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1Academic Journal
المؤلفون: Caroline Sychterz, Hong Shen, Yueping Zhang, Michael Sinz, Amin Rostami‐Hodjegan, Brian J. Schmidt, Lu Gaohua, Aleksandra Galetin
المصدر: CPT: Pharmacometrics & Systems Pharmacology, Vol 13, Iss 11, Pp 1856-1869 (2024)
مصطلحات موضوعية: Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2163-8306
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2
المؤلفون: Matthew D. Hill, Haiquan Fang, Derek Norris, George V. Delucca, Hong Huang, Mikkel DeBenedetto, Claude Quesnelle, William D. Schmitz, John S. Tokarski, Steven Sheriff, Chunhong Yan, Caroline Fanslau, Zuzana Haarhoff, Christine Huang, Melissa Kramer, Shilpa Madari, Krista Menard, Laura Monereau, John Morrison, Nirmala Raghavan, Eric E. Shields, Jean Simmermacher-Mayer, Michael Sinz, Ching Kim Tye, Richard Westhouse, Chunshan Xie, Haiying Zhang, Lisa Zhang, Tatyana Zvyaga, Francis Lee, Ashvinikumar V. Gavai, Andrew P. Degnan
المصدر: ACS Medicinal Chemistry Letters. 13:1165-1171
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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3
المؤلفون: L.V.J. Sankara Sivaprasad, Bokka Venkata Murali, T. Thanga Mariappan, Sushma Basavanthappa, Avinash Annasao Hadambar, Vijaykumar Kuchibhotla, Avisek Deyati, Bradley A. Zinker, Gowtham Raj Gunti, Manjunath Ramarao, Sagnik Chatterjee, Shashyendra Singh Gautam, Yueping Zhang, Tanvi Naik, Hong Shen, Sambuddho Mukherjee, Michael Sinz
المصدر: Journal of Pharmacology and Experimental Therapeutics. 376:29-39
مصطلحات موضوعية: Male, 0301 basic medicine, Coproporphyrins, medicine.medical_specialty, Endogeny, Plasma protein binding, Spodoptera, Rats, Sprague-Dawley, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Non-alcoholic Fatty Liver Disease, Internal medicine, Gene expression, Sf9 Cells, medicine, Animals, Humans, Angiogenic Proteins, Gene, Pharmacology, biology, Chemistry, Transporter, medicine.disease, Rats, Mice, Inbred C57BL, Organic anion-transporting polypeptide, 030104 developmental biology, Endocrinology, biology.protein, Molecular Medicine, Multidrug Resistance-Associated Proteins, Steatosis, Xenobiotic, 030217 neurology & neurosurgery, Protein Binding
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4
المؤلفون: Yueping Zhang, Petia A. Shipkova, Bethanne M Warrack, David M Nelson, Linna Wang, Runlan Huo, Jian Chen, Erika Panfen, Xue-Qing Chen, Marcus Fancher, Qian Ruan, Lisa J. Christopher, Yongjun Xue, Michael Sinz, Hong Shen
المصدر: Drug Metabolism and Disposition. :DMD-AR
مصطلحات موضوعية: Pharmacology, Pharmaceutical Science
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5
المؤلفون: Punit Marathe, Ming Yao, Hong Shen, Michael Sinz, A. David Rodrigues, Mingshe Zhu
المصدر: Molecular Pharmaceutics. 16:4065-4076
مصطلحات موضوعية: Organic Cation Transport Proteins, Organic anion transporter 1, Biological Transport, Active, Pharmaceutical Science, 02 engineering and technology, Organic Anion Transporters, Sodium-Independent, Pharmacology, Transfection, 030226 pharmacology & pharmacy, Madin Darby Canine Kidney Cells, Dabigatran, Inhibitory Concentration 50, 03 medical and health sciences, Dogs, 0302 clinical medicine, Oral administration, Drug Discovery, medicine, Animals, Humans, Drug Interactions, ATP Binding Cassette Transporter, Subfamily B, Member 1, P-glycoprotein, Kidney, Organic cation transport proteins, biology, Chemistry, Organic Cation Transporter 2, 021001 nanoscience & nanotechnology, Quinidine, Renal Elimination, HEK293 Cells, Ketoconazole, medicine.anatomical_structure, Verapamil, Renal physiology, biology.protein, Molecular Medicine, Efflux, 0210 nano-technology, Octamer Transcription Factor-1, medicine.drug
