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1
المؤلفون: Jonathan A. Phillips, Mitchell E. Taub, Matthew S. Bogdanffy, Jing Yuan, Brian Knight, James D. Smith, Warren W. Ku
المصدر: Journal of Applied Toxicology. 42
مصطلحات موضوعية: Toxicology
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2
المؤلفون: Sabrina Wiebe, Ashish Sharma, Martin F. Fromm, Alen Jambrecina, Peter Stopfer, Fabian Müller, Edith Hauel, Kerstin Bader, Mitchell E. Taub, Gerd Mikus, Kathrin Hohl, Sven Schmidt-Gerets, Thomas Giessmann, Thomas Ebner, Naoki Ishiguro
المصدر: Clinical Pharmacokinetics
مصطلحات موضوعية: Male, Organic anion transporter 1, Digoxin, Cmax, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, medicine, Humans, Drug Interactions, Pharmacology (medical), Rosuvastatin, Original Research Article, Cimetidine, biology, Probenecid, Chemistry, Organic anion-transporting polypeptide, Verapamil, Area Under Curve, 030220 oncology & carcinogenesis, biology.protein, Rifampin, medicine.drug
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3
المصدر: Drug Metabolism and Disposition. 48:690-697
مصطلحات موضوعية: Adult, Male, Time Factors, CYP3A, Midazolam, Primary Cell Culture, Drug Evaluation, Preclinical, Pharmaceutical Science, Pharmacology, Hydroxylation, chemistry.chemical_compound, medicine, Cytochrome P-450 CYP3A, Humans, Glucuronosyltransferase, Receptor, Cells, Cultured, Alprazolam, CYP3A4, biology, Chemistry, Cytochrome P-450 CYP3A Inducers, Cytochrome P450, Metabolism, Middle Aged, Coculture Techniques, Uridine, Erythromycin, Hepatobiliary Elimination, medicine.anatomical_structure, Hepatocyte, Hepatocytes, biology.protein, Cytochrome P-450 CYP3A Inhibitors, Female, Rifampin
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4
المؤلفون: Chukwunonso K Nwabufo, Iain Martin, Matthew Segall, Fabio Broccatelli, Emily E. Scott, Eric Gonzalez, Jasleen K. Sodhi, Laura E Russell, Aaron G. Bart, Mary A. Schleiff, W. Griffith Humphreys, Ryan H. Takahashi, Mitchell E. Taub, Volker M. Lauschke, Bhagwat Prasad, Jessica H. Hartman
المصدر: Drug Metab Rev
مصطلحات موضوعية: business.industry, Computational Biology, Congresses as Topic, 030226 pharmacology & pharmacy, Article, Xenobiotics, Machine Learning, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmaceutical Preparations, chemistry, Biochemistry, 030220 oncology & carcinogenesis, Drug Discovery, Quantum Theory, Medicine, Pharmacology (medical), General Pharmacology, Toxicology and Pharmaceutics, Pharmaceutical sciences, Xenobiotic, business, human activities, Drug metabolism
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5
المؤلفون: Jonathan A. Phillips, Mitchell E. Taub, Matthew S. Bogdanffy, Jing Yuan, Brian Knight, James D. Smith, Warren W. Ku
المصدر: Journal of applied toxicology : JATREFERENCES. 42(10)
مصطلحات موضوعية: Male, Toxicology, Kidney, Kidney Neoplasms, Rats, Antigens, CD1, Mice, Diabetes Mellitus, Type 2, Glucosides, Sodium-Glucose Transporter 2, Animals, Humans, Hypoglycemic Agents, Female, Benzhydryl Compounds, Carcinoma, Renal Cell, Sodium-Glucose Transporter 2 Inhibitors
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6
المؤلفون: Bhagwat Prasad, Peter Stopfer, Valerie Nock, Hannah Britz, Thorsten Lehr, Mitchell E. Taub, Éric Fernandez, Ting Wang, Nina Hanke
المصدر: Pharmaceutical Research
مصطلحات موضوعية: Drug, Adult, Male, Physiologically based pharmacokinetic modelling, Organic anion transporter 1, media_common.quotation_subject, Cmax, Pharmaceutical Science, Administration, Oral, Organic Anion Transporters, Drug Elimination Routes, Pharmacology, 030226 pharmacology & pharmacy, Models, Biological, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Furosemide, medicine, Humans, Pharmacology (medical), Computer Simulation, Drug Interactions, Biotransformation, media_common, biology, Chemistry, Probenecid, Organic Chemistry, physiologically based pharmacokinetic modeling (PBPK), Transporter, drug-drug interaction (DDI), organic anion transporter (OAT), 030220 oncology & carcinogenesis, biology.protein, Molecular Medicine, Administration, Intravenous, Female, Rifampin, Biotechnology, medicine.drug, Research Paper
