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المؤلفون: George Kunos, Malliga R. Iyer
المصدر: Expert Opinion on Therapeutic Patents. 31:361-386
مصطلحات موضوعية: Neurotensin receptor 1, Neurotensin receptor 2, Neuropeptide, Biology, 01 natural sciences, Patents as Topic, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, Animals, Humans, Receptors, Neurotensin, Molecular Targeted Therapy, Receptor, Neurotransmitter, Neurotensin, Pharmacology, Drug discovery, Translation (biology), Receptor Cross-Talk, General Medicine, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry, 030220 oncology & carcinogenesis, Neuroscience
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المؤلفون: Lotfi Ferhat, Pascaline Lécorché, Michel Khrestchatisky, Maxime Masse, Grigorios Kyriatzis, Anne Bernard, Angélique Bole, Guillaume Jacquot, Guillaume Pflieger, Petros Chalas
المساهمون: Institut de neurophysiopathologie (INP), Aix Marseille Université (AMU)-Centre National de la Recherche Scientifique (CNRS), Vect-Horus
المصدر: Glia
Glia, 2021, 69 (11), pp.2618-2643. ⟨10.1002/glia.24062⟩مصطلحات موضوعية: kainate, Neurotensin receptor 2, [SDV.NEU.NB]Life Sciences [q-bio]/Neurons and Cognition [q-bio.NC]/Neurobiology, Hippocampus, microglia, Hippocampal formation, Biology, Blood–brain barrier, blood–brain barrier, Cellular and Molecular Neuroscience, Seizures, medicine, Animals, Receptors, Neurotensin, Receptor, Neuroinflammation, Microglia, NTSR2, Pilocarpine, Endothelial Cells, Cell biology, Rats, proinflammatory factors, medicine.anatomical_structure, Neurology, Astrocytes, Neuroinflammatory Diseases, epilepsy, IL1β, Astrocyte
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المؤلفون: Jan J. Enghild, Ebbe Toftgaard Poulsen, Lone Tjener Pallesen, Nádia Gonçalves, Mette Richner, Thomas Hellesøe Holm, Lars Christian Biilmann Rønn, Louis-Etienne Lorenzo, Karin Lykke-Hartmann, Maj Ulrichsen, Christian Bjerggaard Vaegter, Yves De Koninck, Anders Nykjaer, Annie Castonguay, Hande Login, Olav M. Andersen, Ole J. Bjerrum, Ibrahim John Malik
المصدر: Richner, M, Pallesen, L T, Ulrichsen, M, Poulsen, E T, Holm, T H, Login, H, Castonguay, A, Lorenzo, L-E, Gonçalves, N P, Andersen, O M, Lykke-Hartmann, K, Enghild, J J, Rønn, L C B, Malik, I J, De Koninck, Y, Bjerrum, O J, Vægter, C B & Nykjær, A 2019, ' Sortilin gates neurotensin and BDNF signaling to control peripheral neuropathic pain ', Science Advances, vol. 5, no. 6, eaav9946 . https://doi.org/10.1126/sciadv.aav9946
Science Advances
Richner, M, Pallesen, L T, Ulrichsen, M, Poulsen, E T, Holm, T H, Login, H, Castonguay, A, Lorenzo, L E, Gonçalves, N P, Andersen, O M, Lykke-Hartmann, K, Enghild, J J, Rønn, L C B, Malik, I J, De Koninck, Y, Bjerrum, O J, Vægter, C B & Nykjær, A 2019, ' Sortilin gates neurotensin and BDNF signaling to control peripheral neuropathic pain ' Science Advances, vol. 5, no. 6, eaav9946 . https://doi.org/10.1126/sciadv.aav9946مصطلحات موضوعية: Male, PROTEIN, chemistry.chemical_compound, Mice, 0302 clinical medicine, Neurotrophic factors, Peripheral Nerve Injuries, Medicine, Receptors, Neurotensin, BRAIN, Research Articles, Neurotensin, 0303 health sciences, Multidisciplinary, SciAdv r-articles, 3. Good health, Nociception, medicine.anatomical_structure, Hyperalgesia, Peripheral nerve injury, Neuropathic pain, Female, medicine.symptom, SPINAL-CORD, MESSENGER-RNA, Research Article, Signal Transduction, Neurotensin receptor 2, Down-Regulation, 03 medical and health sciences, Animals, Humans, 030304 developmental biology, IDENTIFICATION, RECEPTOR, business.industry, NERVE INJURY, Brain-Derived Neurotrophic Factor, Nerve injury, ANION GRADIENT, Spinal cord, Mice, Inbred C57BL, Adaptor Proteins, Vesicular Transport, MAINTENANCE, chemistry, nervous system, Neuralgia, INTERNALIZATION, business, Neuroscience, 030217 neurology & neurosurgery