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6
المؤلفون: Andrew P. Degnan, Haiquan Fang, Tatyana Zvyaga, Zuzana Haarhoff, Claude A. Quesnelle, Melissa Kramer, Frank Marsilio, Richard A. Westhouse, John S. Tokarski, Shilpa Madari, Jiuqiao Zhao, Amy Wiebesiek, Chunhong Yan, Francis Y. Lee, Michael Sinz, John Morrison, Jean Simmermacher-Mayer, Carolynn Fanslau, Steven Sheriff, Lisa Huang, Ashvinikumar V. Gavai, Chunshan Xie, Matthew D. Hill, Gerry Everlof
المصدر: Bioorganicmedicinal chemistry letters. 51
مصطلحات موضوعية: Stereochemistry, Cell Survival, Clinical Biochemistry, Pharmaceutical Science, Structural diversity, Administration, Oral, Antineoplastic Agents, Triple Negative Breast Neoplasms, Biochemistry, Polar surface area, BET inhibitor, Mice, Structure-Activity Relationship, Drug Development, Drug Discovery, medicine, Animals, Humans, Molecular Biology, Chemotype, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Cancer, Mammary Neoplasms, Experimental, Proteins, medicine.disease, In vitro, Bromodomain, Molecular Medicine, Drug Screening Assays, Antitumor, Carbolines
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7
المؤلفون: R. Marcus Fancher, Hong Shen, Pawel D. Puszczalo, Shen-Jue Chen, Xue-Qing Chen, David J. Shuster, Cliff Chen, Zheng Yang, Yueping Zhang, Michael Sinz
المصدر: The Journal of pharmacology and experimental therapeutics. 375(1)
مصطلحات موضوعية: 0301 basic medicine, Male, Coproporphyrins, Abcg2, CYP3A, Gene Expression, Pharmacology, Kidney, 03 medical and health sciences, Solute Carrier Organic Anion Transporter Family Member 1B3, 0302 clinical medicine, In vivo, Gene expression, Intestine, Small, polycyclic compounds, Animals, Inducer, biology, Chemistry, Multidrug resistance-associated protein 2, Kidney metabolism, biochemical phenomena, metabolism, and nutrition, Hydroxycholesterols, Organic anion-transporting polypeptide, Macaca fascicularis, 030104 developmental biology, Liver, biology.protein, Molecular Medicine, Female, Rifampin, 030217 neurology & neurosurgery, Biomarkers
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8
المؤلفون: Hamza Kandoussi, T. Thanga Mariappan, Jianing Zeng, Vinay K. Holenarsipur, Yueping Zhang, Michael Sinz, Hong Shen
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 48(10)
مصطلحات موضوعية: Male, Coproporphyrins, Organic anion transporter 1, Pharmaceutical Science, Administration, Oral, Endogeny, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, Inhibitory Concentration 50, Solute Carrier Organic Anion Transporter Family Member 1B3, 0302 clinical medicine, Oral administration, In vivo, Furosemide, medicine, Humans, Drug Interactions, biology, Chemistry, Liver-Specific Organic Anion Transporter 1, Probenecid, Transporter, In vitro, Healthy Volunteers, Organic anion-transporting polypeptide, HEK293 Cells, 030220 oncology & carcinogenesis, Area Under Curve, biology.protein, Hepatocytes, Female, medicine.drug
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9
المؤلفون: Mahesh Paschapur, Jeffrey M. Brown, Tanmaya Bastia, Lawrence R. Marcin, Jayakumar Sankara Warrier, Srinivasan Thangathirupathy, Joanne J. Bronson, Raja Reddy Kallem, Huiping Zhang, Jyoti Gulia, Alda Fernandes, Digavalli V. Sivarao, Deborah Keavy, Amy Newton, Jianqing Li, Pattipati S. Naidu, Kuchibhotla Vijaya Kumar, James Kempson, Michael R. Weed, Rick L. Pieschl, Mark Bookbinder, Charlie F. Albright, Kimberly Newberry, Yu-Wen Li, Dalton King, Manjunath Ramarao, Jean Simmermacher, Linda J. Bristow, Meenakshee Sinha, Eric Shields, Lorin A. Thompson, John E. Macor, Charulatha Sanmathi, Imadul Islam, B.N. Srikumar, Richard E. Olson, John D. Graef, Arvind Mathur, Narasimharaju Kalidindi, Joseph Polino, Michael Sinz, Thaddeus F. Molski, Jayant Aher, Reeba K. Vikramadithyan