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7
المصدر: Drug Metabolism and Disposition. 46:770-778
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Methyltransferase, biology, Nicotinamide, Chemistry, Metabolite, Pharmaceutical Science, Kidney metabolism, Methylation, 010402 general chemistry, 030226 pharmacology & pharmacy, 01 natural sciences, 0104 chemical sciences, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Enzyme, Biochemistry, Thiol S-methyltransferase, biology.protein, Microsome
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8
المؤلفون: Jonathan A. Phillips, Hlaing Hlaing Maw, Warren W. Ku, Hongbin Yu, Patricia A. Escobar, William T. Loging, Mitchell E. Taub, Zimei Huang, Pamela Foppiano, James D. Smith
المصدر: International Journal of Toxicology. 36:440-448
مصطلحات موضوعية: Male, 0301 basic medicine, Cell Survival, Sodium, Metabolite, chemistry.chemical_element, Mice, Inbred Strains, Pharmacology, Toxicology, medicine.disease_cause, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Glucosides, Empagliflozin, Animals, Hypoglycemic Agents, Cytotoxic T cell, Medicine, Benzhydryl Compounds, Cytotoxicity, Cells, Cultured, Micronuclei, Chromosome-Defective, Carcinogen, Cell Proliferation, Genetics, Kidney, business.industry, Oxidative Stress, Kidney Tubules, 030104 developmental biology, medicine.anatomical_structure, chemistry, 030220 oncology & carcinogenesis, business, Genotoxicity
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9
المؤلفون: Kathrin Hohl, Naoki Ishiguro, Thomas Giessmann, Ashish Sharma, Arvid Jungnik, Mitchell E. Taub, Dietmar Gansser, Thomas Ebner, Peter Stopfer, Fabian Müller
المصدر: European Journal of Drug Metabolism and Pharmacokinetics
مصطلحات موضوعية: Adult, Male, Adolescent, Digoxin, Biological Availability, Pharmacology, 030226 pharmacology & pharmacy, Young Adult, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Furosemide, medicine, Humans, Hypoglycemic Agents, Drug Interactions, Pharmacology (medical), Rosuvastatin, Original Research Article, Rosuvastatin Calcium, Diuretics, Cross-Over Studies, Dose-Response Relationship, Drug, business.industry, Anticholesteremic Agents, nutritional and metabolic diseases, Middle Aged, Crossover study, Healthy Volunteers, Metformin, Bioavailability, 030220 oncology & carcinogenesis, business, medicine.drug
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10
المؤلفون: Naoki Ishiguro, Mitchell E. Taub, H Zimdahl-Gelling, Dietmar Gansser, Kathrin Hohl, Thomas Giessmann, Thomas Ebner, Ashish Sharma, M Wein, Peter Stopfer, Fabian Müller
المصدر: Clinical Pharmacology and Therapeutics
مصطلحات موضوعية: Adult, Male, Digoxin, Organic Cation Transport Proteins, Metabolic Clearance Rate, Cmax, Organic Anion Transporters, Sodium-Independent, Pharmacology, 030226 pharmacology & pharmacy, Solute Carrier Organic Anion Transporter Family Member 1B3, 03 medical and health sciences, Organic Anion Transport Protein 1, 0302 clinical medicine, Pharmacokinetics, Furosemide, medicine, ATP Binding Cassette Transporter, Subfamily G, Member 2, Humans, Drug Interactions, Pharmacology (medical), Rosuvastatin, ATP Binding Cassette Transporter, Subfamily B, Member 1, Rosuvastatin Calcium, Cation Transport Proteins, Cross-Over Studies, Liver-Specific Organic Anion Transporter 1, business.industry, Research, digestive, oral, and skin physiology, Organic Cation Transporter 2, Articles, Middle Aged, Crossover study, Metformin, Neoplasm Proteins, Area Under Curve, 030220 oncology & carcinogenesis, ATP-Binding Cassette Transporters, business, medicine.drug
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11
المؤلفون: Naoki Ishiguro, Thomas Ebner, Mitchell E. Taub
المصدر: Journal of Pharmaceutical Sciences. 104:3220-3228
مصطلحات موضوعية: Drug, Digoxin, Organic Cation Transport Proteins, Organic anion transporter 1, Abcg2, media_common.quotation_subject, Organic Anion Transporters, Pharmaceutical Science, Pharmacology, Cell Line, Furosemide, In vivo, Cell Line, Tumor, medicine, Humans, Drug Interactions, ATP Binding Cassette Transporter, Subfamily B, Member 1, Rosuvastatin Calcium, media_common, Organic cation transport proteins, biology, Chemistry, Cytochrome P450, Biological Transport, Transporter, Metformin, Neoplasm Proteins, HEK293 Cells, Biochemistry, biology.protein, ATP-Binding Cassette Transporters, Caco-2 Cells, medicine.drug