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa3c302ed3cefcb24aca3ae1644e4f52
https://pure.au.dk/portal/da/publications/sortilin-gates-neurotensin -and-bdnf-signaling-to-control-peripheral-neuropathic-pain(81baa09b-5c54-4b82-91e2-6a5fde210696).html -
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المؤلفون: Steven Ballet, Fanni Tóth, Sándor Benyhe, Magdalena Bujalska-Zadrożny, Patrycja Kleczkowska, Géza Tóth, Dirk Tourwé, Andrzej W. Lipkowski, Jayapal Reddy Mallareddy
المصدر: Neuropeptides. 57:15-20
مصطلحات موضوعية: Male, 0301 basic medicine, Agonist, Neurotensin receptor 2, medicine.drug_class, Stereochemistry, G protein, Ligands, Sulfur Radioisotopes, Tritium, Inhibitory Concentration 50, Radioligand Assay, 03 medical and health sciences, Cellular and Molecular Neuroscience, chemistry.chemical_compound, 0302 clinical medicine, Endocrinology, Opioid receptor, medicine, Animals, Receptors, Neurotensin, Rats, Wistar, Receptor, Neurotensin, Endocrine and Autonomic Systems, Chemistry, Brain, General Medicine, Receptor antagonist, Peptide Fragments, Rats, 030104 developmental biology, Spinal Cord, Neurology, Guanosine 5'-O-(3-Thiotriphosphate), Neuromedin N, 030217 neurology & neurosurgery, Protein Binding
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المؤلفون: Iustin V. Tabarean
المصدر: Neuropharmacology
مصطلحات موضوعية: Male, 0301 basic medicine, Patch-Clamp Techniques, Neurotensin receptor 1, Neurotensin receptor 2, Neuropeptide, Hypothermia, Article, Purinergic P2X Receptor Agonists, Mice, 03 medical and health sciences, Cellular and Molecular Neuroscience, chemistry.chemical_compound, 0302 clinical medicine, Animals, Receptors, Neurotensin, Receptor, Neurotensin, gamma-Aminobutyric Acid, Median preoptic nucleus, Neurons, Pharmacology, Excitatory Postsynaptic Potentials, Preoptic Area, Cell biology, Mice, Inbred C57BL, 030104 developmental biology, nervous system, chemistry, Astrocytes, Neuromedin N, GABAergic, Receptors, Purinergic P2X4, hormones, hormone substitutes, and hormone antagonists, 030217 neurology & neurosurgery
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المؤلفون: Xing Li, Ning Jiang, Xiaodan Niu, Shimiao Zhu, Hao Tian, Yuanjie Niu, Zhiqun Shang, Xuanrong Chen, Amilcar Flores-Morales, Chawnshang Chang, Chuanliang Xu, Shancheng Ren, Yinghao Sun, Simeng Wen, Jiang Wang
المصدر: Oncogene
مصطلحات موضوعية: 0301 basic medicine, Male, Cancer Research, Neurotensin receptor 1, Neurotensin receptor 2, Biology, urologic and male genital diseases, Neuroendocrine differentiation, Article, 03 medical and health sciences, chemistry.chemical_compound, Prostate cancer, Mice, 0302 clinical medicine, Neuroendocrine Cells, Cell Line, Tumor, LNCaP, Genetics, medicine, Animals, Humans, Receptors, Neurotensin, Receptor, Molecular Biology, Neurotensin, Mice, Inbred BALB C, Prostate, Correction, medicine.disease, Adaptor Proteins, Vesicular Transport, Prostatic Neoplasms, Castration-Resistant, Cancer therapeutic resistance, 030104 developmental biology, nervous system, chemistry, 030220 oncology & carcinogenesis, Cell Transdifferentiation, Cancer research, Signal transduction