المصدر: Journal of Pharmacology and Experimental Therapeutics. 363:377-393
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Allosteric modulator, Chemistry, digestive, oral, and skin physiology, Allosteric regulation, Glutamate receptor, Long-term potentiation, Prodrug, stomatognathic diseases, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, In vivo, Molecular Medicine, Receptor, 030217 neurology & neurosurgery, Ex vivo
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10
المؤلفون: Katherine A. Grant-Young, Andrew Nickel, Rajesh Onkardas Bora, Prakash Anjanappa, Bender John A, Kevin Kish, Kap-Sun Yeung, Dawn D. Parker, Joseph Raybon, Mark R. Witmer, Karen Rigat, Matthew G. Soars, Steven Sheriff, Yue-Zhong Shu, Kenneth S. Santone, Prashantha Gunaga, Kyle Parcella, Nicholas A. Meanwell, Jay O. Knipe, Susan B. Roberts, Alicia Ng, Michael Sinz, Kathy Mosure, Ying-Kai Wang, Brett R. Beno, Mengping Liu, Elizabeth Colston, Dennis M. Grasela, John F. Kadow, Qi Gao, Min Gao, Umesh Hanumegowda, Roy Haskell, Julie A. Lemm, Xiaoliang Zhuo, Changhong Wan, Kumaravel Selvakumar
المصدر: Journal of Medicinal Chemistry. 60:4369-4385
مصطلحات موضوعية: Male, 0301 basic medicine, Hepatitis C virus, Allosteric regulation, RNA-dependent RNA polymerase, Hepacivirus, Viral Nonstructural Proteins, medicine.disease_cause, Antiviral Agents, 01 natural sciences, Rats, Sprague-Dawley, 03 medical and health sciences, chemistry.chemical_compound, Dogs, Allosteric Regulation, Drug Discovery, medicine, Animals, Humans, Benzofuran, NS5B, Benzofurans, Ligand efficiency, 010405 organic chemistry, Chemistry, Drug discovery, Haplorhini, Hepatitis C, Rats, 0104 chemical sciences, Molecular Docking Simulation, 030104 developmental biology, Biochemistry, Benzothiadiazine, Molecular Medicine, Allosteric Site
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11
المؤلفون: Michael Sinz, Yang Hong, Jinping Gan, R. Marcus Fancher, Yurong Lai, Xiaomei Gu, Lifei Wang, Yuan Tian, Hong Shen
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 48(8)
مصطلحات موضوعية: Male, Coproporphyrins, Cmax, Drug Evaluation, Preclinical, Pharmaceutical Science, Administration, Oral, Biological Availability, Pharmacology, Kidney, Excretion, Mice, Pharmacokinetics, Cyclosporin a, medicine, Distribution (pharmacology), Animals, Drug Interactions, Tissue Distribution, biology, Chemistry, Liver-Specific Organic Anion Transporter 1, Bioavailability, Probenecid, Organic anion-transporting polypeptide, Macaca fascicularis, Intestinal Absorption, Liver, Area Under Curve, biology.protein, Cyclosporine, Administration, Intravenous, Rifampin, Biomarkers, medicine.drug, Half-Life
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12
المؤلفون: Punit Marathe, Michael Sinz, Erika Panfen, Hong Shen, Yueping Zhang, Marcus Fancher
المصدر: Molecular pharmaceutics. 16(6)
