academic Journal

Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 Inhibitors

المؤلفون: Cherney, Emily C., Zhang, Liping, Guo, Weiwei, Huang, Audris, Williams, David, Seitz, Steven, Shan, Weifang, Zhu, Xiao, Gullo-Brown, Johnni, Maley, Derrick, Lin, Tai-an, Hunt, John T., Huang, Christine, Yang, Zheng, D’Arienzo, Celia J., Discenza, Lorell N., Ranasinghe, Asoka, Grubb, Mary F., Traeger, Sarah C., Li, Xin, Johnston, Kathy A., Kopcho, Lisa, Fereshteh, Mark, Foster, Kimberly A., Stefanski, Kevin, Delpy, Diane, Dhar, Gopal, Anandam, Aravind, Mahankali, Sandeep, Padmanabhan, Shweta, Rajanna, Prabhakar, Murali, Venkata, Mariappan, T. Thanga, Pattasseri, Shabeerali, Nimje, Roshan Y., Hong, Zhenqiu, Kempson, James, Rampulla, Richard, Mathur, Arvind, Gupta, Anuradha, Borzilleri, Robert, Vite, Gregory, Balog, Aaron

المصدر: ACS Medicinal Chemistry Letters ; volume 12, issue 7, page 1143-1150 ; ISSN 1948-5875 1948-5875

الاتاحة: http://dx.doi.org/10.1021/acsmedchemlett.1c00236
https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00236

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3

Academic Journal

Development of a Stereoselective and Scalable Synthesis for the Potent Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor, BMT-297376; N-(( R)-1-((cis)-4-(3-(Difluoromethyl)-2-methoxypyridin-4-yl)cyclohexyl)propyl)-6-methoxynicotinamide

المؤلفون: Nimje, Roshan Y., Kuppusamy, Prakasam, Krishnamoorthy, Suresh, Shanmugam, Yoganand, Ramasamy, Duraisamy, Manoharan, Haridhas, Arunachalam, Pirama Nayagam, Balog, Aaron, Cherney, Emily C., Zhang, Liping, Borzilleri, Robert M., Hong, Zhenqiu, Kempson, James, Rampulla, Richard R., Mathur, Arvind, Gupta, Anuradha

المصدر: Organic Process Research & Development ; volume 25, issue 7, page 1680-1689 ; ISSN 1083-6160 1520-586X

الاتاحة: http://dx.doi.org/10.1021/acs.oprd.1c00142
https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.1c00142

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4

Academic Journal

Practical Synthesis of (3a R, 9b R)-8-Fluoro-7-(perfluoropropan-2-yl)-9b-(phenylsulfonyl)-2,3,3a,4,5,9b-hexahydro-1 H-benzo[e]indole: An Advanced Intermediate to Access the RORγt Inverse Agonist BMT-362265

المؤلفون: Karmakar, Ananta, Nimje, Roshan Y., Silamkoti, Arundutt, Pitchai, Manivel, Basha, Mushkin, Singarayer, Christuraj, Ramasamy, Duraisamy, Babu, G. T. Venkatesh, Samikannu, Ramesh, Subramaniam, Srinath, Anjanappa, Prakash, Vetrichelvan, Muthalagu, Kumar, Hemantha, Dikundwar, Amol G., Gupta, Anuradha, Gupta, Arun Kumar, Rampulla, Richard, Dhar, T. G. Murali, Mathur, Arvind

المصدر: Organic Process Research & Development ; volume 25, issue 4, page 1001-1014 ; ISSN 1083-6160 1520-586X

الاتاحة: http://dx.doi.org/10.1021/acs.oprd.1c00019
https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.1c00019

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5

Academic Journal

Methyl-2,2-difluoro-2-(fluorosulfonyl) acetate (MDFA)/copper (I) iodide mediated and tetrabutylammonium iodide promoted trifluoromethylation of 1-aryl-4-iodo-1,2,3-triazoles

المؤلفون: Panja, Chiradeep, Puttaramu, Jayashankara Vaderapura, Chandran, Thirumurugan Kothandarama, Nimje, Roshan Y., Kumar, Hemantha, Gupta, Anuradha, Arunachalam, Pirama Nayagam, Corte, James R., Mathur, Arvind

المساهمون: Discovery Analytical Department, Biocon Bristol-Myers Squibb Research Centre

المصدر: Journal of Fluorine Chemistry ; volume 236, page 109516 ; ISSN 0022-1139

الاتاحة: http://dx.doi.org/10.1016/j.jfluchem.2020.109516
https://api.elsevier.com/content/article/PII:S0022113920300671?httpAccept=text/xml
https://api.elsevier.com/content/article/PII:S0022113920300671?httpAccept=text/plain

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6

Academic Journal

Synthesis of Differentially Protected Azatryptophan Analogs via Pd 2 (dba) 3 /XPhos Catalyzed Negishi Coupling of N-Ts Azaindole Halides with Zinc Derivative from Fmoc-Protected tert-Butyl ( R)-2-Amino-3-iodopropanoate

