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1Academic Journal
المؤلفون: Mark P. Grillo (2413657), Svetlana Markova (3545603), Marc Evanchik (5806811), Marc Trellu (9650521), Patricia Moliner (9650524), Priscilla Brun (5806805), Anne Perreard-Dumaine (9650527), Pascale Vicat (8053706), Chun Yang (251691), James P. Driscoll (2159146), Tim J. Carlson (9650530)
مصطلحات موضوعية: Biochemistry, Medicine, Microbiology, Cell Biology, Physiology, Pharmacology, Immunology, Developmental Biology, Cancer, Mental Health, Infectious Diseases, Virology, Chemical Sciences not elsewhere classified, Cardiac myosin activator, danicamtiv, MYK-491, pharmacokinetics, allometric scaling, human prediction, metabolites
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2
المؤلفون: Mark P. Grillo
المصدر: Transporters and Drug-Metabolizing Enzymes in Drug Toxicity
مصطلحات موضوعية: chemistry.chemical_classification, Acyl-CoA formation, chemistry.chemical_compound, Transacylation, Chemistry, Stereochemistry, Carboxylic acid, Acyl glucuronidation, Covalent binding, Glutathione, Potential toxicity
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3
المؤلفون: Mark P. Grillo, Svetlana Markova, Marc Evanchik, Marc Trellu, Patricia Moliner, Priscilla Brun, Anne Perreard-Dumaine, Pascale Vicat, Chun Yang, James P. Driscoll, Tim J. Carlson
المصدر: Xenobiotica. 51:222-238
مصطلحات موضوعية: medicine.medical_specialty, Health, Toxicology and Mutagenesis, Toxicology, Left ventricular enlargement, 030226 pharmacology & pharmacy, Biochemistry, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, In vivo, Internal medicine, Myosin, medicine, cardiovascular diseases, Pharmacology, business.industry, Activator (genetics), Dilated cardiomyopathy, General Medicine, medicine.disease, In vitro, 030220 oncology & carcinogenesis, Heart failure, cardiovascular system, Cardiology, business
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4
المؤلفون: Mark P, Grillo, Svetlana, Markova, Marc, Evanchik, Marc, Trellu, Patricia, Moliner, Priscilla, Brun, Anne, Perreard-Dumaine, Pascale, Vicat, James P, Driscoll, Tim J, Carlson
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 51(2)
مصطلحات موضوعية: Cardiomyopathy, Dilated, Male, Mice, Dogs, Hepatocytes, Microsomes, Liver, Animals, Biological Availability, Humans, Caco-2 Cells, Myosins, Protein Binding, Rats
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5Academic Journal
المؤلفون: Mark P. Grillo, Grazia Chiellini, Marco Tonelli, Leslie, Z. Benet
المساهمون: The Pennsylvania State University CiteSeerX Archives
وصف الملف: application/pdf
Relation: http://citeseerx.ist.psu.edu/viewdoc/summary?doi=10.1.1.1027.2582; http://dmd.aspetjournals.org/content/29/9/1210.full.pdf
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6
المؤلفون: Marc J. Evanchik, Priscilla Brun, John C L Erve, Nicole V Haste, Mark P. Grillo, Svetlana Markova, Ryan Dick, Timothy J. Carlson, James P Driscoll
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 49(6)
مصطلحات موضوعية: Male, Benzylamines, Allosteric modulator, Metabolic Clearance Rate, Health, Toxicology and Mutagenesis, Pharmacology, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, Rats, Sprague-Dawley, 03 medical and health sciences, 0302 clinical medicine, Dogs, Pharmacokinetics, Cytochrome P-450 Enzyme System, In vivo, medicine, Animals, Humans, Drug Interactions, Beta (finance), Uracil, Mice, Inbred ICR, Chemistry, Hypertrophic cardiomyopathy, General Medicine, Cardiomyopathy, Hypertrophic, medicine.disease, Small molecule, In vitro, Macaca fascicularis, 030220 oncology & carcinogenesis, Hepatocytes, Microsomes, Liver, Caco-2 Cells, Cardiac Myosins, Drug metabolism
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7
المؤلفون: Mark P. Grillo
المصدر: Expert Opinion on Drug Metabolism & Toxicology. 11:1281-1302
مصطلحات موضوعية: Drug, Magnetic Resonance Spectroscopy, Drug-Related Side Effects and Adverse Reactions, media_common.quotation_subject, Reactive intermediate, Pharmacology, Toxicology, medicine.disease_cause, Pharmacokinetics, Tandem Mass Spectrometry, medicine, Animals, Humans, media_common, Drug discovery, Chemistry, DNA, General Medicine, In vitro, Pharmaceutical Preparations, Drug Design, Toxicity, Carcinogenesis, Drug metabolism, Chromatography, Liquid, Protein Binding