مصطلحات موضوعية: Organic anion transporter 1, Organic Cation Transport Proteins, Estrone, Pharmaceutical Science, Organic Anion Transporters, 02 engineering and technology, Pharmacology, 030226 pharmacology & pharmacy, Cell Line, 03 medical and health sciences, chemistry.chemical_compound, Solute Carrier Organic Anion Transporter Family Member 1B3, 0302 clinical medicine, In vivo, Estrone sulfate, Tandem Mass Spectrometry, Drug Discovery, medicine, Animals, Humans, Rosuvastatin, Drug Interactions, Rosuvastatin Calcium, Pitavastatin, IC50, Sulfonamides, Organic cation transport proteins, biology, Organic Cation Transporter 1, Biological Transport, 021001 nanoscience & nanotechnology, Isoquinolines, Organic anion-transporting polypeptide, Macaca fascicularis, chemistry, biology.protein, Hepatocytes, Molecular Medicine, 0210 nano-technology, medicine.drug
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13
المؤلفون: Weiqi Chen, Jinping Gan, Punit Marathe, Erika Panfen, Hong Shen, Yueping Zhang, Michael Sinz
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 47(11)
مصطلحات موضوعية: Quinidine, Male, Organic anion transporter 1, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, In vivo, medicine, Potency, Humans, Drug Interactions, IC50, Organic cation transport proteins, biology, Chemistry, Organic Cation Transporter 1, Metformin, medicine.anatomical_structure, HEK293 Cells, 030220 oncology & carcinogenesis, Hepatocyte, biology.protein, Cyclosporine, Hepatocytes, medicine.drug
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14
المؤلفون: Heidi J. Einolf, Susanna Tse, Tonika Bohnert, Sirimas Sudsakorn, Ying-Hong Wang, David Moore, Jim Keirns, Ling He, Robert L. Walsky, Rangaraj Narayanan, Wanping Geng, Aarti Patel, Louis Leung, W. George Lai, Xiaoqing Yang, Ralph Stearns, Dieter Lang, Michael Sinz, Yuan Chen, Chuang Lu, Jan Wahlstrom, Ian Templeton
المصدر: Drug Metabolism and Disposition. 44:1399-1423
مصطلحات موضوعية: Drug, Drug Industry, Computer science, media_common.quotation_subject, Population, Decision tree, Pharmaceutical Science, Pharmacology, Risk Assessment, 030226 pharmacology & pharmacy, Substrate Specificity, 03 medical and health sciences, 0302 clinical medicine, Species Specificity, New chemical entity, Drug Discovery, Animals, Humans, Computer Simulation, Drug Interactions, education, Biotransformation, media_common, education.field_of_study, Decision Trees, Perspective (graphical), Models, Theoretical, Enzymes, Kinetics, Identification (information), Drug metabolizing enzymes, Pharmaceutical Preparations, Risk analysis (engineering), 030220 oncology & carcinogenesis, Risk assessment
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15
المؤلفون: Deepak Ahire, Saranjit Singh, Murali Subramanian, Dilip Kumar Singh, Benjamin M. Johnson, Priyadeep Bhutani, Michael Sinz, Amol Patil, Mayurbhai Kathadbhai Ladumor, Shyam H. Kamble, Sivaprasad Putlur
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 49(12)
مصطلحات موضوعية: Male, Allylic rearrangement, Antifungal Agents, Health, Toxicology and Mutagenesis, Reactive intermediate, Alkyne, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, Aldehyde, 03 medical and health sciences, chemistry.chemical_compound, Mice, 0302 clinical medicine, Dogs, Tandem Mass Spectrometry, Animals, Humans, Terbinafine, Pharmacology, chemistry.chemical_classification, General Medicine, Glutathione, Haplorhini, Rats, chemistry, 030220 oncology & carcinogenesis, Toxicity, Michael reaction, Hepatocytes, Microsomes, Liver, Drug metabolism
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16Academic Journal
المؤلفون: Anders Christensen, Mike Cowlishaw, Charles Daney, Stan Murawski, Carl Feinberg, Rainer F. Hauser, Pat Meehan, Paul Heaney, Walter Pachl, Stephen G. Price, Anthony Rudd, David I. Shriver, Michael Sinz, P. Joseph Vertucci, Bebo White, Pete Zybrick
المساهمون: The Pennsylvania State University CiteSeerX Archives
مصطلحات موضوعية: Neil Milsted