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المؤلفون: Peter Gmeiner, Philipp Tripal, Simone Maschauer, Harald Hübner, Cornelia Greff, Jürgen Einsiedel, Olaf Prante, Julian J. Ott
المصدر: Bioorganic & Medicinal Chemistry. 23:4026-4033
مصطلحات موضوعية: Fluorine Radioisotopes, Biodistribution, Neurotensin receptor 2, Clinical Biochemistry, Mice, Nude, Pharmaceutical Science, Chemistry Techniques, Synthetic, Biochemistry, Peptoids, chemistry.chemical_compound, Drug Stability, In vivo, Drug Discovery, medicine, Radioligand, Animals, Humans, Receptors, Neurotensin, Tissue Distribution, Molecular Biology, medicine.diagnostic_test, Chemistry, Organic Chemistry, Radiosynthesis, Glycopeptides, In vitro, Positron emission tomography, Isotope Labeling, Positron-Emission Tomography, Autoradiography, Molecular Medicine, Female, Radiopharmaceuticals, HT29 Cells, Neurotensin
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المصدر: Cellular and Molecular Neurobiology. 35:785-795
مصطلحات موضوعية: MAPK/ERK pathway, Neurotensin receptor 2, MAP Kinase Signaling System, Polymers, media_common.quotation_subject, Cell Cycle Proteins, CHO Cells, Biology, GPI-Linked Proteins, Transfection, Mice, Cellular and Molecular Neuroscience, chemistry.chemical_compound, Cricetulus, Cricetinae, Glioma, medicine, Animals, Protein Isoforms, Receptors, Neurotensin, Neurotensin receptor, Receptor, Internalization, Cells, Cultured, Neurotensin, media_common, Cell Biology, General Medicine, medicine.disease, Molecular biology, Endocytosis, Rats, Cell biology, Animals, Newborn, nervous system, chemistry, Nanoparticles, Protein Binding
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المؤلفون: Amy K. Sutton, Adriana Garcia, Raluca Bugescu, Darren M. Opland, Hillary L. Woodworth, Gina M. Leinninger, Christopher J. Rhodes, Lyndsay Christensen, Martin G. Myers, Juliette A. Brown
المصدر: Molecular Metabolism. 2(4):423-434
مصطلحات موضوعية: medicine.medical_specialty, Leptin receptor, Neurotensin receptor 1, Neurotensin receptor 2, Leptin, digestive, oral, and skin physiology, Cell Biology, Nucleus accumbens, Biology, Orexin, Ventral tegmental area, medicine.anatomical_structure, Endocrinology, nervous system, Dopamine, Internal medicine, medicine, Original Article, Molecular Biology, medicine.drug
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المصدر: Biochemical and Biophysical Research Communications. 439:35-39
مصطلحات موضوعية: medicine.medical_specialty, Neurotensin receptor 1, Neurotensin receptor 2, Calcium pump, Cellular differentiation, Biophysics, chemistry.chemical_element, Biology, Calcium, Biochemistry, chemistry.chemical_compound, Adenosine Triphosphate, Cytosol, Internal medicine, medicine, Humans, Receptors, Neurotensin, Calcium Signaling, RNA, Messenger, Neurotensin receptor, Molecular Biology, Neurotensin, Calcium signaling, Dose-Response Relationship, Drug, Receptors, Purinergic, Cell Differentiation, Cell Biology, Cell biology, Gene Expression Regulation, Neoplastic, Butyrates, Endocrinology, chemistry, Colonic Neoplasms, HT29 Cells, Signal Transduction
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المؤلفون: Thomas Naves, Dominique Bordessoule, Arnaud Jaccard, Nathalie Gachard, Hugo Talbot, Sofiane Saada, Julie Abraham, Anne-Laure Fauchais, Marie-Odile Jauberteau, A. Abbaci
