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1Imatinib does not induce cardiotoxicity at clinically relevant concentrations in preclinical studies
المؤلفون: Francois Pognan, Min Dong, Armin Wolf, Ursula Junker, Jeffrey Tsao, David Ledieu, Ulrich W. Laengle, Danielle Roman, Anja Nussher, Olivier Grenet, Christian Trendelenburg, Gilles-Jacques Riviere, Philippe Couttet, Estelle Marrer, Elke Persohn, Marcia Heron, Daniel Robert Roth
المصدر: Leukemia Research. 34:1180-1188
مصطلحات موضوعية: Male, Cancer Research, medicine.medical_specialty, Cmax, Antineoplastic Agents, Pharmacology, Polymerase Chain Reaction, Piperazines, Mice, hemic and lymphatic diseases, Internal medicine, medicine, Animals, Cytotoxic T cell, Rats, Wistar, neoplasms, DNA Primers, Cardiotoxicity, Base Sequence, business.industry, Endoplasmic reticulum, Heart, Imatinib, Hematology, medicine.disease, Rats, Mice, Inbred C57BL, Pyrimidines, Endocrinology, Imatinib mesylate, Oncology, Apoptosis, Heart failure, Benzamides, Imatinib Mesylate, business, medicine.drug
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2
المؤلفون: Francois Pognan, Elke Persohn, Estelle Marrer, Wei Zhou, Philippe Couttet, Marcia Heron, Ursula Junker, Olivier Grenet, Armin Wolf, David Ledieu, Jeffrey Tsao, Danielle Roman, Andreas Mahl, Min Dong
المصدر: Leukemia research. 35(5)
مصطلحات موضوعية: Male, Cancer Research, medicine.medical_specialty, medicine.drug_class, Heart Ventricles, Drug Evaluation, Preclinical, Pharmacology, Cardiotoxins, Tyrosine-kinase inhibitor, Rats, Sprague-Dawley, Random Allocation, In vivo, Internal medicine, medicine, Animals, Ventricular Function, Myocytes, Cardiac, Rats, Wistar, Cells, Cultured, Cardiotoxicity, Dose-Response Relationship, Drug, business.industry, Heart, Hematology, medicine.disease, Cardiovascular physiology, Rats, Endocrinology, Pyrimidines, Oncology, Nilotinib, Animals, Newborn, Apoptosis, Heart failure, Toxicity, business, medicine.drug
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3Academic Journal
المؤلفون: Daniel P. Becker, Thomas E. Barta, Louis J. Bedell, Terri L. Boehm, Brian R. Bond, Jeffery Carroll, Chris P. Carron, Gary A. DeCrescenzo, Alan M. Easton, John N. Freskos, Chris L. Funckes-Shippy, Marcia Heron, Susan Hockerman, Carol Pearcy Howard, James R. Kiefer, Madeleine H. Li, Karl J. Mathis, Joseph J. McDonald, Pramod P. Mehta, Grace E. Munie
المصدر: Journal of Medicinal Chemistry; Sep2010, Vol. 53 Issue 18, p6653-6680, 28p