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.393.4410; http://www.slac.stanford.edu/pubs/slacreports/reports02/slac-r-401.pdf
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المؤلفون: Arvind Mathur, Rajareddy Kallem, Thaddeus F. Molski, Manjunatha Narayana Rao Kamble, Michelle Nophsker, Huiping Zhang, Murali Subramanian, Dalton King, Linda J. Bristow, Lawrence R. Marcin, B.N. Srikumar, Grandhi Venkat Ram Krishna Mohan Gupta, Kumar Kuchibhotla Vijaya, Jayakumar Sankara Warrier, Michael Sinz, Charulatha Sanmathi, G. Nagaraju, Xiaoliang Zhuo, Raju Mannoori, Imadul Islam, Alicia Ng, Pattipati S. Naidu, Eric Shields, Joanne J. Bronson, Narasimharaju Kalidindi, Reeba K. Vikramadithyan, Gopikishan Tonukunuru, Lorin A. Thompson, James Kempson, Srinivasan Thangathirupathy, Jogi Srinivas, Bradley C. Pearce, Jyoti Gulia, Jean Simmermacher, Srinivas Cheruku, Mahesh Paschapur, Jianliang Shi, John E. Macor, Jayant Aher, Manjunath Ramarao, Charlie F. Albright, Richard E. Olson, Rex Denton, Aliphedi B. Reddy, Hyunsoo Park, Karageorge George N, Tanmaya Bastia, Jianqing Li
المصدر: ACS medicinal chemistry letters. 9(5)
مصطلحات موضوعية: 0301 basic medicine, Allosteric modulator, Chemistry, Organic Chemistry, Allosteric regulation, Pharmacology, Prodrug, medicine.disease, Biochemistry, In vitro, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, In vivo, Drug Discovery, medicine, Major depressive disorder, IC50, 030217 neurology & neurosurgery, Ex vivo
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18
المؤلفون: Y. Amy Siu, Jairam Palamanda, Robert L. Walsky, George Zhang, David B. Buckley, Michael A. Mohutsky, Donald J. Tweedie, Liangfu Chen, Magalie Pardon, Shannon Dallas, Suresh K. Balani, Diane Ramsden, Barry Jones, Heidi J. Einolf, Jane R. Kenny, Odette A. Fahmi, Michael Sinz, Niresh Hariparsad, Joshua G. Dekeyser
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 45(10)
مصطلحات موضوعية: Pharmacology, Medical education, Drug Industry, United States Food and Drug Administration, Drug-drug interaction, MEDLINE, Pharmaceutical Science, Induction time, Positive control, Down-Regulation, 030226 pharmacology & pharmacy, United States, Interaction studies, Food and drug administration, 03 medical and health sciences, Cytochrome P-450 CYP2B6, 0302 clinical medicine, Cytochrome P-450 Enzyme System, Pharmaceutical Preparations, 030220 oncology & carcinogenesis, Agency (sociology), Humans, Drug Interactions, Duration (project management), Psychology
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19
المؤلفون: Michael Sinz
المصدر: Current drug metabolism. 18(1)
مصطلحات موضوعية: Pharmacology, Publishing, Biological Products, Drug Delivery Systems, Pharmaceutical Preparations, Clinical Biochemistry, Proteins, Periodicals as Topic
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20
المؤلفون: Jean Simmermacher, Michael Sinz
المصدر: Drug metabolism letters. 11(2)
مصطلحات موضوعية: Transcriptional Activation, Indoles, medicine.drug_class, Clinical Biochemistry, Primary Cell Culture, Pharmaceutical Science, Receptors, Cytoplasmic and Nuclear, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Downregulation and upregulation, Species Specificity, Coenzyme A Ligases, medicine, Animals, Humans, Pharmacology (medical), RNA, Messenger, Gene, Cells, Cultured, chemistry.chemical_classification, Bile acid, Chemistry, Multidrug resistance-associated protein 2, Biochemistry (medical), Azepines, Isoxazoles, Bile Salt Export Pump, Molecular biology, Amino acid, Rats, Up-Regulation, Nuclear receptor, 030220 oncology & carcinogenesis, Hepatocytes, Farnesoid X receptor, Acyltransferases