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1
المؤلفون: Rhonda M Lachance, Stephen R. Rapp, John J. Parlow, Peter Harris, Rita M. Huff, Case Brenda, Mary W. Burney, Thomas J. Girard, Deborah A. Mischke, Ennis Michael D, Rhonda S. Woerndle, Kerri A. Hall, Ronald R. Hiebsch
المصدر: Journal of Medicinal Chemistry. 53:2010-2037
مصطلحات موضوعية: Adult, Male, Magnetic Resonance Spectroscopy, Adolescent, Platelet Aggregation, Pyridines, Stereochemistry, Administration, Oral, Biological Availability, CHO Cells, Mass Spectrometry, Piperazines, Structure-Activity Relationship, Young Adult, chemistry.chemical_compound, Cricetulus, Glutamates, In vivo, Cricetinae, Drug Discovery, Pyridine, Purinergic P2 Receptor Antagonists, Animals, Humans, Potency, Structure–activity relationship, Aged, Receptors, Purinergic P2, Antagonist, Middle Aged, Receptors, Purinergic P2Y12, Rats, Bioavailability, Piperazine, chemistry, Molecular Medicine, Female, Selectivity, Platelet Aggregation Inhibitors
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2
المؤلفون: John J, Parlow, Mary W, Burney, Brenda L, Case, Thomas J, Girard, Kerri A, Hall, Peter K, Harris, Ronald R, Hiebsch, Rita M, Huff, Rhonda M, Lachance, Deborah A, Mischke, Stephen R, Rapp, Rhonda S, Woerndle, Michael D, Ennis
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1388-1394
مصطلحات موضوعية: Molecular Structure, Platelet Aggregation, Pyridines, Organic Chemistry, Clinical Biochemistry, Administration, Oral, Glutamic Acid, Pharmaceutical Science, CHO Cells, Biochemistry, Receptors, Purinergic P2Y12, Rats, Inhibitory Concentration 50, Structure-Activity Relationship, Cricetulus, Dogs, Fibrinolytic Agents, Piperidines, Cricetinae, Drug Discovery, Purinergic P2 Receptor Antagonists, Animals, Humans, Molecular Medicine, Molecular Biology
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3Piperazinyl-glutamate-pyrimidines as potent P2Y12 antagonists for inhibition of platelet aggregation
المؤلفون: Kerri A. Hall, Rita M. Huff, Rhonda M. Lachance, Ennis Michael D, Rhonda S. Woerndle, Ronald R. Hiebsch, John J. Parlow, Stephen R. Rapp, Deborah A. Mischke, Brenda L. Case, Mary W. Burney, Thomas J. Girard
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:6148-6156
مصطلحات موضوعية: Male, Platelet Aggregation, Pyrimidine, Clinical Biochemistry, Glutamic Acid, Pharmaceutical Science, Pharmacology, Biochemistry, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, Fibrinolytic Agents, Piperidines, In vivo, Drug Discovery, Purinergic P2 Receptor Antagonists, Animals, Humans, Potency, Molecular Biology, Receptors, Purinergic P2, Organic Chemistry, Antagonist, Glutamate receptor, Receptors, Purinergic P2Y12, In vitro, Rats, Bioavailability, Pyrimidines, chemistry, Molecular Medicine, Piperidine
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4
المؤلفون: Mary W. Burney, Louis J. Muglia, Sherri K. Vogt, Paulette M. Johnson
المصدر: American Journal of Physiology-Endocrinology and Metabolism. 282:E650-E656
مصطلحات موضوعية: Lipopolysaccharides, Male, Lipopolysaccharide, Corticotropin-Releasing Hormone, Physiology, Endocrinology, Diabetes and Metabolism, medicine.medical_treatment, Systemic inflammation, Mice, chemistry.chemical_compound, Neuropeptide Y, media_common, Mice, Knockout, Mice, Inbred C3H, Sulfonamides, Leptin, Anorexia, Isoenzymes, Cytokine, Cytokines, medicine.symptom, medicine.medical_specialty, media_common.quotation_subject, Hypothalamus, Inflammation, Biology, Physiology (medical), Internal medicine, Weight Loss, medicine, Animals, Cyclooxygenase Inhibitors, RNA, Messenger, Cyclooxygenase 2 Inhibitors, Immunity, Membrane Proteins, Appetite, Endocrinology, chemistry, Cyclooxygenase 2, Prostaglandin-Endoperoxide Synthases, Cyclooxygenase 1, Prostaglandins, biology.protein, Pyrazoles, Cyclooxygenase, Energy Intake, Energy Metabolism
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5
المصدر: Journal of Virology. 73:3682-3691
مصطلحات موضوعية: CCR1, Muromegalovirus, Time Factors, Chemokine receptor CCR5, viruses, RNA Splicing, Molecular Sequence Data, Immunology, CCR3, CCL7, Microbiology, Cell Line, Mice, Chemokine receptor, Polysaccharides, Virology, Animals, CCR10, Amino Acid Sequence, RNA, Messenger, CX3CL1, CCL13, biology, Fibroblasts, Molecular biology, Eukaryotic Cells, Chemokines, CC, Insect Science, COS Cells, biology.protein, Pathogenesis and Immunity, RNA, Viral, Asparagine, Protein Processing, Post-Translational
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6
المؤلفون: Mary W. Burney, Ted Baginski, Fei Shih, Stephen R. Rapp, Holly Meade, Kimberly Shevlin, Dean Welsch, Mike Baratta, Deborah Knoerzer, Sharon Rouw
المصدر: D61. ANIMAL MODELS OF PULMONARY ARTERIAL HYPERTENSION: NEW IDEAS AND INSIGHTS.
