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1Academic Journal
المؤلفون: Micael Rodrigues Cunha, Maurício Temotheo Tavares, Thais Batista Fernandes, Roberto Parise-Filho
المصدر: Molecules, Vol 26, Iss 6, p 1521 (2021)
مصطلحات موضوعية: peppers, Piper, Capsicum, secondary metabolites, antitumor activity, apoptosis, Organic chemistry, QD241-441
وصف الملف: electronic resource
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2Academic Journal
المؤلفون: Otávio Augusto Chaves, Maurício Temotheo Tavares, Micael Rodrigues Cunha, Roberto Parise-Filho, Carlos Maurício R. Sant’Anna, José Carlos Netto-Ferreira
المصدر: Biomolecules, Vol 8, Iss 3, p 78 (2018)
مصطلحات موضوعية: human serum albumin, RPF101, capsaicin, multi-spectroscopy, molecular docking, Microbiology, QR1-502
وصف الملف: electronic resource
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3
المؤلفون: Rajesh Bhardwaj, Christoph Romanin, Jean-Louis Reymond, Aline Lucie Carrel, Roberto Parise-Filho, Micael Rodrigues Cunha, Matthias A. Hediger, Sonja Lindinger
المصدر: RSC Medicinal Chemistry
Rodrigues Cunha, Micael; Bhardwaj, Rajesh; Carrel, Aline Lucie; Lindinger, Sonja; Romanin, Christoph; Parise-Filho, Roberto; Hediger, Matthias A.; Reymond, Jean-Louis (2020). Natural product inspired optimization of a selective TRPV6 calcium channel inhibitor. RSC Medicinal Chemistry, 11(9), pp. 1032-1040. Royal Society of Chemistry 10.1039/D0MD00145G <http://dx.doi.org/10.1039/D0MD00145G>
Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USPمصطلحات موضوعية: TRPV6, TRPV5, Pharmaceutical Science, 610 Medicine & health, Biochemistry, 03 medical and health sciences, Transient receptor potential channel, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, Calcium flux, 540 Chemistry, Ion channel, 030304 developmental biology, Pharmacology, 0303 health sciences, Natural product, Voltage-dependent calcium channel, Calcium channel, Organic Chemistry, CÁLCIO, 3. Good health, Chemistry, chemistry, 030220 oncology & carcinogenesis, Biophysics, Molecular Medicine, 570 Life sciences, biology
وصف الملف: application/pdf
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4
المؤلفون: Matthias A. Hediger, Rajesh Bhardwaj, Micael Rodrigues Cunha, Appu K. Singh, Jean-Louis Reymond, Isabella Derler, Sonja Lindinger, Christoph Romanin, Arthur Neuberger, Gergely Gyimesi, Kirill D. Nadezhdin, Alexander I. Sobolevsky
المصدر: Bhardwaj, Rajesh; Lindinger, Sonja; Neuberger, Arthur; Nadezhdin, Kirill D.; Singh, Appu K.; R. Cunha, Micael; Derler, Isabella; Gyimesi, Gergely; Reymond, Jean-Louis; Hediger, Matthias A.; Romanin, Christoph; Sobolevsky, Alexander I. (2020). Inactivation-mimicking block of the epithelial calcium channel TRPV6. Science Advances, 6(48), eabe1508. American Association for the Advancement of Science 10.1126/sciadv.abe1508 <http://dx.doi.org/10.1126/sciadv.abe1508>
Science Advancesمصطلحات موضوعية: TRPV6, Calmodulin, TRPV Cation Channels, 610 Medicine & health, 03 medical and health sciences, 0302 clinical medicine, Structural Biology, 540 Chemistry, Humans, Binding site, Ion channel, Research Articles, 030304 developmental biology, Calcium metabolism, 0303 health sciences, Multidisciplinary, biology, Calcium channel, Mutagenesis, Cryoelectron Microscopy, SciAdv r-articles, biology.protein, Molecular mechanism, Biophysics, 570 Life sciences, Calcium, Calcium Channels, 030217 neurology & neurosurgery, Research Article
وصف الملف: application/pdf
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5
المؤلفون: Micael Rodrigues Cunha
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Capsaicin, Capsaicinoid, Pharmacology, Cytotoxicity
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6
المؤلفون: Micael Rodrigues Cunha
المساهمون: Roberto Parise Filho, João Paulo dos Santos Fernandes, Daniel Fabio Kawano, Jean-louis Reymond
المصدر: Biblioteca Digital de Teses e Dissertações da USP
Universidade de São Paulo (USP)
instacron:USP -
7