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12
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 46(7)
مصطلحات موضوعية: Adult, Male, Organic anion transporter 1, Pharmaceutical Science, Organic Anion Transporters, Sodium-Dependent, 030226 pharmacology & pharmacy, Cell Line, 03 medical and health sciences, Solute Carrier Organic Anion Transporter Family Member 1B3, 0302 clinical medicine, In vivo, medicine, Humans, Drug Interactions, Pitavastatin, Pharmacology, biology, Symporters, Chemistry, Liver-Specific Organic Anion Transporter 1, HEK 293 cells, Membrane Transport Proteins, Transporter, Biological Transport, Middle Aged, In vitro, medicine.anatomical_structure, HEK293 Cells, Biochemistry, Liver, Cell culture, 030220 oncology & carcinogenesis, Hepatocyte, biology.protein, Cyclosporine, Hepatocytes, Quinolines, Female, Hydroxymethylglutaryl-CoA Reductase Inhibitors, Rifampin, medicine.drug
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13
المؤلفون: Peter, Stopfer, Thomas, Giessmann, Kathrin, Hohl, Sabine, Hutzel, Sven, Schmidt, Dietmar, Gansser, Naoki, Ishiguro, Mitchell E, Taub, Ashish, Sharma, Thomas, Ebner, Fabian, Müller
المصدر: British Journal of Clinical Pharmacology
مصطلحات موضوعية: Adult, Male, Digoxin, Cross-Over Studies, Dose-Response Relationship, Drug, nutritional and metabolic diseases, Membrane Transport Proteins, drug transporters, Original Articles, drug interactions, Middle Aged, Healthy Volunteers, Metformin, Renal Elimination, Young Adult, Phase I, Drug Development, Furosemide, Area Under Curve, Humans, Original Article, Rosuvastatin Calcium, pharmacokinetics
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14
المؤلفون: Harma Ellens, Mary F. Paine, Maciej J. Zamek-Gliszczynski, Jack Cook, Caroline A. Lee, Mitchell E. Taub, Tasha K. Ritchie, Joseph A. Ware, Bo Feng, Meeghan A O'Connor, Aleksandra Galetin, Isabelle Ragueneau-Majlessi, Joseph W. Polli
المصدر: Drug Metabolism and Disposition. 43:490-509
مصطلحات موضوعية: Drug, Drug-Related Side Effects and Adverse Reactions, media_common.quotation_subject, Pharmaceutical Science, Drug resistance, Pharmacology, Lapatinib, Polymorphism, Single Nucleotide, Intestinal absorption, Substrate Specificity, Efficacy, Pharmacokinetics, Sulfasalazine, medicine, ATP Binding Cassette Transporter, Subfamily G, Member 2, Humans, Drug Interactions, Rosuvastatin, media_common, Clinical Trials as Topic, business.industry, Drug Resistance, Multiple, Neoplasm Proteins, Pharmaceutical Preparations, Research Design, Practice Guidelines as Topic, ATP-Binding Cassette Transporters, business, medicine.drug
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15
المصدر: Drug Metabolism and Pharmacokinetics. 35:S24
مصطلحات موضوعية: Pharmacology, Non specific, Biochemistry, Chemistry, Microsome, Pharmaceutical Science, Pharmacology (medical)
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16
المؤلفون: Lalitha Podila, Rucha S. Sane, Qihong Huang, Jerry O. Stern, Yongmei Li, Tarik Asselah, G. Steinmann, Gerhard Nehmiz, Wulf O. Böcher, Mitchell E. Taub, Stephen Olson, Kirsten Mease, Donald J. Tweedie
المصدر: Journal of Pharmacology and Experimental Therapeutics. 351:403-412
مصطلحات موضوعية: medicine.medical_specialty, Aminoisobutyric Acids, Proline, Bilirubin, Hepatitis C virus, Hepacivirus, medicine.disease_cause, chemistry.chemical_compound, Clinical Trials, Phase II as Topic, Double-Blind Method, Leucine, Internal medicine, medicine, Animals, Humans, Multicenter Studies as Topic, Glucuronosyltransferase, IC50, Hyperbilirubinemia, Randomized Controlled Trials as Topic, Unconjugated hyperbilirubinemia, Pharmacology, Liver injury, Clinical Trials, Phase I as Topic, Chemistry, Multidrug resistance-associated protein 2, medicine.disease, Hepatitis C, Macaca mulatta, Multidrug Resistance-Associated Protein 2, Rats, Thiazoles, Endocrinology, Liver, Faldaprevir, Toxicity, Hepatocytes, Quinolines, Molecular Medicine, Oligopeptides