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8
المؤلفون: Karen Siegler, Bei Shan, Mark P. Grillo, Marion Conn, Jiang Zhu, Jian Ken Zhang, Yingcai Wang, Julio C. Medina, Ming Yu, Peter Coward, Frank Kayser, Jiwen Jim Liu
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:156-160
مصطلحات موضوعية: Agonist, Sulfonamides, Dose-Response Relationship, Drug, Molecular Structure, Pyridines, medicine.drug_class, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Rats, Receptors, G-Protein-Coupled, Structure-Activity Relationship, GPR119, Drug Discovery, Microsomes, Liver, medicine, Animals, Humans, Molecular Medicine, Molecule, Molecular Biology
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9
المؤلفون: Pierre Deprez, Paul M. Wehn, Jeff D. Reagan, Minghan Wang, Paul E. Harrington, Mark P. Grillo, Kanaka Pattabiraman, James Davis, Charles Henley, Sean Morony, Taoues Temal, Christopher H. Fotsch, Steve F. Poon, Timothy J. Carlson, David J. St. Jean, Sarah E. Lively, Yuhua Yang, Jenny Ying-Lin Lu
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:6625-6628
مصطلحات موضوعية: Male, Calcimimetic, Metabolite, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Rats, Sprague-Dawley, chemistry.chemical_compound, Pharmacokinetics, In vivo, Drug Discovery, medicine, Animals, Urea, Potency, Molecular Biology, CYP3A4, Organic Chemistry, medicine.disease, Rats, Bioavailability, Thiazoles, chemistry, Parathyroid Hormone, Molecular Medicine, Hyperparathyroidism, Secondary, Secondary hyperparathyroidism, Receptors, Calcium-Sensing, Half-Life, Protein Binding
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10
المؤلفون: Mark P. Grillo, Michelle Tadano Lohr, Smriti Khera
المصدر: Drug Metabolism and Disposition. 41:111-121
مصطلحات موضوعية: Dipeptidase, Magnetic Resonance Spectroscopy, Stereochemistry, Pharmaceutical Science, Ibuprofen, In Vitro Techniques, Thioester, chemistry.chemical_compound, Tandem Mass Spectrometry, In vivo, Animals, Humans, Mercapturic acid, Pharmacology, chemistry.chemical_classification, Chromatography, biology, organic chemicals, gamma-Glutamyltransferase, Glutathione, In vitro, Enzyme, chemistry, Glycine, biology.protein, Cattle, Chromatography, Liquid
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11
المؤلفون: Mark P. Grillo, Michelle Tadano Lohr, Jill C. M. Wait
المصدر: Drug Metabolism and Disposition. 40:1515-1526
مصطلحات موضوعية: Mefenamic acid, Carboxylic acid, Acyl glucuronidation, Pharmaceutical Science, In Vitro Techniques, Thioester, Mefenamic Acid, chemistry.chemical_compound, Tandem Mass Spectrometry, In vivo, medicine, Animals, Humans, Biotransformation, Pharmacology, chemistry.chemical_classification, Chemistry, Metabolism, Glutathione, Rats, Biochemistry, Hepatocytes, Glucuronide, Chromatography, Liquid, medicine.drug
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12
المؤلفون: Mark P. Grillo, Jessica S. Houghton, Eskouhie Tchaparian, Craig Uyeda, Lixia Jin
المصدر: Drug Metabolism and Disposition. 39:2387-2394
مصطلحات موضوعية: Male, Pharmacology, Abcg2, Organic anion transporter 1, Reverse Transcriptase Polymerase Chain Reaction, Multidrug resistance-associated protein 2, Pharmaceutical Science, Transporter, Articles, Biology, Molecular biology, In vitro, Rats, Rats, Sprague-Dawley, Pharmaceutical Preparations, In vivo, Cell culture, Gene expression, Hepatocytes, biology.protein, Animals, Carrier Proteins, Cells, Cultured
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13
المؤلفون: Mark P. Grillo, Christian Skonberg, Line Olsen
المصدر: Chemical Research in Toxicology. 24:992-1002
مصطلحات موضوعية: chemistry.chemical_classification, Drug, Kava, Chemistry, media_common.quotation_subject, General Medicine, Glutathione, Exanthema, Pharmacology, Toxicology, Plant Roots, In vitro, Lactones, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, In vivo, Toxicity, Animals, Humans, Pipermethystine, Chemical and Drug Induced Liver Injury, Lactone, media_common
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14
المؤلفون: Zice Fu, Yongli Su, Xuemei Wang, Hua Lucy Tang, Timothy J. Sullivan, Lisa Seitz, Felix Gonzalez-Lopez de Turiso, Julio C. Medina, Mark P. Grillo, Shanna Lawlis, Ying Sun, Wang Shen, M.J. Schmitt, Qiuping Ye, Sarah E. Lively, Matthew L. Brown, An-Rong Li, Yingcai Wang, Bettina Van Lengerich, Jill Wait, Sujen Lai, Jiwen Liu, Michael G. Johnson, Jay Danao, Tassie L. Collins, Qingge Xu