المؤلفون: Nimje, Roshan Y, Vytla, Devaiah, Kuppusamy, Prakasam, Velayuthaperumal, Rajeswari, Jarugu, Lokesh Babu, Reddy, China Anki, Chikkananjaiah, Nanjundaswamy Kanikahalli, Rampulla, Richard A., Cavallaro, Cullen L., Li, Jianqing, Mathur, Arvind, Gupta, Anuradha, Roy, Amrita

المصدر: The Journal of Organic Chemistry ; volume 85, issue 17, page 11519-11530 ; ISSN 0022-3263 1520-6904

الاتاحة: http://dx.doi.org/10.1021/acs.joc.0c00973
https://pubs.acs.org/doi/pdf/10.1021/acs.joc.0c00973

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7

Academic Journal

Development of a Scalable Synthesis for the Potent Kinase Inhibitor BMS-986236; 1-(5-(4-(3-Hydroxy-3-methylbutyl)-1 H-1,2,3-triazol-1-yl)-4-(isopropylamino)pyridin-2-yl)-1 H-pyrazolo[3,4-b]pyridine-5-carbonitrile

المصدر: Organic Process Research & Development ; volume 23, issue 5, page 912-918 ; ISSN 1083-6160 1520-586X

الاتاحة: http://dx.doi.org/10.1021/acs.oprd.9b00023
https://pubs.acs.org/doi/pdf/10.1021/acs.oprd.9b00023

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8

Academic Journal

Practical Synthesis of (3aR, 9bR)‑8-Fluoro-7-(perfluoropropan-2-yl)-9b-(phenylsulfonyl)-2,3,3a,4,5,9b-hexahydro‑1H‑benzo[e]indole: An Advanced Intermediate to Access the RORγt Inverse Agonist BMT-362265.

المؤلفون: Karmakar, Ananta, Nimje, Roshan Y., Silamkoti, Arundutt, Pitchai, Manivel, Basha, Mushkin, Singarayer, Christuraj, Ramasamy, Duraisamy, Babu, G. T. Venkatesh, Samikannu, Ramesh, Subramaniam, Srinath, Anjanappa, Prakash, Vetrichelvan, Muthalagu, Kumar, Hemantha, Dikundwar, Amol G., Gupta, Anuradha, Gupta, Arun Kumar, Rampulla, Richard, Dhar, T. G. Murali, Mathur, Arvind

المصدر: Organic Process Research & Development; 4/16/2021, Vol. 25 Issue 4, p1001-1014, 14p

9

Academic Journal

Synthesis of Differentially Protected Azatryptophan Analogs via Pd2(dba)3/XPhos Catalyzed Negishi Coupling of N‑Ts Azaindole Halides with Zinc Derivative from Fmoc-Protected tert-Butyl (R)‑2-Amino-3-iodopropanoate.

المؤلفون: Nimje, Roshan Y, Vytla, Devaiah, Kuppusamy, Prakasam, Velayuthaperumal, Rajeswari, Jarugu, Lokesh Babu, Reddy, China Anki, Chikkananjaiah, Nanjundaswamy Kanikahalli, Rampulla, Richard A., Cavallaro, Cullen L., Li, Jianqing, Mathur, Arvind, Gupta, Anuradha, Roy, Amrita

المصدر: Journal of Organic Chemistry; 9/4/2020, Vol. 85 Issue 17, p11519-11530, 12p

10

Periodical

Synthesis of Differentially Protected Azatryptophan Analogs via Pd2(dba)3/XPhos Catalyzed Negishi Coupling of N-Ts Azaindole Halides with Zinc Derivative from Fmoc-Protected tert-Butyl (R)-2-Amino-3-iodopropanoate

المؤلفون: Nimje, Roshan Y, Vytla, Devaiah, Kuppusamy, Prakasam, Velayuthaperumal, Rajeswari, Jarugu, Lokesh Babu, Reddy, China Anki, Chikkananjaiah, Nanjundaswamy Kanikahalli, Rampulla, Richard A., Cavallaro, Cullen L., Li, Jianqing, Mathur, Arvind, Gupta, Anuradha, Roy, Amrita

المصدر: The Journal of Organic Chemistry; September 2020, Vol. 85 Issue: 17 p11519-11530, 12p

11

Academic Journal

Development of a Scalable Synthesis for the Potent Kinase Inhibitor BMS-986236; 1‑(5-(4-(3-Hydroxy-3-methylbutyl)‑1H‑1,2,3-triazol-1-yl)-4-(isopropylamino)pyridin-2-yl)‑1H‑pyrazolo[3,4‑b]pyridine-5-carbonitrile.

المصدر: Organic Process Research & Development; May2019, Vol. 23 Issue 5, p912-918, 7p

12

Academic Journal

ChemInform Abstract: A Three‐Component Palladium‐Catalyzed Oxidative C—C Coupling Reaction: A Domino Process in Two Dimensions.

المؤلفون: Nimje, Roshan Y., Leskinen, Mikko V., Pihko, Petri M.

المصدر: ChemInform ; volume 44, issue 38 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.201338118
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.201338118
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.201338118

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13

Academic Journal

A Three‐Component Palladium‐Catalyzed Oxidative CC Coupling Reaction: A Domino Process in Two Dimensions

المؤلفون: Nimje, Roshan Y., Leskinen, Mikko V., Pihko, Petri M.