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17
المؤلفون: Mitchell E. Taub, Yongmei Li, Donald J. Tweedie, Diane Ramsden, Tom S. Chan
المصدر: Drug Metabolism and Disposition. 42:394-406
مصطلحات موضوعية: Aminoisobutyric Acids, Proline, Metabolic Clearance Rate, Glucuronidation, Organic Anion Transporters, Pharmaceutical Science, Pharmacology, Biology, Antiviral Agents, Glucuronides, Drug Stability, Leucine, In vivo, medicine, Cytochrome P-450 CYP3A, Humans, Biotransformation, Cells, Cultured, Cryopreservation, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, Liver-Specific Organic Anion Transporter 1, Sodium, Biological Transport, Transporter, Metabolism, Fibroblasts, Coculture Techniques, Culture Media, Kinetics, Thiazoles, Metabolic pathway, medicine.anatomical_structure, Enzyme, Liver, chemistry, Biochemistry, Hepatocyte, Faldaprevir, Hepatocytes, Quinolines, Female, Oligopeptides
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18
المؤلفون: Laurent Salphati, Eric Sands, Praveen Balimane, Caroline A. Lee, Johan E. Palm, Joe Bentz, Lalitha Podila, Jesse Taur, Tetsuo Yamagata, Lei K. Zhang, Kathleen M. Hillgren, Eric L. Reyner, Marie Brännström, Dietmar Weitz, Emile Plise, Jocelyn Yabut, Masoud Jamei, Harma Ellens, Anne Pak, Dallas Bednarczyk, Guangqing Xiao, Mitchell E. Taub, Libin Li, Heleen M. Wortelboer, Elke S Perloff, Andrew K Mason, Michael P. O'Connor, Krisztina Herédi-Szabó, Aarti Patel, Ganesh Rajaraman, Xiaoyan Chu, Evelyn Hollnack-Pusch, Christoph Funk, Joann Coleman, Cindy Q. Xia, Xuena Lin, Imad Hanna, Ailan Guo, Sibylle Neuhoff
المصدر: Drug Metabolism and Disposition. 41:1347-1366
مصطلحات موضوعية: Digoxin, Swine, Pharmaceutical Science, Pharmacology, Risk Assessment, Inhibitory Concentration 50, Dogs, medicine, Animals, Humans, Drug Interactions, ATP Binding Cassette Transporter, Subfamily B, Member 1, IC50, P-glycoprotein, Principal Component Analysis, Isradipine, biology, Chemistry, Biological Transport, Articles, In vitro, biology.protein, LLC-PK1 Cells, Verapamil, Efflux, Caco-2 Cells, Telmisartan, medicine.drug
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19
المؤلفون: Swati Nagar, Masoud Jamei, A Poirier, T Ishikawa, J C Kalvass, Caroline A. Lee, Kenneth R. Korzekwa, Peter W. Swaan, Aleksandra Galetin, Joe Bentz, Maciej J. Zamek-Gliszczynski, Ping Zhao, K S Pang, Mitchell E. Taub, Xiaoyan Chu, Harma Ellens
المصدر: Clinical Pharmacology & Therapeutics. 94:64-79
مصطلحات موضوعية: Biological Availability, Guidelines as Topic, Computational biology, Biology, Pharmacology, Kidney, Models, Biological, Article, Kinetic parameter estimation, Animals, Humans, Drug Interactions, Pharmacokinetics, Tissue Distribution, Pharmacology (medical), Tissue distribution, Brain, Membrane Transport Proteins, Kidney metabolism, Biological Transport, Transporter, Liver metabolism, Liver, Pharmaceutical Preparations, Biological availability
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20
المؤلفون: Eric L. Reyner, Caroline A. Lee, Harma Ellens, Kirsten M Mease, Cory A Watson, Rucha S. Sane, Liangfu Chen, Mitchell E. Taub, Márton Jani, Brad P Hirakawa
المصدر: Drug Metabolism and Disposition. 39:2093-2102
مصطلحات موضوعية: Digoxin, medicine.medical_specialty, Organic anion transporter 1, Organic Anion Transporters, Pharmaceutical Science, ATP-binding cassette transporter, CHO Cells, Organic Anion Transporters, Sodium-Independent, Pharmacology, Substrate Specificity, Solute Carrier Organic Anion Transporter Family Member 1B3, Cricetinae, Internal medicine, polycyclic compounds, medicine, Animals, Humans, Drug Interactions, ATP Binding Cassette Transporter, Subfamily B, Member 1, RNA, Messenger, cardiovascular diseases, IC50, Cells, Cultured, Cardiac glycoside, biology, Liver-Specific Organic Anion Transporter 1, Chemistry, Sodium, digestive, oral, and skin physiology, Biological Transport, Transporter, carbohydrates (lipids), Organic anion-transporting polypeptide, HEK293 Cells, Endocrinology, biology.protein, Efflux, medicine.drug