المصدر: ACS Medicinal Chemistry Letters. 2:326-330
مصطلحات موضوعية: business.industry, Organic Chemistry, Antagonist, Prostanoid, Chemotaxis, Pharmacology, Phenylacetic acid, medicine.disease, Biochemistry, chemistry.chemical_compound, chemistry, Drug Discovery, Medicine, Prostaglandin D2, business, Receptor, G protein-coupled receptor, Asthma
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15
المؤلفون: Mark P. Grillo
المصدر: Current Drug Metabolism. 12:229-244
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Stereochemistry, Metabolite, Clinical Biochemistry, Proteins, Glutathione, Sulfides, Thioester, Combinatorial chemistry, chemistry.chemical_compound, Transacylation, chemistry, Biotransformation, Reagent, Electrophile, Animals, Humans, lipids (amino acids, peptides, and proteins), Acyl Coenzyme A, Glucuronide, Protein Binding
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16
المؤلفون: Leslie Z. Benet, Fengmei Hua, Charles G. Knutson, Mark P. Grillo, Kristi L. March, Joseph A. Ware
المصدر: Chemical Research in Toxicology. 21:1933-1938
مصطلحات موضوعية: Diclofenac, Pharmacology, Toxicology, Rats, Sprague-Dawley, chemistry.chemical_compound, Tandem Mass Spectrometry, In vivo, medicine, Extracellular, Animals, Bile, Incubation, chemistry.chemical_classification, Molecular Structure, Substrate (chemistry), Dipeptides, gamma-Glutamyltransferase, General Medicine, Glutathione, In vitro, Rats, Enzyme, chemistry, Biochemistry, medicine.drug
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17
المؤلفون: Fengmei Hua, Mark P. Grillo
المصدر: Chemical Research in Toxicology. 21:1749-1759
مصطلحات موضوعية: Male, Time Factors, Stereochemistry, Metabolite, Acyl glucuronidation, Molecular Conformation, Glucuronidation, Ibuprofen, Sulfuric Acid Esters, Toxicology, Mass Spectrometry, Rats, Sprague-Dawley, chemistry.chemical_compound, Transacylation, medicine, Animals, Pentanoic Acids, Camphanes, Valproic Acid, organic chemicals, Lauric Acids, Stereoisomerism, General Medicine, Glutathione, Metabolism, Lauric acid, Rats, medicine.anatomical_structure, chemistry, Hepatocyte, Hepatocytes, Chromatography, Liquid
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18
المؤلفون: Mark P. Grillo, Yohannes Teffera, Ji Ma, Daniel J. Waldon
المصدر: Drug Metabolism and Disposition. 36:1740-1744
مصطلحات موضوعية: Diclofenac, Stereochemistry, Carboxylic Acids, Pharmaceutical Science, Sulfaphenazole, chemistry.chemical_compound, Cytochrome P-450 Enzyme System, Tandem Mass Spectrometry, medicine, Animals, Oxidative decarboxylation, Pharmacology, biology, Anti-Inflammatory Agents, Non-Steroidal, Cytochrome P450, Glutathione, Metabolism, Rats, chemistry, Enzyme inhibitor, Microsomes, Liver, Microsome, biology.protein, Oxidation-Reduction, Chromatography, Liquid, medicine.drug
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19
المؤلفون: Daniel J. Waldon, P E Sanders, Fengmei Hua, Joseph A. Ware, Charles G. Knutson, Mark P. Grillo
المصدر: Drug Metabolism and Disposition. 31:1327-1336
مصطلحات موضوعية: Male, Diclofenac, Metabolite, Pharmaceutical Science, Rats, Sprague-Dawley, chemistry.chemical_compound, Glucuronides, Transacylation, In vivo, medicine, Animals, Bile, Incubation, Chromatography, High Pressure Liquid, Pharmacology, Chromatography, biology, Chemistry, Glutathione, In vitro, Rats, Biochemistry, Enzyme inhibitor, biology.protein, medicine.drug
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20
المصدر: Drug Metabolism and Disposition. 31:727-730
مصطلحات موضوعية: Male, Time Factors, Stereochemistry, Serum albumin, Pharmaceutical Science, In Vitro Techniques, Thioester, Mass Spectrometry, Rats, Sprague-Dawley, Palmitic acid, chemistry.chemical_compound, Acyl-CoA, Adenosine Triphosphate, medicine, Animals, Humans, Biotransformation, Chromatography, High Pressure Liquid, Serum Albumin, Pharmacology, chemistry.chemical_classification, Phenylpropionates, biology, Chemistry, Metabolism, Human serum albumin, Rats, Liver, Biochemistry, Enzyme inhibitor, Covalent bond, biology.protein, Acyl Coenzyme A, Protein Binding, medicine.drug