المساهمون: Homéostasie Cellulaire et Pathologies (HCP), Université de Limoges (UNILIM)-CHU Limoges-Génomique, Environnement, Immunité, Santé, Thérapeutique (GEIST FR CNRS 3503), Unité de Catalyse et Chimie du Solide - UMR 8181 (UCCS), Université d'Artois (UA)-Centrale Lille-Institut de Chimie du CNRS (INC)-Université de Lille-Centre National de la Recherche Scientifique (CNRS), Contrôle de la Réponse Immune B et des Lymphoproliférations (CRIBL), Université de Limoges (UNILIM)-Génomique, Environnement, Immunité, Santé, Thérapeutique (GEIST FR CNRS 3503)-Centre National de la Recherche Scientifique (CNRS), Service d'Hématologie biologique [CHU Limoges], CHU Limoges, Service de Médecine interne A et polyclinique médicale [CHU Limoges], Contrôle de l’Activation Cellulaire, Progression Tumorale et Résistance thérapeutique (CAPTuR), Institut Génomique, Environnement, Immunité, Santé, Thérapeutique (GEIST), Université de Limoges (UNILIM)-Université de Limoges (UNILIM), Université de Limoges (UNILIM)-Génomique, Environnement, Immunité, Santé, Thérapeutique (GEIST FR CNRS 3503)-CHU Limoges, Centrale Lille Institut (CLIL)-Université d'Artois (UA)-Centrale Lille-Centre National de la Recherche Scientifique (CNRS)-Institut de Chimie du CNRS (INC)-Université de Lille, Unité de Catalyse et de Chimie du Solide - UMR 8181 (UCCS), Université d'Artois (UA)-Ecole Centrale de Lille-Ecole Nationale Supérieure de Chimie de Lille (ENSCL)-Université de Lille-Centre National de la Recherche Scientifique (CNRS), Institut National de la Santé et de la Recherche Médicale (INSERM)-Centre National de la Recherche Scientifique (CNRS)-Institut Génomique, Environnement, Immunité, Santé, Thérapeutique (GEIST)
المصدر: Oncogene
Oncogene, 2017, 37 (6), pp.756-767. ⟨10.1038/onc.2017.365⟩
Oncogene, Nature Publishing Group, 2017, 37 (6), pp.756-767. ⟨10.1038/onc.2017.365⟩مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Neurotensin receptor 2, Apoptosis, [SDV.CAN]Life Sciences [q-bio]/Cancer, Tropomyosin receptor kinase B, [SDV.BC]Life Sciences [q-bio]/Cellular Biology, Receptor tyrosine kinase, 03 medical and health sciences, Paracrine signalling, 0302 clinical medicine, Biomarkers, Tumor, Tumor Cells, Cultured, Genetics, Humans, Receptor, trkB, Receptors, Neurotensin, Neurotensin receptor, Autocrine signalling, Molecular Biology, ComputingMilieux_MISCELLANEOUS, Cell Proliferation, Brain-derived neurotrophic factor, Membrane Glycoproteins, biology, Brain-Derived Neurotrophic Factor, Leukemia, Lymphocytic, Chronic, B-Cell, Cell biology, 030104 developmental biology, nervous system, 030220 oncology & carcinogenesis, biology.protein, Original Article, Proto-oncogene tyrosine-protein kinase Src
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المؤلفون: Anne-Laure Fauchais, A. Abbaci, Arnaud Jaccard, Dominique Bordessoule, Hugo Talbot, Nathalie Gachard, Sofiane Saada, Julie Abraham, Thomas Naves, Marie-Odile Jauberteau
المصدر: ESMO Open. 3:A19
مصطلحات موضوعية: Cancer Research, Paracrine signalling, Programmed cell death, Oncology, biology, Neurotensin receptor 2, biology.protein, Cancer research, Neurotensin receptor, Tropomyosin receptor kinase B, Receptor, Autocrine signalling, Receptor tyrosine kinase
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المؤلفون: Jordan Walton, Jidong Guo, Kerry J. Ressler, Kenneth M. McCullough, Dennis C. Choi, Donald G. Rainnie, Kelsey Zimmerman