مصطلحات موضوعية: business.industry, Medicine, Pharmacology, business
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7
المؤلفون: Dean Welsch, Mary W. Burney, Stephen R. Rapp, Deborah Knoerzer, Ted Baginski, Kimberly Wade, Connie Fan, Joe Palandra, Karen Regina, Fei Shih, Sharon Rouw
المصدر: A58. ANIMAL MODELS OF PULMONARY FIBROSIS.
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, business.industry, Pulmonary fibrosis, Medicine, Thrombin-Activatable Fibrinolysis Inhibitor, Pharmacology, business, medicine.disease, Bleomycin
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8
المؤلفون: Ted Baginski, Connie Fan, Fei Shih, Deborah Knoerzer, Stephen R. Rapp, Karen Regina, Sharon Rouw, Kimberly Wade, Mary W. Burney, Dean Welsch
المصدر: A58. ANIMAL MODELS OF PULMONARY FIBROSIS.
مصطلحات موضوعية: chemistry.chemical_compound, Pathology, medicine.medical_specialty, Broad spectrum, chemistry, business.industry, Receptor tyrosine kinase inhibitor, Pulmonary fibrosis, Cancer research, Medicine, business, medicine.disease, Bleomycin
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9
المؤلفون: Peter Harris, Kerri A. Hall, Mary W. Burney, Thomas J. Girard, Stephen R. Rapp, Rita M. Huff, Ronald R. Hiebsch, Rhonda M Lachance, Case Brenda, Ennis Michael D, Rhonda S. Woerndle, Deborah A. Mischke, John J. Parlow
المصدر: Bioorganicmedicinal chemistry letters. 19(16)
مصطلحات موضوعية: Male, Platelet Aggregation, Stereochemistry, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Biological Availability, Glutamic Acid, Biochemistry, Chemical synthesis, Piperazines, Rats, Sprague-Dawley, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Oral administration, Drug Discovery, Pyridine, Purinergic P2 Receptor Antagonists, Structure–activity relationship, Animals, Humans, Molecular Biology, Receptors, Purinergic P2, Organic Chemistry, Antagonist, Receptors, Purinergic P2Y12, Recombinant Proteins, Bioavailability, Rats, Piperazine, chemistry, Molecular Medicine, Platelet Aggregation Inhibitors
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10
المؤلفون: David J. Orlicky, Stuart A Ross, Yumi Kasai, Xiaomin Song, Mary W Burney
المصدر: Biochemical and biophysical research communications. 302(2)
مصطلحات موضوعية: Coxsackie and Adenovirus Receptor-Like Membrane Protein, Biophysics, Biology, Biochemistry, Adenoviridae, chemistry.chemical_compound, Mice, Multiplicity of infection, Transduction, Genetic, Adipocyte, Adipocytes, Animals, Receptor, Molecular Biology, Cells, Cultured, 3T3-L1, Cell Biology, Transfection, 3T3 Cells, Virology, Cell biology, Insulin receptor, chemistry, Adipogenesis, biology.protein, Receptors, Virus, GLUT4
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11
المؤلفون: K Wade, F Shih, D Knoerzer, C Fan, T Baginski, K Regina, Stephen R. Rapp, D Welsch, S Rouw, Mary W. Burney
المصدر: Journal of Inflammation (London, England)
مصطلحات موضوعية: Lung, biology, business.industry, Sunitinib, Clinical Biochemistry, Cell Biology, respiratory system, Pharmacology, Bleomycin, medicine.disease, respiratory tract diseases, Vascular endothelial growth factor, chemistry.chemical_compound, medicine.anatomical_structure, chemistry, Fibrosis, Pulmonary fibrosis, Poster Presentation, biology.protein, Medicine, business, Tyrosine kinase, Platelet-derived growth factor receptor, medicine.drug