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المؤلفون: Emily F. Calderwood, Kathleen Aertgeerts, Michael D. Smith, Dylan Bradley England, Roushan Afroze, Ryan Chau, Stepan Vyskocil, Nancy E. Forsyth, Dong Mei Zhang, Ruth Adams, Stephen G. Stroud, O. P. Veiby, Christelle C. Renou, R. Scott Rowland, Erin Paske, Jane X. Liu, Ming Tregay, Michael D. Sintchak, Juliet A Williams, Shih-Chung Huang, Xu Tianlin, Bheemashankar Kulkarni, Sharmila Adhikari, Yuan Tian, Jason Yano, Christopher Blackburn, Paul D. Greenspan, Cheryl A. Farrer, Matthew O. Duffey, Liting Ma, Mi-Sook Kim, Qin Zhang, Sean Harrison, Hirotake Mizutani, Katherine M. Galvin, Alexandra E. Gould, Johnny J. Yang, Steven P. Langston, Dave Janowick, Natalia Iartchouk, Mansoureh Rezaei, Jeffery Gaulin, Khristofer Garcia, Hongbo Zeng, Ribo Guo, Tricia J. Vos, Jouhara Chouitar, Saurabh Menon
المصدر: Journal of Medicinal Chemistry. 54:1836-1846
مصطلحات موضوعية: Models, Molecular, Proto-Oncogene Proteins B-raf, Tetrahydronaphthalenes, Mutant, Melanoma, Experimental, Administration, Oral, Biological Availability, Mice, Nude, Antineoplastic Agents, Pharmacology, Crystallography, X-Ray, Mice, Structure-Activity Relationship, Pharmacokinetics, Mouse xenograft, In vivo, Drug Discovery, medicine, Animals, chemistry.chemical_classification, Chemistry, Melanoma, Stereoisomerism, medicine.disease, Xenograft Model Antitumor Assays, In vitro, Bioavailability, Enzyme, Drug Design, Mutation, Molecular Medicine
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2
المؤلفون: Emily F. Calderwood, Alexandra E. Gould, Nancy E. Forsyth
المصدر: Synthetic Communications. 34:3455-3464
مصطلحات موضوعية: chemistry.chemical_classification, chemistry, Organic Chemistry, Electrophile, Organic chemistry, Imidazoline receptor, chemistry.chemical_element, Alkylation, Protecting group, Nitrogen, Carbon, Alkyl
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المؤلفون: Nancy E. Forsyth, Alexandra E. Gould, Emily F. Calderwood
المصدر: ChemInform. 36
مصطلحات موضوعية: chemistry.chemical_classification, chemistry, Electrophile, Imidazoline receptor, chemistry.chemical_element, Organic chemistry, General Medicine, Alkylation, Protecting group, Carbon, Alkyl
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4
المؤلفون: Nancy E. Forsyth, Thomas H Marsilje, Christopher Blackburn, Lijun Wu, Marie D Bohane, Stephen G. Stroud, David Yowe, Jonathan B Roses, Stacey V Drabic, Michael A. Patane, Christopher F. Claiborne, Ping Li, Wenyan Miao, Emily F. Calderwood, J. Scott Daniels
المصدر: Bioorganicmedicinal chemistry letters. 14(14)
مصطلحات موضوعية: medicine.medical_specialty, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, Melanocortin receptor, Internal medicine, Drug Discovery, medicine, Structure–activity relationship, Animals, Binding site, Receptor, Molecular Biology, Cells, Cultured, Binding Sites, Chemistry, Organic Chemistry, Body Weight, Antagonist, Imidazoles, Small molecule, Rats, Melanocortin 4 receptor, Endocrinology, Molecular Medicine, Receptor, Melanocortin, Type 4, Melanocortin
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المؤلفون: Suresh K. Balani, Tricia J. Vos, Jennifer Lee Che, Martin P. Maguire, Ping Li, Luis E Rodriguez, Cheryl A. Farrer, Michael A. Patane, Christopher F. Claiborne, Stacey V Drabic, Andrei Caracoti, David Yowe, Nancy E. Forsyth, Diana Lamppu, Ingrid B J K Joseph, Hang Zeng, Robert A. Horlick, Mingshi Dai
المصدر: Journal of medicinal chemistry. 47(7)
مصطلحات موضوعية: medicine.medical_specialty, Transplantation, Heterologous, Administration, Cutaneous, Energy homeostasis, Mice, Radioligand Assay, Structure-Activity Relationship, Weight loss, Internal medicine, Neoplasms, Drug Discovery, medicine, Animals, Receptor, Emaciation, Mice, Inbred BALB C, Chemistry, Antagonist, Imidazoles, Biological activity, Benzamidines, Melanocortin 4 receptor, Transplantation, Endocrinology, Molecular Medicine, Receptor, Melanocortin, Type 4, Melanocortin, medicine.symptom, Neoplasm Transplantation