المصدر: Nature Communications
Nature Communications, Vol 7, Iss 1, Pp 1-13 (2016)مصطلحات موضوعية: 0301 basic medicine, General Physics and Astronomy, Bioinformatics, Extinction, Psychological, Stereotaxic Techniques, Mice, 0302 clinical medicine, Piperidines, Genes, Reporter, Receptors, Neurotensin, Clozapine, education.field_of_study, Multidisciplinary, Basolateral Nuclear Complex, Chemogenetics, Fear, medicine.anatomical_structure, Intercellular Signaling Peptides and Proteins, Oligopeptides, Neurotensin receptor 2, Sensory Receptor Cells, Science, Population, Prefrontal Cortex, Optogenetics, Biology, General Biochemistry, Genetics and Molecular Biology, Article, 03 medical and health sciences, Bacterial Proteins, Memory, medicine, Animals, education, Adaptor Proteins, Signal Transducing, Injections, Intraventricular, Integrases, Sequence Analysis, RNA, RNA, General Chemistry, Wnt Proteins, Luminescent Proteins, 030104 developmental biology, nervous system, Gene Expression Regulation, Stereotaxic technique, Thy-1 Antigens, Neuron, Thrombospondins, Neuroscience, 030217 neurology & neurosurgery, Basolateral amygdala
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المؤلفون: Christian E. Elling, Thue W. Schwartz, Nicholas D. Holliday, Anders Bach, Helen M. Cox, Birgitte Holst
المصدر: Journal of Biological Chemistry. 279:53806-53817
مصطلحات موضوعية: Models, Molecular, Receptors, Neuropeptide, DNA, Complementary, Transcription, Genetic, Neurotensin receptor 2, MAP Kinase Signaling System, Protein Conformation, Inositol Phosphates, Motilin receptor, DNA Mutational Analysis, Molecular Sequence Data, Enzyme-Linked Immunosorbent Assay, Biology, Ligands, Phosphatidylinositols, Transfection, GTP-Binding Protein alpha Subunits, G12-G13, Biochemistry, Protein Structure, Secondary, Cell Line, Receptors, G-Protein-Coupled, Receptors, Gastrointestinal Hormone, Cyclic AMP, Enzyme-linked receptor, Animals, Humans, Receptors, Neurotensin, Inverse agonist, Amino Acid Sequence, Receptors, Ghrelin, Receptor, Molecular Biology, Phylogeny, Glucagon-like peptide 1 receptor, Orphan receptor, Microscopy, Dose-Response Relationship, Drug, digestive, oral, and skin physiology, Cell Biology, Protein Structure, Tertiary, Cell biology, Type C Phospholipases, COS Cells, Ghrelin, Signal Transduction
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المؤلفون: Keiji Wada, Ying-Jie Sun, Hiroshi Maeno, Shunsuke Aoki
المصدر: Molecular Brain Research. 95:167-171
مصطلحات موضوعية: Mice, Knockout, Genetics, Neurotensin receptor 1, Transcription, Genetic, Neurotensin receptor 2, Molecular Sequence Data, Alternative splicing, CAAT box, Chromosome Mapping, Promoter, Biology, Molecular biology, Alternative Splicing, Blotting, Southern, Mice, Cellular and Molecular Neuroscience, Exon, Gene Expression Regulation, Animals, Receptors, Neurotensin, Coding region, Promoter Regions, Genetic, Molecular Biology, Gene
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المؤلفون: Zhengwei Cai, Yi Pang, P.G. Rhodes
المصدر: Brain Research. 914:15-22
مصطلحات موضوعية: Lipopolysaccharides, Chemokine, Neurotensin receptor 2, Down-Regulation, Rats, Sprague-Dawley, Complementary DNA, Gene expression, Animals, Growth Substances, Molecular Biology, Transcription factor, Macrophage inflammatory protein, Cells, Cultured, Oligonucleotide Array Sequence Analysis, biology, General Neuroscience, Binding protein, Bacterial Infections, Molecular biology, Rats, Up-Regulation, IRF1, Animals, Newborn, Gene Expression Regulation, Astrocytes, biology.protein, Cytokines, Encephalitis, Neurology (clinical), Transcription Factors, Developmental Biology