المؤلفون: Barbara Behr Martins, Maurício Temotheo Tavares, Rajesh Bhardwaj, Vanessa Zambelli, Euzébio Guimarães Barbosa, Micael Rodrigues Cunha, Roberto Parise-Filho, Ricardo A. Azevedo, Yara Cury, Gustavo José Vasco Pereira, Matthias A. Hediger
المصدر: Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USPمصطلحات موضوعية: MAPK/ERK pathway, Models, Molecular, Programmed cell death, Clinical Biochemistry, TRPV1, Pharmaceutical Science, Apoptosis, Pharmacology, Biochemistry, chemistry.chemical_compound, Drug Discovery, 540 Chemistry, Cytotoxic T cell, Humans, 610 Medicine & health, Molecular Biology, Melanoma, Drug discovery, Organic Chemistry, chemistry, Biological target, Capsaicin, UREIA, Molecular Medicine, 570 Life sciences, biology
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8
المؤلفون: Rajesh Bhardwaj, Jean-Louis Reymond, Matthias A. Hediger, Christoph Romanin, Carmen Butorac, Micael Rodrigues Cunha, Sonja Lindinger
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: TRPV6, 010405 organic chemistry, Calcium channel, Organic Chemistry, Cancer, medicine.disease, 01 natural sciences, Biochemistry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, Transient receptor potential channel, Azobenzene, chemistry, Drug Discovery, 540 Chemistry, Biophysics, medicine, 570 Life sciences, biology, 610 Medicine & health, IC50
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9
المصدر: African Journal of Pharmacy and Pharmacology. 9:1-5
مصطلحات موضوعية: Pharmacology, Analgesic effect, education.field_of_study, biology, medicine.drug_class, business.industry, Ruta graveolens, Population, Analgesic, Pharmaceutical Science, Biological activity, biology.organism_classification, Sedative, medicine, Warm water, Antispasmodic, education, business, medicine.drug
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10
المؤلفون: Marina Candido Primi, Roberto Parise-Filho, Micael Rodrigues Cunha, Maurício Temotheo Tavares, Camila Felix de Carvalho, Nuno Albuquerque Tavares Ferreira da Silva
المصدر: Repositório Institucional da USP (Biblioteca Digital da Produção Intelectual)
Universidade de São Paulo (USP)
instacron:USPمصطلحات موضوعية: 0301 basic medicine, Class (computer programming), Chemistry, Process (engineering), business.industry, In silico, Teaching method, education, 05 social sciences, BASES DE DADOS, 050301 education, Computer-Assisted Instruction, Context (language use), General Chemistry, Pharmacology, Education, 03 medical and health sciences, 030104 developmental biology, Human–computer interaction, Cheminformatics, business, 0503 education, Biomedicine
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11
المؤلفون: Renata Parruca Sakata, Thais B. Fernandes, Wanda P. Almeida, Roberto Parise-Filho, Thalita Marcílio Candido, Micael Rodrigues Cunha, Maurício Temotheo Tavares, Euzébio Guimarães Barbosa, André Rolim Baby
المصدر: Archiv der Pharmazie. 350:1700163
مصطلحات موضوعية: 0301 basic medicine, Molecular model, 010405 organic chemistry, Chemistry, Aché, Pharmaceutical Science, Pharmacology, medicine.disease, 01 natural sciences, Acetylcholinesterase, language.human_language, 0104 chemical sciences, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Biochemistry, Drug Discovery, language, medicine, Dementia, Binding site, Cholinergic neuron, Donepezil, IC50, medicine.drug
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12
المؤلفون: Karinne Esteves Prado
المساهمون: Roberto Parise Filho, Gisele de Freitas Gauze Bandoch, Micael Rodrigues Cunha, Ricardo Augusto Massarico Serafim
المصدر: Biblioteca Digital de Teses e Dissertações da USP
Universidade de São Paulo (USP)
instacron:USP -
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المؤلفون: Vitor de Bastos Navarausckas
المساهمون: Roberto Parise Filho, Micael Rodrigues Cunha, Marcio Vinícius Bertacine Dias, Mauricio Temotheo Tavares
المصدر: Biblioteca Digital de Teses e Dissertações da USP
Universidade de São Paulo (USP)
instacron:USP