المصدر: Angewandte Chemie ; volume 125, issue 18, page 4918-4922 ; ISSN 0044-8249 1521-3757

الاتاحة: http://dx.doi.org/10.1002/ange.201300833
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fange.201300833
https://onlinelibrary.wiley.com/doi/pdf/10.1002/ange.201300833

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14

Academic Journal

Palladium‐Catalyzed Dehydrogenative β′‐Arylation of β‐Keto Esters under Aerobic Conditions: Interplay of Metal and Brønsted Acids

المؤلفون: Yip, Kai‐Tai, Nimje, Roshan Y., Leskinen, Mikko V., Pihko, Petri M.

المصدر: Chemistry – A European Journal ; volume 18, issue 40, page 12590-12594 ; ISSN 0947-6539 1521-3765

الاتاحة: http://dx.doi.org/10.1002/chem.201201988
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchem.201201988
http://onlinelibrary.wiley.com/wol1/doi/10.1002/chem.201201988/fullpdf

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15

Academic Journal

ChemInform Abstract: Organocatalytic Domino Double Michael Reaction of Ethyl (E)‐7‐Oxohept‐2‐enoate and α,β‐Unsaturated Aldehydes: Efficient Asymmetric Synthesis of Cyclohexanes with Four Contiguous Stereocenters.

المؤلفون: Hong, Bor‐Cherng, Sadani, Amit A., Nimje, Roshan Y., Dange, Nitin S., Lee, Gene‐Hsiang

المصدر: ChemInform ; volume 42, issue 43 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.201143049
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.201143049
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.201143049

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16

Academic Journal

Enantioselective Organocatalytic Michael−Wittig−Michael−Michael Reaction: Dichotomous Construction of Pentasubstituted Cyclopentanecarbaldehydes and Pentasubstituted Cyclohexanecarbaldehydes

المؤلفون: Hong, Bor-Cherng, Nimje, Roshan Y., Lin, Cheng-Wei, Liao, Ju-Hsiou

المصدر: Organic Letters ; volume 13, issue 6, page 1278-1281 ; ISSN 1523-7060 1523-7052

الاتاحة: http://dx.doi.org/10.1021/ol1030487
https://pubs.acs.org/doi/pdf/10.1021/ol1030487

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17

Academic Journal

ChemInform Abstract: Enantioselective Synthesis of Highly Functionalized Octahydro‐6‐oxo‐1‐phenylnaphthalene‐2‐carbaldehydes via Organocatalytic Domino Reactions.

المؤلفون: Hong, Bor‐Cherng, Nimje, Roshan Y., Liao, Ju‐Hsiou

المصدر: ChemInform ; volume 40, issue 51 ; ISSN 0931-7597 1522-2667

الاتاحة: http://dx.doi.org/10.1002/chin.200951114
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fchin.200951114
https://onlinelibrary.wiley.com/doi/pdf/10.1002/chin.200951114

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18

Academic Journal

Enantioselective synthesis of highly functionalized octahydro-6-oxo-1-phenylnaphthalene-2-carbaldehydes via organocatalytic domino reactions

المؤلفون: Hong, Bor-Cherng, Nimje, Roshan Y., Liao, Ju-Hsiou

المصدر: Organic & Biomolecular Chemistry ; volume 7, issue 15, page 3095 ; ISSN 1477-0520 1477-0539

الاتاحة: http://dx.doi.org/10.1039/b906205j
http://pubs.rsc.org/en/content/articlepdf/2009/OB/B906205J

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19

Academic Journal

Organocatalytic Enantioselective Cascade Michael−Michael−Wittig Reactions of Phosphorus Ylides: One-Pot Synthesis of the all-cis Trisubstituted Cyclohexenecarboxylates via the [1 + 2 + 3] Annulation

المؤلفون: Hong, Bor-Cherng, Jan, Rei-Hau, Tsai, Chih-Wei, Nimje, Roshan Y., Liao, Ju-Hsiou, Lee, Gene-Hsiang

المصدر: Organic Letters ; volume 11, issue 22, page 5246-5249 ; ISSN 1523-7060 1523-7052

الاتاحة: http://dx.doi.org/10.1021/ol9021832
https://pubs.acs.org/doi/pdf/10.1021/ol9021832

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20

Academic Journal

Organocatalytic Double Michael Reaction of 7‐Oxohept‐2‐enoates and Nitrostyrene – Formal Synthesis of (–)‐α‐ and (–)‐β‐Lycorane

المؤلفون: Hong, Bor‐Cherng, Nimje, Roshan Y., Wu, Ming‐Fun, Sadani, Amit A.

المصدر: European Journal of Organic Chemistry ; volume 2008, issue 8, page 1449-1457 ; ISSN 1434-193X 1099-0690

الاتاحة: http://dx.doi.org/10.1002/ejoc.200701122
https://api.wiley.com/onlinelibrary/tdm/v1/articles/10.1002%2Fejoc.200701122
https://onlinelibrary.wiley.com/doi/full/10.1002/ejoc.200701122

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