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المصدر: PLoS ONE, Vol 9, Iss 1, p e83098 (2014)
PLoS ONEمصطلحات موضوعية: Male, Central Nervous System, Anatomy and Physiology, Lateral hypothalamus, Gene Expression, lcsh:Medicine, Biochemistry, Mice, Behavioral Neuroscience, chemistry.chemical_compound, Neural Pathways, Receptors, Neurotensin, lcsh:Science, Neurotensin, Mice, Inbred ICR, Multidisciplinary, Animal Behavior, Postpartum Period, Brain, Neurochemistry, Animal Models, Neurotransmitters, Immunohistochemistry, Hypothalamus, Medicine, Female, Neurochemicals, Research Article, medicine.drug, medicine.medical_specialty, Neural Networks, Neurotensin receptor 2, Neuropeptide, Biology, Neurological System, Model Organisms, Internal medicine, Animals, Outbred Strains, Genetics, medicine, Animals, RNA, Messenger, Analysis of Variance, Neuropeptides, lcsh:R, Connectomics, Neuroanatomy, Stria terminalis, Endocrinology, Gene Expression Regulation, chemistry, Oxytocin, lcsh:Q, Molecular Neuroscience, Zoology, Postpartum period, Neuroscience
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المؤلفون: P. Ferrara, Gérard Le Fur, Jacques Bonnin, Bruno Delpech, Mourad Kaghad, Pascale Chalon, Natalio Vita, Daniel Caput, Marie Guillemot
المصدر: FEBS Letters. 386:91-94
مصطلحات موضوعية: Neurotensin receptor 1, Neurotensin receptor 2, Molecular Sequence Data, Hypothalamus, Biophysics, Histamine H1 receptor, Biology, Biochemistry, Cell Line, chemistry.chemical_compound, Piperidines, Structural Biology, Complementary DNA, Chlorocebus aethiops, Genetics, medicine, Animals, Receptors, Neurotensin, Tissue Distribution, Amino Acid Sequence, RNA, Messenger, Neurotensin receptor, Binding site, Molecular Biology, Sequence Homology, Amino Acid, Molecular cloning, Cell Biology, Molecular biology, Levocabastine, Rats, chemistry, medicine.drug, Neurotensin
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المؤلفون: Ralf C. Kling, Harald Hübner, Helma Wennemers, Peter Gmeiner, Cornelia Held, Yvonne A. Nagel
المصدر: ChemMedChem. 8(5)
مصطلحات موضوعية: Models, Molecular, Neurotensin receptor 2, Proline, Thiazolidine, Peptide, Ligands, Biochemistry, chemistry.chemical_compound, Peptoids, Structure-Activity Relationship, Drug Discovery, Structure–activity relationship, Humans, Receptors, Neurotensin, General Pharmacology, Toxicology and Pharmaceutics, Receptor, G protein-coupled receptor, Pharmacology, chemistry.chemical_classification, Binding Sites, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Peptoid, Molecular Medicine, Peptides, Neurotensin
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المؤلفون: Peter Gmeiner, Monika Pischetsrieder, Cornelia Held, Jasmin Meltretter, Harald Hübner, Manuel Plomer
المصدر: ChemMedChem. 8(1)
مصطلحات موضوعية: Serum, Neurotensin receptor 2, Pain, Ligands, Biochemistry, Cell Line, chemistry.chemical_compound, Peptoids, Drug Discovery, Inverse agonist, Animals, Humans, Receptors, Neurotensin, Amino Acid Sequence, General Pharmacology, Toxicology and Pharmaceutics, Luciferase reporter gene, Neurotensin, Pharmacology, Organic Chemistry, Metabolic stability, Ligand (biochemistry), chemistry, Molecular Medicine, Selectivity, Molecular probe, Peptides